Page last updated: 2024-08-25

mesulergine and mdl 100907

mesulergine has been researched along with mdl 100907 in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (18.18)18.2507
2000's7 (63.64)29.6817
2010's2 (18.18)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
López-Giménez, JF; Mengod, G; Palacios, JM; Vilaró, MT2
Barwick, VS; Hicks, PB; Jones, DH; Richter, JT; Young, KA1
Gordon, M; Heinz-Esser, K; Kanwal, JS; Peng, JP1
Aloyo, VJ; Harvey, JA1
Goldman, D; Iwata, N; Linnoila, M; Northup, JK; Okada, M; Ozaki, N1
Hietala, J; Majasuo, H; Pälvimäki, EP; Syvälahti, E1
Khan, R; Mohanan, VV; Paulose, CS1
Adams, W; van den Buuse, M1
Haider, S; Haleem, DJ; Khaliq, S; Memon, Z; Saleem, S1

Other Studies

11 other study(ies) available for mesulergine and mdl 100907

ArticleYear
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Selective visualization of rat brain 5-HT2A receptors by autoradiography with [3H]MDL 100,907.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:4

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Fluorobenzenes; Guanylyl Imidodiphosphate; In Situ Hybridization; In Vitro Techniques; Ketanserin; Male; Naphthalenes; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists

1997
[3H]MDL 100,907 labels 5-HT2A serotonin receptors selectively in primate brain.
    Neuropharmacology, 1998, Volume: 37, Issue:9

    Topics: Aged; Aged, 80 and over; Animals; Binding Sites; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Male; Naphthalenes; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Tritium

1998
Subthalamic nucleus microinjections of 5-HT2 receptor antagonists suppress stereotypy in rats.
    Neuroreport, 2000, Feb-07, Volume: 11, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Clozapine; Ergolines; Fluorobenzenes; Male; Mastication; Microinjections; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Stereotypic Movement Disorder; Subthalamic Nucleus

2000
Auditory responses from the frontal cortex in the mustached bat, Pteronotus parnellii.
    Neuroreport, 2000, Feb-07, Volume: 11, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Clozapine; Ergolines; Fluorobenzenes; Male; Mastication; Microinjections; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Stereotypic Movement Disorder; Subthalamic Nucleus

2000
Antagonist binding at 5-HT(2A) and 5-HT(2C) receptors in the rabbit: high correlation with the profile for the human receptors.
    European journal of pharmacology, 2000, Oct-13, Volume: 406, Issue:2

    Topics: Animals; Cerebral Cortex; Ergolines; Female; Fluorobenzenes; Humans; Male; Piperidines; Rabbits; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists

2000
Comparison of G-protein selectivity of human 5-HT2C and 5-HT1A receptors.
    Annals of the New York Academy of Sciences, 2004, Volume: 1025

    Topics: Animals; Cell Line; Dose-Response Relationship, Drug; Ergolines; Heterotrimeric GTP-Binding Proteins; Insecta; Protein Binding; Rats; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2C; Receptors, G-Protein-Coupled; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists

2004
Serotonin 5-HT2C receptor-mediated phosphoinositide hydrolysis in rat choroid plexus after fluoxetine and citalopram treatments.
    Pharmacological research, 2005, Volume: 51, Issue:5

    Topics: Amphetamines; Animals; Choroid Plexus; Citalopram; Dose-Response Relationship, Drug; Ergolines; Fluoxetine; Hydrolysis; Inositol Phosphates; Male; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Second Messenger Systems; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2005
Hypothalamic 5-HT functional regulation through 5-HT1A and 5-HT2C receptors during pancreatic regeneration.
    Life sciences, 2006, Feb-28, Volume: 78, Issue:14

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Down-Regulation; Ergolines; Gene Expression Regulation, Developmental; Hypothalamus; Male; Pancreas; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2C; Regeneration; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2006
Hippocampal serotonin depletion facilitates the enhancement of prepulse inhibition by risperidone: possible role of 5-HT(2C) receptors in the dorsal hippocampus.
    Neuropharmacology, 2011, Volume: 61, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Ergolines; Hippocampus; Male; Nerve Tissue Proteins; Neural Inhibition; Neurons; Organ Specificity; Random Allocation; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Reflex, Startle; Risperidone; Schizophrenia; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2011
Influence of serotonergic 5-HT2C receptor antagonist mesulergine in the reversal of memory deficits induced by mCPP.
    Journal of the College of Physicians and Surgeons--Pakistan : JCPSP, 2012, Volume: 22, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Disease Models, Animal; Ergolines; Male; Maze Learning; Memory Disorders; Memory, Long-Term; Memory, Short-Term; Piperazines; Random Allocation; Rats; Rats, Wistar; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2012