methoctramine and naloxone

methoctramine has been researched along with naloxone in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's3 (75.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Abe, K; Chikuma, T; Hojyo, H; Kato, M; Miyatake, T; Taguchi, K; Utsunomiya, I1
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO1
Bellucci, C; Buccioni, M; Ghelardini, C; Marucci, G; Melchiorre, C; Milelli, A; Minarini, A; Rosini, M; Tumiatti, V1

Reviews

1 review(s) available for methoctramine and naloxone

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993

Other Studies

3 other study(ies) available for methoctramine and naloxone

ArticleYear
Characterization of muscarinic receptor subtypes in the rostral ventrolateral medulla and effects on morphine-induced antinociception in rats.
    European journal of pharmacology, 2003, Apr-04, Volume: 465, Issue:3

    Topics: Analgesics, Opioid; Animals; Atropine; Diamines; Male; Mecamylamine; Medulla Oblongata; Microinjections; Morphine; Naloxone; Narcotic Antagonists; Pain Measurement; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Time Factors

2003
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
    Journal of medicinal chemistry, 2005, Nov-03, Volume: 48, Issue:22

    Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles

2005
Structure-activity relationships of methoctramine-related polyamines as muscarinic antagonist: effect of replacing the inner polymethylene chain with cyclic moieties.
    Bioorganic & medicinal chemistry, 2007, Mar-15, Volume: 15, Issue:6

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Butyrylcholinesterase; Cerebral Cortex; CHO Cells; Cholinesterase Inhibitors; Cricetinae; Cricetulus; Diamines; Drug Design; Drug Evaluation, Preclinical; Guinea Pigs; Heart Atria; Humans; Ileum; Male; Mice; Molecular Structure; Muscarinic Antagonists; Muscle, Skeletal; Parietal Lobe; Photoaffinity Labels; Polyamines; Rabbits; Radioligand Assay; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Vas Deferens

2007