methoctramine has been researched along with aq-ra 741 in 6 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (83.33) | 18.2507 |
2000's | 1 (16.67) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Hamstra, JJ; Roffel, AF; Santing, RE; ten Berge, RE; Zaagsma, J | 1 |
Budriesi, R; Chiarini, A; Melchiorre, C; Minarini, A; Spampinato, S; Tumiatti, V | 1 |
Daniels, DV; Eglen, RM; Ford, AP; Hegde, SS; Meloy, TD | 1 |
Brann, MR; Dörje, F; Lambrecht, G; Mutschler, E; Tacke, R; Wess, J | 1 |
Bolognesi, ML; Budriesi, R; Canossa, M; Chiarini, A; Melchiorre, C; Minarini, A; Spampinato, S | 1 |
Bolognesi, ML; Chiarini, A; Melchiorre, C; Minarini, A; Spampinato, S | 1 |
6 other study(ies) available for methoctramine and aq-ra 741
Article | Year |
---|---|
Dysfunction of muscarinic M2 receptors after the early allergic reaction: possible contribution to bronchial hyperresponsiveness in allergic guinea-pigs.
Topics: Administration, Inhalation; Allergens; Animals; Asthma; Benzodiazepinones; Bronchial Hyperreactivity; Diamines; Disease Models, Animal; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart; Histamine; Hypersensitivity; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle, Smooth; Neuromuscular Junction; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea | 1995 |
The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists.
Topics: Animals; Atrial Function; Benzodiazepines; Benzodiazepinones; Diamines; Drug Design; Guinea Pigs; Heart Atria; Ileum; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Submandibular Gland; Trachea | 1995 |
Functional characterization of rat submaxillary gland muscarinic receptors using microphysiometry.
Topics: Alkaloids; Animals; Atropine; Benzhydryl Compounds; Benzodiazepinones; Binding, Competitive; Biosensing Techniques; Carbachol; Cholinergic Agonists; Cresols; Diamines; Dose-Response Relationship, Drug; Furans; Male; Mandelic Acids; Muscarinic Antagonists; Naphthalenes; Phenethylamines; Phenylpropanolamine; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Submandibular Gland; Tolterodine Tartrate | 2001 |
Antagonist binding profiles of five cloned human muscarinic receptor subtypes.
Topics: Animals; Cells, Cultured; Cricetinae; Humans; N-Methylscopolamine; Parasympatholytics; Receptors, Muscarinic; Scopolamine Derivatives; Transfection | 1991 |
Design, synthesis, and biological activity of methoctramine-related tetraamines bearing an 11-acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4] benzodiazepin-6-one moiety: structural requirements for optimum occupancy of muscarinic receptor subtypes as revealed b
Topics: Animals; Atrial Function; Benzodiazepines; Cells, Cultured; Cerebral Cortex; Drug Design; Female; Guinea Pigs; Heart Atria; Ileum; Male; Molecular Structure; Muscarinic Antagonists; Muscle Contraction; Myocardial Contraction; Myocardium; Polyamines; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Submandibular Gland | 1994 |
Synthesis and biological activity of some methoctramine-related tetraamines bearing a 11-acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]-benzodiazepin-6-one moiety as antimuscarinics: a second generation of highly selective M2 muscarinic receptor antagonists.
Topics: Animals; Benzodiazepines; Diamines; Guinea Pigs; Molecular Structure; Muscarinic Antagonists; Rats; Receptors, Muscarinic; Structure-Activity Relationship | 1993 |