melatonin and colforsin

melatonin has been researched along with colforsin in 133 studies

Research

Studies (133)

TimeframeStudies, this research(%)All Research%
pre-199012 (9.02)18.7374
1990's62 (46.62)18.2507
2000's46 (34.59)29.6817
2010's9 (6.77)24.3611
2020's4 (3.01)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P1
Chik, CL; Ho, AK1
Zatz, M1
Barrett, P; Davidson, G; Hastings, MH; Lawson, W; Morgan, PJ; Thompson, M1
Guerrero, JM; Menendez-Pelaez, A; Reiter, RJ; Santana, C1
Kasper, G; Marquez, CR; Zatz, M1
Hashemi, F; Niles, LP1
Deng, MH; Lopez G-Coviella, I; Lynch, HJ; Wurtman, RJ1
Vanĕcek, J2
Niles, LP; Pickering, DS; Ye, M; Ying, SW1
Janavs, JL; Pierce, ME; Takahashi, JS2
Buzzell, GR; Menendez-Pelaez, A; Nonaka, KO; Reiter, RJ1
Hashemi, FS; Niles, LP1
Besharse, JC; Iuvone, PM1
Guerrero, JM; Reiter, RJ; Santana, C; Troiani, ME1
Barker, D; Harrington, J; Pierce, ME; Takahashi, JS1
Pratt, BL; Takahashi, JS1
Nikaido, SS; Takahashi, JS1
Yuwiler, A1
Guerrero, JM; Reiter, RJ; Santana, C1
Mullen, DA; Zatz, M2
Brun-Marmillon, J; Claustrat, B; Collin, JP; Falcón, J1
Gonzalez-Brito, A; Guerrero, JM; Menendez-Pelaez, A; Reiter, RJ; Santana, C1
Rollag, MD; Sekura, RD; White, BH1
Bubis, M; Zisapel, N1
Gan, J; Iuvone, PM1
Ebisawa, T; Karne, S; Lerner, MR; Reppert, SM1
Barrett, P; Davidson, G; Hazlerigg, D; Lawson, W; MacLean, A; Milligan, G; Morgan, PJ1
Hastings, MH; McNulty, S; Morgan, PJ; Schurov, IL1
Gonzalez-Brito, A; Hastings, MH; Hazlerigg, DG; Lawson, W; Morgan, PJ1
Nash, MS; Osborne, NN2
Florez, JC; Janavs, JL; Pierce, ME; Takahashi, JS1
Barrett, P; Hastings, MH; McNulty, S; Morgan, PJ; Ross, AW1
Chidlow, G; Osborne, NN1
Caignard, DH; Delagrange, P; Depreux, P; Guardiola, B; Howell, HE; Lesieur, D; Mansour, HA; Morgan, P; Pfeiffer, B; Renard, P1
Hastings, MH; Hazlerigg, DG; Morgan, PJ1
Capsoni, S; De Oliveira, AM; Saavedra, JM; Viswanathan, M1
Davidson, G; Hastings, MH; Lawson, W; McNulty, S; Morgan, PJ; Thompson, M1
Barrett, P; Davidson, G; Hazlerigg, D; Lawson, W; Morgan, PJ1
Collin, JP; Falcón, J; Gern, WA; Greenhouse, SS; Lowery, CA; Thibault, C1
Crocker, C; Niles, LP; Ying, SW1
Klein, DC; Vanecek, J1
Hastings, MH; Hazlerigg, DG; Morgan, PJ; Thompson, M1
Fauteck, JD; Fischer, B; Madeja, M; Musshoff, U; Speckmann, EJ; Wittkowski, W1
Baker, J; Ermak, G; Gaudet, SJ; Grande, M; Guisti, LW; Rosano, TG; Slominski, A1
Dubocovich, ML; Witt-Enderby, PA1
Barrett, P; Morgan, PJ; Ross, AW1
Lerchl, A; Niedziela, M; Nieschlag, E1
Barrett, P; Davidson, G; MacLean, A; Morgan, PJ1
Hastings, MH; McNulty, S; Morgan, PJ; Ross, AW; Shiu, KY1
Caillol, M; Martinet, L; Messager, S; Rossano, B1
Barrett, P; Mercer, JG; Morgan, PJ; Ross, AW1
Andersson, RG; Moartensson, LG1
Barrett, P; Canning, SJ; Conway, S; Delagrange, P; Drew, JE; Guardiola-Lemaitre, B; Jockers, R; Morgan, PJ; Strosberg, AD1
Balsamini, C; Di Giacomo, B; Diamantini, G; Fraschini, F; Lucini, V; Mor, M; Nonno, R; Pannacci, M; Plazzi, PV; Rivara, S; Spadoni, G; Stankov, BM; Tarzia, G1
Di Giacomo, B; Diamantini, G; Esposti, D; Fraschini, F; Lucini, V; Nonno, R; Pannacci, M; Spadoni, G; Stankov, BM; Tarzia, G1
Hastings, MH; McNulty, S; McNulty, TJ; Morgan, PJ; Schurov, IL1
Abete, P; Bianco, S; Cacciatore, F; Calabrese, C; Ferrara, N; Napoli, C; Rengo, F1
Duffield, GE; Ebling, FJ; Hastings, MH; Kidd, A; Maywood, ES; Schurov, I1
Barraud, S; Bégay, V; Falcón, J; Thibault, C1
Lamosová, D; Macková, M; Zeman, M1
Dubocovich, ML; Masana, MI; Witt-Enderby, PA1
Adam, C; Barrett, P; Graham, ES; Messager, S; Morgan, PJ; Ross, AW1
Li, L; Pang, SF; Shiu, SY; Wong, JT; Wong, YH; Xu, JN1
Barrett, P; Coon, SL; Fleming, JV; Klein, DC; Morgan, PJ1
Allen, CN; Marino, JL; Nelson, CS1
Cahill, GM; Hasegawa, M1
Flanders, S; Lew, MJ1
Calvo, JR; García-Pergañeda, A; Guerrero, JM; Paz Romero, M; Pozo, D; Rafii-El-Idrissi, M1
Blask, DE; Dauchy, RT; Holowachuk, EW; Kopff, HS; Ruhoff, MS; Sauer, LA1
Graham, ES; Hazlerigg, DG; Morgan, PJ1
Pelisek, V; Slanar, O; Vanecek, J1
Alonso-Bedate, M; Alonso-Gómez, AL; Delgado, MJ; Valenciano, AI1
Beresford, I; Browning, C; Fraser, N; Giles, H1
Jones, MP; Melan, MA; Witt-Enderby, PA1
Beckmann, A; Fauteck, JD; Musshoff, U; Peschke, D; Peschke, E; Schmidt, F1
Gastel, JA; Heath, JR; Klein, DC; Zatz, M1
Korf, HW; Kroeber, S; Maronde, E; Meissl, H1
Pelísek, V; Vanecek, J1
Barrett, P; Choi, WS; Morgan, P; Morris, M1
Karlsson, AM; Lerner, MR; Lundström, I; Svensson, SP; Unett, D1
Abreu, P; Alonso, R; Hernández-Díaz, FJ; López-Coviella, I; Prieto, L; Sánchez, JJ; Tabares, L1
Coon, SL; Klein, DC; Korf, HW; Namboodiri, MA; Rollag, M; Weller, JL1
Blask, DE; Dauchy, RT; Sauer, LA1
Abreu, P; Moujir, F; Reiter, RJ; Sanchez, J; Santana, C1
Pang, SF; Poon, AM; Zhao, H1
Blackhurst, G; Connell, JM; Fraser, R; McElroy, PK; Swan, RL1
MacKenzie, RS; Melan, MA; Passey, DK; Witt-Enderby, PA1
Markowska, M; Mrozkowiak, A; Skwarlo-Sonta, K1
Becq, F; Falcón, J; Gaildrat, P1
Giusti, M; Valenti, S1
Chankiewitz, E; Csernus, VJ; Mühlbauer, E; Musshoff, U; Peschke, D; Peschke, E1
Carpinelli, AR; Cipolla-Neto, J; Curi, R; de Oliveira Carvalho, CR; Haber, EP; Picinato, MC1
Arilla-Ferreiro, E; Boyano-Adánez, Mdel C; Izquierdo-Claros, RM1
Graham, ES; Hazlerigg, DG; Morgan, PJ; Webster, CA1
Chen, J; Deskus, JA; Epperson, JR; Hodges, DB; Iben, L; Li, WS; Luo, G; Mahle, CD; Mattson, RJ; Molstad, D; Ortiz, A; Ryan, E; Sun, LQ; Takaki, K; Xu, C; Yeleswaram, K1
Andrade, LN; Castrucci, AM; Floeter-Winter, LM; Kadekaro, AL; Rollag, MD; Vieira, W; Virador, V1
Angeloni, D; Azeddine, B; Forget, S; Fraschini, F; Grimard, G; Labelle, H; Moreau, A; Poitras, B; Rivard, CH; Wang, DS1
Markowska, M; Mrozkowiak, A; Pawlak, J; Skwarło-Sońta, K1
Jarzynka, MJ; Krawitt, BJ; Melan, MA; Witt-Enderby, PA1
Alonso-Vale, MI; Andreotti, S; Anhê, GF; das Neves Borges-Silva, C; Lima, FB; Neto, JC; Peres, SB1
De Loof, A; Huybrechts, J; Schoofs, L1
Ebadi, M; Govitrapong, P; Santanavanich, C1
Barrett, P; Morgan, PJ; Morris, A; Schuster, C; Williams, LM1
Dubocovich, ML; Masana, MI; Soares, JM1
Ha, DC; Han, S; Kim, KT; Kim, TD1
Csernus, VJ1
Aust, S; Brucker, B; Graf, J; Klimpfinger, M; Thalhammer, T1
Brydon, L; Ignatius, PF; Jarzynka, MJ; Jockers, R; Melan, MA; Passey, DK; Radio, NM; Rasenick, MM; Witt-Enderby, PA1
Azeddine, B; Letellier, K; Moldovan, F; Moreau, A; Wang, da S1
Mühlbauer, E; Peschke, E; Stumpf, I1
Alarma-Estrany, P; Crooke, A; Mediero, A; Peláez, T; Pintor, J1
Genade, S; Genis, A; Huisamen, B; Lochner, A; Ytrehus, K1
Chen, Q; Dong, C; Frasch, T; Hill, SM; Lai, L; Mao, L; Rowan, B; Yuan, L1
Sampaio, Lde F1
Bazwinsky-Wutschke, I; Mühlbauer, E; Peschke, E; Wolgast, S1
Boczek-Leszczyk, E; Juszczak, M1
Guerra, M; Pedreros, M; Ratto, M1
Albrecht, E; Bazwinsky-Wutschke, I; Mühlbauer, E; Peschke, E; Wolgast, S1
Bojunga, J; Fischer, C; Iigo, M; Korf, HW; Yasuo, S1
Juszczak, M; Roszczyk, M1
Hirai, K; Nishiyama, K1
Bojanowska, E; Juszczak, M; Krzyminska, A; Roszczyk, M1
Honma, KI; Honma, S; Yamada, Y; Yamanaka, Y1
Adornetto, A; Bagetta, G; Corasaniti, MT; Morrone, LA; Nucci, C; Rombolà, L; Russo, R1
Asma, A; Marc-André, S1
Ramsay, S; Zagorodnyuk, V1
Aguiar, FLN; Azevedo, VAN; Barrozo, LG; Batista, ALPS; Costa, FC; Donato, MAM; Lopes, EPF; Nascimento, DR; Paulino, LRFM; Peixoto, CA; Rodrigues, APR; Silva, BR; Silva, JRV1

Reviews

2 review(s) available for melatonin and colforsin

ArticleYear
Non-photic signalling in the suprachiasmatic nucleus.
    Biology of the cell, 1997, Volume: 89, Issue:8

    Topics: Afferent Pathways; Age Factors; Animals; Animals, Newborn; Arousal; Calcium; Circadian Rhythm; Colforsin; Cricetinae; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Handling, Psychological; Injections, Subcutaneous; Melatonin; Mesocricetus; Mice; Mice, Inbred C57BL; Neurotransmitter Agents; Phodopus; Phosphorylation; Protein Processing, Post-Translational; Proto-Oncogene Proteins c-fos; Raphe Nuclei; Rodentia; Signal Transduction; Sodium Chloride; Species Specificity; Suprachiasmatic Nucleus; Thalamus

1997
Natural Products: Evidence for Neuroprotection to Be Exploited in Glaucoma.
    Nutrients, 2020, Oct-16, Volume: 12, Issue:10

    Topics: Amides; Biological Products; Colforsin; Curcumin; Cytidine Diphosphate Choline; Dietary Supplements; Ethanolamines; Fatty Acids, Unsaturated; Flavonoids; Ginkgo biloba; Glaucoma; Humans; Melatonin; Neuroprotective Agents; Palmitic Acids; Phytotherapy; Plant Extracts; Resveratrol; Taurine; Tea; Ubiquinone; Vitamins

2020

Other Studies

131 other study(ies) available for melatonin and colforsin

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
    Bioorganic & medicinal chemistry, 2012, Nov-15, Volume: 20, Issue:22

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship

2012
Inhibitors of Na(+)-H+ exchange block stimulus-provoked pineal melatonin synthesis.
    The American journal of physiology, 1992, Volume: 263, Issue:3 Pt 1

    Topics: Amiloride; Animals; Arylamine N-Acetyltransferase; Bucladesine; Carrier Proteins; Colforsin; Cyclic AMP; Hydrogen-Ion Concentration; Male; Melatonin; Pineal Gland; Rats; Rats, Sprague-Dawley; Sodium-Hydrogen Exchangers; Sympathomimetics

1992
Does the circadian pacemaker act through cyclic AMP to drive the melatonin rhythm in chick pineal cells?
    Journal of biological rhythms, 1992,Winter, Volume: 7, Issue:4

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Biological Clocks; Chickens; Circadian Rhythm; Colforsin; Cyclic AMP; Melatonin; Pineal Gland

1992
Intracellular signalling in the ovine pars tuberalis: an investigation using aluminium fluoride and melatonin.
    Journal of molecular endocrinology, 1991, Volume: 7, Issue:2

    Topics: Aluminum; Aluminum Compounds; Animals; Binding Sites; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Fluorides; Inositol Phosphates; Melatonin; Pituitary Gland, Anterior; Sheep; Signal Transduction

1991
Treatment with forskolin for 8 hours during the day increases melatonin synthesis in the Syrian hamster pineal gland in organ culture: the long lag period is required for RNA synthesis.
    Journal of neuroscience research, 1990, Volume: 25, Issue:4

    Topics: Animals; Colforsin; Cricetinae; Male; Melatonin; Mesocricetus; Organ Culture Techniques; Pineal Gland; RNA

1990
Vasoactive intestinal peptide stimulates chick pineal melatonin production and interacts with other stimulatory and inhibitory agents but does not show alpha 1-adrenergic potentiation.
    Journal of neurochemistry, 1990, Volume: 55, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Chickens; Colforsin; Drug Interactions; Isoproterenol; Kinetics; Light; Melatonin; Nitrendipine; Norepinephrine; Phenylephrine; Pineal Gland; Receptors, Adrenergic, alpha; Vasoactive Intestinal Peptide; Yohimbine

1990
Picomolar-affinity binding and inhibition of adenylate cyclase activity by melatonin in Syrian hamster hypothalamus.
    Cellular and molecular neurobiology, 1990, Volume: 10, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclase Inhibitors; Animals; Binding Sites; Colforsin; Cricetinae; Hypothalamus; Iodine Radioisotopes; Male; Melatonin; Mesocricetus; Radioligand Assay; Receptors, Melatonin; Receptors, Neurotransmitter

1990
Melatonin and its precursors in Y79 human retinoblastoma cells: effect of sodium butyrate.
    Brain research, 1991, Oct-11, Volume: 561, Issue:2

    Topics: 5-Hydroxytryptophan; Analysis of Variance; Butyrates; Butyric Acid; Cell Line; Colforsin; Dopamine; Eye Neoplasms; Humans; Kinetics; Levodopa; Melatonin; Retinoblastoma; Serotonin; Spiperone

1991
Melatonin inhibitory effect on luteinizing hormone release is potentiated after long pretreatment with the indole.
    Brain research, 1991, Jan-11, Volume: 538, Issue:2

    Topics: Animals; Animals, Newborn; Colforsin; Cyclic AMP; Female; Gonadotropin-Releasing Hormone; Indoles; Luteinizing Hormone; Melatonin; Pituitary Gland; Rats; Rats, Inbred Strains

1991
Pertussis toxin blocks melatonin-induced inhibition of forskolin-stimulated adenylate cyclase activity in the chick brain.
    Biochemical and biophysical research communications, 1991, Jul-31, Volume: 178, Issue:2

    Topics: Adenylate Cyclase Toxin; Animals; Brain; Cell Membrane; Chickens; Colforsin; Kinetics; Melatonin; Pertussis Toxin; Retina; Synaptosomes; Virulence Factors, Bordetella

1991
N-acetyltransferase and protein synthesis modulate melatonin production by Y79 human retinoblastoma cells.
    Brain research, 1991, Feb-01, Volume: 540, Issue:1-2

    Topics: Acetylserotonin O-Methyltransferase; Anisomycin; Arylamine N-Acetyltransferase; Cell Line; Colforsin; Cycloheximide; Eye Neoplasms; Humans; Kinetics; Melatonin; Neoplasm Proteins; Retinoblastoma

1991
In vivo administration of isoproterenol or forskolin during the light phase induces increases in the melatonin content of the Syrian hamster pineal gland without a rise in N-acetyltransferase activity.
    Neuroscience letters, 1990, Mar-14, Volume: 110, Issue:3

    Topics: Acetyltransferases; Animals; Arylamine N-Acetyltransferase; Circadian Rhythm; Colforsin; Cricetinae; Isoproterenol; Lighting; Melatonin; Mesocricetus; Pineal Gland; Receptors, Adrenergic, beta

1990
Pharmacological inhibition of forskolin-stimulated adenylate cyclase activity in rat brain by melatonin, its analogs, and diazepam.
    Biochemical pharmacology, 1990, Dec-15, Volume: 40, Issue:12

    Topics: Adenylyl Cyclases; Animals; Benzodiazepinones; Brain; Brain Mapping; Cell Membrane; Colforsin; Corpus Striatum; Diazepam; Dose-Response Relationship, Drug; Enzyme Activation; Flumazenil; In Vitro Techniques; Male; Melatonin; Rats; Rats, Inbred Strains

1990
Cyclic AMP stimulates serotonin N-acetyltransferase activity in Xenopus retina in vitro.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Acetyltransferases; Adenosine; Animals; Arylamine N-Acetyltransferase; Bucladesine; Calcium; Circadian Rhythm; Colforsin; Cyclic AMP; Darkness; Fishes; Guinea Pigs; In Vitro Techniques; Light; Melatonin; Retina; Tyrosine 3-Monooxygenase; Xenopus laevis

1986
The in vitro activation of cyclic AMP production by either forskolin or isoproterenol in the Syrian hamster pineal during the day is not accompanied by an increase in melatonin production.
    Biochemical and biophysical research communications, 1988, Dec-30, Volume: 157, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Circadian Rhythm; Colforsin; Cricetinae; Cyclic AMP; Isoproterenol; Kinetics; Male; Melatonin; Mesocricetus; Organ Culture Techniques; Pineal Gland

1988
Cyclic AMP-dependent melatonin production in Y79 human retinoblastoma cells.
    Journal of neurochemistry, 1989, Volume: 53, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 5-Hydroxytryptophan; 8-Bromo Cyclic Adenosine Monophosphate; Colforsin; Cyclic AMP; Humans; Melatonin; Middle Aged; Retinoblastoma; Tumor Cells, Cultured

1989
Vasoactive intestinal polypeptide and alpha 2-adrenoceptor agonists regulate adenosine 3',5'-monophosphate accumulation and melatonin release in chick pineal cell cultures.
    Endocrinology, 1989, Volume: 125, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Amino Acid Sequence; Animals; Brimonidine Tartrate; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Kinetics; Melatonin; Molecular Sequence Data; Pineal Gland; Quinoxalines; Radioimmunoassay; Sequence Homology, Nucleic Acid; Structure-Activity Relationship; Vasoactive Intestinal Peptide

1989
Twenty-four hour oscillation of cAMP in chick pineal cells: role of cAMP in the acute and circadian regulation of melatonin production.
    Neuron, 1989, Volume: 3, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Animals, Newborn; Chickens; Circadian Rhythm; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Male; Melatonin; Pineal Gland

1989
Effects of steroids on serotonin-N-acetyltransferase activity of pineals in organ culture.
    Journal of neurochemistry, 1989, Volume: 52, Issue:1

    Topics: Acetyltransferases; Animals; Arylamine N-Acetyltransferase; Bucladesine; Cholera Toxin; Colforsin; Corticosterone; Dose-Response Relationship, Drug; Hydrocortisone; Indoles; Isoproterenol; Male; Melatonin; Organ Culture Techniques; Pineal Gland; Rats; Rats, Inbred F344; Steroids; Tryptophan

1989
Effects of either forskolin, the 1,9-dideoxy derivative of forskolin, or 8-bromocyclic AMP on cyclic AMP and melatonin production in the Syrian hamster pineal gland in organ culture.
    Neuroscience letters, 1989, Sep-11, Volume: 103, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Colforsin; Cricetinae; Cyclic AMP; Male; Melatonin; Mesocricetus; Organ Culture Techniques; Pineal Gland; Radioimmunoassay; Rats; Rats, Inbred Strains

1989
Photoendocrine transduction in cultured chick pineal cells. II. Effects of forskolin, 8-bromocyclic AMP, and 8-bromocyclic GMP on the melatonin rhythm.
    Brain research, 1988, Jun-21, Volume: 453, Issue:1-2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cells, Cultured; Chickens; Circadian Rhythm; Colforsin; Cyclic GMP; Lighting; Melatonin; Pineal Gland

1988
Melatonin production in organ cultured chicken pineal: modulation by adenosine and its analogs.
    Pflugers Archiv : European journal of physiology, 1988, Volume: 413, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Adenosine Deaminase; Animals; Chickens; Colforsin; Deoxyadenosines; Dipyridamole; Melatonin; Organ Culture Techniques; Phenylisopropyladenosine; Pineal Gland; Thioinosine

1988
Norepinephrine, acting via adenylate cyclase, inhibits melatonin output but does not phase-shift the pacemaker in cultured chick pineal cells.
    Brain research, 1988, May-31, Volume: 450, Issue:1-2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Cells, Cultured; Chickens; Circadian Rhythm; Colforsin; Lighting; Melatonin; Norepinephrine; Photic Stimulation; Pineal Gland

1988
Forskolin, an activator of adenylate cyclase activity, promotes large increases in N-acetyl transferase activity and melatonin production in the Syrian hamster pineal gland only during the late dark period.
    Biochemical and biophysical research communications, 1988, Aug-30, Volume: 155, Issue:1

    Topics: Acetyltransferases; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Circadian Rhythm; Colforsin; Cricetinae; Darkness; Enzyme Activation; Enzyme Induction; Male; Melatonin; Mesocricetus; Pineal Gland

1988
Pertussis toxin blocks melatonin-induced pigment aggregation in Xenopus dermal melanophores.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 1987, Volume: 157, Issue:2

    Topics: Adenylate Cyclase Toxin; Animals; Cell Aggregation; Cells, Cultured; Colforsin; Melanocytes; Melanophores; Melatonin; Pertussis Toxin; Virulence Factors, Bordetella; Xenopus laevis

1987
Modulation by melatonin of protein secretion from melanoma cells: is cAMP involved?
    Molecular and cellular endocrinology, 1995, Aug-11, Volume: 112, Issue:2

    Topics: Animals; Bucladesine; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Isoquinolines; Melanoma, Experimental; Melatonin; Mice; Protein Biosynthesis; Proteins; Sulfonamides; Tumor Cells, Cultured

1995
Melatonin receptor-mediated inhibition of cyclic AMP accumulation in chick retinal cell cultures.
    Journal of neurochemistry, 1994, Volume: 63, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 5-Methoxytryptamine; Animals; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Iodine Radioisotopes; Melatonin; Neurons; Pertussis Toxin; Photoreceptor Cells; Potassium; Receptors, Cell Surface; Receptors, Melatonin; Retina; Second Messenger Systems; Structure-Activity Relationship; Tryptamines; Virulence Factors, Bordetella

1994
Expression cloning of a high-affinity melatonin receptor from Xenopus dermal melanophores.
    Proceedings of the National Academy of Sciences of the United States of America, 1994, Jun-21, Volume: 91, Issue:13

    Topics: Amino Acid Sequence; Animals; Cell Line; Cell Membrane; Cells, Cultured; Chlorocebus aethiops; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Cyclic AMP; DNA; DNA, Complementary; Gene Expression; Kidney; Kinetics; Melanophores; Melatonin; Molecular Sequence Data; Poly A; Protein Structure, Secondary; Receptors, Cell Surface; Receptors, Melatonin; RNA; RNA, Messenger; Skin; Transcription, Genetic; Transfection; Xenopus laevis

1994
Melatonin receptors couple through a cholera toxin-sensitive mechanism to inhibit cyclic AMP in the ovine pituitary.
    Journal of neuroendocrinology, 1995, Volume: 7, Issue:5

    Topics: Adenosine Diphosphate Ribose; Animals; Base Sequence; Blotting, Northern; Cell Membrane; Cholera Toxin; Colforsin; Cyclic AMP; GTP-Binding Proteins; Iodine Radioisotopes; Melatonin; Molecular Sequence Data; NAD; Pertussis Toxin; Pituitary Gland; Receptors, Cell Surface; Receptors, Melatonin; RNA, Messenger; Sheep; Virulence Factors, Bordetella

1995
The inhibitory action of melatonin in the ovine pars tuberalis is not dependent on changes in plasma membrane potential.
    The Journal of endocrinology, 1995, Volume: 145, Issue:3

    Topics: Adenylyl Cyclases; Animals; Cell Membrane; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Female; Male; Melatonin; Membrane Potentials; Pituitary Gland; Potassium; Saponins; Sheep; Stimulation, Chemical; Valinomycin

1995
Prolonged exposure to melatonin leads to time-dependent sensitization of adenylate cyclase and down-regulates melatonin receptors in pars tuberalis cells from ovine pituitary.
    Endocrinology, 1993, Volume: 132, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Aluminum; Aluminum Compounds; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Cycloheximide; Down-Regulation; Fluorides; Iodine Radioisotopes; Kinetics; Melatonin; Pituitary Gland, Anterior; Receptors, Melatonin; Receptors, Neurotransmitter; Sheep

1993
Melatonin inhibits increase of intracellular calcium and cyclic AMP in neonatal rat pituitary via independent pathways.
    Molecular and cellular endocrinology, 1995, Volume: 107, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Calcium; Colforsin; Cyclic AMP; Gonadotropin-Releasing Hormone; GTP-Binding Proteins; Intracellular Fluid; Melatonin; Pituitary Gland, Anterior; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, Melatonin; Second Messenger Systems

1995
Pertussis toxin-sensitive melatonin receptors negatively coupled to adenylate cyclase associated with cultured human and rat retinal pigment epithelial cells.
    Investigative ophthalmology & visual science, 1995, Volume: 36, Issue:1

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adult; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Melatonin; Pertussis Toxin; Pigment Epithelium of Eye; Rats; Receptors, Cell Surface; Receptors, Melatonin; Virulence Factors, Bordetella

1995
Forskolin and camptothecin induce a 30 kDa protein associated with melatonin production in Y79 human retinoblastoma cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:1 Pt 1

    Topics: Camptothecin; Colforsin; Humans; Immunoblotting; Melatonin; Molecular Weight; Neoplasm Proteins; Retinoblastoma; Time Factors; Tumor Cells, Cultured

1995
Melatonin regulates the phosphorylation of CREB in ovine pars tuberalis.
    Journal of neuroendocrinology, 1994, Volume: 6, Issue:5

    Topics: Animals; Base Sequence; Cell Nucleus; Cells, Cultured; Colforsin; Consensus Sequence; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Enzyme Activation; Melatonin; Molecular Sequence Data; Phosphorylation; Pituitary Gland, Anterior; Protein Kinase C; Sheep; Signal Transduction; Tetradecanoylphorbol Acetate

1994
The presence of functional melatonin receptors in the iris-ciliary processes of the rabbit eye.
    Experimental eye research, 1994, Volume: 59, Issue:1

    Topics: Animals; Autoradiography; Ciliary Body; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Iris; Melatonin; Rabbits; Receptors, Cell Surface; Receptors, Melatonin; Serotonin

1994
Synthesis and structure-activity relationships of novel naphthalenic and bioisosteric related amidic derivatives as melatonin receptor ligands.
    Journal of medicinal chemistry, 1994, Sep-30, Volume: 37, Issue:20

    Topics: Acetamides; Animals; Cell Membrane; Colforsin; Cyclic AMP; Iodine Radioisotopes; Ligands; Melatonin; Molecular Structure; Pituitary Gland, Anterior; Receptors, Cell Surface; Receptors, Melatonin; Sheep; Structure-Activity Relationship

1994
The recovery of ovine pars tuberalis cells from melatonin-induced sensitization is a slow, protein synthesis-dependent phenomenon.
    The Journal of endocrinology, 1994, Volume: 142, Issue:1

    Topics: Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Cycloheximide; Drug Synergism; Electrophoresis, Polyacrylamide Gel; Female; Kinetics; Male; Melatonin; Nerve Tissue Proteins; Pituitary Gland, Anterior; Protein Kinases; Sheep

1994
Characterization of melatonin receptors and signal transduction system in rat arteries forming the circle of Willis.
    Endocrinology, 1994, Volume: 135, Issue:1

    Topics: Animals; Arteries; Circle of Willis; Colforsin; Cyclic AMP; Male; Melatonin; Nucleotides; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Melatonin; Signal Transduction

1994
RNA synthesis inhibitors increase melatonin production in Y79 human retinoblastoma cells.
    Brain research. Molecular brain research, 1994, Volume: 23, Issue:1-2

    Topics: Amidohydrolases; Anisomycin; Arylamine N-Acetyltransferase; Calcium; Camptothecin; Colforsin; Cyclic AMP; Dactinomycin; Dopamine; Egtazic Acid; Eye Neoplasms; Humans; Melatonin; Nerve Tissue Proteins; Protein Synthesis Inhibitors; Retinoblastoma; Topoisomerase I Inhibitors; Transcription, Genetic; Tumor Cells, Cultured

1994
Phospholipases and melatonin signal transduction in the ovine pars tuberalis.
    Molecular and cellular endocrinology, 1994, Volume: 99, Issue:1

    Topics: Adenylyl Cyclases; Animals; Arachidonic Acid; Calcimycin; Cells, Cultured; Choline; Colforsin; Cyclic AMP; Female; Lysophospholipids; Male; Melatonin; Membrane Lipids; Phosphatidic Acids; Phospholipases; Phospholipids; Pituitary Gland, Anterior; Second Messenger Systems; Sheep; Signal Transduction; Tetradecanoylphorbol Acetate

1994
p72, a marker protein for melatonin action in ovine pars tuberalis cells: its regulation by protein kinase A and protein kinase C and differential secretion relative to prolactin.
    Neuroendocrinology, 1994, Volume: 59, Issue:4

    Topics: Animals; Autoradiography; Biomarkers; Calcium; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Female; Gonadotropin-Releasing Hormone; Kinetics; Male; Melatonin; Methionine; Microtubules; Nerve Tissue Proteins; Pituitary Gland, Anterior; Prolactin; Protein Kinase C; Receptors, LHRH; Sheep

1994
Regulation of melatonin production by pineal photoreceptor cells: role of cyclic nucleotides in the trout (Oncorhynchus mykiss).
    Journal of neurochemistry, 1993, Volume: 61, Issue:1

    Topics: Animals; Arylamine N-Acetyltransferase; Colforsin; Cyclic AMP; Melatonin; Nucleotides, Cyclic; Photoreceptor Cells; Pineal Gland; Temperature; Theophylline; Trout

1993
Human malignant melanoma cells express high-affinity receptors for melatonin: antiproliferative effects of melatonin and 6-chloromelatonin.
    European journal of pharmacology, 1993, Jul-15, Volume: 246, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Cell Division; Cell Membrane; Colforsin; Cyclic AMP; DNA, Neoplasm; Humans; Indoles; Iodine Radioisotopes; Kinetics; Melanoma; Melatonin; Nucleotides; Receptors, Melatonin; Receptors, Neurotransmitter; Tumor Cells, Cultured

1993
Agonist-induced effects on cyclic AMP metabolism are affected in pigment epithelial cells of the Royal College of Surgeons rat.
    Neurochemistry international, 1995, Volume: 27, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprostadil; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dinoprostone; Fibroblast Growth Factor 2; Imidazoles; Isoproterenol; Kinetics; Melatonin; Pigment Epithelium of Eye; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta-2; Receptors, Purinergic P1; Serotonin

1995
Mechanism of melatonin signal transduction in the neonatal rat pituitary.
    Neurochemistry international, 1995, Volume: 27, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Calcimycin; Calcium; Colforsin; Cyclic AMP; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Melatonin; Nifedipine; Organ Culture Techniques; Pituitary Gland, Anterior; Rats; Receptors, Cell Surface; Receptors, Melatonin; Signal Transduction

1995
Regulation of mitogen-activated protein kinase in the pars tuberalis of the ovine pituitary: interactions between melatonin, insulin-like growth factor-1, and forskolin.
    Endocrinology, 1996, Volume: 137, Issue:1

    Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Colforsin; Cytosol; Enzyme Activation; Humans; Immunohistochemistry; Insulin-Like Growth Factor I; Melatonin; Mitogen-Activated Protein Kinase 1; Myelin Basic Protein; Phosphorylation; Pituitary Gland, Anterior; Protein-Tyrosine Kinases; Receptors, Somatomedin; Recombinant Proteins; Sheep; Tissue Distribution; Tissue Extracts

1996
Expression and functional characterization of a melatonin-sensitive receptor in Xenopus oocytes.
    FEBS letters, 1996, Feb-26, Volume: 381, Issue:1-2

    Topics: Animals; Anthracenes; Autoradiography; Binding Sites; Brain; Caffeine; Colforsin; Cyclic AMP; Female; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Melatonin; Membrane Potentials; Microinjections; Oocytes; Patch-Clamp Techniques; Pertussis Toxin; Rats; Receptors, Cell Surface; Receptors, Melatonin; RNA, Messenger; Virulence Factors, Bordetella

1996
Metabolism of serotonin to N-acetylserotonin, melatonin, and 5-methoxytryptamine in hamster skin culture.
    The Journal of biological chemistry, 1996, May-24, Volume: 271, Issue:21

    Topics: 5-Methoxytryptamine; Animals; Chromatography, High Pressure Liquid; Colforsin; Cricetinae; Gas Chromatography-Mass Spectrometry; Male; Melatonin; Mesocricetus; Organ Culture Techniques; Serotonin; Skin; Tritium

1996
Characterization and regulation of the human ML1A melatonin receptor stably expressed in Chinese hamster ovary cells.
    Molecular pharmacology, 1996, Volume: 50, Issue:1

    Topics: Animals; Binding, Competitive; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Humans; Kinetics; Melatonin; Receptors, Cell Surface; Receptors, Melatonin; Recombinant Proteins; Transfection; Tryptamines

1996
Melatonin regulated gene expression in pars tuberalis cells of the ovine pituitary investigated by differential display.
    Biochemical Society transactions, 1996, Volume: 24, Issue:2

    Topics: Animals; Colforsin; Cycloheximide; DNA-Binding Proteins; Gene Expression; Melatonin; Pituitary Gland; Polymerase Chain Reaction; Proto-Oncogene Proteins c-fos; Sheep; Transcription Factors

1996
Direct effects of the pineal hormone melatonin on testosterone synthesis of Leydig cells in Djungarian hamsters (Phodopus sungorus) in vitro.
    Neuroscience letters, 1995, Dec-15, Volume: 201, Issue:3

    Topics: Animals; Colforsin; Cricetinae; Dose-Response Relationship, Drug; In Vitro Techniques; Leydig Cells; Luteinizing Hormone; Male; Melatonin; Testosterone

1995
Regulation of the Mel 1a melatonin receptor mRNA and protein levels in the ovine pars tuberalis: evidence for a cyclic adenosine 3',5'-monophosphate-independent Mel 1a receptor coupling and an autoregulatory mechanism of expression.
    Molecular endocrinology (Baltimore, Md.), 1996, Volume: 10, Issue:7

    Topics: Animals; Cells, Cultured; Colforsin; Culture Media, Serum-Free; Cyclic AMP; Dactinomycin; Melatonin; Pituitary Gland, Anterior; Protein Synthesis Inhibitors; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; RNA, Messenger; Sheep; Time Factors; Transcription, Genetic; Up-Regulation

1996
Phosphorylation of CREB in ovine pars tuberalis is regulated both by cyclic AMP-dependent and cyclic AMP-independent mechanisms.
    Journal of neuroendocrinology, 1996, Volume: 8, Issue:8

    Topics: Adenosine; Animals; Blood Physiological Phenomena; Blotting, Western; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Dinoprostone; Female; Immunohistochemistry; Male; Melatonin; Phosphorylation; Pituitary Gland, Anterior; Serine; Sheep

1996
Effect of melatonin on the release of gonadotropin-releasing hormone and cyclic AMP from the rat hypothalamus: an in vitro study.
    Journal of neuroendocrinology, 1996, Volume: 8, Issue:10

    Topics: Animals; Colforsin; Cyclic AMP; Gonadotropin-Releasing Hormone; Hypothalamus, Middle; In Vitro Techniques; Male; Melatonin; Preoptic Area; Rats; Rats, Wistar; Reproducibility of Results

1996
Melatonin suppresses the induction of AP-1 transcription factor components in the pars tuberalis of the pituitary.
    Molecular and cellular endocrinology, 1996, Oct-14, Volume: 123, Issue:1

    Topics: Animals; Base Sequence; Blotting, Northern; Cells, Cultured; Colforsin; Female; Gene Expression; Genes, jun; In Situ Hybridization; Insulin-Like Growth Factor I; Male; Melatonin; Oligonucleotide Probes; Pituitary Gland, Anterior; Proto-Oncogene Proteins c-jun; RNA, Messenger; Sheep; Transcription Factor AP-1; Transcription, Genetic

1996
Denervation of pigment cells lead to a receptor that is ultrasensitive to melatonin and noradrenaline.
    Life sciences, 1997, Volume: 60, Issue:18

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Colforsin; Denervation; Fishes; Melanins; Melanophores; Melatonin; Norepinephrine; Peripheral Nervous System; Prazosin; Yohimbine

1997
Identification of Mel1a melatonin receptors in the human embryonic kidney cell line HEK293: evidence of G protein-coupled melatonin receptors which do not mediate the inhibition of stimulated cyclic AMP levels.
    FEBS letters, 1997, Apr-21, Volume: 407, Issue:1

    Topics: Binding, Competitive; Cell Line; Colforsin; Cyclic AMP; Genomic Library; GTP-Binding Proteins; Humans; Kidney; Melatonin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; RNA, Messenger; Sequence Analysis, DNA; Serotonin; Signal Transduction; Tryptamines

1997
Conformationally restrained melatonin analogues: synthesis, binding affinity for the melatonin receptor, evaluation of the biological activity, and molecular modeling study.
    Journal of medicinal chemistry, 1997, Jun-20, Volume: 40, Issue:13

    Topics: Animals; Binding, Competitive; Chickens; Colforsin; Cyclic AMP; Drug Design; Guanosine 5'-O-(3-Thiotriphosphate); Melatonin; Models, Molecular; Quail; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Superior Colliculi

1997
1-(2-Alkanamidoethyl)-6-methoxyindole derivatives: a new class of potent indole melatonin analogues.
    Journal of medicinal chemistry, 1997, Jun-20, Volume: 40, Issue:13

    Topics: Animals; Binding Sites; Binding, Competitive; Chickens; Colforsin; Cyclic AMP; Drug Design; Guanosine 5'-O-(3-Thiotriphosphate); Indoles; Melatonin; Models, Chemical; Quail; Superior Colliculi

1997
Melatonin-sensitive, serum-stimulated signalling in ovine pars tuberalis.
    Journal of pineal research, 1997, Volume: 22, Issue:4

    Topics: Animals; Blood; Cells, Cultured; Colforsin; Cyclic AMP Response Element-Binding Protein; DNA-Binding Proteins; Down-Regulation; Enzyme Inhibitors; Female; Fluorescent Dyes; Fura-2; Genes, Immediate-Early; Immunoenzyme Techniques; Indoles; Male; Melatonin; Phosphorylation; Pituitary Gland, Anterior; Protein Kinase C; Proto-Oncogene Proteins c-fos; Sheep; Signal Transduction; Tetradecanoylphorbol Acetate; Transcription Factors

1997
Effects of melatonin in isolated rat papillary muscle.
    FEBS letters, 1997, Jul-21, Volume: 412, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Calcium; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Isoproterenol; Male; Melatonin; Myocardial Contraction; Papillary Muscles; Rats; Rats, Inbred WKY; Stimulation, Chemical

1997
Inhibitors of messenger RNA and protein synthesis affect differently serotonin arylalkylamine N-acetyltransferase activity in clock-controlled and non clock-controlled fish pineal.
    Brain research, 1998, Jun-22, Volume: 797, Issue:1

    Topics: Acetylserotonin O-Methyltransferase; Animals; Arylamine N-Acetyltransferase; Biological Clocks; Colforsin; Enzyme Activation; Esocidae; Female; Gene Expression Regulation, Enzymologic; Male; Melatonin; Oncorhynchus mykiss; Pineal Gland; RNA, Messenger; Serotonin

1998
Regulation of rhythmic melatonin production in pineal cells of chick embryo by cyclic AMP.
    Cellular and molecular life sciences : CMLS, 1998, Volume: 54, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Chick Embryo; Colforsin; Cyclic AMP; Melatonin; Phosphodiesterase Inhibitors; Pineal Gland

1998
Physiological exposure to melatonin supersensitizes the cyclic adenosine 3',5'-monophosphate-dependent signal transduction cascade in Chinese hamster ovary cells expressing the human mt1 melatonin receptor.
    Endocrinology, 1998, Volume: 139, Issue:7

    Topics: Animals; Catalysis; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; GTP-Binding Proteins; Humans; Melatonin; Pertussis Toxin; Phosphorylation; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Ribose; Signal Transduction; Time Factors; Virulence Factors, Bordetella

1998
oPer1 is an early response gene under photoperiodic regulation in the ovine pars tuberalis.
    Journal of neuroendocrinology, 1998, Volume: 10, Issue:5

    Topics: Animals; Circadian Rhythm; Colforsin; Gene Expression; Gene Expression Regulation; Light; Melatonin; Nuclear Proteins; Photoperiod; Pituitary Gland; RNA, Messenger; Seasons; Sheep

1998
Molecular and cellular analyses of melatonin receptor-mediated cAMP signaling in rat corpus epididymis.
    Journal of pineal research, 1998, Volume: 25, Issue:4

    Topics: Adenylyl Cyclases; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dihydrotestosterone; DNA Primers; Epididymis; Epithelial Cells; GTP-Binding Proteins; In Situ Hybridization; Isoproterenol; Male; Melatonin; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction

1998
Ovine arylalkylamine N-acetyltransferase in the pineal and pituitary glands: differences in function and regulation.
    Endocrinology, 1999, Volume: 140, Issue:2

    Topics: Animals; Arylamine N-Acetyltransferase; Colforsin; Cyclic AMP; Cyclic AMP Response Element Modulator; DNA-Binding Proteins; Female; Gene Expression Regulation; In Vitro Techniques; Male; Melatonin; Pineal Gland; Pituitary Gland; Repressor Proteins; RNA, Messenger

1999
Melatonin receptor potentiation of cyclic AMP and the cystic fibrosis transmembrane conductance regulator ion channel.
    Journal of pineal research, 1999, Volume: 26, Issue:2

    Topics: Adenylate Cyclase Toxin; Animals; Chloride Channels; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Electric Conductivity; Female; Melatonin; Oocytes; Pertussis Toxin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Receptors, Serotonin; Transfection; Virulence Factors, Bordetella; Xenopus laevis

1999
Modulation of rhythmic melatonin synthesis in Xenopus retinal photoreceptors by cyclic AMP.
    Brain research, 1999, Apr-10, Volume: 824, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Circadian Rhythm; Colforsin; Culture Techniques; Cyclic AMP; Enzyme Inhibitors; Male; Melatonin; Photoreceptor Cells, Vertebrate; Retina; Stimulation, Chemical; Thionucleotides; Xenopus laevis

1999
Mechanisms of melatonin-induced vasoconstriction in the rat tail artery: a paradigm of weak vasoconstriction.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Acetamides; Animals; Anticonvulsants; Arteries; Calcium Channel Blockers; Charybdotoxin; Colforsin; Dose-Response Relationship, Drug; Hypnotics and Sedatives; In Vitro Techniques; Indoles; Male; Melatonin; Nifedipine; Nitroprusside; Potassium Channels; Rats; Rats, Sprague-Dawley; Tail; Tryptamines; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents; Vasopressins

1999
Characterization of membrane melatonin receptor in mouse peritoneal macrophages: inhibition of adenylyl cyclase by a pertussis toxin-sensitive G protein.
    Journal of neuroimmunology, 1999, Mar-01, Volume: 95, Issue:1-2

    Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Blotting, Western; Colforsin; Cyclic AMP; GTP-Binding Protein alpha Subunits, Gi-Go; Iodine Radioisotopes; Kinetics; Macrophages, Peritoneal; Melatonin; Mice; Neuroimmunomodulation; Pertussis Toxin; Radioligand Assay; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Serotonin; Signal Transduction; Tryptamines; Virulence Factors, Bordetella

1999
Melatonin inhibition of cancer growth in vivo involves suppression of tumor fatty acid metabolism via melatonin receptor-mediated signal transduction events.
    Cancer research, 1999, Sep-15, Volume: 59, Issue:18

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Biological Transport; Cell Division; Circadian Rhythm; Colforsin; Linoleic Acid; Linoleic Acids; Liver Neoplasms, Experimental; Male; Melatonin; Models, Biological; Naphthalenes; Perfusion; Pertussis Toxin; Rats; Rats, Inbred BUF; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Signal Transduction; Virulence Factors, Bordetella

1999
Evidence for regulation of basic fibroblast growth factor gene expression by photoperiod and melatonin in the ovine pars tuberalis.
    Molecular and cellular endocrinology, 1999, Oct-25, Volume: 156, Issue:1-2

    Topics: Animals; Cell Line; Cells, Cultured; Colforsin; Fibroblast Growth Factor 2; Gene Expression Regulation; Male; Melatonin; Photoperiod; Pituitary Gland, Anterior; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Seasons; Sheep; Tetradecanoylphorbol Acetate; Transcription, Genetic

1999
Melatonin inhibits pituitary adenylyl cyclase-activating polypeptide-induced increase of cyclic AMP accumulation and [Ca2+]i in cultured cells of neonatal rat pituitary.
    Neurochemistry international, 2000, Volume: 36, Issue:3

    Topics: Animals; Animals, Newborn; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Female; Gonadotropin-Releasing Hormone; Melatonin; Neuropeptides; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland, Anterior; Rats; Rats, Wistar

2000
Melatonin synthesis in the greenfrog retina in culture: I. Modulation by the light/dark cycle, forskolin and inhibitors of protein synthesis.
    Life sciences, 2000, Jan-14, Volume: 66, Issue:8

    Topics: Animals; Antioxidants; Arylamine N-Acetyltransferase; Colforsin; Culture Media; Dactinomycin; Light; Melatonin; Organ Culture Techniques; Photoperiod; Protein Synthesis Inhibitors; Radioimmunoassay; Ranidae; Retina; Time Factors

2000
Pharmacological characterization of human recombinant melatonin mt(1) and MT(2) receptors.
    British journal of pharmacology, 2000, Volume: 129, Issue:5

    Topics: Animals; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Humans; Isotope Labeling; Kinetics; Melatonin; Pertussis Toxin; Radioligand Assay; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Recombinant Proteins; Virulence Factors, Bordetella

2000
Melatonin decreases cell proliferation and transformation in a melatonin receptor-dependent manner.
    Cancer letters, 2000, Apr-14, Volume: 151, Issue:2

    Topics: 3T3 Cells; Animals; Binding Sites; Cell Count; Cell Division; Cell Transformation, Neoplastic; Colforsin; Cyclic AMP; DNA; Humans; Melatonin; Mice; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Signal Transduction; Transfection; Tumor Stem Cell Assay

2000
Evidence for a melatonin receptor within pancreatic islets of neonate rats: functional, autoradiographic, and molecular investigations.
    Journal of pineal research, 2000, Volume: 28, Issue:3

    Topics: Animals; Animals, Newborn; Autoradiography; Colforsin; DNA Primers; Dose-Response Relationship, Drug; Female; Gene Expression; Guanosine 5'-O-(3-Thiotriphosphate); Insulin; Insulin Secretion; Islets of Langerhans; Male; Melatonin; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tryptamines

2000
Chick pineal melatonin synthesis: light and cyclic AMP control abundance of serotonin N-acetyltransferase protein.
    Journal of neurochemistry, 2000, Volume: 74, Issue:6

    Topics: Animals; Arylamine N-Acetyltransferase; Cells, Cultured; Chick Embryo; Circadian Rhythm; Colforsin; Cyclic AMP; Cysteine Endopeptidases; Cysteine Proteinase Inhibitors; Enzyme Activation; Leupeptins; Lighting; Melatonin; Multienzyme Complexes; Norepinephrine; Photoreceptor Cells, Vertebrate; Pineal Gland; Proteasome Endopeptidase Complex; Signal Transduction; Sympathomimetics

2000
Analyses of signal transduction cascades reveal an essential role of calcium ions for regulation of melatonin biosynthesis in the light-sensitive pineal organ of the rainbow trout (Oncorhynchus mykiss).
    Journal of neurochemistry, 2000, Volume: 74, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Arylamine N-Acetyltransferase; Calcium; Calcium Signaling; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cysteine Endopeptidases; Female; Gene Expression; Immunohistochemistry; Male; Melatonin; Multienzyme Complexes; Oncorhynchus mykiss; Organ Culture Techniques; Phosphodiesterase Inhibitors; Phosphorylation; Photic Stimulation; Pineal Gland; Proteasome Endopeptidase Complex; Protein Processing, Post-Translational; Signal Transduction; Transcription, Genetic

2000
Different effects of melatonin pretreatment on cAMP and LH responses of the neonatal rat pituitary cells.
    Journal of pineal research, 2000, Volume: 28, Issue:4

    Topics: Animals; Animals, Newborn; Cells, Cultured; Colforsin; Female; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Melatonin; Pituitary Gland, Anterior; Rats; Rats, Wistar

2000
A role for tyrosine phosphorylation in the regulation and sensitization of adenylate cyclase by melatonin.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2000, Volume: 14, Issue:11

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Benzoquinones; Cells, Cultured; Colforsin; Cyclic AMP; Drug Synergism; Enzyme Inhibitors; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Isoenzymes; Lactams, Macrocyclic; Melatonin; Models, Biological; Phosphorylation; Phosphotyrosine; Pituitary Gland; Protein Tyrosine Phosphatases; Protein-Tyrosine Kinases; Quinones; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Rifabutin; RNA, Messenger; Sheep; Signal Transduction; Virulence Factors, Bordetella

2000
Melatonin-induced organelle movement in melanophores is coupled to tyrosine phosphorylation of a high molecular weight protein.
    Cellular signalling, 2000, Volume: 12, Issue:7

    Topics: Adenylate Cyclase Toxin; Animals; Blotting, Western; Cell Aggregation; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Genistein; GTP-Binding Proteins; Kinetics; Melanophores; Melatonin; Pertussis Toxin; Phosphoprotein Phosphatases; Phosphorylation; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Serine; Signal Transduction; Threonine; Time Factors; Tyrosine; Virulence Factors, Bordetella; Xenopus

2000
Estrogen modulates alpha(1)/beta-adrenoceptor- induced signaling and melatonin production in female rat pinealocytes.
    Neuroendocrinology, 2001, Volume: 73, Issue:2

    Topics: Action Potentials; Animals; Arylamine N-Acetyltransferase; Calcium; Cholera Toxin; Colforsin; Cyclic AMP; Estradiol; Female; Hydrogen-Ion Concentration; Hydrolysis; Melatonin; Ovariectomy; Phosphatidylinositols; Pineal Gland; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Estradiol; Signal Transduction

2001
cAmp regulation of arylalkylamine N-acetyltransferase (AANAT, EC 2.3.1.87): a new cell line (1E7) provides evidence of intracellular AANAT activation.
    The Journal of biological chemistry, 2001, Jun-29, Volume: 276, Issue:26

    Topics: Animals; Arylalkylamine N-Acetyltransferase; Arylamine N-Acetyltransferase; Cell Extracts; Cell Line; Colforsin; COS Cells; Cyclic AMP; Cytoplasm; Darkness; Enzyme Activation; Escherichia coli; Humans; Kinetics; Melatonin; Pineal Gland; Rats; Rats, Sprague-Dawley; Tryptamines

2001
Melatonin inhibits fatty acid transport in inguinal fat pads of hepatoma 7288CTC-bearing and normal Buffalo rats via receptor-mediated signal transduction.
    Life sciences, 2001, May-11, Volume: 68, Issue:25

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipose Tissue; Animals; Biological Transport; Circadian Rhythm; Colforsin; Linoleic Acid; Liver Neoplasms, Experimental; Male; Melatonin; Naphthalenes; Neoplasm Transplantation; Pertussis Toxin; Rats; Rats, Inbred BUF; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Signal Transduction; Specific Pathogen-Free Organisms; Time Factors; Virulence Factors, Bordetella

2001
Role of extracellular calcium on the regulation of melatonin synthesis in the Syrian hamster pineal gland.
    Journal of pineal research, 2001, Volume: 31, Issue:4

    Topics: Animals; Arylamine N-Acetyltransferase; Calcium; Colforsin; Cricetinae; Cyclic AMP; Male; Melatonin; Mesocricetus; Organ Culture Techniques; Pineal Gland

2001
mt(1) Receptor-mediated antiproliferative effects of melatonin on the rat uterine antimesometrial stromal cells.
    Molecular reproduction and development, 2002, Volume: 61, Issue:2

    Topics: Adenylate Cyclase Toxin; Animals; Autoradiography; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Endometrium; Female; In Situ Hybridization; Melatonin; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Stromal Cells; Virulence Factors, Bordetella

2002
Seasonal variation in glucocorticoid receptor binding characteristics in human mononuclear leucocytes.
    Clinical endocrinology, 2001, Volume: 55, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Adult; Analysis of Variance; Cells, Cultured; Colforsin; Dexamethasone; Enzyme Inhibitors; Female; Humans; Hydrocortisone; Leukocytes, Mononuclear; Male; Melatonin; Protein Binding; Receptors, Glucocorticoid; Seasons

2001
Dual coupling of MT(1) and MT(2) melatonin receptors to cyclic AMP and phosphoinositide signal transduction cascades and their regulation following melatonin exposure.
    Biochemical pharmacology, 2002, Feb-15, Volume: 63, Issue:4

    Topics: Analysis of Variance; Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Drug Interactions; Humans; Hydrolysis; Melatonin; Phosphatidylinositols; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Signal Transduction; Tetrahydronaphthalenes; Transfection

2002
Influence of melatonin on chicken lymphocytes in vitro: involvement of membrane receptors.
    Neuro endocrinology letters, 2002, Volume: 23 Suppl 1

    Topics: Animals; Antioxidants; Cell Division; Cell Membrane; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Lymphocytes; Male; Melatonin; Phytohemagglutinins; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Signal Transduction; Spleen; Tryptamines

2002
First cloning and functional characterization of a melatonin receptor in fish brain: a novel one?
    Journal of pineal research, 2002, Volume: 32, Issue:2

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Brain; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Cystic Fibrosis Transmembrane Conductance Regulator; Melatonin; Molecular Sequence Data; Phylogeny; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Recombinant Proteins; RNA, Messenger; Sequence Homology, Amino Acid; Superior Colliculi; Tetrahydronaphthalenes

2002
Melatonin participates in the control of testosterone secretion from rat testis: an overview of our experience.
    Annals of the New York Academy of Sciences, 2002, Volume: 966

    Topics: 17-alpha-Hydroxyprogesterone; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Androstenedione; Animals; Calcium Signaling; Cells, Cultured; Colforsin; Cyclic AMP; Gene Expression Regulation; Gonadotropin-Releasing Hormone; GTP-Binding Proteins; Leydig Cells; Luteinizing Hormone; Male; Melatonin; Neuroimmunomodulation; Pertussis Toxin; Prolactin; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Second Messenger Systems; Testosterone; Virulence Factors, Bordetella

2002
Receptor (MT(1)) mediated influence of melatonin on cAMP concentration and insulin secretion of rat insulinoma cells INS-1.
    Journal of pineal research, 2002, Volume: 33, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Biological Transport; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Melatonin; Pancreatic Neoplasms; Phosphodiesterase Inhibitors; Polymerase Chain Reaction; Probenecid; Rats; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Signal Transduction; Tryptamines; Tumor Cells, Cultured

2002
Melatonin inhibits insulin secretion and decreases PKA levels without interfering with glucose metabolism in rat pancreatic islets.
    Journal of pineal research, 2002, Volume: 33, Issue:3

    Topics: Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Melatonin; Protein Kinase C; Protein Subunits; Rats

2002
Effects of subchronic and chronic melatonin treatment on somatostatin binding and its effects on adenylyl cyclase activity in the rat frontoparietal cortex.
    Journal of pineal research, 2002, Volume: 33, Issue:4

    Topics: Adenylyl Cyclases; Animals; Colforsin; Frontal Lobe; Guanylyl Imidodiphosphate; Imidazoles; Melatonin; Parietal Lobe; Rats; Rats, Wistar; Receptors, Somatostatin; Somatostatin

2002
Evidence for the biosynthesis of a prolactin-releasing factor from the ovine pars tuberalis, which is distinct from thyrotropin-releasing hormone.
    Journal of neuroendocrinology, 2002, Volume: 14, Issue:12

    Topics: Animals; Base Sequence; Cells, Cultured; Chromatography, High Pressure Liquid; Colforsin; Cycloheximide; DNA Primers; Immune Sera; In Situ Hybridization; Melatonin; Pituitary Gland, Anterior; Radioimmunoassay; Sheep; Spectrometry, Mass, Electrospray Ionization; Thyrotropin-Releasing Hormone

2002
Heterocyclic aminopyrrolidine derivatives as melatoninergic agents.
    Bioorganic & medicinal chemistry letters, 2003, Dec-15, Volume: 13, Issue:24

    Topics: 3T3 Cells; Aminoquinolines; Animals; Cloning, Molecular; Colforsin; Cyclic AMP; Heterocyclic Compounds; Humans; Kinetics; Ligands; Melatonin; Mice; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Recombinant Proteins; Structure-Activity Relationship

2003
MT-1 melatonin receptor expression increases the antiproliferative effect of melatonin on S-91 murine melanoma cells.
    Journal of pineal research, 2004, Volume: 36, Issue:3

    Topics: Animals; Antineoplastic Agents; Binding Sites; Catalase; Cell Division; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Glutathione Peroxidase; GTP-Binding Protein alpha Subunits, Gi-Go; Male; Melanoma; Melatonin; Mice; Mice, Inbred DBA; Receptor, Melatonin, MT1; Signal Transduction; Transfection; Tumor Cells, Cultured

2004
Melatonin signaling dysfunction in adolescent idiopathic scoliosis.
    Spine, 2004, Aug-15, Volume: 29, Issue:16

    Topics: Adenylyl Cyclases; Adolescent; Cells, Cultured; Colforsin; Cyclic AMP; Female; Guanylyl Imidodiphosphate; Humans; Immunoenzyme Techniques; Male; Melatonin; Osteoblasts; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Scoliosis; Signal Transduction

2004
Intracellular second messengers involved in melatonin signal transduction in chicken splenocytes in vitro.
    Journal of pineal research, 2004, Volume: 37, Issue:3

    Topics: Animals; Cell Proliferation; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Inositol 1,4,5-Trisphosphate; Male; Melatonin; Receptor, Melatonin, MT2; Receptors, Melatonin; Second Messenger Systems; Signal Transduction; Spleen; Tetrahydronaphthalenes; Tryptamines

2004
Knock-down of RGS4 and beta tubulin in CHO cells expressing the human MT1 melatonin receptor prevents melatonin-induced receptor desensitization.
    Life sciences, 2004, Oct-15, Volume: 75, Issue:22

    Topics: Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cycloheximide; GTP-Binding Protein alpha Subunits; Humans; Melatonin; Receptor, Melatonin, MT1; Reverse Transcriptase Polymerase Chain Reaction; RGS Proteins; RNA, Messenger; Tubulin

2004
Melatonin enhances leptin expression by rat adipocytes in the presence of insulin.
    American journal of physiology. Endocrinology and metabolism, 2005, Volume: 288, Issue:4

    Topics: Adipocytes; Animals; Colforsin; Dexamethasone; Dose-Response Relationship, Drug; Drug Interactions; Gene Expression; Glucocorticoids; Inhibitory Concentration 50; Insulin; Leptin; Male; Melatonin; Pertussis Toxin; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Rats; Rats, Wistar; Receptor, Insulin; Receptor, Melatonin, MT1; Reverse Transcriptase Polymerase Chain Reaction; RNA; Tryptamines

2005
Melatonin-induced neuropeptide release from isolated locust corpora cardiaca.
    Peptides, 2005, Volume: 26, Issue:1

    Topics: Animals; Chromatography, High Pressure Liquid; Colforsin; Female; Locusta migratoria; Male; Melatonin; Neuropeptides; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2005
Dopamine receptor activation in bovine pinealocyte via a cAMP-dependent transcription pathway.
    Journal of pineal research, 2005, Volume: 38, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acyltransferases; Animals; Benzazepines; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Melatonin; Phosphorylation; Pineal Gland; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Transcription, Genetic

2005
The human MT1 melatonin receptor stimulates cAMP production in the human neuroblastoma cell line SH-SY5Y cells via a calcium-calmodulin signal transduction pathway.
    Journal of neuroendocrinology, 2005, Volume: 17, Issue:3

    Topics: Calcium-Calmodulin-Dependent Protein Kinases; Colforsin; Cyclic AMP; Enzyme Activators; GTP-Binding Proteins; Humans; Melatonin; Neuroblastoma; Neurons; Receptor, Melatonin, MT1; Signal Transduction; Transfection; Tumor Cells, Cultured

2005
17Beta-estradiol modulates hMT1 melatonin receptor function.
    Neuroendocrinology, 2005, Volume: 81, Issue:2

    Topics: Analysis of Variance; Animals; Blotting, Northern; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Estradiol; Estrogen Receptor alpha; Estrogen Receptor beta; Gene Expression Regulation; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Iodine Isotopes; Melatonin; Protein Binding; Radioligand Assay; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfur Isotopes; Time Factors

2005
Rhythmic expression of adenylyl cyclase VI contributes to the differential regulation of serotonin N-acetyltransferase by bradykinin in rat pineal glands.
    The Journal of biological chemistry, 2005, Nov-18, Volume: 280, Issue:46

    Topics: Adenylyl Cyclases; Animals; Arylalkylamine N-Acetyltransferase; Blotting, Northern; Bradykinin; Calcium; Chelating Agents; Circadian Rhythm; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Inhibitors; Estrenes; Fluorescent Dyes; Fura-2; Gene Expression Regulation, Enzymologic; Immunoblotting; Inositol 1,4,5-Trisphosphate; Ionomycin; Ionophores; Isoproterenol; Male; Melatonin; Norepinephrine; Pertussis Toxin; Phosphodiesterase Inhibitors; Pineal Gland; Protein Isoforms; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA; RNA, Messenger; Signal Transduction; Superior Cervical Ganglion; Time Factors; Transcriptional Activation; Type C Phospholipases

2005
The avian pineal gland.
    Chronobiology international, 2006, Volume: 23, Issue:1-2

    Topics: Animals; Biological Clocks; Chickens; Circadian Rhythm; Colforsin; Female; Light; Male; Melatonin; Photoperiod; Pineal Gland; Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide; Signal Transduction

2006
Melatonin modulates acid/base transport in human pancreatic carcinoma cells.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2006, Volume: 18, Issue:1-3

    Topics: Acids; Antiporters; Bicarbonates; Biological Transport; Cell Line, Tumor; Colforsin; Cyclic AMP; Gene Expression; Humans; Hydrogen-Ion Concentration; Melatonin; Models, Biological; Pancreatic Neoplasms; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Symporters

2006
Modulation of melatonin receptors and G-protein function by microtubules.
    Journal of pineal research, 2006, Volume: 41, Issue:4

    Topics: Animals; Cell Shape; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Heterotrimeric GTP-Binding Proteins; Humans; Melatonin; Microtubules; Protein Kinase C; Receptor, Melatonin, MT1; Rolipram

2006
Molecular determinants of melatonin signaling dysfunction in adolescent idiopathic scoliosis.
    Clinical orthopaedics and related research, 2007, Volume: 462

    Topics: Adenylyl Cyclases; Adolescent; Adult; Cells, Cultured; Child; Child, Preschool; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Combinations; Female; Humans; Male; Melatonin; Osteoblasts; Protein Kinase C-delta; Receptor, Melatonin, MT2; Receptors for Activated C Kinase; Receptors, Cell Surface; Scoliosis; Signal Transduction

2007
Involvement of the cGMP pathway in mediating the insulin-inhibitory effect of melatonin in pancreatic beta-cells.
    Journal of pineal research, 2008, Volume: 45, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Cell Line, Tumor; Colforsin; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 2; Cyclic Nucleotide-Gated Cation Channels; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Glucose; Guanylate Cyclase; Insulin; Insulin Secretion; Insulin-Secreting Cells; Insulinoma; Melatonin; Pineal Gland; Rats; Rats, Wistar; Receptor, Melatonin, MT2; Signal Transduction; Tetrahydronaphthalenes; Tryptamines

2008
Sympathetic nervous system modulates the ocular hypotensive action of MT2-melatonin receptors in normotensive rabbits.
    Journal of pineal research, 2008, Volume: 45, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Administration, Topical; Adrenergic beta-Agonists; Albuterol; Animals; Aqueous Humor; Colforsin; Dose-Response Relationship, Drug; Intraocular Pressure; Isoindoles; Melatonin; Ocular Hypertension; Okadaic Acid; Rabbits; Receptor, Melatonin, MT2; Sympathectomy, Chemical; Sympathetic Nervous System; Terbutaline

2008
Melatonin receptor-mediated protection against myocardial ischaemia/reperfusion injury: role of its anti-adrenergic actions.
    Journal of pineal research, 2008, Volume: 45, Issue:4

    Topics: Adrenergic Antagonists; Animals; Colforsin; Cyclic AMP; Guanylate Cyclase; Heart; Indoles; Isoproterenol; Male; Maleimides; Melatonin; Myocardial Infarction; Myocardial Reperfusion Injury; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oxadiazoles; p38 Mitogen-Activated Protein Kinases; Propranolol; Protein Kinase C; Quinoxalines; Rats; Rats, Wistar; Receptors, Melatonin; Tryptamines

2008
The Galphai and Galphaq proteins mediate the effects of melatonin on steroid/thyroid hormone receptor transcriptional activity and breast cancer cell proliferation.
    Journal of pineal research, 2008, Volume: 45, Issue:4

    Topics: Blotting, Western; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Colforsin; Cyclic AMP; Cyclic GMP; Estrogens; Female; Gene Expression Regulation; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Immunoprecipitation; Luciferases; Melatonin; Phosphorus Radioisotopes; Radioimmunoassay; Receptor, Melatonin, MT1; Receptors, Estrogen; Receptors, Retinoic Acid; Receptors, Thyroid Hormone; Retinoic Acid Receptor alpha; Transcription, Genetic; Transfection

2008
An unexpected effect of 5-MCA-NAT in chick retinal development.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 2009, Volume: 27, Issue:6

    Topics: Aging; Animals; Binding Sites; Chick Embryo; Chickens; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Melatonin; Neurogenesis; Neurons; Organ Culture Techniques; Organogenesis; Quinone Reductases; Receptors, G-Protein-Coupled; Receptors, Melatonin; Retina; Second Messenger Systems; Tryptamines; Up-Regulation

2009
Transcripts of calcium/calmodulin-dependent kinases are changed after forskolin- or IBMX-induced insulin secretion due to melatonin treatment of rat insulinoma beta-cells (INS-1).
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 2009, Volume: 41, Issue:11

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line, Tumor; Colforsin; Gene Expression Regulation, Developmental; Humans; Insulin; Insulin Secretion; Insulin-Secreting Cells; Insulinoma; Islets of Langerhans; Melatonin; Rats; Rats, Wistar

2009
Hypothalamic gonadotropin-releasing hormone receptor activation stimulates oxytocin release from the rat hypothalamo-neurohypophysial system while melatonin inhibits this process.
    Brain research bulletin, 2010, Jan-15, Volume: 81, Issue:1

    Topics: Animals; Colforsin; Cyclic AMP; Gonadotropin-Releasing Hormone; Hypothalamo-Hypophyseal System; Hypothalamus; In Vitro Techniques; Male; Melatonin; Neurons; Oxytocin; Rats; Rats, Wistar; Receptors, LHRH; Signal Transduction

2010
Expression of functional melatonin MT(1) receptors in equine luteal cells: in vitro effects of melatonin on progesterone secretion.
    Reproduction, fertility, and development, 2011, Volume: 23, Issue:3

    Topics: Animals; Blotting, Western; Cholesterol Side-Chain Cleavage Enzyme; Chorionic Gonadotropin; Colforsin; Female; Horses; Luteal Cells; Melatonin; Ovarian Follicle; Progesterone; Receptor, Melatonin, MT1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Statistics, Nonparametric; Tryptamines

2011
Phosphorylation of cyclic AMP-response element-binding protein (CREB) is influenced by melatonin treatment in pancreatic rat insulinoma β-cells (INS-1).
    Journal of pineal research, 2012, Volume: 53, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Cell Line, Tumor; Colforsin; Cyclic AMP Response Element-Binding Protein; Dose-Response Relationship, Drug; Fluorescent Antibody Technique; Humans; Insulin-Secreting Cells; Insulinoma; Melatonin; Microscopy, Confocal; Pancreatic Neoplasms; Phosphorylation; Rats; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Signal Transduction; Tetrahydronaphthalenes; Time Factors; Transfection; Tryptamines

2012
2-Arachidonoyl glycerol sensitizes the pars distalis and enhances forskolin-stimulated prolactin secretion in Syrian hamsters.
    Chronobiology international, 2014, Volume: 31, Issue:3

    Topics: Animals; Arachidonic Acids; Cells, Cultured; Circadian Rhythm; Colforsin; Cricetinae; Endocannabinoids; Glycerides; Male; Melatonin; Photoperiod; Pituitary Gland; Prolactin

2014
Forskolin-stimulated vasopressin and oxytocin release from the rat hypothalamo-neurohypophysial system in vitro is inhibited by melatonin.
    Endokrynologia Polska, 2014, Volume: 65, Issue:2

    Topics: Animals; Colforsin; Cyclic AMP; Hypothalamo-Hypophyseal System; In Vitro Techniques; Male; Melatonin; Oxytocin; Pituitary Gland; Rats; Rats, Wistar; Vasopressins

2014
In vitro comparison of duration of action of melatonin agonists on melatonin MT1 receptor: possible link between duration of action and dissociation rate from receptor.
    European journal of pharmacology, 2015, Jun-15, Volume: 757

    Topics: Animals; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Extracellular Signal-Regulated MAP Kinases; Humans; Kinetics; Melatonin; Phosphorylation; Rats; Receptor, Melatonin, MT1

2015
The role of the cAMP/PKA signalling pathway in the inhibitory influence of melatonin on oxytocin and vasopressin secretion from the rat hypothalamo-neurohypophysial system.
    Endokrynologia Polska, 2018, Volume: 69, Issue:5

    Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Hypothalamo-Hypophyseal System; Male; Melatonin; Oxytocin; Rats; Rats, Wistar; Signal Transduction; Vasopressins

2018
Cryptochrome deficiency enhances transcription but reduces protein levels of pineal Aanat
    Journal of molecular endocrinology, 2018, 10-15, Volume: 61, Issue:4

    Topics: Animals; Blotting, Western; Circadian Rhythm; Colforsin; Cryptochromes; Cyclic AMP; Melatonin; Mice; Period Circadian Proteins; Pineal Gland; Transcription, Genetic

2018
Melatonin Signaling Pathways Implicated in Metabolic Processes in Human Granulosa Cells (KGN).
    International journal of molecular sciences, 2022, Mar-10, Volume: 23, Issue:6

    Topics: Colforsin; Female; Follicular Atresia; Granulosa Cells; Humans; Melatonin; Signal Transduction

2022
Melatonin inhibits muscular-mucosal stretch-sensitive bladder afferents via the MT2 receptors.
    Scientific reports, 2022, 10-21, Volume: 12, Issue:1

    Topics: Animals; Colforsin; Guinea Pigs; Melatonin; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Urinary Bladder

2022
Effects of cyclic adenosine monophosphate modulating agents during oocyte pre-maturation and the role of melatonin on in vitro maturation of bovine cumulus-oocyte complexes.
    Animal reproduction science, 2023, Volume: 257

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Monophosphate; Animals; Cattle; Colforsin; Cumulus Cells; Cyclic AMP; Female; In Vitro Oocyte Maturation Techniques; Melatonin; Natriuretic Peptide, C-Type; Oocytes; RNA, Messenger; Superoxide Dismutase

2023