methadone and saquinavir

methadone has been researched along with saquinavir in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (8.33)18.2507
2000's7 (58.33)29.6817
2010's4 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Brown, AM; Bruening-Wright, A; Kramer, J; Kuryshev, YA; Myatt, G; Obejero-Paz, CA; Verducci, JS1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Berthou, F; Carlhant, D; Dreano, Y; Iribarne, C; Lohezic, F; Picart, D; Riche, C1
Erickson, AD; Geletko, SM1
Aberg, J; Aweeka, F; D'Amico, R; Flexner, C; Gal, J; Gerber, JG; Gulick, R; Hsu, A; Hughes, V; Mildvan, D; Rosenkranz, S; Segal, Y1
Berenson, CS; Buggé, CJ; Cloen, D; de Caprariis, PJ; DiFrancesco, R; Esch, A; Espinosa, O; Hewitt, RG; Ljungqvist, A; Palic, B; Schur, JL; Shelton, MJ1
Coles, LD; Eddington, ND; Hassan, HE; Lee, IJ1
Jamois, C; Morcos, PN; Morrison, R; Patel, A; Riek, M; Schmitt, C; Smith, P; Zhang, X1
Barberan, O; Dubus, E; Ijjaali, I; Petitet, F1

Reviews

1 review(s) available for methadone and saquinavir

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

2 trial(s) available for methadone and saquinavir

ArticleYear
Effect of ritonavir/saquinavir on stereoselective pharmacokinetics of methadone: results of AIDS Clinical Trials Group (ACTG) 401.
    Journal of acquired immune deficiency syndromes (1999), 2001, Jun-01, Volume: 27, Issue:2

    Topics: Adult; Drug Interactions; Female; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Male; Methadone; Middle Aged; Narcotics; Ritonavir; Saquinavir; Stereoisomerism; Substance Abuse, Intravenous

2001
The effects of once-daily saquinavir/minidose ritonavir on the pharmacokinetics of methadone.
    Journal of clinical pharmacology, 2004, Volume: 44, Issue:3

    Topics: Adult; Chromatography, Liquid; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; HIV Protease Inhibitors; Humans; Male; Mass Spectrometry; Metabolic Clearance Rate; Methadone; Middle Aged; Narcotics; Ritonavir; Saquinavir; Stereoisomerism; Time Factors

2004

Other Studies

9 other study(ies) available for methadone and saquinavir

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
MICE models: superior to the HERG model in predicting Torsade de Pointes.
    Scientific reports, 2013, Volume: 3

    Topics: ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Models, Theoretical; Patch-Clamp Techniques; Predictive Value of Tests; Torsades de Pointes

2013
Inhibition of methadone and buprenorphine N-dealkylations by three HIV-1 protease inhibitors.
    Drug metabolism and disposition: the biological fate of chemicals, 1998, Volume: 26, Issue:3

    Topics: Alkylation; Buprenorphine; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; HIV Protease Inhibitors; Humans; Indinavir; Kinetics; Methadone; Microsomes, Liver; Mixed Function Oxygenases; Oxidoreductases, N-Demethylating; Ritonavir; Saquinavir

1998
Decreased methadone effect after ritonavir initiation.
    Pharmacotherapy, 2000, Volume: 20, Issue:1

    Topics: Analgesics, Opioid; Anti-HIV Agents; Diagnosis, Differential; Drug Interactions; Drug Therapy, Combination; HIV Infections; HIV Protease Inhibitors; Humans; Male; Methadone; Middle Aged; Ritonavir; Saquinavir; Stavudine; Substance Withdrawal Syndrome; Substance-Related Disorders

2000
Distribution of saquinavir, methadone, and buprenorphine in maternal brain, placenta, and fetus during two different gestational stages of pregnancy in mice.
    Journal of pharmaceutical sciences, 2009, Volume: 98, Issue:8

    Topics: Animals; Brain; Buprenorphine; Female; Fetal Development; Fetus; Maternal Exposure; Maternal-Fetal Exchange; Methadone; Mice; Placenta; Pregnancy; Pregnancy, Animal; Saquinavir; Tissue Distribution

2009
Effect of saquinavir/ritonavir (1000/100 mg bid) on the pharmacokinetics of methadone in opiate-dependent HIV-negative patients on stable methadone maintenance therapy.
    Addiction biology, 2009, Volume: 14, Issue:3

    Topics: Administration, Oral; Adult; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Female; HIV Protease Inhibitors; HIV Seronegativity; Humans; Male; Methadone; Middle Aged; Narcotics; Opioid-Related Disorders; Protein Binding; Ritonavir; Saquinavir

2009
Drug repositioning using in silico compound profiling.
    Future medicinal chemistry, 2009, Volume: 1, Issue:9

    Topics: Benzimidazoles; Benzoates; Databases, Factual; Drug Repositioning; Methadone; Receptor, Muscarinic M3; Receptors, Cytoplasmic and Nuclear; Receptors, Gastrointestinal Hormone; Receptors, Neurokinin-2; Receptors, Neuropeptide; Saquinavir; Sirolimus; Telmisartan

2009