melatonin and ketanserin

melatonin has been researched along with ketanserin in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (36.36)18.2507
2000's5 (22.73)29.6817
2010's9 (40.91)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X1
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG1
Colau, D; Dolusić, E; Frédérick, R; Larrieu, P; Masereel, B; Moineaux, L; Pilotte, L; Pochet, L; Stroobant, V; Van den Eynde, B; Wouters, J1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E1
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E1
Barrios, VE; Duckles, SP; Krause, DN1
Eison, AS; Mullins, UL1
Münker, M; Olcese, J1
Sandyk, R1
Duckles, SP; Geary, GG; Krause, DN1
Miguez, JM; Pevet, P; Simonneaux, V1
Kennaway, DJ; Moyer, RW1
Buyse, J; Decuypere, E; Herichová, I; Lamosová, D; Zeman, M1
Andorn, AC; Pappolla, MA1
LeMaster, MP; Lutterschmidt, DI; Mason, RT1
Lutterschmidt, DI; Mason, RT1
Jaworek, J; Konturek, SJ; Leja-Szpak, A; Nawrot-Porąbka, K; Reiter, RJ; Szklarczyk, J1
Bonior, J; Goralska, M; Jastrzebska, M; Jaworek, J; Leja-Szpak, A; Link-Lenczowski, P; Nawrot-Porabka, K; Pierzchalski, P1

Other Studies

22 other study(ies) available for melatonin and ketanserin

ArticleYear
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
    Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship

2008
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
    Journal of medicinal chemistry, 2008, Nov-27, Volume: 51, Issue:22

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship

2008
Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators.
    Journal of medicinal chemistry, 2011, Aug-11, Volume: 54, Issue:15

    Topics: Animals; Antineoplastic Agents; Biological Availability; Cell Line; Drug Design; Enzyme Inhibitors; Humans; Immunologic Factors; Indoles; Kinetics; Mice; Neoplasms; Structure-Activity Relationship; Tryptophan Oxygenase

2011
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2013
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
    Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

    Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
    Bioorganic & medicinal chemistry, 2016, Apr-15, Volume: 24, Issue:8

    Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine

2016
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
    Bioorganic & medicinal chemistry, 2017, 01-15, Volume: 25, Issue:2

    Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship

2017
Melatonin receptors mediate potentiation of contractile responses to adrenergic nerve stimulation in rat caudal artery.
    European journal of pharmacology, 1995, Apr-04, Volume: 276, Issue:3

    Topics: Animals; Arteries; Electric Stimulation; In Vitro Techniques; Isometric Contraction; Ketanserin; Male; Melatonin; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Melatonin; Regional Blood Flow; Serotonin; Sympathetic Nervous System; Tail; Tryptamines; Vasoconstriction

1995
Pharmacologic characterization of melatonin-mediated phosphoinositide hydrolysis in pigeon brain.
    Journal of pineal research, 1994, Volume: 17, Issue:1

    Topics: Animals; Brain; Columbidae; Hydrolysis; Ketanserin; Melatonin; Phosphatidylinositols; Second Messenger Systems; Signal Transduction; Tryptamines

1994
Extracellular serotonin promotes melatonin release from cultured rat pinealocytes: evidence for an S2-type receptor-mediated autocrine feedback.
    Brain research, 1994, Apr-18, Volume: 643, Issue:1-2

    Topics: Analysis of Variance; Animals; Bucladesine; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Feedback; Female; Isoproterenol; Ketanserin; Kinetics; Melatonin; Norepinephrine; Pineal Gland; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Time Factors

1994
Bidirectional effect of electromagnetic fields on ketanserin-induced yawning in patients with multiple sclerosis: the role of melatonin.
    The International journal of neuroscience, 1996, Volume: 85, Issue:1-2

    Topics: Adult; Electromagnetic Fields; Female; Humans; Ketanserin; Male; Melatonin; Middle Aged; Multiple Sclerosis; Ritanserin; Serotonin Antagonists; Yawning

1996
Melatonin directly constricts rat cerebral arteries through modulation of potassium channels.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 2

    Topics: Animals; Apamin; Benzimidazoles; Cerebral Arteries; Charybdotoxin; GTP-Binding Proteins; Ketanserin; Male; Melatonin; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Pertussis Toxin; Potassium; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Tetraethylammonium; Tetraethylammonium Compounds; Tryptamines; Vasoconstriction; Virulence Factors, Bordetella

1997
The role of the intracellular and extracellular serotonin in the regulation of melatonin production in rat pinealocytes.
    Journal of pineal research, 1997, Volume: 23, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Arylamine N-Acetyltransferase; Dose-Response Relationship, Drug; Fenclonine; Isoproterenol; Ketanserin; Male; Melatonin; Pineal Gland; Rats; Rats, Wistar; Serotonin; Serotonin Agents; Serotonin Antagonists

1997
Serotonin 5-HT2c agonists mimic the effect of light pulses on circadian rhythms.
    Brain research, 1998, Sep-28, Volume: 806, Issue:2

    Topics: Amphetamines; Animals; Body Temperature; Circadian Rhythm; Ketanserin; Light; Male; Melatonin; Periodicity; Photic Stimulation; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Suprachiasmatic Nucleus

1998
Role of melatonin in the control of growth and growth hormone secretion in poultry.
    Domestic animal endocrinology, 1999, Volume: 17, Issue:2-3

    Topics: Animals; Coturnix; Growth Hormone; Ketanserin; Male; Melatonin; Photoperiod; Quipazine; Radioimmunoassay; Random Allocation; Serotonin Antagonists; Serotonin Receptor Agonists; Thyrotropin-Releasing Hormone

1999
Catecholamines inhibit lipid peroxidation in young, aged, and Alzheimer's disease brain.
    Free radical biology & medicine, 2001, Aug-01, Volume: 31, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adult; Aged; Aging; Alzheimer Disease; Autopsy; Brain; Catecholamines; Caudate Nucleus; Cerebellum; Dopamine; Haloperidol; Humans; Ketanserin; Lipid Peroxidation; Melatonin; Middle Aged; Postmortem Changes; Prefrontal Cortex; Putamen; Serotonin; Thiobarbituric Acid Reactive Substances

2001
Effects of melatonin on the behavioral and hormonal responses of red-sided garter snakes (Thamnophis sirtalis parietalis) to exogenous corticosterone.
    Hormones and behavior, 2004, Volume: 46, Issue:5

    Topics: Analysis of Variance; Animals; Colubridae; Corticosterone; Courtship; Dihydrotestosterone; Ketanserin; Melatonin; Receptors, Serotonin; Serotonin Antagonists; Sexual Behavior, Animal; Testosterone

2004
A serotonin receptor antagonist, but not melatonin, modulates hormonal responses to capture stress in two populations of garter snakes (Thamnophis sirtalis parietalis and Thamnophis sirtalis concinnus).
    General and comparative endocrinology, 2005, May-01, Volume: 141, Issue:3

    Topics: 5-Hydroxytryptophan; Adjuvants, Immunologic; Androgens; Animals; Colubridae; Corticosterone; Endocrine System; Ketanserin; Melatonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Stress, Physiological

2005
Luminal melatonin stimulates pancreatic enzyme secretion via activation of serotonin-dependent nerves.
    Pharmacological reports : PR, 2013, Volume: 65, Issue:2

    Topics: Amylases; Animals; Dose-Response Relationship, Drug; Duodenum; Ketanserin; Melatonin; Pancreas; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Serotonin; Serotonin Antagonists; Time Factors; Tropanes; Tryptophan; Vagus Nerve

2013
Kynuramines induce overexpression of heat shock proteins in pancreatic cancer cells via 5-hydroxytryptamine and MT1/MT2 receptors.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2015, Volume: 66, Issue:5

    Topics: Cell Line, Tumor; Heat-Shock Proteins; Humans; Ketanserin; Kynuramine; Melatonin; Pancreatic Neoplasms; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Serotonin; Tropanes; Tryptamines; Tryptophan

2015