Page last updated: 2024-08-23

metergoline and buspirone

metergoline has been researched along with buspirone in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19901 (7.69)18.7374
1990's7 (53.85)18.2507
2000's4 (30.77)29.6817
2010's1 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA1
Amlaiky, N; Hen, R; Plassat, JL1
Arrang, JM; Diaz, J; Leurs, R; Ruat, M; Schwartz, JC; Tardivel-Lacombe, J; Traiffort, E1
Adkison, KK; Humphreys, JE; Mahar Doan, KM; Polli, JW; Serabjit-Singh, CJ; Shampine, LJ; Webster, LO; Wring, SA1
Duncton, MA; Emerling, DE; Kelly, MG; Nguyen, MT; Vincent, F1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Coccaro, EF; Gabriel, S; Macaluso, J; Mahon, T; Siever, LJ1
Coccaro, EF; Gabriel, S; Siever, LJ1
Anderson, IM; Cowen, PJ; Gregory, CA1
Kellar, KJ; Lumpkin, MD; Mulroney, SE; Shemer, A; Skudlarek, C1
Costall, B; Neill, JC; Wilson, AW1
Mohanakumar, KP; Muralikrishnan, D; Sarkar, S; Thomas, B1
Centurión, D; Gupta, S; MaassenVanDenBrink, A; Mehotra, S; Sánchez-López, A; Villalón, CM1

Reviews

1 review(s) available for metergoline and buspirone

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987

Trials

1 trial(s) available for metergoline and buspirone

ArticleYear
Preliminary evidence of a serotonin (5-HT-1-like) component to the prolactin response to buspirone challenge in humans.
    Archives of general psychiatry, 1990, Volume: 47, Issue:6

    Topics: Adrenocorticotropic Hormone; Adult; Buspirone; Cortisone; Growth Hormone; Humans; Male; Metergoline; Pindolol; Prolactin; Receptors, Dopamine; Receptors, Serotonin

1990

Other Studies

11 other study(ies) available for metergoline and buspirone

ArticleYear
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.
    Molecular pharmacology, 1993, Volume: 44, Issue:2

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Cyclic AMP; DNA; Drosophila; Enzyme Activation; Humans; Intestinal Mucosa; Mice; Molecular Sequence Data; Myocardium; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists

1993
Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Sep-15, Volume: 90, Issue:18

    Topics: Amino Acid Sequence; Animals; Base Sequence; Blotting, Northern; Brain; CHO Cells; Cricetinae; Cyclic AMP; DNA; Genomic Library; Kinetics; Lysergic Acid Diethylamide; Mianserin; Molecular Sequence Data; Multigene Family; Oligodeoxyribonucleotides; Organ Specificity; Rats; Receptors, Serotonin; Restriction Mapping; Serotonin; Serotonin Receptor Agonists; Transfection

1993
Passive permeability and P-glycoprotein-mediated efflux differentiate central nervous system (CNS) and non-CNS marketed drugs.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Cell Line; Cell Membrane Permeability; Central Nervous System Agents; Dogs; Drug Delivery Systems; Permeability; Pharmaceutical Preparations

2002
Mining biologically-active molecules for inhibitors of fatty acid amide hydrolase (FAAH): identification of phenmedipham and amperozide as FAAH inhibitors.
    Bioorganic & medicinal chemistry letters, 2009, Dec-01, Volume: 19, Issue:23

    Topics: Amidohydrolases; Carbamates; Dose-Response Relationship, Drug; Drug Design; Enzyme Inhibitors; Humans; Models, Molecular; Molecular Structure; Piperazines; Stereoisomerism; Structure-Activity Relationship

2009
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Buspirone challenge: preliminary evidence for a role for central 5-HT1a receptor function in impulsive aggressive behavior in humans.
    Psychopharmacology bulletin, 1990, Volume: 26, Issue:3

    Topics: Adult; Aggression; Buspirone; Female; Humans; Male; Metergoline; Personality Disorders; Pindolol; Prolactin; Receptors, Serotonin

1990
Metergoline abolishes the prolactin response to buspirone.
    Psychopharmacology, 1990, Volume: 100, Issue:2

    Topics: Adult; Buspirone; Ergolines; Female; Humans; Male; Metergoline; Prolactin; Radioimmunoassay

1990
Tandospirone stimulates prolactin secretion in the rat by an action at serotonin-1A receptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Dose-Response Relationship, Drug; Isoindoles; Male; Metergoline; Piperazines; Prolactin; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists

1994
An investigation into the effects of 5-HT agonists and receptor antagonists on ethanol self-administration in the rat.
    Alcohol (Fayetteville, N.Y.), 1998, Volume: 16, Issue:3

    Topics: Animals; Buspirone; Dose-Response Relationship, Drug; Ethanol; Female; Fenfluramine; Fluoxetine; Metergoline; Ondansetron; Piperazines; Rats; Rats, Sprague-Dawley; Ritanserin; Selective Serotonin Reuptake Inhibitors; Self Administration; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors

1998
Effects of serotoninergic drugs on tremor induced by physostigmine in rats.
    Behavioural brain research, 2000, Volume: 109, Issue:2

    Topics: Animals; Buspirone; Cholinesterase Inhibitors; Cyproheptadine; Metergoline; N,N-Dimethyltryptamine; Physostigmine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrahydronaphthalenes; Tremor

2000
Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat.
    European journal of pharmacology, 2006, Mar-27, Volume: 535, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Buspirone; Clozapine; Decerebrate State; Dose-Response Relationship, Drug; Drug Interactions; Ergotamine; Heart Rate; Ketanserin; Lisuride; Male; Metergoline; Methiothepin; Methysergide; Phenylephrine; Piperazines; Pizotyline; Prazosin; Pyridines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Serotonin Antagonists; Serotonin Receptor Agonists; Yohimbine

2006