Page last updated: 2024-08-25

mesulergine and piperidines

mesulergine has been researched along with piperidines in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19904 (33.33)18.7374
1990's2 (16.67)18.2507
2000's5 (41.67)29.6817
2010's1 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Engel, G; Hoyer, D; Kalkman, HO1
Hoyer, D; Palacios, JM; Pazos, A; Probst, A1
Ståhle, L; Ungerstedt, U1
Hoyer, D; Palacios, JM; Pazos, A1
López-Giménez, JF; Mengod, G; Palacios, JM; Vilaró, MT2
Barwick, VS; Hicks, PB; Jones, DH; Richter, JT; Young, KA1
Gordon, M; Heinz-Esser, K; Kanwal, JS; Peng, JP1
Aloyo, VJ; Harvey, JA1
Jurzak, M; Leysen, JE; Luyten, WH; Oekelen, DV; Van de Wiel, D; Van Hecke, G1
Feuerbach, D; Loetscher, E; Mahé, C; Müller, W; Schoeffter, P; Seiler, MP1
Capuano, B; Christopoulos, A; Conway, RJ; Crosby, IT; Robertson, AD; Valant, C1

Other Studies

12 other study(ies) available for mesulergine and piperidines

ArticleYear
Molecular pharmacology of 5-HT1 and 5-HT2 recognition sites in rat and pig brain membranes: radioligand binding studies with [3H]5-HT, [3H]8-OH-DPAT, (-)[125I]iodocyanopindolol, [3H]mesulergine and [3H]ketanserin.
    European journal of pharmacology, 1985, Nov-26, Volume: 118, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Chemistry; Choroid Plexus; Ergolines; In Vitro Techniques; Iodocyanopindolol; Ketanserin; Male; Membranes; Pindolol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tetrahydronaphthalenes

1985
Serotonin receptors in the human brain. II. Characterization and autoradiographic localization of 5-HT1C and 5-HT2 recognition sites.
    Brain research, 1986, Jun-18, Volume: 376, Issue:1

    Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Cerebral Cortex; Choroid Plexus; Ergolines; Female; Humans; Ketanserin; Male; Membranes; Middle Aged; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tissue Distribution; Tritium

1986
On the mode of action of six putative dopamine receptor agonists on suppression of exploratory behaviour in rats.
    Psychopharmacology, 1987, Volume: 91, Issue:2

    Topics: Animals; Bromocriptine; Ergolines; Exploratory Behavior; Habituation, Psychophysiologic; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1987
Mesulergine, a selective serotonin-2 ligand in the rat cortex, does not label these receptors in porcine and human cortex: evidence for species differences in brain serotonin-2 receptors.
    European journal of pharmacology, 1984, Nov-27, Volume: 106, Issue:3

    Topics: Animals; Brain Chemistry; Cerebral Cortex; Ergolines; Humans; In Vitro Techniques; Ketanserin; Kinetics; Ligands; Male; Piperidines; Rats; Receptors, Serotonin; Species Specificity; Swine; Tritium

1984
Selective visualization of rat brain 5-HT2A receptors by autoradiography with [3H]MDL 100,907.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:4

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Fluorobenzenes; Guanylyl Imidodiphosphate; In Situ Hybridization; In Vitro Techniques; Ketanserin; Male; Naphthalenes; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists

1997
[3H]MDL 100,907 labels 5-HT2A serotonin receptors selectively in primate brain.
    Neuropharmacology, 1998, Volume: 37, Issue:9

    Topics: Aged; Aged, 80 and over; Animals; Binding Sites; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Male; Naphthalenes; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Tritium

1998
Subthalamic nucleus microinjections of 5-HT2 receptor antagonists suppress stereotypy in rats.
    Neuroreport, 2000, Feb-07, Volume: 11, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Clozapine; Ergolines; Fluorobenzenes; Male; Mastication; Microinjections; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Stereotypic Movement Disorder; Subthalamic Nucleus

2000
Auditory responses from the frontal cortex in the mustached bat, Pteronotus parnellii.
    Neuroreport, 2000, Feb-07, Volume: 11, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Clozapine; Ergolines; Fluorobenzenes; Male; Mastication; Microinjections; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Stereotypic Movement Disorder; Subthalamic Nucleus

2000
Antagonist binding at 5-HT(2A) and 5-HT(2C) receptors in the rabbit: high correlation with the profile for the human receptors.
    European journal of pharmacology, 2000, Oct-13, Volume: 406, Issue:2

    Topics: Animals; Cerebral Cortex; Ergolines; Female; Fluorobenzenes; Humans; Male; Piperidines; Rabbits; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists

2000
Different regulation of rat 5-HT(2A) and rat 5-HT(2C) receptors in NIH 3T3 cells upon exposure to 5-HT and pipamperone.
    European journal of pharmacology, 2001, Aug-03, Volume: 425, Issue:1

    Topics: 3T3 Cells; Animals; Benzamides; Binding Sites; Binding, Competitive; Butyrophenones; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Inositol Phosphates; Iodine Radioisotopes; Membranes; Mice; Piperidines; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Agents; Serotonin Antagonists; Time Factors; Tritium

2001
Differential inverse agonist efficacies of SB-258719, SB-258741 and SB-269970 at human recombinant serotonin 5-HT7 receptors.
    European journal of pharmacology, 2004, Jul-14, Volume: 495, Issue:2-3

    Topics: Animals; Binding, Competitive; CHO Cells; Clozapine; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Ergolines; Humans; Loxapine; Methiothepin; Phenols; Pimozide; Pindolol; Piperidines; Plasmids; Pyrrolidines; Radioligand Assay; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Tosyl Compounds; Transfection

2004
Synthesis and SAR study of 4-arylpiperidines and 4-aryl-1,2,3,6-tetrahydropyridines as 5-HT₂C agonists.
    Bioorganic & medicinal chemistry letters, 2012, Apr-01, Volume: 22, Issue:7

    Topics: Animals; Appetite Depressants; Calcium; Ergolines; Humans; Kinetics; Piperidines; Protein Binding; Pyridines; Radioligand Assay; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship

2012