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methotrimeprazine and acetaminophen

methotrimeprazine has been researched along with acetaminophen in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19903 (30.00)18.7374
1990's0 (0.00)18.2507
2000's5 (50.00)29.6817
2010's2 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Lombardo, F; Obach, RS; Waters, NJ1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Rogers, AG1
Linscott, MS1
Cliff, JM1
Brørs, O; Pettersen, S; Tallaksen, C; Vevelstad, M1

Reviews

1 review(s) available for methotrimeprazine and acetaminophen

ArticleYear
Non-narcotic analgesics--their use and abuse.
    Journal of the Royal Naval Medical Service, 1972,Spring, Volume: 58, Issue:1

    Topics: Acetaminophen; Analgesics; Anti-Inflammatory Agents; Aspirin; Dextropropoxyphene; Drug Synergism; Flufenamic Acid; Humans; Indomethacin; Mefenamic Acid; Methotrimeprazine; Orphenadrine; Oxyphenbutazone; Pentazocine; Phenacetin; Phenylbutazone; Propionates; Tablets

1972

Trials

1 trial(s) available for methotrimeprazine and acetaminophen

ArticleYear
O-demethylation of codeine to morphine inhibited by low-dose levomepromazine.
    European journal of clinical pharmacology, 2009, Volume: 65, Issue:8

    Topics: Acetaminophen; Administration, Oral; Adult; Aged; Analgesics, Non-Narcotic; Analgesics, Opioid; Codeine; Cytochrome P-450 CYP2D6; Drug Administration Schedule; Female; Genotype; Humans; Low Back Pain; Male; Methotrimeprazine; Methylation; Middle Aged; Oxidoreductases, O-Demethylating; Urinalysis

2009

Other Studies

8 other study(ies) available for methotrimeprazine and acetaminophen

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
    Journal of medicinal chemistry, 2001, Jul-19, Volume: 44, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water

2001
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
The use of methotrimeprazine (Levoprome) in a patient sensitive to opioids and possible bowel shutdown.
    Journal of pain and symptom management, 1989, Volume: 4, Issue:1

    Topics: Acetaminophen; Adenocarcinoma; Female; Humans; Intestinal Obstruction; Lung Neoplasms; Methotrimeprazine; Middle Aged; Narcotics; Pain

1989
Analgesics in the management of acute pain.
    Clinical therapeutics, 1986, Volume: 9, Issue:1

    Topics: Acetaminophen; Analgesics; Analgesics, Opioid; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Drug Therapy, Combination; Humans; Methotrimeprazine; Nitrous Oxide; Pain

1986