metaphit has been researched along with mazindol in 2 studies
Studies (metaphit) | Trials (metaphit) | Recent Studies (post-2010) (metaphit) | Studies (mazindol) | Trials (mazindol) | Recent Studies (post-2010) (mazindol) |
---|---|---|---|---|---|
68 | 0 | 4 | 631 | 73 | 31 |
Protein | Taxonomy | metaphit (IC50) | mazindol (IC50) |
---|---|---|---|
Sodium-dependent noradrenaline transporter | Homo sapiens (human) | 0.0029 | |
Sodium-dependent dopamine transporter | Rattus norvegicus (Norway rat) | 0.0454 | |
Sodium-dependent serotonin transporter | Homo sapiens (human) | 0.074 | |
Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | 0.231 | |
Sodium-dependent dopamine transporter | Homo sapiens (human) | 0.0275 | |
Sodium-dependent dopamine transporter | Mus musculus (house mouse) | 0.013 | |
Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | 0.2344 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (50.00) | 18.7374 |
1990's | 1 (50.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Boja, JW; Carroll, FI; Kuhar, MJ; Lewin, AH; Philip, A; Rahman, MA | 1 |
Jacobson, AE; Lajtha, A; Reith, ME; Rice, KC; Zimányi, I | 1 |
2 other study(ies) available for metaphit and mazindol
Article | Year |
---|---|
Isothiocyanate derivatives of cocaine: irreversible inhibition of ligand binding at the dopamine transporter.
Topics: Animals; Benzamides; Binding, Competitive; Brain Stem; Carrier Proteins; Cerebral Cortex; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Ligands; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Paroxetine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Thiocyanates | 1991 |
Long-term blockade of the dopamine uptake complex by metaphit, an isothiocyanate derivative of phencyclidine.
Topics: Animals; Cocaine; Dopamine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Female; Hydrogen-Ion Concentration; Injections, Intraventricular; Kinetics; Male; Mazindol; Membrane Proteins; Mice; Nerve Tissue Proteins; Phencyclidine; Radioligand Assay | 1989 |