Page last updated: 2024-09-03

methylarginyl-lysyl-prolyl-tryptophyl-tert-leucyl-leucyl-ethyl ester and neurotensin

methylarginyl-lysyl-prolyl-tryptophyl-tert-leucyl-leucyl-ethyl ester has been researched along with neurotensin in 5 studies

Compound Research Comparison

Studies
(methylarginyl-lysyl-prolyl-tryptophyl-tert-leucyl-leucyl-ethyl ester)
Trials
(methylarginyl-lysyl-prolyl-tryptophyl-tert-leucyl-leucyl-ethyl ester)
Recent Studies (post-2010)
(methylarginyl-lysyl-prolyl-tryptophyl-tert-leucyl-leucyl-ethyl ester)
Studies
(neurotensin)
Trials
(neurotensin)
Recent Studies (post-2010) (neurotensin)
8004,05445544

Protein Interaction Comparison

ProteinTaxonomymethylarginyl-lysyl-prolyl-tryptophyl-tert-leucyl-leucyl-ethyl ester (IC50)neurotensin (IC50)
Neurotensin receptor type 1Homo sapiens (human)0.0013
Neurotensin receptor type 2Rattus norvegicus (Norway rat)0.0582
SortilinHomo sapiens (human)0.36

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Forgez, P; Hermans, E; Lebeau, A; Lhiaubet, AM; Pelaprat, D; Rostene, W; Skrzydelski, D; Yamada, M1
Machida, R; Tsushima, Y; Watanabe, S; Yamakawa, I1
Abe, K; Machida, R; Sasaki, A; Tanaka, T; Tokumura, T; Tsuchiya, Y1
Abe, K; Machida, R; Saeki, Y; Sasaki, A; Tanaka, T; Tokumura, T; Tsuchiya, Y1
Abe, K; Machida, R; Sasaki, A; Tokumura, T; Tsuchiya, Y1

Other Studies

5 other study(ies) available for methylarginyl-lysyl-prolyl-tryptophyl-tert-leucyl-leucyl-ethyl ester and neurotensin

ArticleYear
Differential involvement of intracellular domains of the rat NTS1 neurotensin receptor in coupling to G proteins: a molecular basis for agonist-directed trafficking of receptor stimulus.
    Molecular pharmacology, 2003, Volume: 64, Issue:2

    Topics: Animals; Arachidonic Acid; CHO Cells; Cricetinae; Cyclic AMP; GTP-Binding Proteins; Oligopeptides; Phosphotransferases (Alcohol Group Acceptor); Protein Structure, Tertiary; Rats; Receptors, Neurotensin; Tritium

2003
Preparation of neurotensin analogue-containing poly(dl-lactic acid) microspheres formed by oil-in-water solvent evaporation.
    Journal of pharmaceutical sciences, 1992, Volume: 81, Issue:9

    Topics: Amino Acid Sequence; Lactates; Lactic Acid; Microspheres; Molecular Sequence Data; Neurotensin; Oligopeptides; Peptide Fragments; Polyesters; Polymers; Solvents

1992
Stability of a novel hexapeptide, (Me)Arg-Lys-Pro-Trp-tert-Leu-Leu-OEt, with neurotensin activity, in aqueous solution and in the solid state.
    Chemical & pharmaceutical bulletin, 1990, Volume: 38, Issue:11

    Topics: Amino Acid Sequence; Drug Stability; Molecular Sequence Data; Neurotensin; Oligopeptides; Psychotropic Drugs; Solutions

1990
Pharmacokinetics of (Me)Arg-Lys-Pro-Trp-tert-Leu-Leu-OEt and (Me)Arg-Lys-Pro-Trp-tert-Leu-Leu administered intravenously to beagle dogs.
    Journal of pharmaceutical sciences, 1993, Volume: 82, Issue:7

    Topics: Amino Acid Sequence; Animals; Blood Proteins; Chemical Phenomena; Chemistry, Physical; Dogs; Half-Life; Injections, Intravenous; Male; Molecular Sequence Data; Neurotensin; Oligopeptides; Peptide Fragments; Protein Binding

1993
Pharmacokinetics of novel hexapeptides with neurotensin activity in rats.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:1

    Topics: Administration, Oral; Amino Acid Sequence; Animals; Biological Availability; Chromatography, High Pressure Liquid; Half-Life; Injections, Intravenous; Intestine, Small; Male; Molecular Sequence Data; Neurotensin; Oligopeptides; Rats; Rats, Wistar; Reproducibility of Results

1993