methysergide and ketanserin
methysergide has been researched along with ketanserin in 200 studies
Research
Studies (200)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 83 (41.50) | 18.7374 |
1990's | 88 (44.00) | 18.2507 |
2000's | 23 (11.50) | 29.6817 |
2010's | 6 (3.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Bull, D; den Daas, I; Foord, S; Goodson, S; Kilpatrick, G; Lee, M; Rees, S | 1 |
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J | 1 |
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR | 1 |
Amlaiky, N; Hen, R; Plassat, JL | 1 |
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R | 1 |
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP | 1 |
Baez, M; Kursar, JD; Lucaites, VL; Nelson, DL; Sasso, DA; Wainscott, DB | 1 |
Egan, CT; Herrick-Davis, K; Teitler, M | 1 |
Bach, T; Krobert, KA; Kvingedal, AM; Levy, FO; Syversveen, T | 1 |
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Hisa, H; Satoh, S; Takahashi, T | 2 |
Gretler, DD; Jones, KC; Murphy, MB | 1 |
Gürdal, H; Onaran, HO; Tulunay, FC | 1 |
Cassuto, J; Jodal, M; Lundgren, O; Sjöqvist, A | 1 |
Contesse, V; Delarue, C; Feuilloley, M; Grise, P; Hery, F; Lefebvre, H; Raynaud, G; Vaudry, H; Verhofstad, AA; Wolf, LM | 1 |
Jørgensen, H; Knigge, U; Warberg, J | 2 |
Miletic, V; Tan, H | 1 |
Fuji, K; Hiramatsu, M; Kameyama, T; Nabeshima, T; Niwa, K | 1 |
Dhasmana, KM; Saxena, PR; Tadipatri, S; Villalón, CM; Zhu, YN | 1 |
Goda, Y; Matsumoto, M; Saito, H; Togashi, H; Yoshioka, M | 1 |
Giordano, J; Schomburg, FM; Sufka, KJ | 1 |
Egashira, K; Hayashi, Y; Nakamura, M; Takeshita, A; Tomoike, H; Yamada, A | 1 |
Alhaider, AA; Mustafa, AA | 1 |
Johnson, JH; Kitts, CS | 2 |
Alhaider, AA | 1 |
Sahin-Erdemli, I; Uma, S | 1 |
Baimbridge, KG; Klancnik, JM; Obenaus, A; Phillips, AG | 1 |
Dhawan, BN; Kumar, A; Raghubir, R | 1 |
Beczkowska, IW; Bodnar, RJ | 1 |
Hyman, PE; Jing, J; Ng, WW; Snape, WJ | 1 |
Horisaka, K; Sugimoto, Y; Yamada, J | 2 |
Danzebrink, RM; Gebhart, GF | 1 |
Bueno, L; Fargeas, MJ; Fioramonti, J; Theodorou, V | 1 |
Arzt, E; Costas, M; Finkielman, S; Nahmod, VE | 1 |
Benito, JM; Conde, MV; Fraile, ML; López de Pablo, AL; Marco, EJ; Moreno, MJ; Sanz, ML | 1 |
Bunce, KT; Burridge, J; Butler, A; Elswood, CJ; Ireland, SJ; Kilpatrick, GJ; Tyers, MB | 1 |
Dewar, KM; Lima, L; Reader, TA | 1 |
Deshpande, SB; Warnick, JE | 1 |
Jackson, DA; White, SR | 1 |
Kamei, J; Kasuya, Y; Tanihara, H | 1 |
Li Volsi, G; Licata, F; Maugeri, G; Santangelo, F | 1 |
Salonen, RO; Webber, SE; Widdicombe, JG | 1 |
Okamura, T; Toda, N | 1 |
Woodman, OL | 1 |
Boeckxstaens, GE; Bogers, JJ; Herman, AG; Pelckmans, PA; Rampart, M; Van Maercke, YM; Verbeuren, TJ | 1 |
Sakurai, Y; Wenk, GL | 1 |
Campbell, AM; Glatfelter, A; Kunkel, RG; Ulevitch, RJ; Wiggins, RC | 1 |
Braimbridge, MV; Erol, C; Hearse, DJ; Maxwell, MP; Saldanha, C; Sonmez, B | 1 |
Kaumann, AJ | 1 |
Dall'Olio, R; Gandolfi, O; Roncada, P | 1 |
Awano, K; Fukuzaki, H; Yokoyama, M | 1 |
DeNoble, VJ; Spencer, KR; Strek, KF | 1 |
Abe, Y; Fukui, K; Iwao, H; Shoji, T; Tamaki, T | 1 |
Bodnar, RJ; Kiefel, JM; Paul, D | 1 |
Horisaka, K; Kimura, I; Sugimoto, Y; Takeuchi, N; Yamada, J | 1 |
Chalmers, JP; Mills, EH; Minson, JB | 1 |
Marín, J; Reviriego, J | 1 |
Hashiba, Y; Ishikawa, N; Satake, T; Sumita, T; Takagi, K | 1 |
Acevedo, CG; Cruz, MA; Gonzalez, C; Rudolph, MI; Sepulveda, WH | 1 |
Alexander, BS; Broadhurst, AM; Wood, MD | 1 |
Costall, B; Gunning, SJ; Naylor, RJ; Tattersall, FD | 1 |
Chiba, S; Sinanović, O | 1 |
Krootila, K; Palkama, A; Uusitalo, H | 1 |
Marek, GJ; Seiden, LS | 1 |
Hewson, G; Hill, RG; Hughes, J; Leighton, GE | 1 |
Ramage, AG | 1 |
Heiligers, J; Mylecharane, EJ; Saxena, PR | 1 |
Janssens, WJ; Van Nueten, JM; Vanhoutte, PM | 1 |
Grekin, RJ; Gross, MD; Shenker, Y | 1 |
Barrett, JE; Brady, LS | 1 |
Lawang, A; Saxena, PR | 1 |
Barrett, JE; Mansbach, RS | 1 |
Connor, HE; Feniuk, W; Humphrey, PP; Perren, MJ | 1 |
Armstrong, ML; Heistad, DD; Marcus, ML; Mark, AL; Piegors, DJ | 1 |
Ferrara, A; Jaffe, BM; Sherlock, DJ | 1 |
Leff, P; Martin, GR | 1 |
Kaumann, AJ; Lemoine, H | 1 |
Knigge, U; Matzen, S; Sleimann, I; Warberg, J | 1 |
Candeletti, S; Ferri, S; Romualdi, P; Spadaro, C; Spampinato, S | 1 |
Kayaalp, SO; Onur, R; Sahin, I; Tuncer, M | 1 |
Blackshear, JL; Hollenberg, NK; Orlandi, C | 1 |
Jandhyala, BS; Kivlighn, SD | 1 |
Barrett, JE; Brady, LS; Witkin, JM | 1 |
Frenken, M; Kaumann, AJ | 3 |
Hole, DR; Hunter, AJ; Wilson, CA | 1 |
Karasawa, A; Kubo, K; Nakamizo, N; Shuto, K | 1 |
Bradley, PB; Humphrey, PP; Williams, RH | 1 |
Heiligers, J; Mylecharane, EJ; Saxena, PR; Tio, R | 1 |
Clarke, KA; Parker, AJ; Stirk, GC | 1 |
Gorzalka, BB; Mendelson, SD | 1 |
Kilbinger, H; Pfeuffer-Friederich, I | 1 |
Burvenich, C; Peeters, G; Vandeputte-Van Messon, G | 1 |
Lin, MT; Won, SJ | 1 |
Connell, LA; Wallis, DI | 1 |
Kannisto, P; Owman, C; Schmidt, G; Sjöberg, NO | 1 |
Davies, M; Roberts, MH; Wilkinson, LS | 1 |
Baird, AW; Cuthbert, AW | 1 |
Emmers, R; Tamir, H; Wilchek, M | 1 |
Furukawa, H; Ishikawa, K; Kameyama, T; Nabeshima, T; Yamaguchi, K | 1 |
Hasegawa, M; Kanaide, H; Kobayashi, S; Nakamura, M | 1 |
de Vries, C; Parmentier, HK; Ruitenberg, EJ; Van Loveren, H | 1 |
Chiba, S; Tsuji, T | 1 |
Clancy, BM; Maayani, S; Osman, R | 1 |
Chu, A; Cobb, FR | 1 |
Kayaalp, SO; Tuncer, M; Uma, S | 1 |
Ishikawa, N; Kamiya, I; Sumita, T | 1 |
Hørby-Petersen, J; Klarskov, P | 1 |
Penington, NJ; Reiffenstein, RJ | 1 |
Johnson, JH; Lenahan, SE; Seibel, HR | 1 |
Edwards, CR; Shaikh, S; Williams, BC | 1 |
Arnold, R; Koop, H | 1 |
Humphrey, PP | 1 |
Van Nueten, JM | 1 |
Eyre, P; Ogunbiyi, PO | 2 |
Feniuk, W | 1 |
Anthony, M | 1 |
Finch, CE; Marcusson, JO; Morgan, DG; Winblad, B | 1 |
Freedman, M; Hamel, L; Luttinger, D; Perrone, M; Ward, SJ | 1 |
Taylor, DA; Yap, CY | 1 |
Janssen, PA; Van Beek, J; Van Nueten, JM | 1 |
Cohen, RA; Shepherd, JT; Vanhoutte, PM | 1 |
Frazer, A; Lucki, I; Nobler, MS | 1 |
Hong, E; Mena, MA; Rión, R | 1 |
de Gaetano, G; Lampugnani, MG | 1 |
Björklund, M; Jäkälä, P; Kaukua, J; Koivisto, E; Riekkinen, P; Sirviö, J | 1 |
Li, S; Pelletier, G | 1 |
Gu, Q; Singer, W | 1 |
Egashira, S; Hayashi, Y; Kuga, T; Mitsuoka, W; Nakamura, M; Tagawa, H; Takeshita, A; Tomoike, H; Yamada, A | 1 |
Dallaire, MJ; Fukuchi, Y; Ludwig, MS; Martin, JG; Nagase, T | 1 |
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI | 1 |
García-Colunga, J; Miledi, R | 1 |
Chiba, S; Vhora, S | 1 |
Hansen, MB; Skadhauge, E | 1 |
Beubler, E; Hansen, MB; Skadhauge, E; Thørboll, JE | 1 |
Garcia de Yebenes, E; Li, S; Pelletier, G | 1 |
Sillar, KT; Wedderburn, JF | 1 |
Camilleri, M; Kost, LJ; Oosterbosch, L; Phillips, SF; Valdovinos, MA; von der Ohe, M | 1 |
Wallis, DI; Wang, XC; Wu, J | 1 |
Horisaka, K; Kimura, I; Sugimoto, Y; Watanabe, Y; Yamada, J | 1 |
Hansen, MB; Jaffe, BM | 1 |
Bach, FW; Iversen, H; Knigge, U; Matzen, S; Pawelczyk, J; Perko, G; Secher, NH; Warberg, J | 1 |
Cholewinski, A; Fitzgibbon, F; Leslie, R; Liu, NP; Nash, M; Osborne, NN | 1 |
Chemineau, P; Le Corre, S | 1 |
Lacosta, S; Roberts, DC | 1 |
Chiba, S; Nakane, T; Noguchi, M | 1 |
Horisaka, K; Kimura, I; Sugimoto, Y; Takeuchi, N; Watanabe, Y; Yamada, J | 1 |
Hamada, S; Hamaguchi, K; Mikuni, M; Niitsu, Y; Okado, N | 1 |
Gidener, S; Güven, H; Kirkali, Z | 1 |
Lacey, MG; Rick, CE; Stanford, IM | 1 |
Becú-Villalobos, D; Lacau-Mengido, IM; Libertun, C | 1 |
Ito, H; Kamato, T; Miyata, K; Nagakura, Y; Nishida, A; Yamano, M | 1 |
Bazzani, C; Bertolini, A; Ferrante, F; Fiore, L; Guarini, S | 1 |
Choi, DS; Launay, JM; Maroteaux, L; Messaddeq, N; Ward, SJ | 1 |
Jäkälä, P; MacDonald, E; Puumala, T; Riekkinen, P; Ruotsalainen, S; Sirviö, J | 1 |
Itoh, Z; Mizumoto, A; Nakajima, M; Sakai, T; Sano, I; Shiba, Y; Shiihara, Y | 1 |
Herges, S; Taylor, DA | 1 |
De Leyn, P; Demedts, MG; Deneffe, G; Dupont, LJ; Pype, JL; Verleden, GM | 1 |
Sugimoto, Y; Yamada, J; Yoshikawa, T | 1 |
Takagi, J; Yonehara, N | 1 |
Aloyo, VJ; Harvey, JA; Hoffman, ME; Salt, GL | 1 |
Avanzi, V; Brandão, ML; Castilho, VM | 1 |
Kaibara, M; Mameya, S; Takada, K; Takemura, K; Taniyama, K | 1 |
Bult, H; Geerts, IS; Herman, AG; Matthys, KE | 1 |
Bisgard, GE; Herman, JK; Mitchell, GS; O'Halloran, KD | 1 |
Placantonakis, DG; Schwarz, C; Welsh, JP | 1 |
Dall'Olio, R; Gaggi, R; Gandolfi, O | 1 |
Bisgard, GE; Herman, JK; O'Halloran, KD | 1 |
Bytautiene, E; Garfield, RE; Marshall, JS; Romero, R; Vedernikov, YP | 1 |
Goto, T; Ochi, T | 1 |
Castro-Souza, C; Coimbra, NC; Garcia-Cairasco, N; Herrero, CF; Nora, JE; Segato, EN; Tedeschi-Filho, W | 1 |
Fozard, JR; Hannon, JP; Mazzoni, L; Tigani, B; Williams, I | 1 |
Hunt, WK; Morrison, AR; Pack, AI; Ross, RJ; Sanford, LD | 1 |
Brandão, ML; Castilho, VM | 1 |
Gebhard, MM; Martin, E; Peter, C; Schmidt, H; Secchi, A; Walther, A | 1 |
Danuser, H; Hauser, DS; Mevissen, M; Portier, CJ; Scholtysik, G; Studer, UE; Weiss, R | 1 |
Collins, JG; Kawamata, M; Koshizaki, M; Saito, Y; Shimada, SG | 1 |
Ling, L; McGuire, M; White, DP; Zhang, Y | 1 |
Adaikan, GP; Adebiyi, A; Prasad, RN | 1 |
Coimbra, NC; Freitas, RL; Kishi, R; Morato, S; Rebouças, EC; Savoldi, M; Segato, EN | 1 |
Centurión, D; Gupta, S; MaassenVanDenBrink, A; Mehotra, S; Sánchez-López, A; Villalón, CM | 1 |
Komada, T; Yano, S | 1 |
Harris, MB; Kober, AM; Leiter, JC; St-John, WM; Toppin, VA | 1 |
Czabanka, M; Martin, E; Peter, C; Petri, E; Walther, A | 1 |
Leiter, JC; St-John, WM | 1 |
Foley, KT; Henderson, DR; Mitchell, GS; Turner, DL | 1 |
Feistel, B; Heimes, K; Verspohl, EJ | 1 |
Gilmour, KM; McDonald, MD; Perry, SF; Walsh, PJ | 1 |
Del Bel, EA; Dias, QM; Prado, WA; Silveira, JW | 1 |
Fedin, AN; Kirilina, VM; Krivchenko, AI; Postnikova, TIu | 1 |
Barchini, J; Jabbur, SJ; Linderoth, B; Meyerson, BA; Saadé, NE; Shamaa, F; Song, Z; Tchachaghian, S | 1 |
Devaud, JM; Farina, WM; Fernández, VM; Giurfa, M | 1 |
Selli, C; Tosun, M | 1 |
Reviews
5 review(s) available for methysergide and ketanserin
Article | Year |
---|---|
Serotonin and vascular reactivity.
Topics: Animals; Blood Platelets; Calcium; Cold Temperature; Electric Stimulation; Hypoxia; Ketanserin; Lidoflazine; Methiothepin; Methysergide; Microcirculation; Models, Biological; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Receptors, Serotonin; Regional Blood Flow; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation | 1985 |
Peripheral 5-hydroxytryptamine receptors and their classification.
Topics: Animals; Dogs; Guinea Pigs; In Vitro Techniques; Ketanserin; Methysergide; Muscle Relaxation; Muscle, Smooth; Neurotransmitter Agents; Piperidines; Rabbits; Rats; Receptors, Serotonin | 1984 |
5-hydroxytryptamine and precapillary vessels.
Topics: Angiotensin II; Animals; Dinoprost; Drug Interactions; Histamine; Ketanserin; Methysergide; Norepinephrine; Piperidines; Prostaglandins F; Receptors, Adrenergic, alpha; Serotonin; Vasoconstriction | 1983 |
An analysis of 5-hydroxytryptamine receptors mediating contraction of isolated smooth muscle.
Topics: Animals; Binding, Competitive; Cats; Cyproheptadine; Dogs; In Vitro Techniques; Ketanserin; Methoxamine; Methysergide; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Piperidines; Rabbits; Rats; Receptors, Serotonin | 1984 |
Serotonin antagonists.
Topics: Cyproheptadine; Depression; Ergotamine; Humans; Hypertension; Ketanserin; Lisuride; Methysergide; Mianserin; Migraine Disorders; Piperidines; Pizotyline; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Diseases | 1984 |
Other Studies
195 other study(ies) available for methysergide and ketanserin
Article | Year |
---|---|
Cloning and characterisation of the human 5-HT5A serotonin receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Genome, Human; GTP-Binding Proteins; Humans; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Serotonin; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid; Serotonin; Tissue Distribution; Transfection | 1994 |
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.
Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction | 1993 |
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection | 1993 |
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Cyclic AMP; DNA; Drosophila; Enzyme Activation; Humans; Intestinal Mucosa; Mice; Molecular Sequence Data; Myocardium; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists | 1993 |
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents | 1996 |
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid | 1997 |
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.
Topics: Adrenergic alpha-Antagonists; Benzofurans; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Imidazoles; Radioligand Assay; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Yohimbine | 1998 |
Creation of a constitutively activated state of the 5-hydroxytryptamine2A receptor by site-directed mutagenesis: inverse agonist activity of antipsychotic drugs.
Topics: Animals; Antipsychotic Agents; COS Cells; Mutagenesis, Site-Directed; Phosphatidylinositols; Protein Conformation; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship | 1998 |
The cloned human 5-HT7 receptor splice variants: a comparative characterization of their pharmacology, function and distribution.
Topics: Adenylyl Cyclases; Alternative Splicing; Binding, Competitive; Brain; Cell Line; Cloning, Organism; Genetic Variation; Humans; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tissue Distribution | 2001 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Serotonin-induced vasoconstriction in dog kidney.
Topics: Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Dogs; Female; Gallic Acid; Indoles; Ketanserin; Kidney; Male; Methysergide; Renal Artery; Renal Circulation; Serotonin; Serotonin Antagonists; Tropisetron; Vasoconstriction | 1992 |
5-Hydroxytryptamine receptor activity of the dopamine receptor agonist fenoldopam in canine tracheal smooth muscle.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Atropine; Benzazepines; Dogs; Dopamine Agents; Drug Interactions; Fenoldopam; In Vitro Techniques; Indomethacin; Ketanserin; Methysergide; Muscle, Smooth; Receptors, Serotonin; Serotonin; Trachea; Vasodilator Agents | 1992 |
Role of alpha-adrenoceptors in the effects of buspirone and 5-carboxamidotryptamine in rabbit isolated thoracic aorta.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Buspirone; Cystamine; Dose-Response Relationship, Drug; Drug Interactions; Ketanserin; Methysergide; Phenylephrine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin; Vasoconstriction | 1992 |
Actions of serotonin antagonists on cholera-toxin-induced intestinal fluid secretion.
Topics: Animals; Body Fluids; Cholera Toxin; Female; Granisetron; Imidazoles; Indazoles; Intestinal Mucosa; Ketanserin; Lysergic Acid Diethylamide; Male; Methysergide; Ondansetron; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Zimeldine | 1992 |
Serotonin-induced stimulation of cortisol secretion from human adrenocortical tissue is mediated through activation of a serotonin4 receptor subtype.
Topics: Adrenal Cortex; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Hydrocortisone; Hydroxyindoleacetic Acid; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Radioimmunoassay; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron | 1992 |
Involvement of 5-HT1, 5-HT2, and 5-HT3 receptors in the mediation of the prolactin response to serotonin and 5-hydroxytryptophan.
Topics: 5-Hydroxytryptophan; Animals; Dose-Response Relationship, Drug; Ergolines; Fluoxetine; Imidazoles; Indoles; Ketanserin; Male; Methysergide; Ondansetron; Prolactin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron | 1992 |
Effect of serotonin 5-HT1, 5-HT2, and 5-HT3 receptor antagonists on the prolactin response to restraint and ether stress.
Topics: Animals; Ergolines; Ether; Indoles; Ketanserin; Male; Methysergide; Ondansetron; Prolactin; Rats; Rats, Wistar; Restraint, Physical; Serotonin Antagonists; Stress, Physiological; Tropisetron | 1992 |
Diverse actions of 5-hydroxytryptamine on frog spinal dorsal horn neurons in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dioxanes; Electric Stimulation; Evoked Potentials; Female; In Vitro Techniques; Ketanserin; Kinetics; Male; Membrane Potentials; Methysergide; Mianserin; Neurons; Rana pipiens; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Synapses; Tetrodotoxin; Tropanes | 1992 |
Effect of naftidrofuryl oxalate on 5-HT2 receptors in mouse brain: evaluation based on quantitative autoradiography and head-twitch response.
Topics: 5-Hydroxytryptophan; Animals; Autoradiography; Behavior, Animal; Binding Sites; Brain Chemistry; Dose-Response Relationship, Drug; Ketanserin; Male; Methysergide; Mice; Nafronyl; Pargyline; Receptors, Serotonin; Ritanserin; Tissue Distribution | 1992 |
Role of 5-HT1-like receptors in the increase in intragastric pressure induced by 5-hydroxytryptamine in the rat.
Topics: Animals; Atropine; Catecholamines; Female; Indoles; Ketanserin; Male; Methiothepin; Methysergide; Pressure; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Stomach; Tropisetron | 1992 |
Pharmacological characterization of 5-hydroxytryptamine-induced apnea in the rat.
Topics: Anesthesia; Animals; Apnea; Bronchoconstriction; Drug Interactions; Imidazoles; Ketanserin; Male; Methysergide; Ondansetron; Phrenic Nerve; Rats; Rats, Inbred Strains; Respiration; Respiratory Function Tests; Serotonin; Serotonin Antagonists; Vagotomy | 1992 |
Receptor mediation of 5-HT-induced inflammation and nociception in rats.
Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Imidazoles; Inflammation; Ketanserin; Male; Methysergide; Ondansetron; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1992 |
Mechanism of ergonovine-induced hyperconstriction of the large epicardial coronary artery in conscious dogs a month after arterial injury.
Topics: Animals; Blood Pressure; Coronary Circulation; Coronary Vasospasm; Coronary Vessels; Diltiazem; Dogs; Electrophysiology; Endothelium, Vascular; Ergonovine; Heart Rate; Indomethacin; Ketanserin; Methysergide; Phenylephrine; Prazosin; Receptors, Serotonin | 1992 |
Enhancement of imipramine-induced rat brain beta-adrenoreceptor desensitization by subacute co-administration of trazodone, zimelidine, quipazine or 5-hydroxytryptophan.
Topics: 5-Hydroxytryptophan; Animals; Brain Chemistry; Drinking Behavior; Female; Fenclonine; Imipramine; Isoproterenol; Ketanserin; Methysergide; Propranolol; Quipazine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Serotonin Antagonists; Trazodone; Zimeldine | 1991 |
Analysis of neurotransmitter receptors mediating changes in LH release induced by electrical stimulation of the dorsal raphe nucleus in the rat.
Topics: Animals; Brain; Electric Stimulation; Estradiol; Female; Ketanserin; Kinetics; Luteinizing Hormone; Metergoline; Methysergide; Naltrexone; Organ Specificity; Ovariectomy; Phenoxybenzamine; Raphe Nuclei; Rats; Receptors, Neurotransmitter; Time Factors | 1991 |
Antinociceptive effect of ketanserin in mice: involvement of supraspinal 5-HT2 receptors in nociceptive transmission.
Topics: Acetates; Acetic Acid; Adrenergic alpha-Antagonists; Analgesics; Animals; Brain Chemistry; Dioxanes; Dopamine; Idazoxan; Ketanserin; Male; Methysergide; Mice; Norepinephrine; Pain; Reaction Time; Receptors, Serotonin; Serotonin; Synaptic Transmission | 1991 |
Receptors mediating the contractile effect of serotonin (5-HT) in the isolated common bile duct of guinea-pig.
Topics: Animals; Atropine; Common Bile Duct; Dose-Response Relationship, Drug; Female; Guinea Pigs; Ketanserin; Male; Methysergide; Muscle Contraction; Receptors, Serotonin; Serotonin | 1991 |
The effects of serotonergic compounds on evoked responses in the dentate gyrus and CA1 region of the hippocampal formation of the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Ketanserin; Male; Methysergide; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes | 1991 |
Effect of monoamine antagonists on pretectal evoked analgesia in rat.
Topics: Analgesia; Animals; Biogenic Monoamines; Electric Stimulation; Haloperidol; Ketanserin; Methysergide; Phenoxybenzamine; Rats; Serotonin Antagonists; Sotalol | 1991 |
Serotonin-induced renin release in the dog kidney.
Topics: Anesthesia; Animals; Blood Pressure; Cyclooxygenase Inhibitors; Dogs; Female; Heart Rate; Indomethacin; Infusions, Intra-Arterial; Ketanserin; Kidney; Male; Methysergide; Norepinephrine; Renal Circulation; Renin; Serotonin | 1991 |
Naloxone and serotonin receptor subtype antagonists: interactive effects upon deprivation-induced intake.
Topics: Animals; Drug Interactions; Feeding Behavior; Food Deprivation; Indoles; Ketanserin; Male; Methysergide; Naloxone; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Tropisetron | 1991 |
Effect of 5-hydroxytryptamine and its antagonists on colonic smooth muscle of the rabbit.
Topics: Animals; Atropine; Colon; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Indoles; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Rabbits; Serotonin; Serotonin Antagonists; Tetrodotoxin; Tropisetron | 1991 |
Activation of peripheral serotonin2 receptors induces hypothermia in mice.
Topics: Animals; Body Temperature Regulation; Hypothermia; Ketanserin; Methysergide; Mice; Mice, Inbred ICR; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1991 |
Evidence that spinal 5-HT1, 5-HT2 and 5-HT3 receptor subtypes modulate responses to noxious colorectal distension in the rat.
Topics: Amidines; Animals; Blood Pressure; Colon; Indoles; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Muscles; Pressure; Rats; Rats, Inbred Strains; Receptors, Serotonin; Rectum; Reflex; Serotonin Antagonists; Spinal Cord; Tropanes; Tropisetron | 1991 |
Involvement of 5-hydroxytryptamine in the intestinal motor disturbances induced by mast cell degranulation in rats.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Duodenum; Gastrointestinal Motility; Indoles; Jejunum; Ketanserin; Lasalocid; Male; Mast Cells; Methysergide; p-Methoxy-N-methylphenethylamine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron | 1991 |
Serotonin inhibition of tumor necrosis factor-alpha synthesis by human monocytes.
Topics: Humans; Ketanserin; Methysergide; Monocytes; Receptors, Serotonin; Serotonin; Tumor Necrosis Factor-alpha | 1991 |
Response of isolated cat middle cerebral artery to platelets: effect of endothelium removal.
Topics: Animals; Blood Platelets; Cats; Cerebral Arteries; Cyproheptadine; Endothelium, Vascular; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth, Vascular; Serotonin | 1991 |
The pharmacological characterization of 5-HT3 receptors in three isolated preparations derived from guinea-pig tissues.
Topics: Animals; Colon; Female; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Kinetics; Male; Methysergide; Receptors, Serotonin; Serotonin; Vagus Nerve | 1990 |
[3H]ketanserin binds to non-5-HT2 sites in rabbit cerebral cortex and neostriatum.
Topics: Animals; Binding, Competitive; Caudate Nucleus; Cell Membrane; Cerebral Cortex; Corpus Striatum; Frontal Lobe; Ketanserin; Kinetics; Male; Methysergide; Mianserin; Piperidines; Putamen; Rabbits; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Interaction of thyrotropin-releasing hormone and methysergide on the monosynaptic reflex in isolated mammalian spinal cord.
Topics: 5,7-Dihydroxytryptamine; Animals; Animals, Newborn; Cyproheptadine; Drug Interactions; In Vitro Techniques; Indoles; Ketanserin; Male; Methysergide; Rats; Rats, Inbred Strains; Reflex; Serotonin Antagonists; Spinal Cord; Spiperone; Synapses; Thyrotropin-Releasing Hormone; Tropisetron | 1990 |
Receptor subtypes mediating facilitation by serotonin of excitability of spinal motoneurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; In Vitro Techniques; Injections, Intravenous; Iontophoresis; Ketanserin; Male; Methysergide; Microelectrodes; Motor Neurons; Piperidines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes | 1990 |
Antitussive effects of two specific kappa-opioid agonists, U-50,488H and U-62,066E, in rats.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Antitussive Agents; Cisterna Magna; Cough; Injections; Ketanserin; Male; Methysergide; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rats; Rats, Inbred Strains; Reflex | 1990 |
Effects of 5-hydroxytryptamine on the firing rates of neurons of the lateral vestibular nucleus in the rat.
Topics: Action Potentials; Animals; Ketanserin; Male; Metergoline; Methysergide; Rats; Rats, Inbred Strains; Serotonin; Vestibular Nuclei | 1990 |
Receptors mediating the effects of 5-hydroxytryptamine on the tracheal vasculature and smooth muscle of sheep.
Topics: Animals; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle Tonus; Muscle, Smooth; Perfusion; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sheep; Trachea | 1990 |
Comparison of the response to 5-carboxamidotryptamine and serotonin in isolated human, monkey and dog coronary arteries.
Topics: Animals; Coronary Vessels; Dogs; Drug Interactions; Female; Humans; Ketanserin; Macaca; Male; Methysergide; Muscle, Smooth, Vascular; Serotonin; Serotonin Antagonists; Species Specificity; Vasoconstriction | 1990 |
Enhanced coronary vasoconstrictor responses to 5-hydroxytryptamine in the presence of a coronary artery stenosis in anaesthetized dogs.
Topics: Anesthesia; Animals; Coronary Circulation; Coronary Disease; Coronary Vessels; Dogs; Electrocardiography; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Serotonin; Serotonin Antagonists; Vasoconstriction | 1990 |
Pharmacological characterization of 5-hydroxytryptamine receptors in the canine terminal ileum and ileocolonic junction.
Topics: Animals; Colon; Culture Techniques; Dogs; Female; Ileum; Indoles; Intestinal Mucosa; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron | 1990 |
The interaction of acetylcholinergic and serotonergic neural systems on performance in a continuous non-matching to sample task.
Topics: Acetylcholine; Acoustic Stimulation; Animals; Brain; Discrimination, Psychological; Ketanserin; Male; Memory; Methysergide; Neurons; p-Chloroamphetamine; Photic Stimulation; Rats; Reinforcement, Psychology; Serotonin | 1990 |
Acute hypotension due to platelet serotonin-induced chemoreflexes after intravenous injection of dextran sulfate in the rabbit.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Autonomic Nervous System; Blood Platelets; Bradycardia; Chemoreceptor Cells; Cimetidine; Complement C3; Dextran Sulfate; Dextrans; Factor XII; Histamine; Histamine Release; Hypotension; Injections, Intravenous; Ketanserin; Leukocyte Count; Lung; Male; Methysergide; Piperidines; Rabbits; Serotonin | 1985 |
Particle-induced coronary vasoconstriction in the rat heart: pharmacological investigation of underlying mechanisms.
Topics: Animals; Bicarbonates; Calcium Chloride; Cimetidine; Coronary Circulation; Drug Contamination; Filtration; Heart Arrest, Induced; Isoproterenol; Ketanserin; Magnesium; Male; Methysergide; Phenylephrine; Potassium Chloride; Pyrilamine; Rats; Rats, Inbred Strains; Serotonin; Sodium Chloride | 1986 |
A two-state model for the 5-HT2 receptor: effects of alpha-adrenoceptor ligands.
Topics: Animals; Binding, Competitive; Cattle; Coronary Vessels; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth, Vascular; Phenethylamines; Phentolamine; Receptors, Adrenergic; Receptors, Serotonin; Serotonin; Tetralones | 1988 |
Single or repeated administrations of SCH 23390 fail to affect serotonergic neurotransmission.
Topics: Animals; Benzazepines; Dose-Response Relationship, Drug; Frontal Lobe; Hydroxyindoleacetic Acid; Ketanserin; Male; Methysergide; Mianserin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Synaptic Transmission; Synaptosomes | 1988 |
Role of serotonin, histamine, and thromboxane A2 in platelet-induced contractions of coronary arteries and aortae from rabbits.
Topics: Animals; Aorta, Thoracic; Aspirin; Blood Platelets; Coronary Vessels; Diphenhydramine; Endothelium, Vascular; Female; Histamine; In Vitro Techniques; Isometric Contraction; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Rabbits; Serotonin; Thromboxane A2 | 1989 |
Manipulation of serotonin protects against an hypoxia-induced deficit of a passive avoidance response in rats.
Topics: Animals; Avoidance Learning; Cyproheptadine; Dose-Response Relationship, Drug; Fluoxetine; Hypoxia; Ketanserin; Male; Methysergide; Mianserin; Rats; Rats, Inbred Strains; Serotonin; Zimeldine | 1989 |
Renal hemodynamic responses to 5-hydroxytryptamine (5-HT): involvement of the 5-HT receptor subtypes in the canine kidney.
Topics: Adrenergic alpha-Antagonists; Animals; Dogs; Female; Ketanserin; Kidney; Male; Methysergide; Prazosin; Receptors, Serotonin; Renal Circulation; Renin; Serotonin | 1989 |
Reduction in opioid and non-opioid forms of swim analgesia by 5-HT2 receptor antagonists.
Topics: Analgesia; Endorphins; Ketanserin; Methysergide; Physical Exertion; Piperidines; Receptors, Serotonin; Serotonin Antagonists | 1989 |
The evidence for the involvement of the 5-HT1A receptor in 5-HT syndrome induced in mice by tryptamine.
Topics: Animals; Behavior, Animal; Haloperidol; Ketanserin; Male; Methysergide; Mice; Mice, Inbred DBA; Propranolol; Receptors, Serotonin; Serotonin; Spiperone; Tryptamines | 1989 |
Serotonin-induced hypoglycemia and increased serum insulin levels in mice.
Topics: Animals; Blood Glucose; Hypoglycemia; Indoles; Insulin; Ketanserin; Male; Methysergide; Mice; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron | 1989 |
The effect of intrathecal serotonergic antagonists on the pressor response to stimulation of the brainstem in the rat.
Topics: Animals; Blood Pressure; Electric Stimulation; Glutamates; Indoles; Injections, Spinal; Ketanserin; Medulla Oblongata; Methysergide; Microinjections; Rats; Rats, Inbred WKY; Receptors, Serotonin; Spinal Cord; Tropanes; Tropisetron | 1989 |
Effects of 5-hydroxytryptamine on human isolated placental chorionic arteries and veins.
Topics: Arteries; Calcium; Calcium Radioisotopes; Female; Humans; In Vitro Techniques; Ketanserin; Methysergide; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Placenta; Pregnancy; Regional Blood Flow; Serotonin; Veins | 1989 |
5-Hydroxytryptamine receptor subtypes participating in pulmonary edema in dogs.
Topics: Animals; Capillary Permeability; Dogs; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Methysergide; Perfusion; Pulmonary Circulation; Pulmonary Edema; Receptors, Serotonin; Serotonin; Vascular Resistance | 1989 |
Effects of histamine and serotonin on the contractility of isolated pregnant and nonpregnant human myometrium.
Topics: Cimetidine; Dose-Response Relationship, Drug; Drug Interactions; Female; Histamine; Humans; In Vitro Techniques; Ketanserin; Methysergide; Myometrium; Pregnancy; Pyrilamine; Serotonin; Uterine Contraction | 1989 |
Heterogeneous 3H-rauwolscine binding sites in rat cortex: two alpha 2-adrenoceptor subtypes or an additional non-adrenergic interaction?
Topics: Animals; Binding Sites; Binding, Competitive; Cerebral Cortex; Creatinine; Dioxanes; Drug Combinations; Hippocampus; Ketanserin; Male; Methysergide; Phentolamine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Spiperone; Spiro Compounds; Yohimbine | 1988 |
Modification of electrical field stimulation-induced contractions in the guinea-pig ileum by metoclopramide and ICS 205-930 depends on the integrity of the mucosa.
Topics: Animals; Drug Interactions; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Intestinal Mucosa; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Muscle, Smooth; Serotonin Antagonists; Tropisetron | 1986 |
Pharmacological analysis of 5-HT-induced vasoconstriction in isolated, perfused dog skeletal muscle arteries.
Topics: Adrenergic alpha-Antagonists; Animals; Arteries; Cold Temperature; Diltiazem; Dogs; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Quinazolines; Serotonin; Vasoconstriction | 1987 |
Effect of alpha-adrenergic and serotonergic blockers on the acute irritative response in the rabbit eye.
Topics: Adrenergic alpha-Antagonists; Animals; Aqueous Humor; Blood Pressure; Eye Diseases; Eye Proteins; Female; Formaldehyde; Intraocular Pressure; Ketanserin; Male; Methysergide; Phentolamine; Prazosin; Pupil; Rabbits; Serotonin Antagonists; Yohimbine | 1987 |
Effects of selective 5-hydroxytryptamine-2 and nonselective 5-hydroxytryptamine antagonists on the differential-reinforcement-of-low-rate 72-second schedule.
Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Dose-Response Relationship, Drug; Ketanserin; Male; Methysergide; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reinforcement Schedule; Reinforcement, Psychology; Serotonin Antagonists | 1988 |
Quipazine reduces food intake in the rat by activation of 5-HT2-receptors.
Topics: Animals; Diet; Dose-Response Relationship, Drug; Eating; Histamine H2 Antagonists; Imidazoles; Ketanserin; Methysergide; Ondansetron; Pindolol; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1988 |
The effects of ketanserin, methysergide and LY 53857 on sympathetic nerve activity.
Topics: Anesthesia; Animals; Blood Pressure; Cats; Ergolines; Heart Rate; Hemodynamics; Ketanserin; Lactates; Lactic Acid; Male; Methysergide; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Sympathetic Nervous System | 1985 |
Analysis of the heart rate effects of 5-hydroxytryptamine in the cat; mediation of tachycardia by 5-HT1-like receptors.
Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Isoproterenol; Ketanserin; Male; Methysergide; Piperidines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tropanes; Vagus Nerve | 1985 |
Peripheral serotonin2 receptor blockade does not inhibit 5-hydroxytryptophan-induced aldosterone stimulation.
Topics: 5-Hydroxytryptophan; Adult; Aldosterone; Humans; Ketanserin; Male; Methysergide; Piperidines; Potassium; Renin; Serotonin; Serotonin Antagonists | 1985 |
Effects of serotonin receptor agonists and antagonists on schedule-controlled behavior of squirrel monkeys.
Topics: 5-Hydroxytryptophan; Animals; Cinanserin; Conditioning, Operant; Cyproheptadine; Electroshock; Female; Ketanserin; Male; Metergoline; Methysergide; Piperazines; Piperidines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri | 1985 |
A comparison of cardiovascular and smooth muscle effects of 5-hydroxytryptamine and 5-carboxamidotryptamine, a selective agonist of 5-HT1 receptors.
Topics: Airway Resistance; Animals; Cyproheptadine; Guinea Pigs; Heart Rate; Hemodynamics; Ileum; In Vitro Techniques; Ketanserin; Male; Mecamylamine; Methysergide; Muscle, Smooth; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Urinary Bladder | 1985 |
Effects of MK-212 (6-chloro-2[1-piperazinyl]pyrazine) on schedule-controlled behavior and their reversal by 5-HT antagonists in the pigeon.
Topics: Animals; Columbidae; Conditioning, Operant; Cues; Generalization, Stimulus; Ketanserin; Male; Metergoline; Methysergide; Piperidines; Pyrazines; Receptors, Serotonin; Reinforcement Schedule | 1986 |
5-Carboxamidotryptamine is a selective agonist at 5-hydroxytryptamine receptors mediating vasodilatation and tachycardia in anaesthetized cats.
Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Ketanserin; Male; Methiothepin; Methysergide; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasodilation | 1986 |
Potentiation of vasoconstrictor responses to serotonin in the limb of atherosclerotic monkeys.
Topics: Animals; Arteriosclerosis; Hindlimb; Hypercholesterolemia; Ketanserin; Macaca fascicularis; Methysergide; Piperidines; Serotonin; Vasoconstriction | 1986 |
Comparative effects of ketanserin, atropine and methysergide on the gastrointestinal effects of hyperserotoninemia in the awake dog.
Topics: Animals; Atropine; Digestive System; Dogs; Gastrointestinal Motility; Ketanserin; Methysergide; Piperidines; Receptors, Serotonin; Serotonin; Water-Electrolyte Balance | 1986 |
Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?
Topics: Animals; Aorta, Thoracic; In Vitro Techniques; Jugular Veins; Ketanserin; Male; Methysergide; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Trazodone | 1986 |
Allosteric properties of 5-HT2 receptors in tracheal smooth muscle.
Topics: Allosteric Regulation; Animals; Binding, Competitive; Cattle; Female; Guinea Pigs; Ketanserin; Kinetics; Male; Methysergide; Models, Biological; Muscle Relaxation; Muscle, Smooth; Piperidines; Potassium; Receptors, Serotonin; Serotonin; Species Specificity; Trachea | 1986 |
Histaminergic regulation of prolactin secretion: involvement of serotoninergic neurons.
Topics: Dimaprit; Histamine; Ketanserin; Methysergide; Neurons; Prolactin; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Thiourea | 1988 |
Studies on the antinociceptive effect of intrathecal salmon calcitonin.
Topics: Analgesics; Animals; Benzomorphans; Calcitonin; Enkephalin, Leucine; Haloperidol; Ketanserin; Male; Methysergide; Nociceptors; Phentolamine; Piperidines; Rats; Receptors, Opioid | 1985 |
Are there any presynaptic 5-HT receptors in frog atria?
Topics: Animals; Anura; Calcium; Electric Stimulation; Epinephrine; Heart Atria; In Vitro Techniques; Ketanserin; Male; Methysergide; Myocardial Contraction; Neuromuscular Junction; Phentolamine; Receptors, Neurotransmitter; Receptors, Serotonin; Synaptic Transmission | 1986 |
Serotonin and the renal blood supply: role of prostaglandins and the 5HT-2 receptor.
Topics: Angiotensin II; Animals; Blood Pressure; Cyclooxygenase Inhibitors; Dogs; Dose-Response Relationship, Drug; Indomethacin; Ketanserin; Kidney; Methysergide; Prostaglandins; Receptors, Serotonin; Renal Circulation; Serotonin | 1986 |
Antagonism by methysergide of neurogenic vasoconstriction in the dog forelimb.
Topics: Animals; Dogs; Electric Stimulation; Forelimb; Ketanserin; Median Nerve; Methysergide; Phentolamine; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasoconstriction; Vasodilation | 1987 |
Antagonism by ketanserin of the behavioral effects of quipazine but not l-5-hydroxytryptophan in squirrel monkeys.
Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Female; Ketanserin; Male; Methysergide; Quinolines; Quipazine; Saimiri | 1988 |
Effects of tryptamine mediated through 2 states of the 5-HT2 receptor in calf coronary artery.
Topics: Animals; Cattle; Coronary Vessels; Endothelium, Vascular; In Vitro Techniques; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Serotonin; Selegiline; Tryptamines | 1988 |
Studies into the dual effects of serotonergic pharmacological agents on female sexual behaviour in the rat: preliminary evidence that endogenous 5HT is stimulatory.
Topics: 5-Hydroxytryptophan; Adrenalectomy; Alanine; Animals; Castration; Cinanserin; Female; Ketanserin; Metergoline; Methysergide; Mianserin; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal; Zimeldine | 1985 |
A paradox: the 5-HT2-receptor antagonist ketanserin restores the 5-HT-induced contraction depressed by methysergide in large coronary arteries of calf. Allosteric regulation of 5-HT2-receptors.
Topics: Allosteric Regulation; Animals; Cattle; Coronary Vessels; In Vitro Techniques; Ketanserin; Methysergide; Models, Biological; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vasoconstriction | 1985 |
Interaction of 5-hydroxytryptamine and ketanserin in rat vas deferens subjected to low frequency field stimulation.
Topics: Animals; Drug Interactions; Electric Stimulation; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth; Piperidines; Prazosin; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Vas Deferens | 1985 |
Tryptamine-induced vasoconstrictor responses in rat caudal arteries are mediated predominantly via 5-hydroxytryptamine receptors.
Topics: Animals; Arteries; In Vitro Techniques; Ketanserin; Male; Methysergide; Monoamine Oxidase Inhibitors; Phentolamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tryptamines; Vasoconstriction | 1985 |
Excitatory 5-hydroxytryptamine receptors in the cat urinary bladder are of the M- and 5-HT2-type.
Topics: Animals; Atropine; Cats; Cyproheptadine; Dimethylphenylpiperazinium Iodide; Drug Interactions; Female; Guanethidine; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Urinary Bladder | 1985 |
Potentiation of motoneurone excitability by combined administration of 5-HT agonist and TRH analogue.
Topics: Animals; Anterior Horn Cells; Drug Synergism; Female; Fenclonine; Ketanserin; Methoxydimethyltryptamines; Methysergide; Motor Neurons; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Serotonin; Stimulation, Chemical; Thyrotropin-Releasing Hormone | 1985 |
A facilitatory role for serotonin in the sexual behavior of the female rat.
Topics: Animals; Castration; Estradiol; Female; Ketanserin; Methysergide; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Sexual Behavior, Animal; Spiperone | 1985 |
Two types of receptors for 5-hydroxytryptamine on the cholinergic nerves of the guinea-pig myenteric plexus.
Topics: Acetylcholine; Animals; Binding, Competitive; Cocaine; Electric Stimulation; Female; Guinea Pigs; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Myenteric Plexus; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes | 1985 |
Effect of serotonin on the motility of smooth muscles in teats of lactating cows.
Topics: Animals; Cattle; Female; Ketanserin; Lactation; Mammary Glands, Animal; Methysergide; Mianserin; Milk Ejection; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Piperidines; Pregnancy; Serotonin; Serotonin Antagonists | 1985 |
Serotonergic mediation of a negative feedback effect of estrogen on luteinizing hormone release in ovariectomized rats.
Topics: Animals; Estradiol; Estrogens; Feedback; Female; Ketanserin; Luteinizing Hormone; Metergoline; Methysergide; Ovariectomy; Quipazine; Rats; Receptors, Serotonin; Serotonin; Software | 1988 |
5-Hydroxytryptamine receptors in the hypothalamus mediate thermoregulatory responses in rabbits.
Topics: Animals; Body Temperature Regulation; Cyproheptadine; Ketanserin; Male; Methysergide; Preoptic Area; Rabbits; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1988 |
Responses to 5-hydroxytryptamine evoked in the hemisected spinal cord of the neonate rat.
Topics: Animals; Animals, Newborn; Citalopram; Electrodes; In Vitro Techniques; Ketanserin; Male; Methysergide; Neuromuscular Depolarizing Agents; Norepinephrine; Pargyline; Rats; Serotonin; Serotonin Antagonists; Spinal Cord | 1988 |
Is serotonin involved in the ovulatory process of the rat ovary perfused in vitro?
Topics: Animals; Female; Ketanserin; Luteinizing Hormone; Methysergide; Nifedipine; Ovary; Ovulation; Perfusion; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin | 1988 |
Evidence for depressant 5-HT1-like receptors on rat brainstem neurones.
Topics: Animals; Brain Stem; Ketanserin; Male; Membrane Potentials; Metergoline; Methysergide; Neurons; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tropanes | 1988 |
Neuronal involvement in type 1 hypersensitivity reactions in gut epithelia.
Topics: Animals; Cyproheptadine; Epithelium; Guinea Pigs; Hypersensitivity, Immediate; In Vitro Techniques; Indoles; Intestinal Mucosa; Ketanserin; Methysergide; Neurons; Serotonin Antagonists; Tetrodotoxin; Tropisetron | 1987 |
Influence of a serotonin receptor antagonist, 5-HTP-DP-hex, on spinal and thalamic nociceptive neurons in rats.
Topics: 5-Hydroxytryptophan; Action Potentials; Animals; Ketanserin; Male; Methysergide; Naloxone; Nerve Fibers; Pain; Periaqueductal Gray; Rats; Reaction Time; Sciatic Nerve; Spinothalamic Tracts; Thalamic Nuclei | 1987 |
Phencyclidine-induced head-twitch response in rats treated chronically with methysergide.
Topics: Animals; Brain; Drug Interactions; Drug Tolerance; Ketanserin; Male; Methoxydimethyltryptamines; Methysergide; Phencyclidine; Rats; Rats, Inbred F344; Receptors, Serotonin; Stereotyped Behavior | 1987 |
Serotonin-induced cytosolic free calcium transients in cultured vascular smooth muscle cells.
Topics: Aminoquinolines; Animals; Calcium; Cells, Cultured; Ketanserin; Methysergide; Muscle, Smooth, Vascular; Rats; Receptors, Serotonin; Serotonin | 1987 |
Involvement of serotonin in intestinal mastocytopoiesis and inflammation during a Trichinella spiralis infection in mice.
Topics: Animals; Cell Division; Cells, Cultured; Female; Hematopoiesis; Inflammation; Intestinal Diseases; Intestinal Mucosa; Ketanserin; Mast Cells; Methysergide; Mice; Mice, Inbred Strains; Mice, Nude; Serotonin; Stem Cells; Trichinella; Trichinellosis | 1987 |
Vasoconstrictor mechanism of 5-hydroxytryptamine in isolated and perfused canine basilar arteries.
Topics: Animals; Basilar Artery; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; Ketanserin; Male; Methysergide; Potassium Chloride; Receptors, Serotonin; Saponins; Serotonin; Vasoconstriction | 1987 |
Kinetics of competitive drug action at 5-hydroxytryptamine2 receptors in isolated rabbit aorta.
Topics: Animals; Aorta; Binding, Competitive; Diffusion; Indoles; Ketanserin; Kinetics; Male; Methysergide; Muscle, Smooth, Vascular; Rabbits; Receptors, Serotonin; Serotonin; Spiperone; Tryptamines | 1987 |
Interconversion into a low active state protects vascular 5-HT2-receptors against irreversible antagonism by phenoxybenzamine.
Topics: Allosteric Regulation; Animals; Binding Sites; Cattle; Coronary Vessels; In Vitro Techniques; Ketanserin; Methysergide; Models, Biological; Muscle, Smooth, Vascular; Phenoxybenzamine; Pulmonary Artery; Receptors, Serotonin | 1987 |
Vasoactive effects of serotonin on proximal coronary arteries in awake dogs.
Topics: Animals; Coronary Circulation; Coronary Vessels; Dogs; Endothelium; Ketanserin; Kinetics; Methysergide; Receptors, Serotonin; Serotonin; Vasoconstriction; Vasodilation | 1987 |
The subtype of serotonin (5-HT) receptors in the rat pulmonary artery.
Topics: Animals; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Mianserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Pizotyline; Prazosin; Pulmonary Artery; Rats; Receptors, Serotonin | 1987 |
S1-receptor participation in serotonin-induced pulmonary edema in the dog.
Topics: Animals; Blood Pressure; Body Water; Capillary Permeability; Dogs; Histamine; In Vitro Techniques; Ketanserin; Lung; Methysergide; Pulmonary Edema; Receptors, Serotonin; Serotonin | 1987 |
Influence of serotonin on lower urinary tract smooth muscle in vitro.
Topics: Animals; Cyproheptadine; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Serotonin; Serotonin Antagonists; Swine; Urethra; Urinary Bladder | 1986 |
Lack of effect of antagonists on serotonin-induced inhibition in rat hippocampus.
Topics: Action Potentials; Animals; Cyproheptadine; Halothane; Hippocampus; Ketanserin; Lysergic Acid Diethylamide; Metergoline; Methysergide; Neural Inhibition; Picrotoxin; Rats; Serotonin; Serotonin Antagonists; Urethane | 1986 |
Opiate-serotonin synergism stimulating luteinizing hormone release in estrogen-progesterone-primed ovariectomized rats: mediation by serotonin2 receptors.
Topics: Animals; Estradiol; Female; Ketanserin; Luteinizing Hormone; Methysergide; Morphine; Ovariectomy; Progesterone; Quinolines; Quipazine; Rats; Receptors, Serotonin; Serotonin | 1987 |
The specificity of ketanserin in the inhibition of serotonin-induced steroidogenesis in the rat adrenal zona glomerulosa.
Topics: Adrenal Cortex; Aldosterone; Animals; Corticosterone; Cyclic AMP; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Methysergide; Piperidines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1984 |
Serotoninergic control of somatostatin and gastrin release from the isolated rat stomach.
Topics: Animals; Gastric Mucosa; Gastrins; In Vitro Techniques; Ketanserin; Male; Methysergide; Perfusion; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Receptors, Serotonin; Serotonin; Somatostatin | 1984 |
Tryptaminergic receptors in the bovine pulmonary vasculature: effects of ketanserin.
Topics: Animals; Cattle; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pulmonary Artery; Pulmonary Veins; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists | 1984 |
Serotonin-2 binding sites in human frontal cortex and hippocampus. Selective loss of S-2A sites with age.
Topics: Adolescent; Adult; Aged; Aging; Cerebral Cortex; Hippocampus; Humans; Ketanserin; Kinetics; Methysergide; Middle Aged; Organ Specificity; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone | 1984 |
The effects of serotonin antagonists in a behavioral despair procedure in mice.
Topics: Animals; Behavior, Animal; Cyproheptadine; Guinea Pigs; Ketanserin; Male; Methysergide; Mice; Muscle, Smooth; Piperidines; Pizotyline; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Trazodone; Tritium | 1984 |
Involvement of 5-HT2 receptors in the wet-dog shake behaviour induced by 5-hydroxytryptophan in the rat.
Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Female; Ketanserin; Methysergide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists | 1983 |
Inhibitory effect of ketanserin on ergonovine-induced contractions of isolated canine coronary arteries.
Topics: Animals; Coronary Vessels; Dogs; Ergonovine; In Vitro Techniques; Ketanserin; Methysergide; Piperidines; Serotonin Antagonists; Vasoconstriction | 1983 |
5-Hydroxytryptamine can mediate endothelium-dependent relaxation of coronary arteries.
Topics: Animals; Blood Platelets; Coronary Vessels; Dogs; In Vitro Techniques; Isometric Contraction; Ketanserin; Methysergide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Piperidines; Serotonin; Serotonin Antagonists; Thromboxane B2 | 1983 |
Differential actions of serotonin antagonists on two behavioral models of serotonin receptor activation in the rat.
Topics: Animals; Behavior, Animal; Butyrophenones; Ketanserin; Male; Metergoline; Methysergide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists | 1984 |
Effects of tryptamine antagonists on the anaphylactic contractions of the bovine pulmonary smooth muscles.
Topics: Anaphylaxis; Animals; Cattle; Horses; In Vitro Techniques; Ketanserin; Lung; Methysergide; Muscle Contraction; Muscle, Smooth; Piperidines; Pulmonary Artery; Pulmonary Veins; Serotonin Antagonists; Trachea; Tryptamines | 1984 |
On the mechanism of action of ketanserin, a selective antagonist of the S2 receptors with antihypertensive activity.
Topics: Animals; Antihypertensive Agents; Dogs; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Norepinephrine; Piperidines; Rats; Serotonin Antagonists; Vasodilation | 1983 |
Comparative effects of ketanserin, a novel serotonergic receptor antagonist, on 5HT-induced shape change and 5HT uptake in rat and human platelets.
Topics: Adenosine Diphosphate; Animals; Blood Platelets; Clomipramine; Female; Humans; In Vitro Techniques; Ketanserin; Kinetics; Male; Methysergide; Piperidines; Rats; Serotonin; Serotonin Antagonists | 1982 |
Modulation of rat neocortical high-voltage spindle activity by 5-HT1/5-HT2 receptor subtype specific drugs.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Analysis of Variance; Animals; Cerebral Cortex; Electroencephalography; Infusions, Parenteral; Ketanserin; Male; Methiothepin; Methysergide; Neural Pathways; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin; Thalamus | 1995 |
Involvement of serotonin in the regulation of GnRH gene expression in the male rat brain.
Topics: Animals; Evaluation Studies as Topic; Gene Expression Regulation; Gonadotropin-Releasing Hormone; In Situ Hybridization; Ketanserin; Male; Methysergide; Neurons; Ondansetron; Preoptic Area; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists | 1995 |
Involvement of serotonin in developmental plasticity of kitten visual cortex.
Topics: 5,7-Dihydroxytryptamine; Aging; Animals; Animals, Newborn; Cats; Functional Laterality; Ketanserin; Methysergide; Neuronal Plasticity; Ocular Physiological Phenomena; Serotonin; Serotonin Antagonists; Vision, Monocular; Visual Cortex | 1995 |
Augmentation of coronary responsiveness to serotonin at the site of X-ray-induced intimal thickening in miniature pigs.
Topics: Animals; Coronary Vasospasm; Coronary Vessels; Endothelium, Vascular; Histamine; Ketanserin; Male; Methysergide; Myocardial Ischemia; Phenylephrine; Serotonin; Serotonin Antagonists; Swine; Swine, Miniature; Tunica Intima; Vasoconstriction; X-Rays | 1995 |
In vitro airway and tissue response to antigen in sensitized rats. Role of serotonin and leukotriene D4.
Topics: Airway Resistance; Animals; Bronchi; Bronchial Provocation Tests; Bronchoconstriction; Indoles; Ketanserin; Leukotriene D4; Lipoxygenase Inhibitors; Lung; Methysergide; Ovalbumin; Propionates; Quinolines; Rats; Rats, Inbred BN; Receptors, Immunologic; Respiratory Hypersensitivity; Serotonin | 1995 |
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach | 1995 |
Effects of serotonergic agents on neuronal nicotinic acetylcholine receptors.
Topics: Animals; Cells, Cultured; Electric Conductivity; Female; Ketanserin; Membrane Potentials; Methysergide; Neurons; Oocytes; Patch-Clamp Techniques; Rats; Receptors, Nicotinic; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tetrahydronaphthalenes; Xenopus laevis | 1995 |
Functional 5-HT receptor subtypes in the isolated canine common carotid artery.
Topics: Adrenergic alpha-Antagonists; Animals; Carotid Artery, Common; Diltiazem; Dogs; Female; Ketanserin; Male; Methysergide; Norepinephrine; Potassium Chloride; Quinazolines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Spiperone; Vasoconstriction | 1994 |
Ketanserin and granisetron reduce cholera toxin-induced hypersecretion in pig jejunum.
Topics: Animals; Animals, Newborn; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cholera Toxin; Diarrhea; Dose-Response Relationship, Drug; Drug Therapy, Combination; Granisetron; Indoles; Intestinal Secretions; Jejunum; Ketanserin; Methysergide; Serotonin Antagonists; Swine; Tropisetron | 1994 |
Effect of indomethacin, renzapride, methysergide, ketanserin, granisetron and citalopram on serotonin-induced fluid accumulation in pig jejunum.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Citalopram; Dose-Response Relationship, Drug; Granisetron; Indomethacin; Intestinal Absorption; Jejunum; Ketanserin; Methysergide; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Swine | 1994 |
Role of serotonin in the regulation of prolactin gene expression in the male rat as evaluated by in situ hybridization.
Topics: Animals; Autoradiography; Gene Expression Regulation; Growth Hormone; In Situ Hybridization; Ketanserin; Male; Methysergide; Prolactin; Rats; Rats, Sprague-Dawley; RNA, Messenger; Serotonin | 1994 |
Modulation of rhythmic swimming activity in post-embryonic Xenopus laevis tadpoles by 5-hydroxytryptamine acting at 5HT1a receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Animals; Cyproheptadine; Ergolines; Ketanserin; Metamorphosis, Biological; Methysergide; Motor Activity; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming; Xenopus laevis | 1994 |
Effects of serotonin on rat ileocolonic transit and fluid transfer in vivo: possible mechanisms of action.
Topics: Animals; Atropine; Benzamides; Bethanechol; Bethanechol Compounds; Biological Transport; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Colon; Gastrointestinal Transit; Heterocyclic Compounds; Ileum; Ketanserin; Male; Methysergide; Models, Biological; Pyrroles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists | 1993 |
Is 5-hydroxytryptamine mediating descending inhibition in the neonatal rat spinal cord through different receptor subtypes?
Topics: Animals; Animals, Newborn; Citalopram; Dioxanes; Dopamine Antagonists; Electric Stimulation; Ketanserin; Lumbar Vertebrae; Methiothepin; Methysergide; Rats; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Spinal Cord; Spinal Nerve Roots; Spiperone; Spiro Compounds; Sulpiride; Sumatriptan | 1993 |
Inhibitory effects of tryptamine on tolbutamide-induced hypoglycemia in mice: mediation by 5-HT receptors.
Topics: Animals; Blood Glucose; Hypoglycemia; Indoles; Ketanserin; Male; Methysergide; Mice; Mice, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Time Factors; Tolbutamide; Tropisetron; Tryptamines | 1994 |
5-HT receptor subtypes involved in luminal serotonin-induced secretion in rat intestine in vivo.
Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Ileum; Indoles; Jejunum; Ketanserin; Male; Methysergide; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Tropisetron; Water-Electrolyte Balance | 1994 |
Effect of serotonin receptor blockade on endocrine and cardiovascular responses to head-up tilt in humans.
Topics: Adrenocorticotropic Hormone; beta-Endorphin; Blood Pressure; Heart Rate; Hemodynamics; Hormones; Humans; Hydrocortisone; Ketanserin; Male; Methysergide; Norepinephrine; Ondansetron; Posture; Prolactin; Reference Values; Renin; Serotonin Antagonists; Vagus Nerve; Vascular Resistance | 1993 |
Serotonergic, 5-HT2, receptor-mediated phosphoinositide turnover and mobilization of calcium in cultured rat retinal pigment epithelium cells.
Topics: Animals; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Inositol Phosphates; Ketanserin; Methysergide; Phosphatidylinositols; Pigment Epithelium of Eye; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1993 |
Serotonergic 5HT2 receptors mediate the inhibitory action of serotonin on luteinizing hormone secretion in ovariectomized, estradiol-treated ewes that are refractory to short days.
Topics: Animals; Cyproheptadine; Dose-Response Relationship, Drug; Estradiol; Female; Ketanserin; Light; Luteinizing Hormone; Methysergide; Ovariectomy; Ovary; Periodicity; Receptors, Serotonin; Sheep | 1993 |
MDL 72222, ketanserin, and methysergide pretreatments fail to alter breaking points on a progressive ratio schedule reinforced by intravenous cocaine.
Topics: Animals; Cocaine; Conditioning, Operant; Injections, Intravenous; Ketanserin; Male; Methysergide; Rats; Rats, Wistar; Reinforcement Schedule; Self Administration; Serotonin Antagonists; Tropanes | 1993 |
Characterization of 5-HT receptors in simian isolated gastroepiploic artery.
Topics: Animals; Arteries; Diltiazem; Endothelium, Vascular; Female; In Vitro Techniques; Ketanserin; Macaca; Male; Methysergide; Norepinephrine; Omentum; Perfusion; Phentolamine; Potassium Chloride; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Stomach; Vasoconstriction | 1993 |
Peripherally administered serotonin induces hyperglucagonemia in mice.
Topics: Animals; Glucagon; Indoles; Injections, Intraperitoneal; Ketanserin; Male; Methysergide; Mice; Mice, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Tropisetron | 1993 |
Regulation of synapse density by 5-HT2A receptor agonist and antagonist in the spinal cord of chicken embryo.
Topics: Amphetamines; Animals; Chick Embryo; Ketanserin; Methysergide; Microscopy, Electron; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synapses | 1995 |
Influence of serotonin on the human ureter: an in vitro pharmacological study.
Topics: Adult; Aged; Atropine; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Indoles; Ketanserin; Male; Methysergide; Middle Aged; Muscle Contraction; Serotonin; Serotonin Antagonists; Tropisetron; Ureter | 1995 |
Excitation of rat substantia nigra pars reticulata neurons by 5-hydroxytryptamine in vitro: evidence for a direct action mediated by 5-hydroxytryptamine2C receptors.
Topics: Animals; Electrophysiology; In Vitro Techniques; Ketanserin; Male; Methysergide; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Substantia Nigra | 1995 |
Different serotonin receptor types participate in 5-hydroxytryptophan-induced gonadotropins and prolactin release in the female infantile rat.
Topics: 5-Hydroxytryptophan; Animals; Female; Follicle Stimulating Hormone; Ketanserin; Luteinizing Hormone; Methysergide; Ondansetron; Prolactin; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1996 |
Characterization of 5-hydroxytryptamine (5-HT) receptor subtypes influencing colonic motility in conscious dogs.
Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Benzimidazoles; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dogs; Dose-Response Relationship, Drug; Gastrointestinal Motility; Hexamethonium; Injections, Intravenous; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Transducers | 1996 |
Serotonin is involved in the ACTH-induced reversal of hemorrhagic shock in anesthetized rats.
Topics: Animals; Cosyntropin; Female; Fenclonine; Ketanserin; Male; Methysergide; Rats; Serotonin Agents; Shock, Hemorrhagic | 1996 |
5-HT2B receptor-mediated serotonin morphogenetic functions in mouse cranial neural crest and myocardiac cells.
Topics: Animals; Binding Sites; Brain; Cell Differentiation; DNA Primers; Embryo, Mammalian; Embryonic and Fetal Development; Embryonic Induction; Gene Expression Regulation, Developmental; Heart; Humans; In Situ Hybridization; Ketanserin; Methysergide; Mice; Microscopy, Electron, Scanning; Morphogenesis; Neural Crest; Organ Culture Techniques; Paroxetine; Polymerase Chain Reaction; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Ritanserin; RNA, Messenger; Serotonin; Serotonin Antagonists; Signal Transduction; Transcription, Genetic | 1997 |
Differential effects of three 5-HT receptor antagonists on the performance of rats in attentional and working memory tasks.
Topics: Animals; Attention; Dose-Response Relationship, Drug; Ketanserin; Male; Memory; Methysergide; Rats; Rats, Wistar; Serotonin Antagonists; Task Performance and Analysis | 1997 |
Effect of 5-hydroxytryptamine on gastrointestinal motility in conscious guinea-pigs.
Topics: Animals; Atropine; Consciousness; Duodenum; Eating; Fasting; Female; Gastrointestinal Motility; Guinea Pigs; Ileum; Infusions, Intravenous; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Pyloric Antrum; Serotonin; Serotonin Antagonists | 1997 |
Involvement of serotonin in the modulation of cocaine-induced locomotor activity in the rat.
Topics: Animals; Behavior, Animal; Cocaine; Drug Interactions; Female; Fluoxetine; Ketanserin; Methysergide; Motor Activity; Narcotics; Piperazines; Pyridines; Rats; Rats, Wistar; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists | 1998 |
The effects of 8-hydroxy-2-(di-n-propylamino)tetralin on the cholinergic contraction in guinea pig and human airways in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Bronchi; Bronchoconstriction; Capsaicin; Cholinergic Fibers; Culture Techniques; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Humans; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Neuropeptides; Pindolol; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles; Trachea; Tropisetron | 1998 |
p-Chloroamphetamine, a serotonin-releasing drug, elicited in rats a hyperglycemia mediated by the 5-HT1A and 5-HT2B/2C receptors.
Topics: 4-Aminobenzoic Acid; Adrenal Medulla; Adrenalectomy; Aminopyridines; Animals; Blood Glucose; Dose-Response Relationship, Drug; Ergolines; Fenclonine; Hyperglycemia; Indoles; Ketanserin; Male; Methysergide; p-Chloroamphetamine; para-Aminobenzoates; Piperazines; Propranolol; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Ritanserin; Serotonin; Serotonin Agents; Serotonin Antagonists; Tropisetron | 1998 |
Serotonin receptor subtypes involved in modulation of electrical acupuncture.
Topics: Animals; Dental Pulp; Electric Stimulation; Electroacupuncture; Evoked Potentials; Indoles; Injections, Intravenous; Ketanserin; Male; Methysergide; Nociceptors; Pain; Pindolol; Piperazines; Rabbits; Receptors, Serotonin; Serotonin Antagonists; Trigeminal Caudal Nucleus; Tropisetron | 1998 |
Agonist and antagonist binding to rabbit cortical 5-HT2A receptors: opposite effects of magnesium.
Topics: Amphetamines; Animals; Cerebral Cortex; Fluorobenzenes; Guanylyl Imidodiphosphate; Ketanserin; Magnesium; Methysergide; Piperidines; Prazosin; Rabbits; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone | 1998 |
Antinociception elicited by aversive stimulation of the inferior colliculus.
Topics: Algorithms; Analgesia; Animals; Arousal; Behavior, Animal; Electric Stimulation; Escape Reaction; GABA Modulators; Inferior Colliculi; Ketanserin; Male; Methysergide; Midazolam; Naltrexone; Narcotic Antagonists; Pain Measurement; Rats; Rats, Wistar; Serotonin Antagonists; Stress, Psychological | 1999 |
Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach.
Topics: Animals; Atropine; Dioxanes; Enzyme Inhibitors; Female; Gastric Fundus; Granisetron; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscarinic Antagonists; Muscle Relaxation; Muscle Tonus; Nitroarginine; Piperidines; Pyloric Antrum; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Tetrodotoxin | 1999 |
Involvement of 5-HT1B receptors in collar-induced hypersensitivity to 5-hydroxytryptamine of the rabbit carotid artery.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Braces; Carotid Arteries; Dose-Response Relationship, Drug; Hypersensitivity; In Vitro Techniques; Ketanserin; Male; Methysergide; Oxadiazoles; Piperazines; Potassium Chloride; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sumatriptan; Tryptamines; Vasoconstriction | 1999 |
Methysergide augments the acute, but not the sustained, hypoxic ventilatory response in goats.
Topics: Acclimatization; Animals; Blood Pressure; Carbon Dioxide; Female; Goats; Heart Rate; Hypoxia; Ketanserin; Methysergide; Partial Pressure; Respiratory Mechanics; Serotonin Antagonists; Time Factors; Wakefulness | 1999 |
Serotonin suppresses subthreshold and suprathreshold oscillatory activity of rat inferior olivary neurones in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Amphetamines; Animals; Cardiovascular Agents; Electric Impedance; Electrophysiology; Ketanserin; Methysergide; Neurons; Olivary Nucleus; Periodicity; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pyrimidines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
Blockade of the serotonergic system counteracts the dizocilpine-induced changes in dopaminergic function.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Behavior, Animal; Dizocilpine Maleate; Dopamine; Dopamine Agonists; Excitatory Amino Acid Antagonists; Grooming; Ketanserin; Male; Methysergide; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Stereotyped Behavior | 2000 |
Serotonin and the hypoxic ventilatory response in awake goats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acclimatization; Animals; Carotid Body; Chemoreceptor Cells; Female; Goats; Hypoxia; Ketanserin; Methysergide; Oxygen; Respiration; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2000 |
Modulation of rat uterine contractility by mast cells and their mediators.
Topics: Animals; Antibodies, Anti-Idiotypic; Blood; Carbachol; Female; Histamine; Immunoglobulin E; Ketanserin; Mast Cells; Metalloendopeptidases; Methysergide; Ovalbumin; p-Methoxy-N-methylphenethylamine; Pregnancy; Rabbits; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Uterine Contraction; Uterus | 2000 |
The antinociceptive effect induced by FR140423 is mediated through spinal 5-HT2A and 5-HT3 receptors.
Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Methysergide; Mice; Pain; Pain Measurement; Piperazines; Pyrazoles; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Sulfoxides; Tropanes | 2000 |
Post-ictal analgesia: involvement of opioid, serotoninergic and cholinergic mechanisms.
Topics: Analgesia; Animals; Atropine; Convulsants; Disease Models, Animal; Injections, Intraperitoneal; Ketanserin; Methysergide; Motor Activity; Muscarinic Antagonists; Naloxone; Narcotic Antagonists; Pain Measurement; Pentylenetetrazole; Rats; Rats, Wistar; Reaction Time; Reflex; Seizures; Serotonin Antagonists | 2001 |
Mechanism of airway hyperresponsiveness to adenosine induced by allergen challenge in actively sensitized Brown Norway rats.
Topics: Adenosine; Allergens; Animals; Atropine; Bradykinin; Bronchoconstriction; Bronchoconstrictor Agents; Capsaicin; Cardiovascular System; Cell Degranulation; Cromolyn Sodium; Dose-Response Relationship, Drug; Histamine; In Vitro Techniques; Ketanserin; Lung; Male; Mast Cells; Methacholine Chloride; Methysergide; Ovalbumin; p-Methoxy-N-methylphenethylamine; Rats; Rats, Inbred BN; Respiratory Hypersensitivity; Serotonin; Serotonin Antagonists; Time Factors; Vagotomy; Vasoconstrictor Agents | 2001 |
Central administration of a 5-HT2 receptor agonist and antagonist: lack of effect on rapid eye movement sleep and pgo waves.
Topics: Analysis of Variance; Animals; Arousal; Cats; Electroencephalography; Female; Ketanserin; Methysergide; Pons; Receptors, Serotonin; Serotonin Antagonists; Sleep; Sleep, REM; Wakefulness | 1998 |
Conditioned antinociception and freezing using electrical stimulation of the dorsal periaqueductal gray or inferior colliculus as unconditioned stimulus are differentially regulated by 5-HT2A receptors in rats.
Topics: Animals; Autonomic Nervous System; Avoidance Learning; Behavior, Animal; Conditioning, Psychological; Electric Stimulation; Inferior Colliculi; Ketanserin; Male; Methysergide; Microinjections; Pain; Pain Measurement; Pain Threshold; Periaqueductal Gray; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Tectum Mesencephali | 2001 |
Selective serotonin receptor antagonism and leukocyte-independent plasma extravasation during endotoxemia.
Topics: Animals; Binding Sites; Cinanserin; Endothelium, Vascular; Endotoxemia; Extravasation of Diagnostic and Therapeutic Materials; Ketanserin; Leukocytes; Methysergide; Microcirculation; Protein Binding; Rats; Receptors, Serotonin; Serotonin Antagonists; Time Factors | 2002 |
Effects of ketanserin and DOI on spontaneous and 5-HT-evoked peristalsis of the pig ureter in vivo.
Topics: Animals; Female; Indophenol; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swine; Ureter | 2002 |
5-HT3 receptors partially mediate halothane depression of spinal dorsal horn sensory neurons.
Topics: Anesthetics, Inhalation; Animals; Decerebrate State; Depression, Chemical; Halothane; Indoles; Ketanserin; Methiothepin; Methysergide; Neurons, Afferent; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Spinal Cord; Tropisetron | 2003 |
Serotonin receptor subtypes required for ventilatory long-term facilitation and its enhancement after chronic intermittent hypoxia in awake rats.
Topics: Animals; Chronic Disease; Clozapine; Hypoxia; Ketanserin; Male; Methysergide; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Respiration; Respiratory Mechanics; Serotonin Antagonists | 2004 |
Oxytocic activity of thrombin: modulation of thrombin-induced gravid rat myometrial contractions by 5-hydroxytryptamine receptor antagonists.
Topics: Animals; Dose-Response Relationship, Drug; Female; Ketanserin; Male; Methysergide; Myometrium; Oxytocics; Pregnancy; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Thrombin; Uterine Contraction | 2004 |
Effect of the blockade of mu1-opioid and 5HT2A-serotonergic/alpha1-noradrenergic receptors on sweet-substance-induced analgesia.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Analgesia; Animals; Dose-Response Relationship, Drug; Ketanserin; Male; Methysergide; Naloxone; Naltrexone; Pain Measurement; Pain Threshold; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Opioid, mu; Serotonin Antagonists; Sucrose; Taste | 2005 |
Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Buspirone; Clozapine; Decerebrate State; Dose-Response Relationship, Drug; Drug Interactions; Ergotamine; Heart Rate; Ketanserin; Lisuride; Male; Metergoline; Methiothepin; Methysergide; Phenylephrine; Piperazines; Pizotyline; Prazosin; Pyridines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Serotonin Antagonists; Serotonin Receptor Agonists; Yohimbine | 2006 |
Pharmacological characterization of 5-Hydroxytryptamine-receptor subtypes in circular muscle from the rat stomach.
Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Synergism; Gastric Emptying; Gastric Fundus; In Vitro Techniques; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Ondansetron; Oxadiazoles; Phenols; Piperazines; Piperidines; Protein Isoforms; Pyloric Antrum; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin | 2007 |
Persistence of eupnea and gasping following blockade of both serotonin type 1 and 2 receptors in the in situ juvenile rat preparation.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Decerebrate State; Disease Models, Animal; Dose-Response Relationship, Drug; Hypoglossal Nerve; Ischemia; Ketanserin; Lung; Methysergide; Peripheral Nerves; Phrenic Nerve; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT1; Respiratory Mechanics; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors; Vagus Nerve | 2007 |
Selective serotonin-receptor antagonism and microcirculatory alterations during experimental endotoxemia.
Topics: Animals; Blood Flow Velocity; Cell Communication; Endothelium, Vascular; Endotoxemia; Ketanserin; Leukocytes; Male; Methysergide; Rats; Rats, Wistar; Serotonin Antagonists; Stress, Mechanical; Venules | 2007 |
Maintenance of gasping and restoration of eupnea after hypoxia is impaired following blockers of alpha1-adrenergic receptors and serotonin 5-HT2 receptors.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amphetamines; Animals; Decerebrate State; Diaphragm; Dioxanes; Disease Models, Animal; Dose-Response Relationship, Drug; Hypoxia; Ketanserin; Methoxamine; Methysergide; Periodicity; Phrenic Nerve; Rats; Receptors, Adrenergic, alpha-1; Receptors, Serotonin, 5-HT2; Respiratory Mechanics; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2008 |
Spinal serotonin receptor activation modulates the exercise ventilatory response with increased dead space in goats.
Topics: Animals; Blood Gas Analysis; Carbon Dioxide; Dose-Response Relationship, Drug; Female; Goats; Ketanserin; Methysergide; Physical Conditioning, Animal; Pulmonary Ventilation; Receptors, Serotonin; Respiration, Artificial; Respiratory Dead Space; Serotonin Antagonists; Spinal Cord; Tidal Volume | 2008 |
Impact of the 5-HT3 receptor channel system for insulin secretion and interaction of ginger extracts.
Topics: Animals; Blood Glucose; Cells, Cultured; Diabetes Mellitus; Guanidine; Indoles; Insulin; Insulin Secretion; Insulin-Secreting Cells; Ion Channels; Ketanserin; Methysergide; Plant Extracts; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Tropisetron; Zingiber officinale | 2009 |
Cardiovascular and respiratory reflexes of the gulf toadfish (Opsanus beta) during acute hypoxia.
Topics: Analysis of Variance; Animals; Batrachoidiformes; Bradycardia; Cardiovascular System; Disease Models, Animal; Enzyme Inhibitors; Heart Rate; Hypoxia; Ketanserin; Methysergide; Reflex; Respiration; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium Cyanide | 2010 |
Serotonin receptors are involved in the spinal mediation of descending facilitation of surgical incision-induced increase of Fos-like immunoreactivity in rats.
Topics: Animals; Atropine; Cholinergic Antagonists; Immunohistochemistry; Ketanserin; Male; Methiothepin; Methysergide; Neurons; Norepinephrine; Pain; Pain Measurement; Pain, Postoperative; Phenoxybenzamine; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Spinal Cord | 2010 |
[Heterogeneity of the rat respiratory way responses to serotonin].
Topics: Animals; Atropine; Bronchi; Electric Stimulation; Hexamethonium; Isometric Contraction; Ketanserin; Male; Methysergide; Muscle, Smooth; Nerve Fibers; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Tissue Culture Techniques; Trachea | 2011 |
Spinal segmental and supraspinal mechanisms underlying the pain-relieving effects of spinal cord stimulation: an experimental study in a rat model of neuropathy.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Baclofen; Bicuculline; Disease Models, Animal; Dopamine Antagonists; Electrodes; Female; GABA Antagonists; Hyperalgesia; Ketanserin; Methysergide; Neuralgia; Pain Measurement; Pain Threshold; Phentolamine; Propranolol; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Spinal Cord; Sulpiride; Time Factors; Transcutaneous Electric Nerve Stimulation | 2012 |
Latent inhibition in an insect: the role of aminergic signaling.
Topics: Analysis of Variance; Animals; Bees; Conditioning, Classical; Dibenzazepines; Dopamine; Dopamine Antagonists; Ethylketocyclazocine; Extinction, Psychological; Fluphenazine; Habituation, Psychophysiologic; Histamine H1 Antagonists; Imidazoles; Inhibition, Psychological; Ketanserin; Methysergide; Odorants; Serotonin; Serotonin Antagonists; Smell | 2012 |
Effects of cyclopiazonic acid and dexamethasone on serotonin-induced calcium responses in vascular smooth muscle cells.
Topics: Animals; Anti-Inflammatory Agents; Calcium Channel Blockers; Calcium Signaling; Cell Line; Dexamethasone; Enzyme Inhibitors; Indoles; Ketanserin; Methysergide; Muscle, Smooth, Vascular; Protein Kinase C; Protein Kinase Inhibitors; Rats; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vasoconstrictor Agents; Vasodilator Agents | 2016 |