Page last updated: 2024-08-25

mesulergine and ergoline

mesulergine has been researched along with ergoline in 212 studies

Research

Studies (212)

TimeframeStudies, this research(%)All Research%
pre-199070 (33.02)18.7374
1990's100 (47.17)18.2507
2000's31 (14.62)29.6817
2010's11 (5.19)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beauchamp, RD; Greeley, GH; Ishizuka, J; Thompson, JC; Townsend, CM1
Esterle, TM; Sanders-Bush, E1
Gorospe, E; Hoffman, BJ; Leonhardt, S; Teitler, M1
Donatsch, P; Ettlin, RA; Prentice, DE; Qureshi, S; Siegel, RA1
Pawlikowski, M; Pisarek, H; Stepien, H1
Aulakh, CS; Hill, JL; Murphy, DL1
Choudhary, MS; Craigo, S; Roth, BL2
Crompton, MR; De Paermentier, F; Horton, RW; Lowther, S1
Griebel, G; Haefely, WE; Jenck, F; Martin, JR; Moreau, JL; Widmer, U1
Havlik, S; Peroutka, SJ1
Emanuelsson, H1
Bartyzel, P; Glennon, RA; Leonhardt, S; Raghupathi, R; Teitler, M1
Murthy, JN; Pluchino, RS; Pranzatelli, MR1
Pisarek, H; Stepien, H1
Dahlgren, IL; Klint, T; Larsson, K1
Miller, KJ; Teitler, M1
Adham, N; Branchek, TA; Hartig, PR; Kao, HT; Olsen, MA; Weinshank, RL1
Breeding, M; Sanders-Bush, E1
Kagaya, A; Mikuni, M; Takahashi, K1
Katoh, F; Kuroda, Y; Mikuni, M; Takahashi, K1
Boulenguez, P; Chauveau, J; Delaage, M; Lanoir, J; Morel, A; Segu, L1
Brown, AM; Kaumann, AJ; Patch, TL1
Hicks, PB; Young, KA; Zavodny, R1
Gershon, MD; Hsiung, SC; Kirchgessner, AL; Liu, KP; Tamir, H; Yu, PY1
Robertson, DW; Threlkeld, PG; Wong, DT1
McQuade, RD; Taylor, LA; Tedford, CE1
Goldstein, M; Gopinathan, G; Lieberman, AN; Pasternack, P1
Canton, H; Colpaert, FC; Verrièle, L1
Lucot, JB1
Pranzatelli, MR1
Axel, R; Huang, KN; Jessell, TM; Julius, D; Livelli, TJ1
Le, H; Lübbert, H; Mengod, G; Nguyen, H; Palacios, JM; Waeber, C1
Hamik, A; Peroutka, SJ; Switzer, JA1
Herrick-Davis, K; Titeler, M2
Palacios, JM; Waeber, C1
Dietl, MM; Hoyer, D; Palacios, JM; Waeber, C1
Brazell, C; Dourish, CT; King, BH; Middlemiss, DN1
Chojnacka-Wójcik, E; Jaros, T; Kłodzińska, A; Maj, J1
Chiodini, PG; Dallabonzana, D; Liuzzi, A; Oppizzi, G; Verde, GG1
Glennon, RA; McKenney, JD; Pierson, ME1
Curzon, G; Kennett, GA1
Engel, G; Hoyer, D; Kalkman, HO1
Hoyer, D; Palacios, JM; Pazos, A; Probst, A1
Heuring, RE; Peroutka, SJ1
Palacios, JM; Pazos, A; Probst, A1
Goldstein, M; Gopinathan, G; Lieberman, AN; Neophytides, A1
Huang, JC; Peroutka, SJ1
Amedro, J; Brown, L; Smith, D; Williams, G1
Hoyer, D; Palacios, JM; Pazos, A; Probst, A; Waeber, C1
Hoyer, D; Palacios, JM; Schoeffter, P; Waeber, C1
Markstein, R; Palacios, JM; Pazos, A1
Rinne, UK2
Churg, A; Fleetham, JA; McElvaney, NG; Wilcox, PG1
Lang, AE1
Begaud, B; Dang Tran, L; Montastruc, JL; Montastruc, P1
Dupont, E; Jakobsen, J; Mikkelsen, B1
Crosignani, PG; Ferrari, C1
Lees, AJ; Stern, GM; Wright, A1
Chang, RJ; Goodman, LA; Hesla, JS; Molitch, ME; Rodman, EF1
Ståhle, L; Ungerstedt, U1
Montastruc, JL; Rascol, A; Rascol, O; Senard, JM1
Engel, G; Hoyer, D; Palacios, JM; Pazos, A; Srivatsa, S1
Blackwell, RE1
Jankovic, J; Jansson, B; Orman, J1
Pfeiffer, RF1
Buchhave, J; Eskildsen, PC; Hommel, E1
Glaeske, C; Pfeiffer, RF; Wilken, K1
Bratty, PJ; Burton, K; Calne, DB; Larsen, TA; Martin, WR; Robinson, RG; Schulzer, M1
Buvat, J; Dewailly, D; Fossati, P; Fourlinnie, JC; Lemaitre, G; Mazzuca, M; Thomas, P; Wemeau, JL1
Pepperell, RJ1
Gopinathan, G; Lieberman, AN; Neophytides, A1
Hietanen, M; Huttunen, J; Teräväinen, H1
Agnati, L; Fuxe, K; Goldstein, M; Helmer-Matyjek, E; Kuga, S; Mascagni, F1
Baas, H; Fischer, PA; Japp, G; Schneider, E2
Besser, GM; Bouloux, PM; Grossman, A; Loneragan, R; Rees, LH; Wass, JA1
Adams, CB; Besser, GM; Charlesworth, M; Doniach, I; Grossman, A; Ross, R; Wass, JA1
Brabant, G; Brennecke, I; Friedrich, H; Herrmann, H; Hesch, RD; von zur Mühlen, A; Wagner, TO1
Burton, K; Calne, DB1
Enz, A1
Bystritsky, A; Engel, J; Goldstein, M; Lieberman, A; Mino, S; Regev, I1
Closse, A; Jaton, AL1
Esplugues, J; Morales-Olivas, FJ; Palop, V; Rubio, E1
Jellinger, K1
Biesemeyer, H; Ludin, HP; Ringwald, E1
Markstein, R1
Beckman, J; Burton, K; Calne, DB; Martin, WR1
Jensen, I; Pakkenberg, H1
Borges, JL; Boyett, RL; Elton, RL; Evans, WS; Kaiser, DL; MacLeod, RM; Rogol, AD; Schran, HF; Thorner, MO1
Markó, M1
Klÿn, JG; Lamberts, SW; Oosterom, R1
Hoyer, D; Palacios, JM; Pazos, A2
Donatsch, P; Enz, A; Nordmann, R1
Agid, Y; Bonnet, AM; Esteguy, M; Guimaraes, J; Lhermitte, F1
Fischer, PA; Hubener, K; Schneider, E2
Kvist Poulsen, H; Møller Pedersen, S; Rasmussen, P; Riber Petersen, M1
Closse, A1
Reynolds, GP; Riederer, P1
Fiorella, D; Johnson, RG; Rabin, RA1
Fiorella, D; Rabin, RA; Winter, JC1
Grignaschi, G; Samanin, R; Sironi, F1
Aulakh, CS; Hulihan-Giblin, BA; Park, YD1
Katusić, ZS; Krstić, MK1
Hietala, J; Kuoppamäki, M; Seppälä, T; Syvälahti, E1
de Boer, T; Klomp, J; Olijve, W; Stam, NJ; van Alebeek, C; van Delft, AM; Vanderheyden, P1
Barker, EL; Sanders-Bush, E; Schmidt, D; Westphal, RS1
Grotewiel, MS; Sanders-Bush, E1
Esposito, E; Pagannone, S; Prisco, S1
Sanders-Bush, E; Westphal, RS1
Hietala, J; Kuoppamäki, M; Pälvimäki, EP; Syvälahti, E1
Callahan, PM; Cunningham, KA1
Sillar, KT; Wedderburn, JF1
Borsini, F; Ceci, A; Cesana, R; Ciprandi, C1
Aulakh, CS; Goldman, D; Hulihan-Giblin, BA; Park, YD1
Gregory, CM; Pranzatelli, MR1
Di Scala, G; Hoyer, D; Rigo, M; Rocha, B; Sandner, G1
Davis, JM; Dubey, MP; Pandey, GN; Pandey, SC; Piano, MR; Schwertz, DW1
Barone, P; Fillion, G; Millet, S; Moret, C; Prudhomme, N1
Beer, MS; Hawkins, LM; Middlemiss, DN; Stanton, JA1
Craig, DA; Martin, GR1
Doble, A; Flamand, F; Malgouris, C1
Briley, M; Palmier, C; Pauwels, PJ1
Cynader, MS; Dyck, RH1
Murthy, JN; Pranzatelli, MR; Tailor, PT1
Bruinvels, AT; Hoyer, D; Palacios, JM1
Aulakh, CS; Hulihan-Giblin, BA; Mazzola-Pomietto, P; Murphy, DL1
Almaula, N; Ballesteros, JA; Ebersole, BJ; Sealfon, SC; Weinstein, H1
Akiyoshi, J; Fujii, I; Isogawa, K; Nagayama, H; Yamada, K1
Hartman, JL; Northup, JK1
Kellermann, O; Launay, JM; Loric, S; Maroteaux, L1
Hietala, J; Kuoppamäki, M; Laakso, A; Pälvimäki, EP; Syvälahti, E1
Li, TK; Lumeng, L; Pandey, SC1
Baron, BM; Freedman, J; Siegel, BW; Vaal, MJ1
Cooke, BA; Dirami, G; Teerds, KJ1
Carey, JE; Chen, C; Elliott, JM; Flanigan, TP; Kumar, C; McDonald, B; Newberry, NR; Newton, RA; Phipps, SL1
Imada-Shirakata, Y; Kotera, T; Okuma, M; Ueda, S1
Curtis, MJ; Ellwood, AJ1
Cynader, MS; Gu, Q; Wang, Y1
Cadavid, MI; Calleja, JM; Dominguez, R; Honrubia, MA; Loza, MI; Lozoya, E; Maayani, S; Manaut, F; Rodriguez, J; Sanz, F; Seijas, JA; Villaverde, MC1
Cenarruzabeitia, E; Del Rio, J; Lasheras, B; Ramírez, MJ1
De Vries, P; Heiligers, JP; Saxena, PR; Villalón, CM1
Elliott, JM; Newton, RA1
Egan, C; Herrick-Davis, K; Teitler, M1
Castillo, MJ; Castro, ME; del Arco, C; del Olmo, E; Pazos, A; Romón, T1
López-Giménez, JF; Mengod, G; Palacios, JM; Vilaró, MT4
Giovannini, MG; Pepeu, G; Zhelyazkova-Savova, M2
Boess, FG; Bourson, A; Kapps, V; Rudler, A; Sleight, AJ; Zwingelstein, C1
Ijzerman, AP; Kuipers, W; Oliveira, L; Vriend, G1
Grill, HJ; Kaplan, JM; Song, S1
Belden, M; Carvey, PM; Goetz, CG; Pappert, EJ; Stebbins, GT1
Cooke, BA; Dirami, G1
Di Giovanni, G; Di Mascio, M; Di Matteo, V; Esposito, E1
Couvaris, C; Daifotis, Z; Galanopoulou, P; Giannakopoulos, G1
Centurión, D; De Vries, P; Heiligers, JP; Sánchez-López, A; Saxena, PR; Villalón, CM1
Applegate, CD; Tecott, LH1
Bloem, LJ; Hurley, JH; Liu, J; Pavalko, F; Simon, JR; Tian, M; Yu, L1
Carvey, PM; Goetz, CG; Leurgans, S; Ling, ZD; Pappert, EJ; Raman, R; Vu, TQ1
Gauthier, C; Grinde, E; Herrick-Davis, K; Teitler, M1
Coupar, IM; Hemedah, M; Mitchelson, FJ2
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP1
Grinde, E; Herrick-Davis, K; Niswender, CM1
Alberts, GL; Gill, GS; Im, WB; Pregenzer, JF; Zaworski, PG1
Cassano, GB; Dell'Osso, L; Giannaccini, G; Lucacchini, A; Marazziti, D; Rossi, A; Zavaglia, KM1
Barwick, VS; Hicks, PB; Jones, DH; Richter, JT; Young, KA1
Gordon, M; Heinz-Esser, K; Kanwal, JS; Peng, JP1
Cussac, D; Millan, MJ; Newman-Tancredi, A; Quentric, Y1
Aloyo, VJ; Harvey, JA1
Cordi, AA; Ragonnet, C; Vayssettes-Courchay, C; Verbeuren, TJ1
Brotchie, JM; Fox, SH1
Ebersole, BJ; Rosendorff, A; Sealfon, SC1
Honda, M; Ono, H1
Berg, KA; Clarke, WP; Cropper, JD; Emeson, RB; Niswender, CM; Sanders-Bush, E1
Jurzak, M; Leysen, JE; Luyten, WH; Oekelen, DV; Van de Wiel, D; Van Hecke, G1
Alberts, GL; Chio, CL; Im, WB1
Alloui, A; Bardin, L; Chassaing, C; Courade, JP; Eschalier, A1
Chen, Y; Hertz, L; Kong, EK; Peng, L; Yu, AC1
Martín-Cora, FJ; Pazos, A1
Clifton, PG; Dourish, CT; Kennett, GA; Lee, MD; Somerville, EM1
Feuerbach, D; Loetscher, E; Mahé, C; Müller, W; Schoeffter, P; Seiler, MP1
Christopoulos, A; Devlin, MG; Guida, E; Ryan, OM; Sexton, PM; Smith, NJ1
Goldman, D; Iwata, N; Linnoila, M; Northup, JK; Okada, M; Ozaki, N1
Hietala, J; Majasuo, H; Pälvimäki, EP; Syvälahti, E1
Chathu, F; Mohanan, VV; Paulose, CS1
Antonatos, S; Galanopoulou, P1
Khan, R; Mohanan, VV; Paulose, CS1
Brunden, K; Doucette, C; Graham, E; Hanniford, D; Harrington, J; Poole, MF; Sherf, B; Song, J; Stricker-Krongrad, A; Ting, A1
Hietala, J; Laakso, A; Majasuo, H; Pälvimäki, EP; Penttilä, J; Syvälahti, E1
Andressen, KW; Krobert, KA; Levy, FO1
Bell, W; Deng, C; du Bois, TM; Huang, XF1
Ackley, DC; Holbert, JK; Hu, XE; Kim, N; Klopfenstein, SR; Méndez-Andino, JL; Meyers, KM; Mitchell, MC; Mittelstadt, SW; Mumin, RN; Paris, JL; Reizes, O; Wos, JA1
García, M; Martín, ML; Morán, A; Ortizde Urbina, AV; San Román, L1
Krishnakumar, A; Nandhu, MS; Paulose, CS1
Haleem, DJ; Shireen, E1
Bönisch, H; Brüss, M; Göthert, M; Steinhagen, F; Walstab, J1
Adams, W; van den Buuse, M1
Haider, S; Haleem, DJ; Khaliq, S; Memon, Z; Saleem, S1
Capuano, B; Christopoulos, A; Conway, RJ; Crosby, IT; Robertson, AD; Valant, C1
Jahnsen, JA; Uhlén, S1
Booth, RG; Kondabolu, K; Kuipers, A; Morgan, D; Robertson, KL; Rowland, NE; Sakhuja, R1
Andreeva, LA; Khashaba, EY; Kost, NV; Meshavkin, VK; Myasoedov, NF; Sokolov, OY; Voevodina, ME; Zolotarev, YA1
Andressen, KW; Brevik, CH; Krobert, KA; Levy, FO; Manfra, O; Ulsund, AH; Vanhoenacker, P1
Bojarski, AJ; Duszyńska, B; Lenda, T; Nowak, G; Satała, G1

Reviews

6 review(s) available for mesulergine and ergoline

ArticleYear
Medical treatment of pituitary adenomas: effects on tumor growth.
    Journal of endocrinological investigation, 1985, Volume: 8, Issue:3

    Topics: Adenoma; Adrenocorticotropic Hormone; Bromocriptine; Dihydroergotoxine; Dopamine; Drug Administration Schedule; Ergolines; Growth Hormone; Levodopa; Lisuride; Metergoline; Methysergide; Pergolide; Pituitary Neoplasms; Prolactin; Tomography, X-Ray Computed

1985
D-1 and D-2 agonists in Parkinson's disease.
    The Canadian journal of neurological sciences. Le journal canadien des sciences neurologiques, 1987, Volume: 14, Issue:3 Suppl

    Topics: Aged; Aged, 80 and over; Antiparkinson Agents; Dopamine; Ergolines; Female; Humans; Male; Middle Aged; Parkinson Disease; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1987
Update on dopamine agonists in Parkinson's disease: "beyond bromocriptine".
    The Canadian journal of neurological sciences. Le journal canadien des sciences neurologiques, 1987, Volume: 14, Issue:3 Suppl

    Topics: Antiparkinson Agents; Bromocriptine; Dopamine; Ergolines; Humans; Parkinson Disease; Piperazines

1987
Medical treatment of hyperprolactinaemic disorders.
    Human reproduction (Oxford, England), 1986, Volume: 1, Issue:8

    Topics: Acromegaly; Bromocriptine; Delayed-Action Preparations; Dopamine; Ergolines; Female; Humans; Hyperprolactinemia; Lisuride; Pergolide; Pituitary Neoplasms; Pregnancy; Prolactin; Psychoses, Substance-Induced; Tamoxifen

1986
Diagnosis and management of prolactinomas.
    Fertility and sterility, 1985, Volume: 43, Issue:1

    Topics: Adenoma; Adult; Diagnosis, Differential; Ergolines; Female; Follow-Up Studies; Galactorrhea; Genital Diseases, Female; Humans; Hypophysectomy; Hypothyroidism; Infertility, Female; Pergolide; Pituitary Neoplasms; Pregnancy; Pregnancy Complications, Neoplastic; Prolactin; Sella Turcica; Tomography, X-Ray Computed; Visual Field Tests

1985
The pharmacology of mesulergine.
    Clinical neuropharmacology, 1985, Volume: 8, Issue:1

    Topics: Animals; Antiparkinson Agents; Ergolines; Humans; Parkinson Disease; Receptors, Dopamine

1985

Trials

10 trial(s) available for mesulergine and ergoline

ArticleYear
Mesulergine: a dopamine agonist with novel properties in Parkinson's disease.
    Advances in neurology, 1990, Volume: 53

    Topics: Aged; Dopamine Agents; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ergolines; Female; Humans; Levodopa; Male; Middle Aged; Neurologic Examination; Parkinson Disease

1990
Mesulergine in early Parkinson's disease: a double blind controlled trial.
    Journal of neurology, neurosurgery, and psychiatry, 1986, Volume: 49, Issue:4

    Topics: Aged; Antiparkinson Agents; Benserazide; Clinical Trials as Topic; Double-Blind Method; Drug Combinations; Ergolines; Female; Humans; Levodopa; Male; Middle Aged; Parkinson Disease; Random Allocation

1986
Placebo-controlled study of mesulergine in Parkinson's disease.
    Neurology, 1985, Volume: 35, Issue:2

    Topics: Aged; Antiparkinson Agents; Clinical Trials as Topic; Ergolines; Female; Humans; Male; Middle Aged; Parkinson Disease; Placebos

1985
The effect of a new ergoline derivative, CU 32-085, in the treatment of acromegaly. A controlled study.
    Clinical endocrinology, 1985, Volume: 22, Issue:2

    Topics: Acromegaly; Adult; Aged; Blood Pressure; Clinical Trials as Topic; Ergolines; Female; Growth Hormone; Hormones; Humans; Hydrocortisone; Male; Middle Aged; Prolactin

1985
Mesulergine (CU32-085) in the treatment of Parkinson's disease.
    Annals of neurology, 1985, Volume: 17, Issue:4

    Topics: Aged; Antiparkinson Agents; Clinical Trials as Topic; Double-Blind Method; Ergolines; Female; Humans; Male; Middle Aged; Parkinson Disease; Random Allocation

1985
Parkinson's disease: a comparison of mesulergine and bromocriptine.
    Neurology, 1985, Volume: 35, Issue:8

    Topics: Adult; Aged; Bromocriptine; Clinical Trials as Topic; Ergolines; Female; Humans; Male; Middle Aged; Movement; Nervous System; Parkinson Disease

1985
Treatment of human hyperprolactinaemia with a new dopamine agonist: CU 32085 (mesulergin).
    Acta endocrinologica, 1985, Volume: 110, Issue:4

    Topics: Administration, Oral; Adolescent; Adult; Aged; Bromocriptine; Clinical Trials as Topic; Ergolines; Female; Gonads; Humans; Hyperprolactinemia; Male; Middle Aged; Pituitary Gland; Pituitary Neoplasms; Prolactin; Receptors, Dopamine; Tomography, X-Ray Computed

1985
Mesulergine and bromocriptine in long-term treatment of advanced parkinsonism.
    Journal of neural transmission, 1985, Volume: 64, Issue:1

    Topics: Adult; Aged; Blood Pressure; Bromocriptine; Drug Administration Schedule; Ergolines; Female; Heart Rate; Humans; Levodopa; Male; Middle Aged; Parkinson Disease; Time Factors

1985
Adjuvant treatment of Parkinson's disease with dopamine agonists: open trial with bromocriptine and CU 32-085.
    Journal of neurology, 1982, Volume: 227, Issue:2

    Topics: Aged; Bromocriptine; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ergolines; Female; Humans; Levodopa; Male; Middle Aged; Parkinson Disease; Receptors, Dopamine

1982
Treatment of Parkinson's disease with the ergoline derivatives CQ 32-084 and CU 32-085.
    Advances in neurology, 1983, Volume: 37

    Topics: Adult; Aged; Blood Pressure; Clinical Trials as Topic; Disability Evaluation; Ergolines; Female; Humans; Male; Middle Aged; Parkinson Disease; Pilot Projects

1983

Other Studies

196 other study(ies) available for mesulergine and ergoline

ArticleYear
Receptor-mediated autocrine growth-stimulatory effect of 5-hydroxytryptamine on cultured human pancreatic carcinoid cells.
    Journal of cellular physiology, 1992, Volume: 150, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Cell Division; Cyclic AMP; Cyclic GMP; Ergolines; Humans; Pancreatic Neoplasms; Pertussis Toxin; Phosphatidylinositols; Pindolol; Receptors, Serotonin; Second Messenger Systems; Serotonin; Serotonin Antagonists; Tumor Cells, Cultured; Virulence Factors, Bordetella

1992
Serotonin agonists increase transferrin levels via activation of 5-HT1C receptors in choroid plexus epithelium.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:12

    Topics: Amino Acid Isomerases; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Choroid Plexus; Cyclosporins; Epithelium; Ergolines; Fibroblasts; Kinetics; Male; Mianserin; Peptidylprolyl Isomerase; Phosphatidylinositols; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA Probes; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Thymidine; Time Factors; Transferrin

1992
Molecular pharmacological differences in the interaction of serotonin with 5-hydroxytryptamine1C and 5-hydroxytryptamine2 receptors.
    Molecular pharmacology, 1992, Volume: 42, Issue:2

    Topics: 3T3 Cells; Amphetamines; Animals; Binding, Competitive; Brain; Cell Membrane; Choroid Plexus; Ergolines; Fibroblasts; GTP-Binding Proteins; Inositol Phosphates; Iodine Radioisotopes; Kinetics; Mice; Neurotransmitter Agents; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stimulation, Chemical; Swine; Transfection; Tritium

1992
Mesulergine induced Leydig cell tumours, a syndrome involving the pituitary-testicular axis of the rat.
    Archives of toxicology. Supplement. = Archiv fur Toxikologie. Supplement, 1992, Volume: 15

    Topics: Animals; Dihydropyridines; Ergolines; Isradipine; Leydig Cell Tumor; Male; Pituitary Hormones; Rats; Rats, Inbred Strains; Syndrome; Testicular Hormones; Time Factors

1992
Effect of mesulergine on prolactin secretion and dopamine D2 receptors-adaptive changes in diethylstilbestrol-induced hyperplasia of the rat anterior pituitary.
    Endocrine regulations, 1992, Volume: 26, Issue:1

    Topics: Animals; Antiparkinson Agents; Bromocriptine; Diethylstilbestrol; Dose-Response Relationship, Drug; Ergolines; Female; Hyperplasia; Hyperprolactinemia; Pergolide; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine D2; Spiperone; Time Factors; Tritium

1992
Effects of various serotonin receptor subtype-selective antagonists alone and on m-chlorophenylpiperazine-induced neuroendocrine changes in rats.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Corticosterone; Ergolines; Male; Metergoline; Mianserin; Neurosecretory Systems; Piperazines; Prolactin; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone

1992
Identification of receptor domains that modify ligand binding to 5-hydroxytryptamine2 and 5-hydroxytryptamine1c serotonin receptors.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Base Sequence; Binding, Competitive; Ergolines; Haloperidol; In Vitro Techniques; Ketanserin; Molecular Sequence Data; Oligodeoxyribonucleotides; Receptors, Serotonin; Recombinant Fusion Proteins; Spiperone; Structure-Activity Relationship; Transfection

1992
The distribution of 5-HT1D and 5-HT1E binding sites in human brain.
    European journal of pharmacology, 1992, Nov-03, Volume: 222, Issue:1

    Topics: Adult; Aged; Antiparkinson Agents; Brain; Brain Chemistry; Ergolines; Female; Humans; In Vitro Techniques; Kinetics; Male; Membranes; Middle Aged; Pindolol; Receptors, Serotonin

1992
Behavioral profile of the 5HT1A receptor antagonist (S)-UH-301 in rodents and monkeys.
    Brain research bulletin, 1992, Volume: 29, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acoustic Stimulation; Animals; Brain; Cerebral Ventricles; Conditioning, Operant; Conflict, Psychological; Ergolines; Exploratory Behavior; Feeding Behavior; Injections, Intraventricular; Ketanserin; Learning; Mice; Mice, Inbred DBA; Motor Activity; N-Methylaspartate; Rats; Receptors, Serotonin; Seizures; Serotonin; Serotonin Antagonists

1992
Differential radioligand binding properties of [3H]5-hydroxytryptamine and [3H]mesulergine in a clonal 5-hydroxytryptamine1C cell line.
    Brain research, 1992, Jul-03, Volume: 584, Issue:1-2

    Topics: Animals; Antiparkinson Agents; Cell Line; Centrifugation; Clone Cells; Cold Temperature; Ergolines; Filtration; Guanosine Triphosphate; Mice; Radioligand Assay; Receptors, Serotonin; Serotonin

1992
Autoradiographic localization in polychaete embryos of tritiated mesulergine, a selective antagonist of serotonin receptors that inhibits early polychaete development.
    The International journal of developmental biology, 1992, Volume: 36, Issue:2

    Topics: Animals; Autoradiography; Cell Division; Cell Movement; Cell Nucleus; Chromosomes; Cytoplasm; Ergolines; Gestational Age; Polychaeta; Receptors, Serotonin; Serotonin Antagonists; Tritium

1992
Binding of phenylalkylamine derivatives at 5-HT1C and 5-HT2 serotonin receptors: evidence for a lack of selectivity.
    Journal of medicinal chemistry, 1992, Feb-21, Volume: 35, Issue:4

    Topics: Animals; Binding Sites; Binding, Competitive; Ergolines; Ketanserin; Male; Molecular Structure; Propylamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Structure-Activity Relationship; Tritium

1992
Identification of spinal 5-HT1C binding sites in the rat: characterization of [3H]mesulergine binding.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:1

    Topics: Animals; Antiparkinson Agents; Binding Sites; Binding, Competitive; Ergolines; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spinal Cord

1992
The effect of mesulergine on prolactin secretion and anterior pituitary cells morphology in diethylstilboestrol-treated female Wistar rats.
    Histology and histopathology, 1992, Volume: 7, Issue:1

    Topics: Animals; Antiparkinson Agents; Bromocriptine; Cell Division; Diethylstilbestrol; Drug Interactions; Ergolines; Female; Hyperprolactinemia; Immunohistochemistry; Pergolide; Pituitary Gland, Anterior; Prolactin; Rats

1992
The selective 5-HT2 receptor antagonist amperozide attenuates 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane-induced inhibition of male rat sexual behavior.
    European journal of pharmacology, 1992, Mar-03, Volume: 212, Issue:2-3

    Topics: Alprenolol; Amphetamines; Animals; Ergolines; Ketanserin; Male; Piperazines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Sexual Behavior, Animal

1992
Quantitative autoradiography of 5-CT-sensitive (5-HT1D) and 5-CT-insensitive (5-HT1E) serotonin receptors in human brain.
    Neuroscience letters, 1992, Mar-02, Volume: 136, Issue:2

    Topics: Antiparkinson Agents; Autoradiography; Brain Chemistry; Ergolines; Humans; In Vitro Techniques; Pindolol; Receptors, Serotonin; Serotonin

1992
Site-directed mutagenesis of a single residue changes the binding properties of the serotonin 5-HT2 receptor from a human to a rat pharmacology.
    FEBS letters, 1992, Aug-03, Volume: 307, Issue:3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; DNA; Ergolines; Humans; Ketanserin; Molecular Sequence Data; Mutagenesis, Site-Directed; Rats; Receptors, Serotonin; Sequence Homology, Nucleic Acid; Species Specificity; Transfection

1992
Choroid plexus epithelial cells in primary culture: a model of 5HT1C receptor activation by hallucinogenic drugs.
    Psychopharmacology, 1991, Volume: 105, Issue:3

    Topics: 3,4-Methylenedioxyamphetamine; Amphetamines; Animals; Antiparkinson Agents; Cells, Cultured; Choroid Plexus; DOM 2,5-Dimethoxy-4-Methylamphetamine; Epithelial Cells; Ergolines; Hallucinogens; Male; Phosphatidylinositols; Quipazine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stereoisomerism

1991
Modulation of 5-HT2 receptor-mediated intracellular calcium movement in platelets and its function in affective disorders.
    The Japanese journal of psychiatry and neurology, 1991, Volume: 45, Issue:1

    Topics: Animals; Antiparkinson Agents; Corticosterone; Ergolines; Hippocampus; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1991
Rat hippocampal 5-HT1c receptor binding and 5-HT1c receptor mediated rat blood corticosterone responses.
    The Japanese journal of psychiatry and neurology, 1991, Volume: 45, Issue:1

    Topics: Animals; Antiparkinson Agents; Corticosterone; Ergolines; Hippocampus; Male; Piperazines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin

1991
Pharmacological characterization of serotonin-O-carboxymethyl-glycyl-tyrosinamide, a new selective indolic ligand for 5-hydroxytryptamine (5-HT)1B and 5-HT1D binding sites.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:3

    Topics: Animals; Binding Sites; Brain; Dipeptides; Ergolines; Guinea Pigs; Male; Membranes; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium

1991
The antimigraine drugs ergotamine and dihydroergotamine are potent 5-HT1C receptor agonists in piglet choroid plexus.
    British journal of pharmacology, 1991, Volume: 104, Issue:1

    Topics: Animals; Binding, Competitive; Choroid Plexus; Dihydroergotamine; Ergolines; Ergotamine; In Vitro Techniques; Inositol Phosphates; Migraine Disorders; Piperazines; Receptors, Serotonin; Serotonin; Swine; Thermodynamics

1991
Subchronic buspirone, mesulergine, and ICS 205-930 lack effects on D1 and D2 dopamine binding in the rat striatum during chronic haloperidol treatment.
    Journal of neural transmission. General section, 1991, Volume: 86, Issue:3

    Topics: Animals; Apomorphine; Buspirone; Corpus Striatum; Ergolines; Haloperidol; In Vitro Techniques; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Serotonin Antagonists; Stereotyped Behavior; Tropisetron; Up-Regulation

1991
Identification of serotonin receptors recognized by anti-idiotypic antibodies.
    Journal of neurochemistry, 1991, Volume: 57, Issue:3

    Topics: Androstadienes; Animals; Antibodies, Anti-Idiotypic; Antiparkinson Agents; Brain; Carrier Proteins; Cell Line; Chromatography, Affinity; Enzyme-Linked Immunosorbent Assay; Ergolines; Fibroblasts; Fluorescent Antibody Technique; HeLa Cells; Humans; Immunohistochemistry; Iodine Radioisotopes; Iodocyanopindolol; Ketanserin; Mineralocorticoid Receptor Antagonists; Pindolol; Rabbits; Receptors, Serotonin; Serotonin; Thyroid Neoplasms; Tritium

1991
Affinities of fluoxetine, its enantiomers, and other inhibitors of serotonin uptake for subtypes of serotonin receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1991, Volume: 5, Issue:1

    Topics: Animals; Antidepressive Agents; Binding, Competitive; Cattle; Choroid Plexus; Ergolines; Fluoxetine; In Vitro Techniques; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stereoisomerism; Synaptosomes

1991
The binding of SCH 39166 and SCH 23390 to 5-HT1C receptors in porcine choroid plexus.
    Life sciences, 1991, Volume: 49, Issue:20

    Topics: Animals; Antiparkinson Agents; Benzazepines; Binding, Competitive; Choroid Plexus; Dopamine; Dopamine Antagonists; Ergolines; Receptors, Serotonin; Serotonin Antagonists; Swine

1991
Binding of typical and atypical antipsychotics to 5-HT1C and 5-HT2 sites: clozapine potently interacts with 5-HT1C sites.
    European journal of pharmacology, 1990, Nov-20, Volume: 191, Issue:1

    Topics: Animals; Antipsychotic Agents; Binding Sites; Choroid Plexus; Clozapine; Ergolines; In Vitro Techniques; Ketanserin; Kinetics; Receptors, Serotonin; Swine

1990
Effects of serotonin antagonists on motion sickness and its suppression by 8-OH-DPAT in cats.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cats; Dose-Response Relationship, Drug; Ergolines; Female; Metergoline; Motion Sickness; Piperazines; Propranolol; Serotonin Antagonists; Stereoisomerism; Tetrahydronaphthalenes

1990
Neonatal 5,7-DHT lesions upregulate [3H]mesulergine-labelled spinal 5-HT1C binding sites in the rat.
    Brain research bulletin, 1990, Volume: 25, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Animals; Animals, Newborn; Antiparkinson Agents; Cisterna Magna; Ergolines; Female; In Vitro Techniques; Injections; Injections, Intraperitoneal; Kinetics; Male; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spinal Cord; Up-Regulation

1990
The 5HT2 receptor defines a family of structurally distinct but functionally conserved serotonin receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1990, Volume: 87, Issue:3

    Topics: Amino Acid Sequence; Animals; Antiparkinson Agents; Brain; DNA; Ergolines; Fibroblasts; Gene Library; Genes; Mice; Molecular Sequence Data; Organ Specificity; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Nucleic Acid; Spiperone; Transfection; Type C Phospholipases

1990
The distribution and cellular localization of the serotonin 1C receptor mRNA in the rodent brain examined by in situ hybridization histochemistry. Comparison with receptor binding distribution.
    Neuroscience, 1990, Volume: 35, Issue:3

    Topics: Animals; Antiparkinson Agents; Autoradiography; Blotting, Northern; Brain; Ergolines; Male; Mice; Mice, Inbred Strains; Nucleic Acid Hybridization; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, Serotonin; RNA Probes; RNA, Messenger; Tritium

1990
Identification of 5-hydroxytryptamine1D binding sites in human brain membranes.
    Synapse (New York, N.Y.), 1989, Volume: 3, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adolescent; Adult; Aged; Binding, Competitive; Caudate Nucleus; Ergolines; Frontal Lobe; Globus Pallidus; Humans; Middle Aged; Receptors, Serotonin; Subcellular Fractions; Tetrahydronaphthalenes

1989
Detection and characterization of a 5HT1D serotonin receptor-GTP binding protein interaction in porcine and bovine brain.
    Synapse (New York, N.Y.), 1989, Volume: 3, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Brain; Cattle; Ergolines; GTP-Binding Proteins; In Vitro Techniques; Receptors, Serotonin; Swine; Tetrahydronaphthalenes

1989
Serotonin-1 receptor binding sites in the human basal ganglia are decreased in Huntington's chorea but not in Parkinson's disease: a quantitative in vitro autoradiography study.
    Neuroscience, 1989, Volume: 32, Issue:2

    Topics: Aged; Basal Ganglia; Ergolines; Female; Humans; Huntington Disease; Male; Middle Aged; Parkinson Disease; Receptors, Serotonin

1989
5.HT1 receptors in the vertebrate brain. Regional distribution examined by autoradiography.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aged; Animals; Autoradiography; Brain; Cats; Disease Models, Animal; Dogs; Ergolines; Female; Guinea Pigs; Humans; Macaca mulatta; Male; Mice; Movement Disorders; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Tritium

1989
MK-212 increases rat plasma ACTH concentration by activation of the 5-HT1C receptor subtype.
    Neuroscience letters, 1989, Oct-23, Volume: 105, Issue:1-2

    Topics: Adrenocorticotropic Hormone; Animals; Antiparkinson Agents; Ergolines; Ketanserin; Male; Metergoline; Pindolol; Piperazines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1989
Exploratory hypoactivity induced by m-trifluoromethylphenylpiperazine (TFMPP) and m-chlorophenylpiperazine (m-CPP).
    Journal of neural transmission. Parkinson's disease and dementia section, 1989, Volume: 1, Issue:3

    Topics: Animals; Ergolines; Exploratory Behavior; Male; Metergoline; Mianserin; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1989
Stimulus generalization of 1-(3-trifluoromethylphenyl)piperazine (TFMPP) to propranolol, pindolol, and mesulergine.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Antiparkinson Agents; Drug Interactions; Ergolines; Generalization, Stimulus; Male; Pindolol; Piperazines; Propranolol; Rats; Rats, Inbred Strains

1988
Evidence that hypophagia induced by mCPP and TFMPP requires 5-HT1C and 5-HT1B receptors; hypophagia induced by RU 24969 only requires 5-HT1B receptors.
    Psychopharmacology, 1988, Volume: 96, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Ergolines; Feeding Behavior; Food Deprivation; Indoles; Male; Mianserin; Motor Activity; Pindolol; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tropisetron

1988
Molecular pharmacology of 5-HT1 and 5-HT2 recognition sites in rat and pig brain membranes: radioligand binding studies with [3H]5-HT, [3H]8-OH-DPAT, (-)[125I]iodocyanopindolol, [3H]mesulergine and [3H]ketanserin.
    European journal of pharmacology, 1985, Nov-26, Volume: 118, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Chemistry; Choroid Plexus; Ergolines; In Vitro Techniques; Iodocyanopindolol; Ketanserin; Male; Membranes; Pindolol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tetrahydronaphthalenes

1985
Serotonin receptors in the human brain. II. Characterization and autoradiographic localization of 5-HT1C and 5-HT2 recognition sites.
    Brain research, 1986, Jun-18, Volume: 376, Issue:1

    Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Cerebral Cortex; Choroid Plexus; Ergolines; Female; Humans; Ketanserin; Male; Membranes; Middle Aged; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Swine; Tissue Distribution; Tritium

1986
Characterization of a novel 3H-5-hydroxytryptamine binding site subtype in bovine brain membranes.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding Sites; Binding, Competitive; Brain; Calcium; Cattle; Caudate Nucleus; Ergolines; Membranes; Nucleotides; Osmolar Concentration; Serotonin; Tetrahydronaphthalenes; Tritium

1987
Serotonin receptors in the human brain--III. Autoradiographic mapping of serotonin-1 receptors.
    Neuroscience, 1987, Volume: 21, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adult; Aged; Aged, 80 and over; Autoradiography; Brain; Ergolines; Female; Humans; Male; Mianserin; Middle Aged; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1987
Identification of 5-hydroxytryptamine binding site subtypes in rat spinal cord.
    Brain research, 1987, Dec-08, Volume: 436, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding Sites; Binding, Competitive; Ergolines; In Vitro Techniques; Indoles; Rats; Receptors, Serotonin; Serotonin; Spinal Cord; Tetrahydronaphthalenes

1987
A pharmacological analysis of the rat spinal cord serotonin (5-HT) autoreceptor.
    European journal of pharmacology, 1988, Jan-12, Volume: 145, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Male; Piperazines; Potassium; Quipazine; Rats; Receptors, Serotonin; Serotonin; Spinal Cord; Spiperone; Tetrahydronaphthalenes; Tritium

1988
Identification of a 5-HT1 recognition site in human brain membranes different from 5-HT1A, 5-HT1B and 5-HT1C sites.
    Neuroscience letters, 1988, Mar-10, Volume: 85, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Binding, Competitive; Brain Chemistry; Caudate Nucleus; Cerebral Cortex; Ergolines; Humans; Receptors, Serotonin; Tetrahydronaphthalenes

1988
Molecular pharmacology of 5-HT1D recognition sites: radioligand binding studies in human, pig and calf brain membranes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antiparkinson Agents; Brain; Cattle; Caudate Nucleus; Ergolines; Humans; In Vitro Techniques; Kinetics; Membranes; Receptors, Serotonin; Serotonin Antagonists; Species Specificity; Swine; Tetrahydronaphthalenes

1988
Serotonin-1C sites in the choroid plexus are not linked in a stimulatory or inhibitory way to adenylate cyclase.
    Brain research, 1986, Aug-13, Volume: 380, Issue:1

    Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cerebral Cortex; Choroid Plexus; Colforsin; Cyclic AMP; Dopamine; Ergolines; Hippocampus; Histamine; Kinetics; Mianserin; Rats; Receptors, Serotonin; Serotonin; Swine

1986
Dopamine agonists as primary treatment in Parkinson's disease.
    Advances in neurology, 1987, Volume: 45

    Topics: Antiparkinson Agents; Bromocriptine; Disability Evaluation; Drug Therapy, Combination; Ergolines; Humans; Levodopa; Lisuride; Long-Term Care; Parkinson Disease; Pergolide; Receptors, Dopamine

1987
Pleuropulmonary disease during bromocriptine treatment of Parkinson's disease.
    Archives of internal medicine, 1988, Volume: 148, Issue:10

    Topics: Aged; Antiparkinson Agents; Bromocriptine; Ergolines; Humans; Lung Diseases; Male; Middle Aged; Parkinson Disease; Pleural Diseases; Radiography

1988
Detection and characterization of the serotonin 5-HT 1D receptor in rat and human brain.
    Journal of neurochemistry, 1988, Volume: 50, Issue:5

    Topics: Animals; Binding, Competitive; Brain; Brain Chemistry; Caudate Nucleus; Cerebral Cortex; Ergolines; Humans; Kinetics; Male; Middle Aged; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tissue Distribution

1988
Antihypertensive effects of mesulergine: further evidence for a peripheral site of action of dopamine agonists.
    Fundamental & clinical pharmacology, 1987, Volume: 1, Issue:3

    Topics: Animals; Antihypertensive Agents; Antiparkinson Agents; Blood Pressure; Cisterna Magna; Dogs; Ergolines; Female; Injections; Injections, Intravenous; Male; Receptors, Dopamine

1987
Mesulergine and pergolide in previously untreated Parkinson's disease.
    Journal of neurology, neurosurgery, and psychiatry, 1987, Volume: 50, Issue:4

    Topics: Aged; Antiparkinson Agents; Domperidone; Ergolines; Female; Humans; Male; Parkinson Disease; Pergolide

1987
The effect of the ergoline derivative, CU 32-085, on prolactin secretion in hyperprolactinemic women.
    Fertility and sterility, 1987, Volume: 48, Issue:4

    Topics: Adenoma; Adult; Ergolines; Female; Humans; Hyperprolactinemia; Kinetics; Menstruation Disturbances; Pituitary Neoplasms; Prolactin

1987
On the mode of action of six putative dopamine receptor agonists on suppression of exploratory behaviour in rats.
    Psychopharmacology, 1987, Volume: 91, Issue:2

    Topics: Animals; Bromocriptine; Ergolines; Exploratory Behavior; Habituation, Psychophysiologic; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1987
Mesulergine (CU 32-085) in the treatment of Parkinson's disease.
    Clinical neuropharmacology, 1986, Volume: 9, Issue:2

    Topics: Adult; Aged; Antiparkinson Agents; Drug Administration Schedule; Ergolines; Female; Humans; Levodopa; Male; Middle Aged; Movement Disorders; Parkinson Disease; Time Factors

1986
[125I]LSD labels 5-HT1C recognition sites in pig choroid plexus membranes. Comparison with [3H]mesulergine and [3H]5-HT binding.
    Neuroscience letters, 1986, Sep-12, Volume: 69, Issue:3

    Topics: Animals; Cell Membrane; Cerebral Cortex; Choroid Plexus; Ergolines; Kinetics; Lysergic Acid Diethylamide; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin; Species Specificity; Swine

1986
Management of prolactinomas. A reappraisal.
    The Australian & New Zealand journal of obstetrics & gynaecology, 1985, Volume: 25, Issue:3

    Topics: Adenoma; Bromocriptine; Ergolines; Female; Humans; Lisuride; Metergoline; Pergolide; Pituitary Neoplasms; Pregnancy; Prolactin; Radiotherapy Dosage; Radiotherapy, High-Energy; Time Factors

1985
Efficacy of pergolide and mesulergine.
    European neurology, 1986, Volume: 25, Issue:2

    Topics: Aged; Antiparkinson Agents; Drug Therapy, Combination; Dyskinesia, Drug-Induced; Ergolines; Humans; Levodopa; Middle Aged; Parkinson Disease; Pergolide

1986
Initial treatment of parkinsonism with 8-alpha-amino-ergoline.
    Neurology, 1985, Volume: 35, Issue:1

    Topics: Adult; Aged; Ergolines; Female; Humans; Male; Middle Aged; Neurologic Examination; Parkinson Disease; Psychomotor Performance

1985
Central dopamine agonist activity on the 8-alpha-amino-ergoline CU 32-085.
    Brain research, 1985, Mar-04, Volume: 328, Issue:2

    Topics: Animals; Antiparkinson Agents; Brain; Chlorocebus aethiops; Corpus Striatum; Dopamine; Ergolines; Female; Male; Mice; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tremor

1985
Three-year observation of mesulergine (CU 32-085) in advanced and newly treated parkinsonism.
    Journal of neurology, 1985, Volume: 232, Issue:1

    Topics: Adult; Aged; Antiparkinson Agents; Bromocriptine; Drug Therapy, Combination; Ergolines; Female; Humans; Levodopa; Male; Middle Aged; Parkinson Disease

1985
Comparison of the clinical activity of mesulergine and pergolide in the treatment of hyperprolactinaemia.
    Clinical endocrinology, 1985, Volume: 22, Issue:5

    Topics: Adenoma; Adult; Ergolines; Female; Humans; Male; Middle Aged; Pergolide; Pituitary Neoplasms; Pregnancy; Prolactin

1985
The effect of dopamine agonist therapy on large functionless pituitary tumours.
    Clinical endocrinology, 1985, Volume: 22, Issue:5

    Topics: Adenoma, Chromophobe; Adult; Bromocriptine; Dopamine; Ergolines; Female; Humans; Male; Middle Aged; Pergolide; Pituitary Neoplasms; Prolactin; Prospective Studies

1985
[Hyperprolactinemia and prolactinomas. Results of surgical and drug therapy].
    Deutsche medizinische Wochenschrift (1946), 1985, Oct-11, Volume: 110, Issue:41

    Topics: Adolescent; Adult; Aged; Bromocriptine; Dopamine; Drug Therapy, Combination; Ergolines; Female; Humans; Hyperprolactinemia; Lisuride; Male; Middle Aged; Paraneoplastic Endocrine Syndromes; Prolactin

1985
Dopamine agonists and Parkinson's disease.
    Clinical neurology and neurosurgery, 1984, Volume: 86, Issue:3

    Topics: Antiparkinson Agents; Apomorphine; Brain; Bromocriptine; Ergolines; Ergot Alkaloids; Humans; Levodopa; Lisuride; Neurons; Parkinson Disease; Pergolide; Piribedil; Receptors, Dopamine

1984
Biphasic influence of a 8 alpha-amino ergoline, CU 32-085, on striatal dopamine synthesis and turnover in vivo in the rat.
    Life sciences, 1981, Nov-23, Volume: 29, Issue:21

    Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; alpha-Methyltyrosine; Animals; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Ergolines; Homovanillic Acid; Male; Methyltyrosines; Rats; Time Factors; Tyrosine 3-Monooxygenase

1981
Therapeutic potentials of centrally acting dopamine and alpha 2-adrenoreceptor agonists.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Adrenergic alpha-Agonists; Animals; Dopamine; Ergolines; Haplorhini; Humans; Neurons; Norepinephrine; Parkinson Disease; Pergolide; Quinpirole; Rats

1983
Investigation of the influence of lithium upon the down-regulation of serotonin2 receptors in rat frontal cortex induced by long-term treatment with dibenzepin, an antidepressant without appreciable affinity to serotonin2 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 326, Issue:4

    Topics: Animals; Dibenzazepines; Ergolines; Frontal Lobe; Lithium; Male; Radioligand Assay; Rats; Receptors, Serotonin; Time Factors

1984
Hypotensive action and alpha-adrenolytic properties of a new dopaminergic agonist, CU 32-085, in the rat.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 272, Issue:1

    Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Antihypertensive Agents; Antiparkinson Agents; Blood Pressure; Bromocriptine; Clonidine; Epinephrine; Ergolines; Female; Heart Rate; Hemodynamics; Male; Methoxamine; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Dopamine

1984
Therapeutic experience with the new dopamine agonist CU 32-085 in advanced Parkinson's disease.
    Journal of neurology, 1983, Volume: 230, Issue:1

    Topics: Adult; Aged; Amantadine; Antiparkinson Agents; Bromocriptine; Carboxy-Lyases; Drug Therapy, Combination; Ergolines; Female; Humans; Levodopa; Male; Middle Aged; Parasympatholytics; Parkinson Disease

1983
Mesulergine and its 1,20-N,N-bidemethylated metabolite interact directly with D1- and D2-receptors.
    European journal of pharmacology, 1983, Nov-11, Volume: 95, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Antiparkinson Agents; Chemical Phenomena; Chemistry; Choline; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1983
Dopamine agonists in Parkinson's disease.
    The Canadian journal of neurological sciences. Le journal canadien des sciences neurologiques, 1984, Volume: 11, Issue:1 Suppl

    Topics: Bromocriptine; Dopamine; Drug Therapy, Combination; Ergolines; Ergot Alkaloids; Humans; Levodopa; Lisuride; Parkinson Disease; Pergolide; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1984
Dopamine agonists in the treatment of Parkinson's disease.
    Advances in neurology, 1983, Volume: 37

    Topics: Blood Pressure; Bromocriptine; Disability Evaluation; Domperidone; Dopamine; Ergolines; Follow-Up Studies; Humans; Levodopa; Parkinson Disease; Pleural Effusion; Receptors, Neurotransmitter; Time Factors

1983
Mesulergine, a new dopamine agonist: effects on anterior pituitary function and kinetics.
    Clinical pharmacology and therapeutics, 1984, Volume: 36, Issue:5

    Topics: Absorption; Adult; Analysis of Variance; Biological Availability; Bromocriptine; Ergolines; Humans; Male; Pituitary Gland, Anterior; Pituitary Hormone-Releasing Hormones; Prolactin; Radioimmunoassay

1984
Dopamine agonistic potency of two novel prolactin release-inhibiting ergolines.
    European journal of pharmacology, 1984, Jun-01, Volume: 101, Issue:3-4

    Topics: Animals; Cells, Cultured; Dopamine; Ergolines; Male; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains

1984
Mechanism of action and tolerance of mesulergine.
    Clinical pharmacology and therapeutics, 1984, Volume: 36, Issue:5

    Topics: Adenoma; Administration, Oral; Adult; Animals; Blood Pressure; Bromocriptine; Cells, Cultured; Dopamine Antagonists; Drug Evaluation; Ergolines; Female; Humans; Hypotension; Male; Menstruation; Middle Aged; Nausea; Pituitary Neoplasms; Prolactin; Radioimmunoassay; Random Allocation; Rats

1984
Mesulergine, a selective serotonin-2 ligand in the rat cortex, does not label these receptors in porcine and human cortex: evidence for species differences in brain serotonin-2 receptors.
    European journal of pharmacology, 1984, Nov-27, Volume: 106, Issue:3

    Topics: Animals; Brain Chemistry; Cerebral Cortex; Ergolines; Humans; In Vitro Techniques; Ketanserin; Kinetics; Ligands; Male; Piperidines; Rats; Receptors, Serotonin; Species Specificity; Swine; Tritium

1984
The binding of serotonergic ligands to the porcine choroid plexus: characterization of a new type of serotonin recognition site.
    European journal of pharmacology, 1984, Nov-27, Volume: 106, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Choroid Plexus; Ergolines; Frontal Lobe; In Vitro Techniques; Kinetics; Ligands; Receptors, Serotonin; Serotonin; Swine

1984
Dopaminergic properties of mesulergine (CU 32-085) and its metabolites.
    Journal of neural transmission, 1984, Volume: 60, Issue:3-4

    Topics: Animals; Corpus Striatum; Dopamine; Ergolines; Kinetics; Male; Rats; Receptors, Dopamine

1984
Low-dose CU 32-085 (mesulergine) in previously untreated Parkinson's disease.
    Neurology, 1984, Volume: 34, Issue:8

    Topics: Ergolines; Female; Humans; Male; Middle Aged; Parkinson Disease

1984
Treatment of Parkinson's disease with 8-alpha-amino-ergoline, CU 32-085.
    Neurology, 1983, Volume: 33, Issue:4

    Topics: Activities of Daily Living; Adult; Aged; Antiparkinson Agents; Bromocriptine; Drug Therapy, Combination; Ergolines; Female; Humans; Hypotension, Orthostatic; Levodopa; Male; Middle Aged; Nausea; Parkinson Disease; Psychomotor Performance; Receptors, Dopamine

1983
Therapeutic results with a new ergoline derivate (8-alpha-amino-ergoline, CU 32-085) in parkinsonian patients.
    Advances in neurology, 1984, Volume: 40

    Topics: Aged; Antiparkinson Agents; Bromocriptine; Drug Therapy, Combination; Ergolines; Female; Humans; Levodopa; Male; Middle Aged; Parkinson Disease

1984
Puerperal lactation inhibition with a novel 8 alpha-aminoergoline (CU 32-085).
    Gynecologic and obstetric investigation, 1984, Volume: 17, Issue:3

    Topics: Adolescent; Adult; Chemical Phenomena; Chemistry; Depression, Chemical; Ergolines; Female; Humans; Lactation; Postpartum Period; Pregnancy; Prolactin

1984
[3H]Mesulergine, a selective ligand for serotonin-2 receptors.
    Life sciences, 1983, May-23, Volume: 32, Issue:21

    Topics: Animals; Cations; Cerebral Cortex; Ergolines; Kinetics; Lithium; Male; Rats; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1983
The effects of lisuride and some other dopaminergic agonists on receptor binding in human brain.
    Journal of neural transmission, 1981, Volume: 51, Issue:1-2

    Topics: Brain; Bromocriptine; Ergolines; Humans; Kinetics; Lisuride; Receptors, Dopamine; Spiperone

1981
Effects of chronic cocaine administration on the serotonergic system in the rat brain.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 46, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Antiparkinson Agents; Brain; Brain Chemistry; Cocaine; Ergolines; Hydroxyindoleacetic Acid; Ketanserin; Male; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin

1993
The role of the 5-HT2A and 5-HT2C receptors in the stimulus effects of m-chlorophenylpiperazine.
    Psychopharmacology, 1995, Volume: 119, Issue:2

    Topics: Animals; Antiparkinson Agents; Binding, Competitive; Dose-Response Relationship, Drug; Ergolines; Male; Piperazines; Rats; Rats, Inbred F344; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
The 5-HT1B receptor mediates the effect of d-fenfluramine on eating caused by intra-hypothalamic injection of neuropeptide Y.
    European journal of pharmacology, 1995, Feb-14, Volume: 274, Issue:1-3

    Topics: Analysis of Variance; Animals; Antiparkinson Agents; Drug Interactions; Eating; Ergolines; Fenfluramine; Hyperphagia; Hypothalamus; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Male; Metergoline; Neuropeptide Y; Paraventricular Hypothalamic Nucleus; Pindolol; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists

1995
Differential effects of chronic antidepressant treatment on 5-HT1C receptor binding sites in Wistar rat brain.
    European journal of pharmacology, 1994, Sep-22, Volume: 263, Issue:1-2

    Topics: Animals; Brain; Clomipramine; Clorgyline; Ergolines; Imipramine; Male; Rats; Rats, Wistar; Receptors, Serotonin

1994
Further evidence that the tachycardiac response to 5-hydroxytryptamine in rats is not mediated via typical 5-HT2 receptors.
    General pharmacology, 1994, Volume: 25, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Ergolines; Female; Heart Rate; Ketanserin; Male; Methiothepin; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin

1994
Regulation of serotonin 5-HT2C receptors in the rat choroid plexus after acute clozapine treatment.
    European journal of pharmacology, 1994, Oct-14, Volume: 269, Issue:2

    Topics: Amphetamines; Animals; Antiparkinson Agents; Autoradiography; Cerebral Cortex; Choroid Plexus; Clozapine; Ergolines; Haloperidol; Image Processing, Computer-Assisted; Injections, Subcutaneous; Male; Neostriatum; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Serotonin; Serotonin Receptor Agonists

1994
Genomic organisation and functional expression of the gene encoding the human serotonin 5-HT2C receptor.
    European journal of pharmacology, 1994, Nov-15, Volume: 269, Issue:3

    Topics: 3T3 Cells; Amino Acid Sequence; Animals; Antiparkinson Agents; Base Sequence; Binding, Competitive; Blotting, Southern; Cloning, Molecular; DNA Primers; DNA, Complementary; Ergolines; Exons; Gene Expression Regulation; Hippocampus; Humans; Mice; Molecular Sequence Data; Polymerase Chain Reaction; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Restriction Mapping; RNA, Messenger; Transfection; Type C Phospholipases

1994
Constitutively active 5-hydroxytryptamine2C receptors reveal novel inverse agonist activity of receptor ligands.
    The Journal of biological chemistry, 1994, Apr-22, Volume: 269, Issue:16

    Topics: 3T3 Cells; Animals; Antiparkinson Agents; Cell Membrane; Cells, Cultured; Choroid Plexus; Cloning, Molecular; DNA, Complementary; DOM 2,5-Dimethoxy-4-Methylamphetamine; Epithelium; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Lysergic Acid Diethylamide; Mianserin; Mice; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin Antagonists; Transfection

1994
Regulation of serotonin2A receptors in heterologous expression systems.
    Journal of neurochemistry, 1994, Volume: 63, Issue:4

    Topics: 3T3 Cells; Animals; Antiparkinson Agents; Binding, Competitive; Cell Line; Dogs; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ergolines; Gene Expression Regulation; Ketanserin; Kidney; Kinetics; Mice; Pituitary Neoplasms; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Recombinant Proteins; Transfection; Tumor Cells, Cultured

1994
Serotonin-dopamine interaction in the rat ventral tegmental area: an electrophysiological study in vivo.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dopamine; Ergolines; Male; Motor Activity; Pindolol; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Ventral Tegmental Area

1994
Reciprocal binding properties of 5-hydroxytryptamine type 2C receptor agonists and inverse agonists.
    Molecular pharmacology, 1994, Volume: 46, Issue:5

    Topics: 3T3 Cells; Animals; Binding, Competitive; Cell Line; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ergolines; Guanine Nucleotides; Hydrolysis; Mice; Phosphatidylinositols; Radioligand Assay; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists

1994
5-HT1C receptor-mediated phosphoinositide hydrolysis in the rat choroid plexus after chronic treatment with clozapine.
    European journal of pharmacology, 1994, Apr-01, Volume: 255, Issue:1-3

    Topics: Amphetamines; Animals; Autoradiography; Choroid Plexus; Clozapine; Ergolines; Haloperidol; Hydrolysis; Image Processing, Computer-Assisted; In Vitro Techniques; Male; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Second Messenger Systems; Serotonin Receptor Agonists

1994
Involvement of 5-HT2C receptors in mediating the discriminative stimulus properties of m-chlorophenylpiperazine (mCPP).
    European journal of pharmacology, 1994, May-12, Volume: 257, Issue:1-2

    Topics: Animals; Discrimination, Psychological; Dopamine Antagonists; Ergolines; Fenfluramine; Lysergic Acid Diethylamide; Male; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Trazodone

1994
Modulation of rhythmic swimming activity in post-embryonic Xenopus laevis tadpoles by 5-hydroxytryptamine acting at 5HT1a receptors.
    Proceedings. Biological sciences, 1994, Jul-22, Volume: 257, Issue:1348

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Animals; Cyproheptadine; Ergolines; Ketanserin; Metamorphosis, Biological; Methysergide; Motor Activity; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming; Xenopus laevis

1994
Mesulergine antagonism towards the fluoxetine anti-immobility effect in the forced swimming test in mice.
    The Journal of pharmacy and pharmacology, 1993, Volume: 45, Issue:5

    Topics: Animals; Behavior, Animal; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Fluoxetine; Immobilization; Male; Mice; Neurotransmitter Uptake Inhibitors; Receptors, Serotonin; Swimming

1993
Analysis of the 5-HT1C receptor and the serotonin uptake site in fawn-hooded rat brain.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: Animals; Binding Sites; Brain; Brain Stem; Corpus Striatum; Ergolines; Frontal Lobe; Hippocampus; Hypothalamus; Male; Paroxetine; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Serotonin; Serotonin

1993
High and low affinity 5-HT2 and 5-HT1C binding sites: responses to neonatal 5,7-DHT lesions in rat brain.
    Cytobios, 1993, Volume: 75, Issue:302-303

    Topics: 5,7-Dihydroxytryptamine; Analysis of Variance; Animals; Animals, Newborn; Binding Sites; Brain Neoplasms; Brain Stem; Cerebellum; Cerebral Cortex; Diencephalon; Dose-Response Relationship, Drug; Ergolines; Female; Hippocampus; Injections, Intraperitoneal; Mianserin; Pregnancy; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin; Time Factors; Tritium

1993
Effect of 5,7-dihydroxytryptamine lesion on mianserin-induced conditioned place aversion and on 5-hydroxytryptamine1C receptors in the rat brain.
    Neuroscience, 1993, Volume: 56, Issue:3

    Topics: 5,7-Dihydroxytryptamine; Animals; Antiparkinson Agents; Autoradiography; Brain Chemistry; Carbolines; Conditioning, Operant; Ergolines; In Situ Hybridization; Male; Mianserin; Rats; Receptors, GABA-A; Receptors, Serotonin; RNA, Messenger; Transcription, Genetic

1993
Modulation of 5-HT1C receptors and phosphoinositide system by ethanol consumption in rat brain and choroid plexus.
    European journal of pharmacology, 1993, Sep-15, Volume: 247, Issue:1

    Topics: Animals; Antiparkinson Agents; Binding Sites; Brain; Cerebral Cortex; Choroid Plexus; Ergolines; Ethanol; Hippocampus; Hydrolysis; Male; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Up-Regulation

1993
Quantitative autoradiography of 5-HT1E binding sites in rodent brains: effect of lesion of serotonergic neurones.
    European journal of pharmacology, 1993, Nov-09, Volume: 249, Issue:2

    Topics: 5,7-Dihydroxytryptamine; Animals; Autoradiography; Binding, Competitive; Brain; Brain Chemistry; Ergolines; Guinea Pigs; In Vitro Techniques; Male; Membranes; Mice; Neurons; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists

1993
5-Carboxamidotryptamine-insensitive 5-HT1-like receptors are concentrated in guinea pig but not rat, claustrum.
    European journal of pharmacology, 1993, May-12, Volume: 236, Issue:1

    Topics: Animals; Antiparkinson Agents; Autoradiography; Basal Ganglia; Brain Mapping; Ergolines; Guinea Pigs; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Species Specificity

1993
5-HT1B receptors mediate potent contractile responses to 5-HT in rat caudal artery.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Arteries; Ergolines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Pindolol; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Vasoconstrictor Agents

1993
Autoradiographic studies of RP 62203, a potent 5-HT2 receptor antagonist. In vitro and ex vivo selectivity profile.
    European journal of pharmacology, 1993, Mar-16, Volume: 233, Issue:1

    Topics: Animals; Antiparkinson Agents; Autoradiography; Cerebellum; Choroid Plexus; Cyclic S-Oxides; Ergolines; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Naphthalenes; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Serotonin Antagonists; Thalamus

1993
A single point mutation (Phe340-->Leu340) of a conserved phenylalanine abolishes 4-[125I]iodo-(2,5-dimethoxy)phenylisopropylamine and [3H]mesulergine but not [3H]ketanserin binding to 5-hydroxytryptamine2 receptors.
    Molecular pharmacology, 1993, Volume: 43, Issue:5

    Topics: Amino Acid Sequence; Amphetamines; Animals; Base Sequence; Cell Line, Transformed; Chlorocebus aethiops; Ergolines; Hydrolysis; Ketanserin; Leucine; Molecular Sequence Data; Mutagenesis, Site-Directed; Phenylalanine; Phosphatidylinositols; Point Mutation; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1993
Identification of 5-hydroxytryptamine1D binding sites in sheep caudate nucleus membranes.
    Biochemical pharmacology, 1993, Aug-03, Volume: 46, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding Sites; Caudate Nucleus; Cell Membrane; Cerebral Cortex; Ergolines; Humans; Indoles; Rats; Selective Serotonin Reuptake Inhibitors; Serotonin; Sheep; Sulfonamides; Sumatriptan; Tritium

1993
Autoradiographic localization of serotonin receptor subtypes in cat visual cortex: transient regional, laminar, and columnar distributions during postnatal development.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Animals; Animals, Newborn; Antiparkinson Agents; Autoradiography; Cats; Ergolines; Granisetron; Organ Specificity; Receptors, Serotonin; Serotonin; Tritium; Visual Cortex

1993
Novel regulation of 5-HT1C receptors: down-regulation induced both by 5-HT1C/2 receptor agonists and antagonists.
    European journal of pharmacology, 1993, Jan-04, Volume: 244, Issue:1

    Topics: Analysis of Variance; Animals; Binding Sites; Down-Regulation; Ergolines; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Regression Analysis; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord

1993
5-hydroxytryptamine1 recognition sites in rat brain: heterogeneity of non-5-hydroxytryptamine1A/1C binding sites revealed by quantitative receptor autoradiography.
    Neuroscience, 1993, Volume: 53, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antiparkinson Agents; Autoradiography; Binding, Competitive; Brain Chemistry; Dipeptides; Ergolines; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Male; Mesencephalon; Prosencephalon; Rats; Receptors, Serotonin; Serotonin

1993
Lack of cross-tolerance for hypophagia induced by DOI versus m-CPP suggests separate mediation by 5-HT2A and 5-HT2C receptors, respectively.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1995, Volume: 13, Issue:1

    Topics: Amphetamines; Animals; Binding, Competitive; Drug Tolerance; Eating; Ergolines; Frontal Lobe; Injections, Intraperitoneal; Ketanserin; Male; Piperazines; Propane; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Receptor Agonists; Time Factors

1995
Contribution of a helix 5 locus to selectivity of hallucinogenic and nonhallucinogenic ligands for the human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors: direct and indirect effects on ligand affinity mediated by the same locus.
    Molecular pharmacology, 1996, Volume: 50, Issue:1

    Topics: Amino Acid Sequence; Animals; Binding Sites; Binding, Competitive; Cell Line; Chlorocebus aethiops; Ergolines; Hallucinogens; Humans; Ketanserin; Kinetics; Ligands; Lysergic Acid Diethylamide; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Phosphatidylinositols; Point Mutation; Protein Structure, Secondary; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Sequence Homology, Amino Acid; Structure-Activity Relationship; Transfection

1996
Effects of antidepressants on intracellular Ca2+ mobilization in CHO cells transfected with the human 5-HT2C receptors.
    Biological psychiatry, 1996, Jun-15, Volume: 39, Issue:12

    Topics: Animals; Antidepressive Agents; Antidepressive Agents, Second-Generation; Calcium; Calcium Channels; CHO Cells; Cricetinae; Ergolines; Humans; Intracellular Fluid; Mianserin; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction; Transfection

1996
Functional reconstitution in situ of 5-hydroxytryptamine2c (5HT2c) receptors with alphaq and inverse agonism of 5HT2c receptor antagonists.
    The Journal of biological chemistry, 1996, Sep-13, Volume: 271, Issue:37

    Topics: Animals; Binding, Competitive; Cattle; Cell Line; Decapodiformes; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Ketanserin; Mianserin; Photoreceptor Cells, Invertebrate; Rats; Receptor, Serotonin, 5-HT2C; Receptors, Cell Surface; Receptors, Serotonin; Recombinant Proteins; Serotonin

1996
Sequential onset of three 5-HT receptors during the 5-hydroxytryptaminergic differentiation of the murine 1C11 cell line.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Animals; Antiparkinson Agents; Cells, Cultured; Colforsin; Cyclic AMP; Ergolines; Gene Expression; Quinoxalines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Time Factors

1996
Chronic citalopram and fluoxetine treatments upregulate 5-HT2c receptors in the rat choroid plexus.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1996, Volume: 15, Issue:2

    Topics: Amphetamines; Animals; Antiparkinson Agents; Autoradiography; Choroid Plexus; Citalopram; Ergolines; Fluoxetine; Image Processing, Computer-Assisted; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Up-Regulation

1996
Serotonin2C receptors and serotonin2C receptor-mediated phosphoinositide hydrolysis in the brain of alcohol-preferring and alcohol-nonpreferring rats.
    Alcoholism, clinical and experimental research, 1996, Volume: 20, Issue:6

    Topics: Alcohol Drinking; Alcoholism; Animals; Brain; Brain Mapping; Choroid Plexus; Ergolines; Hydrolysis; Male; Phosphatidylinositols; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin

1996
Activities of novel aryloxyalkylimidazolines on rat 5-HT2A and 5-HT2C receptors.
    European journal of pharmacology, 1996, Feb-05, Volume: 296, Issue:3

    Topics: 3T3 Cells; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Lysergic Acid Diethylamide; Mice; Phosphatidylinositols; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Effect of a dopamine agonist on the development of Leydig cell hyperplasia in Sprague-Dawley rats.
    Toxicology and applied pharmacology, 1996, Volume: 141, Issue:1

    Topics: Adenoma; Animals; Antiparkinson Agents; Body Weight; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Extracellular Space; Hyperplasia; Leydig Cell Tumor; Leydig Cells; Male; Organ Size; Rats; Rats, Sprague-Dawley; Testicular Neoplasms

1996
Characterisation of human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors expressed in the human neuroblastoma cell line SH-SY5Y: comparative stimulation by hallucinogenic drugs.
    Journal of neurochemistry, 1996, Volume: 67, Issue:6

    Topics: Adrenergic alpha-Agonists; Amphetamines; Antiparkinson Agents; Calcium; Choroid Plexus; Electrophysiology; Ergolines; Ergotamine; Frontal Lobe; Hallucinogens; Humans; Hydrolysis; Ketanserin; Lysergic Acid Diethylamide; Mescaline; Methoxydimethyltryptamines; Neuroblastoma; Phosphatidylinositols; Piperazines; Quipazine; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium; Tumor Cells, Cultured

1996
Serotonin activates electrolyte transport via 5-HT2A receptor in rat colonic crypt cells.
    Biochemical and biophysical research communications, 1997, Jan-13, Volume: 230, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Biological Transport; Calcium; Cells, Cultured; Chlorides; Colon; Egtazic Acid; Electrolytes; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Intestinal Mucosa; Male; Membrane Potentials; Patch-Clamp Techniques; Potassium; Protein Kinase Inhibitors; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin

1997
Mechanism of actions of sumatriptan on coronary flow before and after endothelial dysfunction in guinea-pig isolated heart.
    British journal of pharmacology, 1997, Volume: 120, Issue:6

    Topics: Animals; Coronary Circulation; Coronary Vessels; Endothelium, Vascular; Enzyme Inhibitors; Ergolines; Guinea Pigs; Heart; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Piperazines; Saponins; Serotonin Receptor Agonists; Sumatriptan; Vasoconstrictor Agents

1997
Blockade of serotonin-2C receptors by mesulergine reduces ocular dominance plasticity in kitten visual cortex.
    Experimental brain research, 1997, Volume: 114, Issue:2

    Topics: Animals; Cats; Dominance, Cerebral; Electric Stimulation; Ergolines; Functional Laterality; Microelectrodes; Neuronal Plasticity; Neurons; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Vision, Monocular; Visual Cortex; Visual Perception

1997
Synthesis, affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors and structure-activity relationships of a series of cyproheptadine analogues.
    Chemical & pharmaceutical bulletin, 1997, Volume: 45, Issue:5

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Choroid Plexus; Cyproheptadine; Ergolines; Gastric Fundus; In Vitro Techniques; Ketanserin; Kinetics; Male; Models, Molecular; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Swine

1997
5-HT2 receptor regulation of acetylcholine release induced by dopaminergic stimulation in rat striatal slices.
    Brain research, 1997, May-16, Volume: 757, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Benzazepines; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Ergolines; Haloperidol; In Vitro Techniques; Ketanserin; Male; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Physalaemin; Potassium; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Substance P

1997
Nature of 5-HT1-like receptors mediating depressor responses in vagosympathectomized rats; close resemblance to the cloned 5-ht7 receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: 5-Methoxytryptamine; Adrenergic beta-Agonists; Animals; Blood Pressure; Clozapine; Ergolines; Heart Rate; Isoproterenol; Lisuride; Male; Metergoline; Methiothepin; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathectomy

1997
Mianserin-induced down-regulation of human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors stably expressed in the human neuroblastoma cell line SH-SY5Y.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: Cell Membrane; DNA, Complementary; Down-Regulation; Ergolines; Humans; Ketanserin; Kinetics; Mianserin; Neuroblastoma; Phosphatidylinositols; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Serotonin; Time Factors; Transfection; Tumor Cells, Cultured

1997
Activating mutations of the serotonin 5-HT2C receptor.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: Animals; Binding Sites; COS Cells; Ergolines; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Kinetics; Lysine; Methysergide; Mianserin; Mutagenesis, Site-Directed; Phenylalanine; Phosphatidylinositols; Point Mutation; Protein Conformation; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Serine; Serotonin; Serotonin Antagonists; Signal Transduction; Transfection

1997
Identification and characterization of a new serotonergic recognition site with high affinity for 5-carboxamidotryptamine in mammalian brain.
    Journal of neurochemistry, 1997, Volume: 69, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Cerebral Cortex; Ergolines; Ergotamine; Female; Guinea Pigs; Humans; Kinetics; Male; Mammals; Middle Aged; Organ Specificity; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium

1997
Selective visualization of rat brain 5-HT2A receptors by autoradiography with [3H]MDL 100,907.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:4

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Fluorobenzenes; Guanylyl Imidodiphosphate; In Situ Hybridization; In Vitro Techniques; Ketanserin; Male; Naphthalenes; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists

1997
Increase of cortical acetylcholine release after systemic administration of chlorophenylpiperazine in the rat: an in vivo microdialysis study.
    Neuroscience letters, 1997, Nov-07, Volume: 236, Issue:3

    Topics: Acetylcholine; Animals; Antihypertensive Agents; Aporphines; Cerebral Cortex; Ergolines; Male; Microdialysis; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Substantia Innominata

1997
Correlation between 5-HT7 receptor affinity and protection against sound-induced seizures in DBA/2J mice.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:6

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; CHO Cells; Cricetinae; Ergolines; Male; Methysergide; Mianserin; Mice; Mice, Inbred DBA; Receptors, Serotonin; Seizures; Serotonin Antagonists

1997
Identification of class-determining residues in G protein-coupled receptors by sequence analysis.
    Receptors & channels, 1997, Volume: 5, Issue:3-4

    Topics: Amino Acid Sequence; Binding Sites; Chlorpromazine; Ergolines; GTP-Binding Proteins; Ligands; Molecular Sequence Data; Molecular Structure; Pindolol; Propranolol; Receptors, Cell Surface; Receptors, Muscarinic; Receptors, Serotonin; Sequence Analysis; Sequence Homology, Amino Acid; Serotonin Receptor Agonists

1997
Serotonin receptors in the caudal brainstem are necessary and sufficient for the anorectic effect of peripherally administered mCPP.
    Psychopharmacology, 1998, Volume: 137, Issue:1

    Topics: Animals; Appetite Depressants; Brain Stem; Decerebrate State; Dose-Response Relationship, Drug; Ergolines; Injections, Intraventricular; Male; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists

1998
5-Hydroxytryptophan-induced myoclonus in guinea pigs: mediation through 5-HT1/2 receptor subtypes.
    European journal of pharmacology, 1998, Apr-17, Volume: 347, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Guinea Pigs; Male; Methiothepin; Myoclonus; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Substrate Specificity

1998
Effect of a dopamine agonist on luteinizing hormone receptors, cyclic AMP production and steroidogenesis in rat Leydig cells.
    Toxicology and applied pharmacology, 1998, Volume: 150, Issue:2

    Topics: Administration, Oral; Animals; Aromatase; Cell Separation; Chorionic Gonadotropin; Cyclic AMP; Dopamine Agonists; Ergolines; Hydroxycholesterols; Iodine Radioisotopes; Leydig Cells; Male; Pregnenolone; Rats; Rats, Sprague-Dawley; Receptors, LH; Serotonin Antagonists; Signal Transduction; Testosterone

1998
Selective blockade of serotonin2C/2B receptors enhances dopamine release in the rat nucleus accumbens.
    Neuropharmacology, 1998, Volume: 37, Issue:2

    Topics: Animals; Apomorphine; Cyclic S-Oxides; Dopamine; Dopamine Agonists; Ergolines; Indoles; Microdialysis; Naphthalenes; Nucleus Accumbens; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1998
Effects of mesulergine treatment on diet selection, brain serotonin (5-HT) and dopamine (DA) turnover in free feeding rats.
    Progress in neuro-psychopharmacology & biological psychiatry, 1998, Volume: 22, Issue:5

    Topics: Animals; Body Weight; Brain Chemistry; Dietary Carbohydrates; Dopamine; Dopamine Agonists; Ergolines; Food Preferences; Male; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists

1998
[3H]MDL 100,907 labels 5-HT2A serotonin receptors selectively in primate brain.
    Neuropharmacology, 1998, Volume: 37, Issue:9

    Topics: Aged; Aged, 80 and over; Animals; Binding Sites; Binding, Competitive; Brain; Cyclic S-Oxides; Ergolines; Female; Fluorobenzenes; Humans; In Situ Hybridization; Ketanserin; Macaca fascicularis; Male; Naphthalenes; Piperidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Tritium

1998
The canine external carotid vasoconstrictor 5-HT1 receptor: blockade by 5-HT1B (SB224289), but not by 5-HT1D (BRL15572) receptor antagonists.
    European journal of pharmacology, 1998, Nov-27, Volume: 362, Issue:1

    Topics: Anesthesia; Animals; Biphenyl Compounds; Blood Pressure; Carotid Artery, External; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Heart Rate; Norepinephrine; Piperazines; Piperidones; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiro Compounds; Sumatriptan; Sympathectomy; Vagotomy; Vasoconstriction

1998
Global increases in seizure susceptibility in mice lacking 5-HT2C receptors: a behavioral analysis.
    Experimental neurology, 1998, Volume: 154, Issue:2

    Topics: Animals; Behavior, Animal; Brain Chemistry; Convulsants; Cornea; Disease Susceptibility; Dopamine Agonists; Electroshock; Epilepsies, Myoclonic; Epilepsy; Ergolines; Flurothyl; Kindling, Neurologic; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Knockout; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin

1998
Structure-function studies of the eighth hydrophobic domain of a serotonin receptor.
    Journal of neurochemistry, 1999, Volume: 72, Issue:1

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Biological Transport; Chlorides; Ergolines; Fluorescent Antibody Technique; Gene Expression; GTP-Binding Proteins; Ligands; Molecular Sequence Data; Mutagenesis; Oocytes; Protein Structure, Secondary; Protein Structure, Tertiary; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Xenopus laevis

1999
Animal model of posthypoxic myoclonus: effects of serotonergic antagonists.
    Neurology, 1999, Jan-01, Volume: 52, Issue:1

    Topics: Acoustic Stimulation; Animals; Brain Chemistry; Disease Models, Animal; Dose-Response Relationship, Drug; Ergolines; Heart Arrest; Hypoxia; Hypoxia, Brain; Male; Methiothepin; Myoclonus; Oxadiazoles; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists

1999
Pharmacological characterization of the constitutively activated state of the serotonin 5-HT2C receptor.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: 3T3 Cells; Amino Acid Substitution; Animals; Cell Membrane; Ergolines; Kinetics; Lysine; Mice; Mutagenesis, Site-Directed; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Serine; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Transfection

1998
[3H]-Mesulergine labels 5-HT7 sites in rat brain and guinea-pig ileum but not rat jejunum.
    British journal of pharmacology, 1999, Volume: 126, Issue:1

    Topics: 5-Methoxytryptamine; Animals; Binding Sites; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Ergolines; Female; Free Radical Scavengers; Guinea Pigs; Ileum; In Vitro Techniques; Jejunum; Male; Muscle Contraction; Ondansetron; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Sumatriptan; Tritium

1999
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
    Journal of neurochemistry, 1999, Volume: 72, Issue:5

    Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1999
Systemic chlorophenylpiperazine increases acetylcholine release from rat hippocampus-implication of 5-HT2C receptors.
    Pharmacological research, 1999, Volume: 40, Issue:2

    Topics: Acetylcholine; Animals; Aporphines; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Routes; Ergolines; Haloperidol; Hippocampus; Male; Piperazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Serotonin 5-HT2C receptor RNA editing alters receptor basal activity: implications for serotonergic signal transduction.
    Journal of neurochemistry, 1999, Volume: 73, Issue:4

    Topics: Animals; COS Cells; Ergolines; Humans; Inositol Phosphates; Kinetics; Mianserin; Mutagenesis, Site-Directed; Pargyline; Rats; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; RNA Editing; Serotonin; Serotonin Antagonists; Signal Transduction; Transfection

1999
Agonist-induced GTPgamma35S binding mediated by human 5-HT(2C) receptors expressed in human embryonic kidney 293 cells.
    European journal of pharmacology, 1999, Nov-03, Volume: 383, Issue:3

    Topics: Cyclic AMP; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Inositol 1,4,5-Trisphosphate; Kidney; Pertussis Toxin; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Virulence Factors, Bordetella

1999
Distribution and characterization of [3H]mesulergine binding in human brain postmortem.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1999, Volume: 10, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Binding Sites; Binding, Competitive; Brain; Cell Membrane; Choroid Plexus; Dopamine Antagonists; Ergolines; Female; Humans; Male; Middle Aged; Postmortem Changes; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Substantia Nigra; Substrate Specificity; Tissue Distribution; Tritium

1999
Characterisation of a 5-HT(7) binding site in mouse ileum.
    European journal of pharmacology, 2000, Jan-17, Volume: 387, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding Sites; Ergolines; Female; Ileum; Male; Mice; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Antagonists

2000
Subthalamic nucleus microinjections of 5-HT2 receptor antagonists suppress stereotypy in rats.
    Neuroreport, 2000, Feb-07, Volume: 11, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Clozapine; Ergolines; Fluorobenzenes; Male; Mastication; Microinjections; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Stereotypic Movement Disorder; Subthalamic Nucleus

2000
Auditory responses from the frontal cortex in the mustached bat, Pteronotus parnellii.
    Neuroreport, 2000, Feb-07, Volume: 11, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Clozapine; Ergolines; Fluorobenzenes; Male; Mastication; Microinjections; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Stereotypic Movement Disorder; Subthalamic Nucleus

2000
An innovative method for rapid characterisation of phospholipase C activity: SB242,084 competitively antagonises 5-HT2C receptor-mediated [3H]phosphatidylinositol depletion.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 361, Issue:2

    Topics: Aminopyridines; Animals; CHO Cells; Cricetinae; Ergolines; Humans; Indoles; Phosphatidylinositols; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Type C Phospholipases

2000
Antagonist binding at 5-HT(2A) and 5-HT(2C) receptors in the rabbit: high correlation with the profile for the human receptors.
    European journal of pharmacology, 2000, Oct-13, Volume: 406, Issue:2

    Topics: Animals; Cerebral Cortex; Ergolines; Female; Fluorobenzenes; Humans; Male; Piperidines; Rabbits; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists

2000
In vivo analysis of adrenergic and serotoninergic constrictions of the rabbit saphenous vein.
    European journal of pharmacology, 2000, Nov-24, Volume: 408, Issue:3

    Topics: Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anesthesia; Animals; Benzazepines; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Indoles; Injections, Intravenous; Isoindoles; Oxadiazoles; Peripheral Nervous System; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Agents; Serotonin Receptor Agonists; Sumatriptan; Tetrahydronaphthalenes; Time Factors; Ultrasonography, Doppler; Vasoconstrictor Agents

2000
5-HT2C receptor binding is increased in the substantia nigra pars reticulata in Parkinson's disease.
    Movement disorders : official journal of the Movement Disorder Society, 2000, Volume: 15, Issue:6

    Topics: Aged; Aged, 80 and over; Antiparkinson Agents; Autoradiography; Binding Sites; Brain; Dopamine Agonists; Dyskinesia, Drug-Induced; Ergolines; Female; Humans; Male; Parkinson Disease; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Substantia Nigra

2000
Conserved helix 7 tyrosine functions as an activation relay in the serotonin 5HT(2C) receptor.
    Brain research. Molecular brain research, 2000, Dec-08, Volume: 84, Issue:1-2

    Topics: Amino Acid Motifs; Amphetamines; Binding, Competitive; Cell Line; Conserved Sequence; Ergolines; Humans; Indoles; Inositol Phosphates; Ligands; Mianserin; Mutation; Protein Structure, Secondary; Pyridines; Quipazine; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Transfection; Tyrosine

2000
No involvement of 5-HT(7) or 5-HT(1D) receptors in the (R)-8-OH-DPAT-induced depression of the monosynaptic reflex in spinalized rats.
    European journal of pharmacology, 2001, Sep-14, Volume: 427, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Clozapine; Decerebrate State; Dose-Response Relationship, Drug; Ergolines; Indoles; Male; Methiothepin; Oxadiazoles; Phenols; Piperazines; Pyridines; Rats; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Time Factors

2001
RNA-editing of the 5-HT(2C) receptor alters agonist-receptor-effector coupling specificity.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: Amphetamines; Animals; Arachidonic Acid; Binding, Competitive; Bufotenin; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Ergolines; Inositol Phosphates; Lysergic Acid Diethylamide; Piperazines; Protein Isoforms; Quipazine; Radioligand Assay; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; RNA Editing; Serotonin; Serotonin Receptor Agonists; Tritium

2001
Regional distribution and cellular localization of 5-HT2C receptor mRNA in monkey brain: comparison with [3H]mesulergine binding sites and choline acetyltransferase mRNA.
    Synapse (New York, N.Y.), 2001, Volume: 42, Issue:1

    Topics: Animals; Binding Sites; Brain; Choline O-Acetyltransferase; Ergolines; Female; Macaca fascicularis; Macaca mulatta; Male; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; RNA, Messenger; Serotonin Antagonists

2001
Different regulation of rat 5-HT(2A) and rat 5-HT(2C) receptors in NIH 3T3 cells upon exposure to 5-HT and pipamperone.
    European journal of pharmacology, 2001, Aug-03, Volume: 425, Issue:1

    Topics: 3T3 Cells; Animals; Benzamides; Binding Sites; Binding, Competitive; Butyrophenones; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Inositol Phosphates; Iodine Radioisotopes; Membranes; Mice; Piperidines; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin; Serotonin Agents; Serotonin Antagonists; Time Factors; Tritium

2001
Allosteric modulation of the human 5-HT(7A) receptor by lipidic amphipathic compounds.
    Molecular pharmacology, 2001, Volume: 60, Issue:6

    Topics: Allosteric Regulation; Cells, Cultured; Ergolines; HeLa Cells; Humans; Oleic Acid; Oleic Acids; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium

2001
5-HT receptor subtypes involved in the spinal antinociceptive effect of acetaminophen in rats.
    European journal of pharmacology, 2001, Nov-30, Volume: 432, Issue:1

    Topics: Acetaminophen; Analgesics; Animals; Ergolines; Granisetron; Injections, Spinal; Ketanserin; Male; Pain Threshold; Penbutolol; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Time Factors; Vocalization, Animal

2001
Up-regulation of 5-HT2B receptor density and receptor-mediated glycogenolysis in mouse astrocytes by long-term fluoxetine administration.
    Neurochemical research, 2002, Volume: 27, Issue:1-2

    Topics: Animals; Astrocytes; Carrier Proteins; Cells, Cultured; Drug Administration Schedule; Ergolines; Fluoxetine; Glycogen; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Protein Isoforms; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Up-Regulation

2002
Autoradiographic distribution of 5-HT7 receptors in the human brain using [3H]mesulergine: comparison to other mammalian species.
    British journal of pharmacology, 2004, Volume: 141, Issue:1

    Topics: 5-Methoxytryptamine; Amphetamines; Animals; Autoradiography; Brain; Cerebral Cortex; Corpus Striatum; Ergolines; Guinea Pigs; Humans; Male; Mammals; Radioligand Assay; Radionuclide Imaging; Rats; Rats, Wistar; Receptors, Serotonin; Tritium

2004
Reduced hypophagic effects of d-fenfluramine and the 5-HT2C receptor agonist mCPP in 5-HT1B receptor knockout mice.
    Psychopharmacology, 2004, Volume: 176, Issue:1

    Topics: Animals; Binding Sites; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Evaluation, Preclinical; Eating; Ergolines; Fenfluramine; Genotype; Injections, Intraperitoneal; Injections, Subcutaneous; Isomerism; Mianserin; Mice; Mice, Knockout; Piperazines; Piperidones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Satiation; Satiety Response; Serotonin 5-HT2 Receptor Agonists; Species Specificity; Spiperone; Spiro Compounds; Time Factors; Tritium; United Kingdom

2004
Differential inverse agonist efficacies of SB-258719, SB-258741 and SB-269970 at human recombinant serotonin 5-HT7 receptors.
    European journal of pharmacology, 2004, Jul-14, Volume: 495, Issue:2-3

    Topics: Animals; Binding, Competitive; CHO Cells; Clozapine; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Ergolines; Humans; Loxapine; Methiothepin; Phenols; Pimozide; Pindolol; Piperidines; Plasmids; Pyrrolidines; Radioligand Assay; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Tosyl Compounds; Transfection

2004
Regulation of serotonin 5-HT2C receptors by chronic ligand exposure.
    European journal of pharmacology, 2004, Sep-13, Volume: 498, Issue:1-3

    Topics: Algorithms; Analysis of Variance; Animals; Binding, Competitive; Cell Membrane; Chlorpromazine; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Ergolines; Humans; Indoles; Indophenol; Inositol Phosphates; Kinetics; Ligands; Lisuride; Mianserin; Radioligand Assay; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium; Tryptamines

2004
Comparison of G-protein selectivity of human 5-HT2C and 5-HT1A receptors.
    Annals of the New York Academy of Sciences, 2004, Volume: 1025

    Topics: Animals; Cell Line; Dose-Response Relationship, Drug; Ergolines; Heterotrimeric GTP-Binding Proteins; Insecta; Protein Binding; Rats; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2C; Receptors, G-Protein-Coupled; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists

2004
Serotonin 5-HT2C receptor-mediated phosphoinositide hydrolysis in rat choroid plexus after fluoxetine and citalopram treatments.
    Pharmacological research, 2005, Volume: 51, Issue:5

    Topics: Amphetamines; Animals; Choroid Plexus; Citalopram; Dose-Response Relationship, Drug; Ergolines; Fluoxetine; Hydrolysis; Inositol Phosphates; Male; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Second Messenger Systems; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2005
Decreased 5-HT2C receptor binding in the cerebral cortex and brain stem during pancreatic regeneration in rats.
    Molecular and cellular biochemistry, 2005, Volume: 272, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain Stem; Cerebral Cortex; Ergolines; Pancreas; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Regeneration; Serotonin; Serotonin Antagonists

2005
Effects of mu-CPP and mesulergine on dietary choices in deprived rats: possible mechanisms of their action.
    Progress in neuro-psychopharmacology & biological psychiatry, 2006, Volume: 30, Issue:1

    Topics: Animals; Apomorphine; Behavior, Animal; Choice Behavior; Diet; Dopamine Agonists; Dose-Response Relationship, Drug; Eating; Ergolines; Food Deprivation; Male; Piperazines; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists

2006
Hypothalamic 5-HT functional regulation through 5-HT1A and 5-HT2C receptors during pancreatic regeneration.
    Life sciences, 2006, Feb-28, Volume: 78, Issue:14

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Down-Regulation; Ergolines; Gene Expression Regulation, Developmental; Hypothalamus; Male; Pancreas; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2C; Regeneration; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2006
Development of homogeneous high-affinity agonist binding assays for 5-HT2 receptor subtypes.
    Assay and drug development technologies, 2005, Volume: 3, Issue:6

    Topics: Amphetamines; Binding, Competitive; Calcium Signaling; Cell Line; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Ergolines; Humans; Ketanserin; Lysergic Acid Diethylamide; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Transfection

2005
Combined treatment with citalopram and buspirone: effects on serotonin 5-HT2A and 5-HT2C receptors in the rat brain.
    Pharmacopsychiatry, 2006, Volume: 39, Issue:1

    Topics: Amphetamines; Animals; Anti-Anxiety Agents; Antidepressive Agents; Autoradiography; Brain Chemistry; Buspirone; Cerebral Cortex; Choroid Plexus; Citalopram; Ergolines; Hydrolysis; Image Processing, Computer-Assisted; Ketanserin; Male; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists

2006
Heterologous desensitization is evoked by both agonist and antagonist stimulation of the human 5-HT(7) serotonin receptor.
    European journal of pharmacology, 2006, Feb-17, Volume: 532, Issue:1-2

    Topics: Adenylyl Cyclases; Alternative Splicing; Binding, Competitive; Cell Line; Cell Membrane; Clozapine; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Ergolines; Gene Expression; Humans; Isoproterenol; Isoquinolines; Methiothepin; Multivariate Analysis; Phenols; Protein Isoforms; Protein Kinase Inhibitors; Radioligand Assay; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Time Factors; Tritium

2006
Fatty acids differentially affect serotonin receptor and transporter binding in the rat brain.
    Neuroscience, 2006, Volume: 139, Issue:4

    Topics: Analysis of Variance; Animals; Brain; Ergolines; Fatty Acids; Ketanserin; Male; Paroxetine; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins

2006
Aminomethyl tetrahydronaphthalene biphenyl carboxamide MCH-R1 antagonists--Increasing selectivity over hERG.
    Bioorganic & medicinal chemistry letters, 2007, Feb-01, Volume: 17, Issue:3

    Topics: Biphenyl Compounds; ERG1 Potassium Channel; Ergolines; Ether-A-Go-Go Potassium Channels; Humans; Indicators and Reagents; Mianserin; Naphthalenes; Potassium Channel Blockers; Receptor, Serotonin, 5-HT2C; Receptors, Somatostatin; Serotonin Antagonists; Structure-Activity Relationship

2007
Diabetes-induced changes in 5-hydroxytryptamine modulation of vagally-induced bradycardia in rat heart.
    Clinical and experimental pharmacology & physiology, 2007, Volume: 34, Issue:11

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Biphenyl Compounds; Blood Glucose; Bradycardia; Cholinergic Agents; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Electric Stimulation; Ergolines; Heart; Heart Rate; Injections, Intravenous; Male; Methiothepin; Oxadiazoles; Piperazines; Pyridines; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tryptamines; Vagus Nerve

2007
Upregulation of 5-HT2C receptors in hippocampus of pilocarpine-induced epileptic rats: antagonism by Bacopa monnieri.
    Epilepsy & behavior : E&B, 2009, Volume: 16, Issue:2

    Topics: Animals; Anticonvulsants; Bacopa; Carbamazepine; Disease Models, Animal; Epilepsy; Ergolines; Hippocampus; Inositol 1,4,5-Trisphosphate; Male; Pilocarpine; Plant Preparations; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Serotonin Antagonists; Statistics, Nonparametric; Swimming; Tritium; Up-Regulation

2009
Reversal of haloperidol-induced motor deficits by mianserin and mesulergine in rats.
    Pakistan journal of pharmaceutical sciences, 2011, Volume: 24, Issue:1

    Topics: Animals; Antipsychotic Agents; Catalepsy; Dopamine Agonists; Dyskinesia, Drug-Induced; Ergolines; Haloperidol; Male; Mianserin; Motor Activity; Parkinson Disease, Secondary; Psychomotor Performance; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Selective Serotonin Reuptake Inhibitors

2011
Differences between human wild-type and C23S variant 5-HT2C receptors in inverse agonist-induced resensitization.
    Pharmacological reports : PR, 2011, Volume: 63, Issue:1

    Topics: Adult; Aequorin; Base Sequence; Calcium; DNA, Complementary; Drug Inverse Agonism; Ergolines; HEK293 Cells; Humans; Indoles; Luminescent Measurements; Protein Binding; Pyridines; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin Antagonists; Time Factors

2011
Hippocampal serotonin depletion facilitates the enhancement of prepulse inhibition by risperidone: possible role of 5-HT(2C) receptors in the dorsal hippocampus.
    Neuropharmacology, 2011, Volume: 61, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Ergolines; Hippocampus; Male; Nerve Tissue Proteins; Neural Inhibition; Neurons; Organ Specificity; Random Allocation; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2C; Reflex, Startle; Risperidone; Schizophrenia; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2011
Influence of serotonergic 5-HT2C receptor antagonist mesulergine in the reversal of memory deficits induced by mCPP.
    Journal of the College of Physicians and Surgeons--Pakistan : JCPSP, 2012, Volume: 22, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Disease Models, Animal; Ergolines; Male; Maze Learning; Memory Disorders; Memory, Long-Term; Memory, Short-Term; Piperazines; Random Allocation; Rats; Rats, Wistar; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2012
Synthesis and SAR study of 4-arylpiperidines and 4-aryl-1,2,3,6-tetrahydropyridines as 5-HT₂C agonists.
    Bioorganic & medicinal chemistry letters, 2012, Apr-01, Volume: 22, Issue:7

    Topics: Animals; Appetite Depressants; Calcium; Ergolines; Humans; Kinetics; Piperidines; Protein Binding; Pyridines; Radioligand Assay; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Agonists; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship

2012
The N-terminal region of the human 5-HT₂C receptor has as a cleavable signal peptide.
    European journal of pharmacology, 2012, Jun-05, Volume: 684, Issue:1-3

    Topics: Amino Acid Sequence; Animals; Cell Membrane; Chlorocebus aethiops; COS Cells; Ergolines; Gene Expression Regulation; Humans; Molecular Sequence Data; Polymorphism, Single Nucleotide; Protein Sorting Signals; Protein Structure, Secondary; Proteolysis; Receptor, Serotonin, 5-HT2C; Transfection

2012
Molecular and behavioral pharmacology of two novel orally-active 5HT2 modulators: potential utility as antipsychotic medications.
    Neuropharmacology, 2013, Volume: 72

    Topics: Amphetamines; Animals; Antipsychotic Agents; Cell Line, Transformed; Dose-Response Relationship, Drug; Ergolines; Food Preferences; Glycolates; Head Movements; Humans; Ketanserin; Mice; Mice, Inbred C57BL; Motor Activity; Protein Binding; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium

2013
Multiple conformations of 5-HT2A and 5-HT 2C receptors in rat brain: an autoradiographic study with [125I](±)DOI.
    Experimental brain research, 2013, Volume: 230, Issue:4

    Topics: Aminopyridines; Animals; Autoradiography; Brain; Ergolines; Indoles; Ketanserin; Male; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Serotonin

2013
Neurotensin-like peptides as potential antipsychotics: modulation of the serotonin system.
    Bulletin of experimental biology and medicine, 2014, Volume: 157, Issue:6

    Topics: Animals; Antipsychotic Agents; Cell Membrane; Ergolines; Frontal Lobe; Ketanserin; Male; Mice; Neurotensin; Oligopeptides; Piperazines; Platelet Aggregation; Radioligand Assay; Rats; Serotonin; Serotonin Antagonists; Statistics, Nonparametric

2014
The atypical antipsychotics clozapine and olanzapine promote down-regulation and display functional selectivity at human 5-HT7 receptors.
    British journal of pharmacology, 2015, Volume: 172, Issue:15

    Topics: Antipsychotic Agents; Arrestins; Benzodiazepines; beta-Arrestins; Cells, Cultured; Chloroquine; Clozapine; Down-Regulation; Drug Inverse Agonism; Ergolines; HEK293 Cells; Humans; Ligands; Lysosomes; Olanzapine; Phenols; Radioligand Assay; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction; Sulfonamides

2015
Allosteric Inhibition of Serotonin 5-HT
    Molecular neurobiology, 2018, Volume: 55, Issue:4

    Topics: Allosteric Regulation; Cell Death; Cell Survival; Cyclic AMP; Ergolines; HEK293 Cells; Humans; Ions; Kinetics; Ligands; Phenols; Receptors, Serotonin; Sulfonamides; Zinc

2018