mesalamine and indomethacin

mesalamine has been researched along with indomethacin in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19908 (25.00)18.7374
1990's6 (18.75)18.2507
2000's9 (28.13)29.6817
2010's8 (25.00)24.3611
2020's1 (3.13)2.80

Authors

AuthorsStudies
Strassburg, CP; Tukey, RH1
Doman, TN; McGovern, SL; Seidler, J; Shoichet, BK1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Lombardo, F; Obach, RS; Waters, NJ1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Bansal, Y; Kaur, M; Silakari, O1
Farhat, M; George, RF; Girgis, AS; Katritzky, AR; Naumov, RN; Panda, SS1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Gaginella, TS; Gullikson, GW; Moummi, C1
Bostwick, JS; Decktor, DL; Fitzpatrick, LR; Pendleton, RG; Renzetti, M1
Guarner, F; Malagelada, JR; Rodriguez, R; Salas, A; Vilaseca, J1
Bertovich, MJ; MacDermott, RP; Nash, GS; Peters, M; Schloemann, SR; Stenson, WF1
Bazzocchi, G; Brignola, C; Campieri, M; Del Soldato, P; Gionchetti, P; Lanfranchi, GA; Tamba, M1
Gibson, PR; Jewell, DP1
Hoppe, U; Kleemeyer, K; Peskar, BA; Peskar, BM; Wittenberg, HR1
Bartholomew, TC; Jewell, DP; Rhodes, JM1
Chastenay, BF; Holdstock, G; Krawitt, EL1
Lobos, E; Stenson, WF1
Hawkey, CJ; Lo Casto, M1
Hata, Y; Nagata, T; Ota, S; Sugimoto, T; Terano, A; Uehara, Y1
Jewell, D; Lowes, J; Radwan, P; Skrzydło-Radomańska, B1
Rao, JP; Robert, FS1
Johnson, LK; Kim, YS; MacGregor, DJ; Sleisenger, MH1
Harada, K; Inoue, T; Nagakura, N; Oketani, K1
Valentine, JF1
Levine, RA; Nandi, J; Palma, DT; Saud, B; Zinkievich, JM1
Jagtap, AG; Niphadkar, PV; Phadke, AS1
Bures, J; Kholova, D; Kunes, M; Kvetina, J; Pavlik, M; Tlaskalova-Hogenova, H1
Almási, A; Fischer, E; Fischer, T; Simon, H1
Hong, EM; Jang, HJ; Jung, ES; Kae, SH; Lee, J; Lee, SP; Lim, HL1

Reviews

2 review(s) available for mesalamine and indomethacin

ArticleYear
Human UDP-glucuronosyltransferases: metabolism, expression, and disease.
    Annual review of pharmacology and toxicology, 2000, Volume: 40

    Topics: Autoimmunity; Chromosome Mapping; Glucuronides; Glucuronosyltransferase; Humans; Hyperbilirubinemia; Neoplasms; Steroids; Terminology as Topic

2000
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

30 other study(ies) available for mesalamine and indomethacin

ArticleYear
Identification and prediction of promiscuous aggregating inhibitors among known drugs.
    Journal of medicinal chemistry, 2003, Oct-09, Volume: 46, Issue:21

    Topics: Antifungal Agents; beta-Lactamase Inhibitors; Chemical Phenomena; Chemistry, Physical; Chymotrypsin; Enzyme Inhibitors; Kinetics; Light; Malate Dehydrogenase; Models, Molecular; Molecular Conformation; Scattering, Radiation; Structure-Activity Relationship

2003
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Benzimidazole--ibuprofen/mesalamine conjugates: potential candidates for multifactorial diseases.
    European journal of medicinal chemistry, 2015, Jan-07, Volume: 89

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Rheumatoid; Benzimidazoles; Edema; Ibuprofen; Immunomodulation; Mesalamine; Mice; Molecular Structure; Neoplasms; Rats; Rats, Wistar; Sheep

2015
Synthesis and QSAR study of novel anti-inflammatory active mesalazine-metronidazole conjugates.
    Bioorganic & medicinal chemistry letters, 2015, Jun-01, Volume: 25, Issue:11

    Topics: Animals; Anti-Inflammatory Agents; Indomethacin; Mesalamine; Metronidazole; Mice; Molecular Structure; Quantitative Structure-Activity Relationship; Stomach Ulcer

2015
Monochloramine induces contraction of guinea pig gallbladder via two different pathways.
    The American journal of physiology, 1991, Volume: 260, Issue:6 Pt 1

    Topics: Aminosalicylic Acids; Animals; Chloramines; Gallbladder; Guinea Pigs; Hydrogen Peroxide; Hypochlorous Acid; In Vitro Techniques; Indomethacin; Isometric Contraction; Male; Mesalamine; Models, Biological; Muscle, Smooth; Piroxicam; Tetrodotoxin; Verapamil; Virulence Factors, Bordetella

1991
Antiinflammatory effects of various drugs on acetic acid induced colitis in the rat.
    Agents and actions, 1990, Volume: 30, Issue:3-4

    Topics: Acetates; Acetic Acid; Aminosalicylic Acids; Animals; Anti-Inflammatory Agents; Colitis, Ulcerative; Dexamethasone; Disease Models, Animal; Gossypol; Hydrocortisone; Indomethacin; Intestinal Mucosa; Leukocyte Count; Male; Masoprocol; Mesalamine; Neutrophils; Peroxidase; Rats; Rats, Inbred Strains; Sulfasalazine

1990
Participation of thromboxane and other eicosanoid synthesis in the course of experimental inflammatory colitis.
    Gastroenterology, 1990, Volume: 98, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Aminosalicylic Acids; Animals; Colitis; Dinoprostone; Indomethacin; Leukotriene B4; Male; Mesalamine; Methacrylates; Pentanoic Acids; Prednisone; Pyridines; Rats; Rats, Inbred Strains; Thromboxane B2; Thromboxane-A Synthase; Trinitrobenzenesulfonic Acid

1990
Inhibition of antibody secretion by 5-aminosalicylic acid.
    Gastroenterology, 1989, Volume: 96, Issue:2 Pt 1

    Topics: Aminosalicylic Acids; Antibodies; Cell Division; Cell Survival; Humans; Immunoglobulin A; Indomethacin; Intestinal Mucosa; Intestines; Mesalamine; Monocytes; Pokeweed Mitogens; Sulfapyridine; Sulfasalazine

1989
A possible mechanism of action of sulfasalazine and 5-aminosalicylic acid in inflammatory bowel diseases: interaction with oxygen free radicals.
    Gastroenterology, 1985, Volume: 89, Issue:5

    Topics: Aminosalicylic Acids; Animals; Chemical Phenomena; Chemistry; Colitis; Free Radicals; Humans; Indomethacin; Mesalamine; Rats; Sulfasalazine; Superoxides

1985
Sulphasalazine and derivatives, natural killer activity and ulcerative colitis.
    Clinical science (London, England : 1979), 1985, Volume: 69, Issue:2

    Topics: Aminosalicylic Acids; Catechols; Cytotoxicity, Immunologic; Humans; In Vitro Techniques; Indomethacin; Killer Cells, Natural; Lipoxygenase Inhibitors; Masoprocol; Mesalamine; Monocytes; Sulfapyridine; Sulfasalazine

1985
Release of eicosanoids from human synovial tissue and the effect of anti-inflammatory drugs.
    Progress in clinical and biological research, 1987, Volume: 242

    Topics: Aminosalicylic Acids; Animals; Calcimycin; Chromones; Guinea Pigs; Humans; In Vitro Techniques; Indomethacin; Mesalamine; Muscle Contraction; Prostaglandins; SRS-A; Sulfanilamides; Sulfapyridine; Synovial Membrane

1987
Inhibition of leucocyte motility by drugs used in ulcerative colitis.
    Gut, 1981, Volume: 22, Issue:8

    Topics: Aminosalicylic Acids; Cell Movement; Chemotaxis, Leukocyte; Colitis, Ulcerative; Dose-Response Relationship, Drug; Humans; Indomethacin; Leukocytes; Mesalamine; Prednisolone; Sulfapyridine; Sulfasalazine

1981
Increased suppressor cell activity in inflammatory bowel disease.
    Gut, 1981, Volume: 22, Issue:12

    Topics: Aminosalicylic Acids; Colitis, Ulcerative; Crohn Disease; Humans; Hydrocortisone; In Vitro Techniques; Indomethacin; Lymphocyte Activation; Mesalamine; Mitogens; Sulfapyridine; Sulfasalazine; T-Lymphocytes, Regulatory

1981
Sulfasalazine inhibits the synthesis of chemotactic lipids by neutrophils.
    The Journal of clinical investigation, 1982, Volume: 69, Issue:2

    Topics: Aminosalicylic Acids; Arachidonic Acid; Arachidonic Acids; Calcimycin; Dose-Response Relationship, Drug; Humans; Hydroxyeicosatetraenoic Acids; Indomethacin; Leukotriene B4; Mesalamine; Neutrophils; Sulfasalazine

1982
Inhibition of prostaglandin synthetase in human rectal mucosa.
    Gut, 1983, Volume: 24, Issue:3

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents; Colitis, Ulcerative; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Flurbiprofen; Humans; Indomethacin; Intestinal Mucosa; Mesalamine; Prednisolone; Rectum; Sulfapyridine; Sulfasalazine

1983
Primary colonic epithelial cell culture of the rabbit producing prostaglandins.
    Prostaglandins, 1993, Volume: 45, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Aminosalicylic Acids; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cells, Cultured; Chromatography, High Pressure Liquid; Colon; Dinoprost; Dinoprostone; Epithelium; Female; Indomethacin; Male; Mesalamine; Prostaglandin D2; Prostaglandins; Rabbits; Thromboxane B2

1993
The effect of 5-aminosalicylic acid, hydrocortisone and indomethacin on gamma interferon induced expression of HLA-DR antigens on colonic epithelium.
    Annales Universitatis Mariae Curie-Sklodowska. Sectio D: Medicina, 1993, Volume: 48

    Topics: Aminosalicylic Acids; Anti-Inflammatory Agents, Non-Steroidal; Cells, Cultured; Colon; Epithelium; HLA-DR Antigens; Humans; Hydrocortisone; Indomethacin; Interferon-gamma; Mesalamine; Recombinant Proteins

1993
Mechanism of purgative effect of magnesium sulphate on mouse colon.
    Journal of diarrhoeal diseases research, 1997, Volume: 15, Issue:4

    Topics: Animals; Anthracenes; Cathartics; Chloride Channels; Colon; Diarrhea; Disease Models, Animal; Drug Interactions; Enzyme Inhibitors; Indomethacin; Intestinal Mucosa; Magnesium Sulfate; Male; Mesalamine; Methylene Blue; Mice; Mice, Inbred Strains; Premedication; Random Allocation; Reference Values; Sodium Chloride

1997
Chemoprevention of colon cancer carcinogenesis by balsalazide: inhibition of azoxymethane-induced aberrant crypt formation in the rat colon and intestinal tumor formation in the B6-Min/+ mouse.
    International journal of oncology, 2000, Volume: 17, Issue:1

    Topics: Aminosalicylic Acids; Animals; Anti-Ulcer Agents; Anticarcinogenic Agents; Azoxymethane; Cell Division; Colonic Neoplasms; Genes, APC; Humans; Indomethacin; Intestinal Mucosa; Intestinal Neoplasms; Mesalamine; Mice; Mice, Mutant Strains; Phenylhydrazines; Prodrugs; Rats; Rats, Inbred F344; Tumor Cells, Cultured

2000
In vitro effects of E3040, a dual inhibitor of 5-lipoxygenase and thromboxane A(2) synthetase, on eicosanoid production.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Animals; Arachidonate 5-Lipoxygenase; Benzothiazoles; Dinoprostone; Dose-Response Relationship, Drug; Eicosanoids; Humans; Hydroxyurea; Indomethacin; Leukocytes; Leukotriene B4; Lipoxygenase Inhibitors; Male; Mesalamine; Methacrylates; Neutrophils; Peritoneal Cavity; Prostaglandin-Endoperoxide Synthases; Pyridines; Rats; Rats, Inbred F344; Sheep; Sulfasalazine; Thiazoles; Thromboxane B2; Thromboxane-A Synthase

2001
Mesalamine induces manganese superoxide dismutase in rat intestinal epithelial cell lines and in vivo.
    American journal of physiology. Gastrointestinal and liver physiology, 2001, Volume: 281, Issue:4

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cell Line; Cycloheximide; Cyclooxygenase Inhibitors; Dactinomycin; Enzyme Induction; Free Radical Scavengers; Humans; Immunoblotting; Indoles; Indomethacin; Intestinal Mucosa; Lipopolysaccharides; Lipoxygenase Inhibitors; Mesalamine; Nucleic Acid Synthesis Inhibitors; Protein Synthesis Inhibitors; Rats; Superoxide Dismutase; Tumor Necrosis Factor-alpha

2001
5-aminosalicylic acid improves indomethacin-induced enteropathy by inhibiting iNOS transcription in rats.
    Digestive diseases and sciences, 2008, Volume: 53, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Biomarkers; Blotting, Western; Cyclooxygenase Inhibitors; Disease Models, Animal; Disease Progression; Electrophoresis, Polyacrylamide Gel; Enteritis; Ileitis; Indomethacin; Jejunal Diseases; Male; Mesalamine; Nitric Oxide Synthase Type II; Rats; Rats, Sprague-Dawley; Severity of Illness Index; Transcription, Genetic

2008
Protective effect of aqueous extract of Bombax malabaricum DC on experimental models of inflammatory bowel disease in rats and mice.
    Indian journal of experimental biology, 2011, Volume: 49, Issue:5

    Topics: Acetic Acid; Animals; Bombax; Colitis; Disease Models, Animal; Female; India; Indomethacin; Inflammatory Bowel Diseases; Iodoacetamide; Male; Medicine, Traditional; Mesalamine; Mice; Phytotherapy; Plant Extracts; Plants, Medicinal; Prednisolone; Rats; Rats, Sprague-Dawley

2011
Absorption kinetics of 5-aminosalicylic acid in rat: influence of indomethacin-induced gastrointestinal lesions and Escherichia Coli Nissle 1917 medication.
    Neuro endocrinology letters, 2011, Volume: 32 Suppl 1

    Topics: Absorption; Animals; Anti-Inflammatory Agents, Non-Steroidal; Escherichia coli; Gastrointestinal Diseases; Gastrointestinal Tract; Indomethacin; Kinetics; Male; Mesalamine; Osmolar Concentration; Probiotics; Rats; Rats, Wistar

2011
Effects of Mesalazine on Morphological and Functional Changes in the Indomethacin-Induced Inflammatory Bowel Disease (Rat Model of Crohn's Disease).
    Pathology oncology research : POR, 2017, Volume: 23, Issue:1

    Topics: Animals; Crohn Disease; Disease Models, Animal; Glucuronates; Indomethacin; Inflammation; Inflammatory Bowel Diseases; Intestine, Small; Liver; Male; Mesalamine; Nitrobenzenes; Nitrophenols; Rats; Rats, Wistar

2017
The Protective Effect of 5-Aminosalicylic Acid Against Non-Steroidal Anti-Inflammatory Drug-Induced Injury Through Free Radical Scavenging in Small Intestinal Epithelial Cells.
    Medicina (Kaunas, Lithuania), 2020, Oct-01, Volume: 56, Issue:10

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Epithelial Cells; Indomethacin; Mesalamine; Pharmaceutical Preparations

2020