meproadifen has been researched along with proadifen in 8 studies
| Studies (meproadifen) | Trials (meproadifen) | Recent Studies (post-2010) (meproadifen) | Studies (proadifen) | Trials (proadifen) | Recent Studies (post-2010) (proadifen) |
|---|---|---|---|---|---|
| 8 | 0 | 0 | 1,481 | 0 | 35 |
| Protein | Taxonomy | meproadifen (IC50) | proadifen (IC50) |
|---|---|---|---|
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | 1.5849 | |
| Aldehyde oxidase 1 | Rattus norvegicus (Norway rat) | 1.1 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 6 (75.00) | 18.7374 |
| 1990's | 1 (12.50) | 18.2507 |
| 2000's | 1 (12.50) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Boyd, ND; Cohen, JB; Krodel, EK; Neubig, RR | 1 |
| Bouet, F; Changeux, JP; Galzi, JL; Goeldner, M; Hirth, C; Ménez, A; Revah, F | 1 |
| Boyd, ND; Leeman, SE | 1 |
| Bloch, RJ | 1 |
| Albuquerque, EX; Aracava, Y | 1 |
| Albuquerque, EX; Cohen, JB; Maleque, MA; Souccar, C | 1 |
| Changeux, JP; Heidmann, T; Oswald, RE | 1 |
| Barrantes, GE; Ortells, MO | 1 |
8 other study(ies) available for meproadifen and proadifen
| Article | Year |
|---|---|
Acetylcholine and local anesthetic binding to Torpedo nicotinic postsynaptic membranes after removal of nonreceptor peptides.
Topics: Acetylcholine; Anesthetics, Local; Animals; Cell Membrane Permeability; Electric Organ; Fishes; Hydrogen-Ion Concentration; Ion Channels; Isoquinolines; Kinetics; Membrane Proteins; Molecular Weight; Proadifen; Receptors, Cholinergic; Receptors, Nicotinic; Sodium; Synaptic Membranes | 1979 |
Allosteric transitions of the acetylcholine receptor probed at the amino acid level with a photolabile cholinergic ligand.
Topics: Affinity Labels; Allosteric Regulation; Amino Acid Sequence; Animals; Diazonium Compounds; Kinetics; Macromolecular Substances; Models, Structural; Molecular Sequence Data; Peptide Fragments; Proadifen; Protein Conformation; Receptors, Cholinergic; Sequence Homology, Nucleic Acid; Torpedo; Tubocurarine | 1991 |
Multiple actions of substance P that regulate the functional properties of acetylcholine receptors of clonal rat PC12 cells.
Topics: Animals; Carbachol; Cell Line; Clone Cells; Ion Channels; Kinetics; Models, Biological; Proadifen; Receptors, Cholinergic; Sodium; Substance P | 1987 |
Loss of acetylcholine receptor clusters induced by treatment of cultured rat myotubes with carbachol.
Topics: Animals; Calcium; Carbachol; Chlorides; Dose-Response Relationship, Drug; Fluphenazine; Lidocaine; Muscles; Potassium; Proadifen; Protease Inhibitors; Protein Conformation; Rats; Receptors, Cholinergic; Sodium | 1986 |
Meproadifen enhances activation and desensitization of the acetylcholine receptor-ionic channel complex (AChR): single channel studies.
Topics: Acetylcholine; Animals; Animals, Newborn; Electric Conductivity; Ion Channels; Muscles; Proadifen; Rats; Receptors, Cholinergic | 1984 |
Meproadifen reaction with the ionic channel of the acetylcholine receptor: potentiation of agonist-induced desensitization at the frog neuromuscular junction.
Topics: Animals; Electric Stimulation; Electrophysiology; In Vitro Techniques; Ion Channels; Membrane Potentials; Motor Endplate; Muscles; Neuromuscular Junction; Proadifen; Rana pipiens; Receptors, Cholinergic; Time Factors | 1982 |
Multiple sites of action for noncompetitive blockers on acetylcholine receptor rich membrane fragments from torpedo marmorata.
Topics: Alkanes; Allosteric Regulation; Amphibian Venoms; Animals; Binding Sites; Chlorpromazine; Electric Organ; Isoquinolines; Membrane Lipids; Neuromuscular Junction; Parasympatholytics; Phencyclidine; Polyethylene Glycols; Proadifen; Receptors, Cholinergic; Torpedo | 1983 |
Understanding channel blocking in the nicotinic acetylcholine receptor.
Topics: Acetylcholine; Animals; Binding Sites; Chlorisondamine; Ethidium; Hexamethonium; Lidocaine; Mice; Nicotinic Antagonists; Onium Compounds; Pempidine; Proadifen; Quinacrine; Receptors, Nicotinic; Trityl Compounds | 2001 |