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melarsomine dihydrochloride and diminazene aceturate

melarsomine dihydrochloride has been researched along with diminazene aceturate in 15 studies

Compound Research Comparison

Studies
(melarsomine dihydrochloride)
Trials
(melarsomine dihydrochloride)
Recent Studies (post-2010)
(melarsomine dihydrochloride)
Studies
(diminazene aceturate)
Trials
(diminazene aceturate)
Recent Studies (post-2010) (diminazene aceturate)
5336903
533656216194

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (53.33)18.2507
2000's3 (20.00)29.6817
2010's4 (26.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Al-Salabi, MI; Ali, JA; de Koning, HP; El-Sabbagh, N; Ho, W; Ibrahim, HM; Koomen, GJ; Rodenko, B; Teka, IA; Wanner, MJ1
Holmes, PH; Jennings, FW; Osman, AS1
Adams, JH; Hunter, CA; Jennings, FW; Kennedy, PG; Murray, M1
Jennings, FW1
Huang, D; Huang, YT; Liang, JX; Lun, ZR; Min, ZP; Yang, XF1
Baltz, T; Giroud, C; Zhang, ZQ2
Baltz, T; Barrett, MP; Denise, H; Giroud, C; Zhang, ZQ1
Scott, AG; Tait, A; Turner, CM1
Martin, RJ; Ross, CA; Suswam, EA; Taylor, DW1
Martin, RJ; Ross, CA; Suswam, EA1
Aliyu, MM; Ibrahim, UI; Mbaya, AW; Nwosu, CO; Taiwo, VO1
Alemu, T; Claes, F; Feseha, G; Fikru, R; Goddeeris, BM; Hagos, A; Yacob, HT; Yilkal, K1
Kumshe, HA; Mbaya, AW; Nwosu, CO1
Birhanu, H; Büscher, P; Kidane, W; Mekonnen, G; Mohammed, EF; Nesibu, A; Van Reet, N; Yohannes, H1

Trials

2 trial(s) available for melarsomine dihydrochloride and diminazene aceturate

ArticleYear
Effects of melarsamine hydrochloride (Cymelarsan) and diminazene aceturate (Berenil) on the pathology of experimental Trypanosoma brucei infection in red fronted gazelles (Gazella rufifrons).
    Veterinary parasitology, 2009, Jul-07, Volume: 163, Issue:1-2

    Topics: Animals; Antelopes; Arsenicals; Diminazene; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2009
Efficacy of Cymelarsan and Diminasan against Trypanosoma equiperdum infections in mice and horses.
    Veterinary parasitology, 2010, Aug-04, Volume: 171, Issue:3-4

    Topics: Animals; Arsenicals; Diminazene; Female; Horse Diseases; Horses; Mice; Parasitemia; Time Factors; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2010

Other Studies

13 other study(ies) available for melarsomine dihydrochloride and diminazene aceturate

ArticleYear
Synthesis of marine-derived 3-alkylpyridinium alkaloids with potent antiprotozoal activity.
    ACS medicinal chemistry letters, 2011, Dec-08, Volume: 2, Issue:12

    Topics:

2011
The rapid development of drug-resistance by Trypanosoma evansi in immunosuppressed mice.
    Acta tropica, 1992, Volume: 50, Issue:3

    Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Immunosuppression Therapy; Mice; Phenanthridines; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

1992
Subcurative chemotherapy and fatal post-treatment reactive encephalopathies in African trypanosomiasis.
    Lancet (London, England), 1992, Apr-18, Volume: 339, Issue:8799

    Topics: Adolescent; Adult; Animals; Arsenicals; Brain; Brain Diseases; Child; Child, Preschool; Diminazene; Female; Humans; Male; Mice; Nitroimidazoles; Polymerase Chain Reaction; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1992
Chemotherapy of CNS-trypanosomiasis: the combined use of diminazene aceturate or pentamidine with DL-alpha-difluoromethylornithine (DFMO).
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1992, Volume: 43, Issue:2

    Topics: Animals; Arsenicals; Central Nervous System Diseases; Diminazene; Drug Administration Schedule; Drug Therapy, Combination; Eflornithine; Female; Mice; Pentamidine; Treatment Outcome; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1992
Cymelarsan in the treatment of buffaloes naturally infected with Trypanosoma evansi in south China.
    Acta tropica, 1991, Volume: 49, Issue:3

    Topics: Animals; Arsenicals; Buffaloes; Diminazene; Female; Injections, Intramuscular; Male; Muscles; Necrosis; Recurrence; Skin; Trypanocidal Agents; Trypanosomiasis

1991
In vivo and in vitro sensitivity of Trypanosoma evansi and T. equiperdum to diminazene, suramin, MelCy, quinapyramine and isometamidium.
    Acta tropica, 1991, Volume: 50, Issue:2

    Topics: Animals; Arsenicals; Diminazene; Female; Mice; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

1991
Trypanosoma evansi: in vivo and in vitro determination of trypanocide resistance profiles.
    Experimental parasitology, 1993, Volume: 77, Issue:4

    Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma

1993
A diamidine-resistant Trypanosoma equiperdum clone contains a P2 purine transporter with reduced substrate affinity.
    Molecular and biochemical parasitology, 1995, Volume: 73, Issue:1-2

    Topics: Adenosine; Animals; Arsenicals; Biological Transport, Active; Carrier Proteins; Diminazene; Drug Resistance; Kinetics; Pentamidine; Receptors, Purinergic P2; Trypanocidal Agents; Trypanosoma

1995
Trypanosoma brucei: lack of cross-resistance to melarsoprol in vitro by cymelarsan-resistant parasites.
    Experimental parasitology, 1997, Volume: 86, Issue:3

    Topics: Adenine; Adenosine; Animals; Arsenicals; Diminazene; Dose-Response Relationship, Drug; Drug Resistance; Enzyme Inhibitors; Female; Inosine; Melarsoprol; Mice; Pentamidine; Trypanocidal Agents; Trypanosoma brucei brucei

1997
Changes in properties of adenosine transporters in Trypanosoma evansi and modes of selection of resistance to the melaminophenyl arsenical drug, Mel Cy.
    Veterinary parasitology, 2001, Dec-13, Volume: 102, Issue:3

    Topics: Adenine; Adenosine; Animals; Arsenicals; Biological Transport; Biomarkers; Carrier Proteins; Diminazene; Dose-Response Relationship, Drug; Drug Resistance; Inosine; Membrane Transport Proteins; Nucleoside Transport Proteins; Parasitic Sensitivity Tests; Trypanocidal Agents; Trypanosoma

2001
Changes in adenosine transport associated with melaminophenyl arsenical (Mel CY) resistance in Trypanosoma evansi: down-regulation and affinity changes of the P2 transporter.
    Parasitology, 2003, Volume: 127, Issue:Pt 6

    Topics: Adenine; Adenosine; Animals; Arsenicals; Diminazene; Down-Regulation; Drug Resistance; Inosine; Kinetics; Nucleoside Transport Proteins; Trypanocidal Agents; Trypanosoma

2003
Genital lesions in male red fronted gazelles (Gazella rufifrons) experimentally infected with Trypanosoma brucei and the effect of melarsamine hydrochloride (Cymelarsan®) and diminazene aceturate (Berenil®) in its treatment.
    Theriogenology, 2011, Sep-01, Volume: 76, Issue:4

    Topics: Animals; Antelopes; Arsenicals; Body Temperature; Diminazene; Genital Diseases, Male; Hematocrit; Histocytochemistry; Male; Parasitemia; Semen; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2011
Isometamidium chloride and homidium chloride fail to cure mice infected with Ethiopian Trypanosoma evansi type A and B.
    PLoS neglected tropical diseases, 2018, Volume: 12, Issue:9

    Topics: Animals; Arsenicals; Diminazene; Disease Models, Animal; Ethiopia; Female; Injections; Mice; Phenanthridines; Recurrence; Treatment Outcome; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2018