melatonin and guanosine 5'-o-(3-thiotriphosphate)

melatonin has been researched along with guanosine 5'-o-(3-thiotriphosphate) in 51 studies

Research

Studies (51)

Timeframe	Studies, this research(%)	All Research%
pre-1990	1 (1.96)	18.7374
1990's	31 (60.78)	18.2507
2000's	17 (33.33)	29.6817
2010's	2 (3.92)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Capsoni, S; Cozzi, B; Fauteck, J; Fraschini, F; Fumagalli, P; Lucini, V; Stankov, B	1
Niles, LP; Ying, SW	1
Laitinen, JT; Saavedra, JM	1
Flügge, G; Laitinen, JT; Saavedra, JM	1
Conron, RW; Reppert, SM; Rivkees, SA	1
Davidson, G; Howell, HE; Lawson, W; Morgan, PJ	1
Bubis, M; Zisapel, N	1
Brown, GM; Pang, SF; Poon, AM; Song, Y; Tam, PC	1
Dubocovich, ML; Popova, JS	1
Barrett, P; MacLean, A; Morgan, PJ	1
Bromage, N; Davies, B; Hannah, LT; Randall, CF; Williams, LM	1
Bergmann, M; Fauteck, JD; Fraschini, F; Lerchl, A; Møller, M; Stankov, B; Wittkowski, W	1
Pang, SF; Poon, AM	2
Helliwell, RJ; Williams, LM	1
Biella, G; Capsoni, S; Cozzi, B; Fauteck, J; Fraschini, F; Gatti, S; Gridelli, B; Lucini, V; Stankov, B	1
Aste, N; Capsoni, S; Cozzi, B; Fraschini, F; Lucini, V; Panzica, GC; Stankov, B; Viglietti-Panzica, C	1
Brown, GM; Pang, CS; Pang, SF; Song, Y; Tang, PL	1
Barrett, P; Davidson, G; Hannah, L; Lawson, W; MacLean, A; Morgan, PJ; Williams, LM	1
Brown, GM; Liao, M; Pang, SF; Wan, Q	1
Eison, AS; Fernandes, PB; Mullins, UL	1
Balsamini, C; Di Giacomo, B; Diamantini, G; Fraschini, F; Lucini, V; Mor, M; Nonno, R; Pannacci, M; Plazzi, PV; Rivara, S; Spadoni, G; Stankov, BM; Tarzia, G	1
Di Giacomo, B; Diamantini, G; Esposti, D; Fraschini, F; Lucini, V; Nonno, R; Pannacci, M; Spadoni, G; Stankov, BM; Tarzia, G	1
Barrett, P; Clarke, IJ; Lincoln, GA; Mercer, JG; Morgan, PJ; Williams, LM	1
Aida, K; Hara, M; Hirata, K; Iigo, M; Ohtani-Kaneko, R; Sánchez-Vázquez, FJ; Shinohara, H; Tabata, M	1
Brown, GM; Delagrange, P; Guardiola-Lemaitre, B; Ng, KW; Pang, CS; Pang, SF; Song, Y; Tang, PL	1
Angeloni, D; Fraschini, F; Lucini, V; Mazzucchelli, C; Nonno, R; Pannacci, M; Stankov, BM	1
Falcón, J; Gaildrat, P; Ron, B	1
Balsamini, C; Bedini, A; Di Giacomo, B; Diamantini, G; Fraschini, F; Lucini, V; Mor, M; Nonno, R; Pannacci, M; Plazzi, PV; Rivara, S; Spadoni, G; Stankov, BM; Tarzia, G; Tontini, A	1
Beresford, IJ; Giles, H; Hall, DA; Harvey, FJ	1
Bassett, JM; Hannah, LT; Williams, LM	1
Angeloni, D; Fraschini, F; Lucini, V; Nonno, R; Pannacci, M; Stankov, BM	1
Beckmann, A; Fauteck, JD; Musshoff, U; Peschke, D; Peschke, E; Schmidt, F	1
Balsamini, C; Croce, A; Esposti, D; Fraschini, F; Lucini, V; Nonno, R; Pannacci, M; Spadoni, G; Stankov, BM; Tarzia, G	1
Bedini, A; Di Giacomo, B; Diamantini, G; Fraschini, F; Lucini, V; Mor, M; Nonno, R; Pannacci, M; Plazzi, PV; Rivara, S; Spadoni, G; Stankov, BM; Tarzia, G	1
Dubocovich, ML; Erşahin, C; Masana, MI	1
Kravtsov, G; Pang, CS; Pang, SF; Shiu, SY; Yau, MY	1
Kravtsov, GM; Pang, SF; Poon, AM	1
Audinot, V; Bennejean, C; Bochu, C; Boutin, JA; Delagrange, P; Durieux-Poissonnier, S; Guelzim, H; Lesieur, D; Lipka-Belloli, E; Renard, P; Yous, S	1
Amano, M; Iigo, M; Ikuta, K; Kitamura, S; Yamamori, K	1
Alonso-Bedate, M; Alonso-Gómez, AL; Delgado, MJ; Guijarro, A; Isorna, E	1
Bayarri, MJ; Garcia-Allegue, R; Iigo, M; Madrid, JA; Muñoz-Cueto, JA; Sánchez-Vázquez, FJ; Tabata, M	1
Alonso-Bedate, M; Alonso-Gómez, AL; Delgado, MJ; Guijarro, A; Isorna, E; López-Patiño, MA	1
Dubocovich, ML; Masana, MI; Soares, JM	1
Delgado, MJ; Guijarro, AI; Isorna, E; López-Patiño, MA; Luis Alonso-Gómez, A; Pedro, Nd	1
Bogdanovic, N; Karelson, E; Land, T; Reis, K; Zharkovsky, A	1
Bedini, A; Di Giacomo, B; Fraschini, F; Lucini, V; Pannacci, M; Spadoni, G; Tarzia, G	1
Alonso-Gómez, AL; Delgado, MJ; Guijarro, A; Isorna, E; López Patiño, MA	1
Bennett, JM; Bondi, CD; Brydon, L; Ignatius, PF; Jockers, R; McKeon, RM; Melan, MA; Witt-Enderby, PA	1
Bettler, B; Clement, N; Daulat, AM; Delagrange, P; Galès, C; Guillaume, JL; Ivankova-Susankova, K; Jockers, R; Kamal, M; Maurice, P; Turecek, R; Zamponi, F	1
Boutin, JA; Caignard, S; Delagrange, P; Devavry, S; Legros, C; Nosjean, O; Ouvry, C; Tessier, C	1

Other Studies

51 other study(ies) available for melatonin and guanosine 5'-o-(3-thiotriphosphate)

Article	Year
Localization and characterization of melatonin binding sites in the brain of the rabbit (Oryctolagus cuniculus) by autoradiography and in vitro ligand-receptor binding. Neuroscience letters, 1991, Nov-25, Volume: 133, Issue:1 Topics: Animals; Autoradiography; Brain Chemistry; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Hypothalamus; In Vitro Techniques; Iodine Radioisotopes; Ligands; Male; Melatonin; Rabbits; Receptors, Melatonin; Receptors, Neurotransmitter	1991
3-[(3-cholamidopropyl)dimethylammonio]-1-propane sulfonate-solubilized binding sites for 2-[125I]iodomelatonin in chick brain retain sensitivity to guanine nucleotides. Journal of neurochemistry, 1991, Volume: 56, Issue:2 Topics: Animals; Binding Sites; Brain; Cell Membrane; Chickens; Cholic Acids; Cytosol; Detergents; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Iodine Radioisotopes; Kinetics; Male; Melatonin; Receptors, Melatonin; Receptors, Neurotransmitter; Solubility	1991
Characterization of melatonin receptors in the rat suprachiasmatic nuclei: modulation of affinity with cations and guanine nucleotides. Endocrinology, 1990, Volume: 126, Issue:4 Topics: Animals; Autoradiography; Binding Sites; Binding, Competitive; Cations; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Male; Melatonin; Rats; Rats, Inbred Strains; Receptors, Melatonin; Receptors, Neurotransmitter; Suprachiasmatic Nucleus; Thionucleotides	1990
Characterization of melatonin receptors in the rat area postrema: modulation of affinity with cations and guanine nucleotides. Neuroendocrinology, 1990, Volume: 51, Issue:6 Topics: Animals; Autoradiography; Binding Sites; Binding, Competitive; Calcium Chloride; Cations, Divalent; Cerebral Ventricles; GTP-Binding Proteins; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Magnesium Chloride; Male; Melatonin; Rats; Rats, Inbred Strains; Receptors, Melatonin; Receptors, Neurotransmitter; Serotonin; Thionucleotides	1990
Solubilization and purification of melatonin receptors from lizard brain. Endocrinology, 1990, Volume: 127, Issue:3 Topics: Animals; Brain Chemistry; Cell Membrane; Chromatography, Affinity; Chromatography, Gel; Digitonin; Freezing; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Hot Temperature; Iodine Radioisotopes; Kinetics; Lizards; Melatonin; Molecular Structure; Receptors, Melatonin; Receptors, Neurotransmitter; Solubility; Thionucleotides	1990
Guanine nucleotides regulate the affinity of melatonin receptors on the ovine pars tuberalis. Neuroendocrinology, 1989, Volume: 50, Issue:3 Topics: Animals; Cell Membrane; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Melatonin; Pituitary Gland, Anterior; Receptors, Melatonin; Receptors, Neurotransmitter; Sheep; Thionucleotides	1989
Facilitation and inhibition of G-protein regulated protein secretion by melatonin. Neurochemistry international, 1995, Volume: 27, Issue:2 Topics: Aluminum Compounds; Animals; Cholera Toxin; Fluorides; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Melatonin; Mice; Neoplasm Proteins; Tumor Cells, Cultured	1995
2-[125I]iodomelatonin-binding sites in the human kidney and the effect of guanosine 5'-O-(3-thiotriphosphate). The Journal of clinical endocrinology and metabolism, 1995, Volume: 80, Issue:5 Topics: Adult; Aged; Autoradiography; Binding Sites; Carcinoma, Renal Cell; Carcinoma, Transitional Cell; Female; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Iodine Radioisotopes; Kidney Cortex; Kidney Neoplasms; Male; Melatonin; Middle Aged; Tissue Distribution	1995
Melatonin receptor-mediated stimulation of phosphoinositide breakdown in chick brain slices. Journal of neurochemistry, 1995, Volume: 64, Issue:1 Topics: Animals; Brain; Calcium; Chickens; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Melatonin; Phosphatidylinositols; Receptors, Cell Surface; Receptors, Melatonin; Receptors, Serotonin; Time Factors; Type C Phospholipases	1995
Evidence for multiple forms of melatonin receptor-G-protein complexes by solubilization and gel electrophoresis. Journal of neuroendocrinology, 1994, Volume: 6, Issue:5 Topics: Animals; Brain Chemistry; Chickens; Digitonin; Electrophoresis, Polyacrylamide Gel; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Iodine Radioisotopes; Lizards; Macromolecular Substances; Melatonin; Molecular Weight; Receptors, Cell Surface; Receptors, Melatonin; Sheep; Signal Transduction; Solubility	1994
Central melatonin binding sites in rainbow trout (Onchorhynchus mykiss). General and comparative endocrinology, 1994, Volume: 96, Issue:1 Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Kinetics; Melatonin; Oncorhynchus mykiss; Receptors, Cell Surface; Receptors, Melatonin; Serotonin; Temperature	1994
The adult human cerebellum is a target of the neuroendocrine system involved in the circadian timing. Neuroscience letters, 1994, Sep-26, Volume: 179, Issue:1-2 Topics: Adult; Aged; Aged, 80 and over; Autoradiography; Binding, Competitive; Cerebellar Cortex; Circadian Rhythm; Female; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Melatonin; Middle Aged; Neurosecretory Systems	1994
Differential effects of guanosine 5'-O-(3-thiotriphosphate) (GTP gamma S) on the 2-[125I]iodomelatonin binding sites in the chicken bursa of Fabricius and spleen. Neuroscience letters, 1994, May-23, Volume: 173, Issue:1-2 Topics: Animals; Bursa of Fabricius; Chickens; Down-Regulation; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Melatonin; Membranes; Receptors, Cell Surface; Receptors, Melatonin; Spleen	1994
The development of melatonin-binding sites in the ovine fetus. The Journal of endocrinology, 1994, Volume: 142, Issue:3 Topics: Animals; Autoradiography; Binding, Competitive; Fetus; Guanosine 5'-O-(3-Thiotriphosphate); Melatonin; Protein Binding; Receptors, Cell Surface; Receptors, Melatonin; Sheep; Tissue Distribution	1994
Modulation of 2-[125I]iodomelatonin binding in the guinea pig spleen by guanine nucleotides and cations. Neuroendocrinology, 1994, Volume: 59, Issue:2 Topics: Animals; Binding, Competitive; Calcium; Cations; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Guinea Pigs; Iodine Radioisotopes; Melatonin; Sodium; Spleen	1994
Autoradiographic localization of putative melatonin receptors in the brains of two Old World primates: Cercopithecus aethiops and Papio ursinus. Neuroscience, 1993, Volume: 52, Issue:2 Topics: Animals; Autoradiography; Binding, Competitive; Brain; Brain Chemistry; Chlorocebus aethiops; Female; Guanosine 5'-O-(3-Thiotriphosphate); Male; Melatonin; Papio; Pituitary Gland; Receptors, Melatonin; Receptors, Neurotransmitter	1993
Distribution and characterization of melatonin receptors in the brain of the Japanese quail, Coturnix japonica. Neuroscience letters, 1993, Feb-19, Volume: 150, Issue:2 Topics: Animals; Autoradiography; Brain; Coturnix; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Ligands; Male; Melatonin; Receptors, Melatonin; Receptors, Neurotransmitter; Signal Transduction	1993
2-[125I]Iodomelatonin binding sites in the quail heart: characteristics, distribution and modulation by guanine nucleotides and cations. Life sciences, 1996, Volume: 58, Issue:13 Topics: Animals; Autoradiography; Binding Sites; Binding, Competitive; Calcium Chloride; Cell Membrane; Choline; Coturnix; Female; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Kinetics; Magnesium Chloride; Male; Melatonin; Myocardium; Radioligand Assay; Receptors, Cell Surface; Receptors, Melatonin; Sensitivity and Specificity; Structure-Activity Relationship	1996
Differential regulation of melatonin receptors in sheep, chicken and lizard brains by cholera and pertussis toxins and guanine nucleotides. Neurochemistry international, 1996, Volume: 28, Issue:3 Topics: Animals; Autoradiography; Binding, Competitive; Brain Chemistry; Chickens; Cholera Toxin; GTP-Binding Proteins; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Kinetics; Lizards; Melatonin; Radioligand Assay; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Sheep; Species Specificity; Virulence Factors, Bordetella	1996
Localization and characterization of melatonin receptors in the rabbit spinal cord. Neuroscience letters, 1996, Feb-02, Volume: 204, Issue:1-2 Topics: Animals; Autoradiography; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Male; Melatonin; Rabbits; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Spinal Cord	1996
Melatonin agonists induce phosphoinositide hydrolysis in Xenopus laevis melanophores. Cellular signalling, 1997, Volume: 9, Issue:2 Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Cells, Cultured; Cricetinae; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Hydrolysis; Melanophores; Melatonin; Pertussis Toxin; Phosphatidylinositols; Prazosin; Signal Transduction; Virulence Factors, Bordetella; Xenopus laevis	1997
Conformationally restrained melatonin analogues: synthesis, binding affinity for the melatonin receptor, evaluation of the biological activity, and molecular modeling study. Journal of medicinal chemistry, 1997, Jun-20, Volume: 40, Issue:13 Topics: Animals; Binding, Competitive; Chickens; Colforsin; Cyclic AMP; Drug Design; Guanosine 5'-O-(3-Thiotriphosphate); Melatonin; Models, Molecular; Quail; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Superior Colliculi	1997
1-(2-Alkanamidoethyl)-6-methoxyindole derivatives: a new class of potent indole melatonin analogues. Journal of medicinal chemistry, 1997, Jun-20, Volume: 40, Issue:13 Topics: Animals; Binding Sites; Binding, Competitive; Chickens; Colforsin; Cyclic AMP; Drug Design; Guanosine 5'-O-(3-Thiotriphosphate); Indoles; Melatonin; Models, Chemical; Quail; Superior Colliculi	1997
Melatonin receptors in the brain and pituitary gland of hypothalamo-pituitary disconnected Soay rams. Journal of neuroendocrinology, 1997, Volume: 9, Issue:8 Topics: Animals; Autoradiography; Brain; Goats; Guanosine 5'-O-(3-Thiotriphosphate); Hypothalamus; In Situ Hybridization; Iodine Radioisotopes; Male; Melatonin; Neurons; Photoperiod; Pituitary Gland; Pituitary Gland, Anterior; Prolactin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Seasons	1997
Characterization, guanosine 5'-O-(3-thiotriphosphate) modulation, daily variation, and localization of melatonin-binding sites in the catfish (Silurus asotus) brain. General and comparative endocrinology, 1997, Volume: 108, Issue:1 Topics: Animals; Binding Sites; Brain; Brain Chemistry; Catfishes; Circadian Rhythm; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Kinetics; Lighting; Melatonin; Membranes; Protein Binding	1997
Differential inhibitory effects of melatonin analogs and three naphthalenic ligands on 2-[125I]iodomelatonin binding to chicken tissues. Journal of pineal research, 1997, Volume: 23, Issue:3 Topics: Aging; Animals; Binding, Competitive; Brain; Chickens; Female; Guanosine 5'-O-(3-Thiotriphosphate); Kidney; Ligands; Lung; Male; Melatonin; Membranes; Naphthalenes; Radioligand Assay; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Spleen; Tryptamines	1997
Pharmacological characterization of the human melatonin Mel1a receptor following stable transfection into NIH3T3 cells. British journal of pharmacology, 1998, Volume: 124, Issue:3 Topics: 3T3 Cells; Animals; Binding, Competitive; Cell Membrane; Cloning, Molecular; DNA; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Ligands; Melatonin; Mice; Pertussis Toxin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Thermodynamics; Transfection; Virulence Factors, Bordetella	1998
Daily and circadian variations in 2-[125I]-iodomelatonin binding sites in the pike brain (Esox lucius). Journal of neuroendocrinology, 1998, Volume: 10, Issue:7 Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Circadian Rhythm; Esocidae; Female; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Kinetics; Male; Melatonin; Pineal Gland	1998
2-[N-Acylamino(C1-C3)alkyl]indoles as MT1 melatonin receptor partial agonists, antagonists, and putative inverse agonists. Journal of medicinal chemistry, 1998, Sep-10, Volume: 41, Issue:19 Topics: 3T3 Cells; Animals; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indoles; Ligands; Melatonin; Mice; Rats; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Sodium Chloride; Structure-Activity Relationship	1998
Pharmacological characterisation of melatonin mt1 receptor-mediated stimulation of [35S]-GTPgammaS binding. Biochemical pharmacology, 1998, Nov-01, Volume: 56, Issue:9 Topics: Animals; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Humans; Melatonin; Pertussis Toxin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Virulence Factors, Bordetella	1998
Melatonin receptors in neonatal pig brain and pituitary gland. Journal of pineal research, 1999, Volume: 26, Issue:1 Topics: Animals; Animals, Newborn; Binding, Competitive; Brain; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Melatonin; Pituitary Gland; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Swine; Tissue Distribution	1999
Ligand efficacy and potency at recombinant human MT2 melatonin receptors: evidence for agonist activity of some mt1-antagonists. British journal of pharmacology, 1999, Volume: 127, Issue:5 Topics: 3T3 Cells; Animals; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Melatonin; Mice; Pertussis Toxin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Recombinant Proteins; Tryptamines; Virulence Factors, Bordetella	1999
Evidence for a melatonin receptor within pancreatic islets of neonate rats: functional, autoradiographic, and molecular investigations. Journal of pineal research, 2000, Volume: 28, Issue:3 Topics: Animals; Animals, Newborn; Autoradiography; Colforsin; DNA Primers; Dose-Response Relationship, Drug; Female; Gene Expression; Guanosine 5'-O-(3-Thiotriphosphate); Insulin; Insulin Secretion; Islets of Langerhans; Male; Melatonin; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tryptamines	2000
A new melatonin receptor ligand with mt1-agonist and MT2-antagonist properties. Journal of pineal research, 2000, Volume: 29, Issue:4 Topics: 3T3 Cells; Animals; Cell Membrane; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Indoles; Ligands; Melatonin; Mice; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin	2000
Synthesis, pharmacological characterization and QSAR studies on 2-substituted indole melatonin receptor ligands. Bioorganic & medicinal chemistry, 2001, Volume: 9, Issue:4 Topics: 3T3 Cells; Algorithms; Animals; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indoles; Least-Squares Analysis; Ligands; Melatonin; Mice; Models, Molecular; Protein Conformation; Quantitative Structure-Activity Relationship; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Regression Analysis	2001
Constitutively active melatonin MT(1) receptors in male rat caudal arteries. European journal of pharmacology, 2002, Mar-29, Volume: 439, Issue:1-3 Topics: Animals; Arteries; Autoradiography; Binding, Competitive; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Male; Melatonin; Rats; Rats, Inbred F344; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Sulfur Radioisotopes; Tetrahydronaphthalenes	2002
2[125I]Iodomelatonin binding sites in guinea pig platelets. Journal of pineal research, 2002, Volume: 32, Issue:2 Topics: Adenosine Diphosphate; Age Factors; Animals; Binding Sites; Binding, Competitive; Blood Platelets; Cyclic AMP; Female; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Iodine Radioisotopes; Light; Male; Melatonin; Platelet Aggregation; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Serotonin; Sex Factors	2002
Receptor-mediated modulation of avian caecal muscle contraction by melatonin: role of tyrosine protein kinase. Journal of pineal research, 2002, Volume: 32, Issue:3 Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Apamin; Binding, Competitive; Cecum; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Indoles; Melatonin; Muscle Contraction; Muscle, Smooth; Naphthalenes; Potassium Channels; Protein-Tyrosine Kinases; Quail; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Tetrahydronaphthalenes; Tryptamines	2002
Design and synthesis of 3-phenyl tetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands. Bioorganic & medicinal chemistry, 2003, Mar-06, Volume: 11, Issue:5 Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Drug Design; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Humans; Indicators and Reagents; Ligands; Magnetic Resonance Spectroscopy; Melatonin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Structure-Activity Relationship; Tetrahydronaphthalenes	2003
Characterization and maturational differences of melatonin binding sites in the masu salmon brain. General and comparative endocrinology, 2003, Volume: 131, Issue:3 Topics: Animals; Binding Sites; Brain; Brain Chemistry; Cell Membrane; Female; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Male; Melatonin; Oncorhynchus; Photoperiod; Radioligand Assay; Receptors, Melatonin	2003
Characterization of melatonin binding sites in the brain and retina of the frog Rana perezi. General and comparative endocrinology, 2004, Volume: 135, Issue:3 Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cell Membrane; Diencephalon; Guanosine 5'-O-(3-Thiotriphosphate); Intracellular Membranes; Kinetics; Magnesium; Melatonin; Pertussis Toxin; Radioligand Assay; Ranidae; Receptors, Melatonin; Retina; Sodium; Subcellular Fractions; Superior Colliculi; Telencephalon; Tetrahydronaphthalenes; Tryptamines	2004
Melatonin binding sites in the brain of European sea bass (Dicentrarchus labrax). Zoological science, 2004, Volume: 21, Issue:4 Topics: Animals; Bass; Binding Sites; Brain; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Kinetics; Melatonin; Photoperiod; Radioligand Assay	2004
Effects of temperature on 2-[125I]-iodomelatonin binding to melatonin receptors in the neural retina of the frog Rana perezi. Journal of pineal research, 2005, Volume: 38, Issue:3 Topics: Acclimatization; Animals; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Kinetics; Melatonin; Ranidae; Receptors, Melatonin; Retina; Seasons; Signal Transduction; Temperature	2005
17Beta-estradiol modulates hMT1 melatonin receptor function. Neuroendocrinology, 2005, Volume: 81, Issue:2 Topics: Analysis of Variance; Animals; Blotting, Northern; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Estradiol; Estrogen Receptor alpha; Estrogen Receptor beta; Gene Expression Regulation; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Iodine Isotopes; Melatonin; Protein Binding; Radioligand Assay; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfur Isotopes; Time Factors	2005
Ontogeny of central melatonin receptors in tadpoles of the anuran Rana perezi: modulation of dopamine release. Journal of comparative physiology. A, Neuroethology, sensory, neural, and behavioral physiology, 2005, Volume: 191, Issue:12 Topics: Animals; Brain; Cyclic AMP; Dopamine; Eye; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Larva; Melatonin; Metamorphosis, Biological; Ranidae; Receptors, Melatonin	2005
Critical role of methionine-722 in the stimulation of human brain G-proteins and neurotoxicity induced by London familial Alzheimer's disease (FAD) mutated V717G-APP(714-723). Neuroscience, 2007, Jan-19, Volume: 144, Issue:2 Topics: Aged; Alzheimer Disease; Amyloid beta-Protein Precursor; Animals; Case-Control Studies; Cell Differentiation; Cells, Cultured; Deferoxamine; Dose-Response Relationship, Drug; Estradiol; Female; Glutathione; Glycine; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Melatonin; Methionine; Middle Aged; Peptides; Protein Binding; Rats; Temporal Lobe; Valine	2007
Synthesis and biological activity of new melatonin dimeric derivatives. Bioorganic & medicinal chemistry, 2007, Jul-01, Volume: 15, Issue:13 Topics: 3T3 Cells; Animals; Fibroblasts; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indicators and Reagents; Ligands; Magnetic Resonance Spectroscopy; Melatonin; Mice; Rats; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2	2007
Melatonin receptors in brain areas and ocular tissues of the teleost Tinca tinca: characterization and effect of temperature. General and comparative endocrinology, 2008, Feb-01, Volume: 155, Issue:3 Topics: Animals; Binding Sites; Body Temperature; Brain; Cyprinidae; Eye; Female; Guanosine 5'-O-(3-Thiotriphosphate); Iodine Radioisotopes; Male; Melatonin; Protein Binding; Receptors, Melatonin; Sodium; Temperature	2008
MT1 melatonin receptor internalization underlies melatonin-induced morphologic changes in Chinese hamster ovary cells and these processes are dependent on Gi proteins, MEK 1/2 and microtubule modulation. Journal of pineal research, 2008, Volume: 44, Issue:3 Topics: Animals; Cadaverine; Cell Differentiation; CHO Cells; Clathrin; Cricetinae; Cricetulus; Demecolcine; Extracellular Signal-Regulated MAP Kinases; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Lumicolchicines; MAP Kinase Kinase 1; MAP Kinase Kinase Kinase 2; Melatonin; Microtubules; Pertussis Toxin; Receptor, Melatonin, MT1; Tryptamines	2008
Molecular organization and dynamics of the melatonin MT₁ receptor/RGS20/G(i) protein complex reveal asymmetry of receptor dimers for RGS and G(i) coupling. The EMBO journal, 2010, Nov-03, Volume: 29, Issue:21 Topics: Amino Acid Sequence; Cells, Cultured; Electrophysiology; Energy Transfer; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GTP-Binding Protein alpha Subunits, Gi-Go; GTPase-Activating Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Immunoprecipitation; Kidney; Melatonin; Membrane Proteins; Molecular Sequence Data; Nerve Tissue Proteins; Promoter Regions, Genetic; Protein Binding; Protein Conformation; Protein Multimerization; Receptor, Melatonin, MT1; RGS Proteins; Signal Transduction	2010
Melatonin MT₁ and MT₂ receptors display different molecular pharmacologies only in the G-protein coupled state. British journal of pharmacology, 2014, Volume: 171, Issue:1 Topics: Animals; Binding Sites; Cell Line, Tumor; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); HEK293 Cells; Humans; Kinetics; Ligands; Melatonin; Mice; Molecular Sequence Data; Radioligand Assay; Rats; Receptor, Melatonin, MT2; Sheep; Sodium Chloride; Species Specificity; Transfection	2014