Page last updated: 2024-08-23

metergoline and methiothepin

metergoline has been researched along with methiothepin in 46 studies

Research

Studies (46)

TimeframeStudies, this research(%)All Research%
pre-199016 (34.78)18.7374
1990's22 (47.83)18.2507
2000's7 (15.22)29.6817
2010's1 (2.17)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beer, MS; Charlesworth, A; Iversen, LL; McAllister, G; Middlemiss, DN; Noble, AJ; Snodin, C; Whiting, P1
Hamblin, MW; Metcalf, MA1
Hamblin, MW; Monsma, FJ; Shen, Y; Sibley, DR; Ward, RP1
Bull, D; den Daas, I; Foord, S; Goodson, S; Kilpatrick, G; Lee, M; Rees, S1
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J1
Adham, N; Bard, J; Branchek, TA; Durkin, M; Hartig, PR; Kao, HT; Olsen, M; Schecter, LE; Urquhart, D; Weinshank, RL1
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR1
Amlaiky, N; Hen, R; Plassat, JL1
Druck, T; Hamblin, MW; Huebner, K; Khan, N; Kohen, R; Lachowicz, JE; Meltzer, HY; Metcalf, MA; Roth, BL; Sibley, DR1
Izzarelli, DG; Lewis-Higgins, L; Palmer, D; Parker, EM; Shapiro, RA1
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R1
Boess, FG; Meyer, V; Monsma, FJ; Sleight, AJ; Zwingelstein, C1
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP1
Beleta, J; Doménech, T; Palacios, JM1
Bentley, J; Boess, FG; Bös, M; Bourson, A; Riemer, C; Sleight, AJ1
Boess, FG; Monsma, FJ; Sleight, AJ1
Bach, T; Krobert, KA; Kvingedal, AM; Levy, FO; Syversveen, T1
Bai, F; Johnstone, EM; Little, SP; Nelson, DL; Su, C; Varga, G; Yin, T1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Bergeron, C; Bolton, JL; Budzinski, JW; Dietz, BM; Foster, BC; Gafner, S; Glinski, JA; McCollom, MM; McPhail, KL; Rhyu, MR; Russell, FE; Scott, IM1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Lepailleur, A; Rochais, C; Thirumaran, SL1
Artaud, F; Bockaert, J; Bourgoin, S; Glowinski, J; Hamon, M; Héry, F1
Deicher, R; Limberger, N; Starke, K1
Buda, M; Devau, G; Multon, MF; Pujol, JF1
Feuerstein, TJ; Hertting, G; Lupp, A1
Houston, DS; Vanhoutte, PM1
Eide, PK; Tjølsen, A1
Ramage, AG1
Lis, EV; Martin, GE1
Svensson, L1
Choquet, D; Korn, H1
Cohen, RA1
Ristine, LA; Spear, LP1
Berge, OG1
Buda, C; Janin, M; Jouvet, M; Sallanon, M1
Ahlenius, S; Larsson, K1
Laguzzi, R1
Aghajanian, GK; McCall, RB1
Duncan, J; Fong, PP; Ram, JL1
Castillo, C; Castillo, E; López-Muñoz, FJ; Ramírez-San Juan, E; Terrón, JA; Villalón, CM1
Beattie, DT; Connor, HE; Walsh, DM1
Masek, K; Ruzicka, V; Sevcík, J; Slánsky, J1
De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM1
Centurión, D; Gupta, S; MaassenVanDenBrink, A; Mehotra, S; Sánchez-López, A; Villalón, CM1
Bray, JK; Goddard, WA1

Reviews

1 review(s) available for metergoline and methiothepin

ArticleYear
Structure-activity relationships of serotonin 5-HT
    European journal of medicinal chemistry, 2019, Dec-01, Volume: 183

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

2019

Other Studies

45 other study(ies) available for metergoline and methiothepin

ArticleYear
Molecular cloning of a serotonin receptor from human brain (5HT1E): a fifth 5HT1-like subtype.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Jun-15, Volume: 89, Issue:12

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Base Sequence; Binding, Competitive; Cell Line; Cloning, Molecular; Colforsin; DNA; Frontal Lobe; Gene Library; GTP-Binding Proteins; Hippocampus; Humans; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Receptors, Serotonin; Recombinant Proteins; Restriction Mapping; Sequence Homology, Nucleic Acid; Serotonin; Transfection

1992
Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor.
    Molecular pharmacology, 1991, Volume: 40, Issue:2

    Topics: Amino Acid Sequence; Base Sequence; Cloning, Molecular; Cyclic AMP; GTP-Binding Proteins; Humans; Molecular Sequence Data; Pertussis Toxin; Receptors, Serotonin; Virulence Factors, Bordetella

1991
Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain Chemistry; Cell Line; Cloning, Molecular; DNA; GTP-Binding Proteins; Lysergic Acid Diethylamide; Molecular Sequence Data; Polymerase Chain Reaction; Psychotropic Drugs; Rats; Receptors, Serotonin; RNA; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Transfection

1993
Cloning and characterisation of the human 5-HT5A serotonin receptor.
    FEBS letters, 1994, Dec-05, Volume: 355, Issue:3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Genome, Human; GTP-Binding Proteins; Humans; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Serotonin; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid; Serotonin; Tissue Distribution; Transfection

1994
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.
    The Journal of biological chemistry, 1993, Nov-05, Volume: 268, Issue:31

    Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction

1993
Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Jan-15, Volume: 90, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Colforsin; Dose-Response Relationship, Drug; Gene Library; Guinea Pigs; Humans; Indoles; Lymphocytes; Molecular Sequence Data; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Serotonin; Serotonin Receptor Agonists; Spiperone; Sulfonamides; Sumatriptan; Tissue Distribution

1993
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
    The Journal of biological chemistry, 1993, Aug-25, Volume: 268, Issue:24

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection

1993
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.
    Molecular pharmacology, 1993, Volume: 44, Issue:2

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Cyclic AMP; DNA; Drosophila; Enzyme Activation; Humans; Intestinal Mucosa; Mice; Molecular Sequence Data; Myocardium; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists

1993
Cloning, characterization, and chromosomal localization of a human 5-HT6 serotonin receptor.
    Journal of neurochemistry, 1996, Volume: 66, Issue:1

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line, Transformed; Chlorocebus aethiops; Chromosome Mapping; Chromosomes, Human, Pair 1; Cloning, Molecular; Clozapine; DNA, Complementary; Genes; Humans; Kinetics; Molecular Sequence Data; Open Reading Frames; Protein Conformation; Rats; Receptors, Serotonin; Recombinant Proteins; Sequence Alignment; Sequence Homology, Nucleic Acid; Serotonin Agents; Signal Transduction; Species Specificity

1996
Two amino acid differences in the sixth transmembrane domain are partially responsible for the pharmacological differences between the 5-HT1D beta and 5-HT1E 5-hydroxytryptamine receptors.
    Journal of neurochemistry, 1996, Volume: 67, Issue:5

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Binding, Competitive; Chlorocebus aethiops; Cloning, Molecular; COS Cells; DNA Primers; Ergolines; Glutamic Acid; Humans; Isoleucine; Kinetics; Ligands; Lysine; Models, Structural; Molecular Sequence Data; Point Mutation; Polymerase Chain Reaction; Protein Structure, Secondary; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombinant Fusion Proteins; Sequence Homology, Amino Acid; Serine; Serotonin; Transfection

1996
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
    Molecular pharmacology, 1996, Volume: 50, Issue:6

    Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents

1996
Interaction of tryptamine and ergoline compounds with threonine 196 in the ligand binding site of the 5-hydroxytryptamine6 receptor.
    Molecular pharmacology, 1997, Volume: 52, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding Sites; Cells, Cultured; Cloning, Molecular; Cricetinae; Dogs; Drug Interactions; Ergolines; Guinea Pigs; Humans; Kidney; Ligands; Lysergic Acid Diethylamide; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Rats; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin; Threonine; Tryptamines

1997
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
    British journal of pharmacology, 1997, Volume: 122, Issue:1

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid

1997
Characterization of human serotonin 1D and 1B receptors using [3H]-GR-125743, a novel radiolabelled serotonin 5HT1D/1B receptor antagonist.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:3

    Topics: Benzamides; Binding, Competitive; Gene Expression; HeLa Cells; Humans; Kinetics; Ligands; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Substantia Nigra; Tritium

1997
The 5-hydroxytryptamine6 receptor-selective radioligand [3H]Ro 63-0563 labels 5-hydroxytryptamine receptor binding sites in rat and porcine striatum.
    Molecular pharmacology, 1998, Volume: 54, Issue:3

    Topics: Aminopyridines; Animals; Binding Sites; Corpus Striatum; HeLa Cells; Humans; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin Antagonists; Species Specificity; Swine; Tritium

1998
Identification of residues in transmembrane regions III and VI that contribute to the ligand binding site of the serotonin 5-HT6 receptor.
    Journal of neurochemistry, 1998, Volume: 71, Issue:5

    Topics: Adenylyl Cyclases; Amino Acid Substitution; Binding Sites; Binding, Competitive; Cell Line; Cyclic AMP; Humans; Ligands; Lysergic Acid Diethylamide; Mutagenesis, Site-Directed; Mutation; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists

1998
The cloned human 5-HT7 receptor splice variants: a comparative characterization of their pharmacology, function and distribution.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:6

    Topics: Adenylyl Cyclases; Alternative Splicing; Binding, Competitive; Brain; Cell Line; Cloning, Organism; Genetic Variation; Humans; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tissue Distribution

2001
Molecular cloning and pharmacological characterization of the guinea pig 5-HT1E receptor.
    European journal of pharmacology, 2004, Jan-26, Volume: 484, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Chickens; Cloning, Molecular; Cricetinae; Dose-Response Relationship, Drug; Gerbillinae; Guinea Pigs; Haplorhini; Humans; Molecular Sequence Data; Protein Binding; Rabbits; Receptors, Serotonin; Serotonin Agents; Swine

2004
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Alkaloids from Eschscholzia californica and their capacity to inhibit binding of [3H]8-Hydroxy-2-(di-N-propylamino)tetralin to 5-HT1A receptors in Vitro.
    Journal of natural products, 2006, Volume: 69, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alkaloids; Benzylisoquinolines; Dioxoles; Eschscholzia; Humans; Molecular Structure; Receptor, Serotonin, 5-HT1A; Serotonin Receptor Agonists

2006
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Paradoxical decrease of brain 5-HT turnover by metergoline, a central 5-HT receptor blocker.
    Naunyn-Schmiedeberg's archives of pharmacology, 1978, Volume: 302, Issue:3

    Topics: Adenylyl Cyclases; Animals; Brain; Ergolines; In Vitro Techniques; Indoles; Lysergic Acid Diethylamide; Male; Membranes; Metergoline; Methiothepin; Potassium; Rats; Receptors, Serotonin; Serotonin; Synaptosomes

1978
Species differences in presynaptic serotonin autoreceptors: mainly 5-HT1B but possibly in addition 5-HT1D in the rat, 5-HT1D in the rabbit and guinea-pig brain cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:4

    Topics: Animals; Brain; Dioxanes; Electric Stimulation; Female; Guinea Pigs; Idazoxan; Male; Metergoline; Methiothepin; Rabbits; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Species Specificity; Tritium

1991
Inhibition of tyrosine hydroxylase activity by serotonin in explants of newborn rat locus ceruleus.
    Journal of neurochemistry, 1987, Volume: 49, Issue:3

    Topics: Amanitins; Animals; Animals, Newborn; Cycloheximide; Locus Coeruleus; Metergoline; Methiothepin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tyrosine 3-Monooxygenase

1987
The serotonin (5-HT) autoreceptor in the hippocampus of the rabbit: role of 5-HT biophase concentration.
    Neuropharmacology, 1987, Volume: 26, Issue:8

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Hippocampus; Mathematics; Metergoline; Methiothepin; Methoxydimethyltryptamines; Methysergide; Phentolamine; Pindolol; Quipazine; Rabbits; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1987
Comparison of serotonergic receptor subtypes on the smooth muscle and endothelium of the canine coronary artery.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Coronary Vessels; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Ketanserin; Male; Metergoline; Methiothepin; Muscle, Smooth, Vascular; Pindolol; Receptors, Serotonin; Tetrahydronaphthalenes; Vasodilation

1988
Effects of serotonin receptor antagonists and agonists on the tail-flick response in mice involve altered tail-skin temperature.
    Neuropharmacology, 1988, Volume: 27, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Hypothermia, Induced; Male; Metergoline; Methiothepin; Methoxydimethyltryptamines; Mice; Mice, Inbred Strains; Reaction Time; Receptors, Serotonin; Skin Temperature; Tetrahydronaphthalenes

1988
Examination of the effects of some 5-HT2 receptor antagonists on central sympathetic outflow and blood pressure in anaesthetised cats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:6

    Topics: Anesthesia; Animals; Blood Pressure; Cats; Cinanserin; Cyproheptadine; Male; Metergoline; Methiothepin; Piperidines; Quinolines; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System

1988
Hypotensive action of 8-hydroxy-2-(di-N-propylamino)tetralin (8-OH-DPAT) in spontaneously hypertensive rats.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 273, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Administration, Oral; Animals; Antihypertensive Agents; Blood Pressure; Cyproheptadine; Heart Rate; Injections, Intraperitoneal; Injections, Intraventricular; Male; Metergoline; Methiothepin; Naphthalenes; Rats; Rats, Inbred SHR; Tetrahydronaphthalenes

1985
Effects of 8-OH-DPAT, lisuride and some ergot-related compounds on the acoustic startle response in the rat.
    Psychopharmacology, 1985, Volume: 85, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bromocriptine; Ergolines; Lisuride; Male; Metergoline; Methiothepin; Naphthalenes; Pergolide; Quinpirole; Rats; Rats, Inbred Strains; Reflex, Startle; Tetrahydronaphthalenes

1985
Dual effects of serotonin on a voltage-gated conductance in lymphocytes.
    Proceedings of the National Academy of Sciences of the United States of America, 1988, Volume: 85, Issue:12

    Topics: Abelson murine leukemia virus; Animals; B-Lymphocytes; Cell Line, Transformed; Electric Conductivity; Indoles; Ketanserin; Membrane Potentials; Metergoline; Methiothepin; Mice; Potassium; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1988
Serotonergic prejunctional inhibition of canine coronary adrenergic nerves.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:1

    Topics: Acetylcholine; Animals; Coronary Vessels; Dogs; Electric Stimulation; Epinephrine; Ergolines; Heart Conduction System; Metergoline; Methiothepin; Neuromuscular Junction; Serotonin; Vasoconstriction

1985
Suckling behavior in neonatal rats: psychopharmacological investigations.
    Journal of comparative and physiological psychology, 1982, Volume: 96, Issue:2

    Topics: Animals; Animals, Newborn; Haloperidol; Metergoline; Methiothepin; Methysergide; Naloxone; Neurotransmitter Agents; Phentolamine; Propranolol; Rats; Rats, Inbred Strains; Scopolamine; Sucking Behavior

1982
Effects of 5-HT receptor agonists and antagonists on a reflex response to radiant heat in normal and spinally transected rats.
    Pain, 1982, Volume: 13, Issue:3

    Topics: 5-Hydroxytryptophan; Animals; Carbidopa; Circadian Rhythm; Hot Temperature; Male; Metergoline; Methiothepin; Mianserin; Neurotransmitter Agents; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Spinal Cord

1982
5-HT antagonists suppress sleep and delay its restoration after 5-HTP in p-chlorophenylalanine-pretreated cats.
    European journal of pharmacology, 1982, Aug-13, Volume: 82, Issue:1-2

    Topics: 5-Hydroxytryptophan; Animals; Cats; Female; Fenclonine; Humans; Male; Metergoline; Methiothepin; Serotonin Antagonists; Sleep; Sleep Initiation and Maintenance Disorders; Sleep, REM

1982
Failure to antagonize the 8-hydroxy-2-di-n-propylamino)tetralin-induced facilitation of male rat sexual behavior by the administration of 5-HT receptor antagonists.
    European journal of pharmacology, 1984, Apr-06, Volume: 99, Issue:4

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Female; Male; Metergoline; Methiothepin; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Sexual Behavior, Animal; Tetrahydronaphthalenes

1984
[Effects of the intraventricular injection of methiothepin and methergoline on the sleep of rats].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1981, Volume: 175, Issue:2

    Topics: Animals; Dibenzothiepins; Ergolines; Injections, Intraventricular; Male; Metergoline; Methiothepin; Rats; Sleep; Sleep Stages; Sleep, REM

1981
Pharmacological characterization of serotonin receptors in the facial motor nucleus: a microiontophoretic study.
    European journal of pharmacology, 1980, Jul-25, Volume: 65, Issue:2-3

    Topics: Animals; Cinanserin; Cyproheptadine; Facial Nerve; Iontophoresis; Male; Metergoline; Methiothepin; Methysergide; Motor Neurons; Norepinephrine; Propranolol; Rats; Receptors, Serotonin

1980
Inhibition and sex specific induction of spawning by serotonergic ligands in the zebra mussel Dreissena polymorpha (Pallas).
    Experientia, 1994, May-15, Volume: 50, Issue:5

    Topics: Animals; Dose-Response Relationship, Drug; Female; Male; Metergoline; Methiothepin; Mollusca; Reproduction; Serotonin

1994
Pharmacological profile of the receptors that mediate external carotid vasoconstriction by 5-HT in vagosympathectomized dogs.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: Animals; Carotid Artery, External; Dogs; Dose-Response Relationship, Drug; Female; Hemodynamics; Male; Metergoline; Methiothepin; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathectomy; Vagus Nerve; Vasoconstriction

1995
The activity of 5-HT1D receptor ligands at cloned human 5-HT1D alpha and 5-HT1D beta receptors.
    European journal of pharmacology, 1995, Dec-04, Volume: 287, Issue:1

    Topics: Cyclic AMP; HeLa Cells; Humans; Metergoline; Methiothepin; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan

1995
Which type of 5-hydroxytryptamine receptor mediates relaxation of the longitudinal muscle of guinea pig proximal colon in vitro?
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:7

    Topics: Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Metergoline; Methiothepin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron

1996
Nature of 5-HT1-like receptors mediating depressor responses in vagosympathectomized rats; close resemblance to the cloned 5-ht7 receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: 5-Methoxytryptamine; Adrenergic beta-Agonists; Animals; Blood Pressure; Clozapine; Ergolines; Heart Rate; Isoproterenol; Lisuride; Male; Metergoline; Methiothepin; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathectomy

1997
Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat.
    European journal of pharmacology, 2006, Mar-27, Volume: 535, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Buspirone; Clozapine; Decerebrate State; Dose-Response Relationship, Drug; Drug Interactions; Ergotamine; Heart Rate; Ketanserin; Lisuride; Male; Metergoline; Methiothepin; Methysergide; Phenylephrine; Piperazines; Pizotyline; Prazosin; Pyridines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Serotonin Antagonists; Serotonin Receptor Agonists; Yohimbine

2006
The structure of human serotonin 2c G-protein-coupled receptor bound to agonists and antagonists.
    Journal of molecular graphics & modelling, 2008, Volume: 27, Issue:1

    Topics: Amino Acid Sequence; Binding Sites; Humans; Kinetics; Metergoline; Methiothepin; Molecular Sequence Data; Mutagenesis; Protein Structure, Secondary; Psilocybin; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Structure-Activity Relationship; Thermodynamics

2008