melarsomine dihydrochloride has been researched along with arsenic in 48 studies
Studies (melarsomine dihydrochloride) | Trials (melarsomine dihydrochloride) | Recent Studies (post-2010) (melarsomine dihydrochloride) | Studies (arsenic) | Trials (arsenic) | Recent Studies (post-2010) (arsenic) |
---|---|---|---|---|---|
53 | 3 | 6 | 27,806 | 280 | 13,049 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (2.08) | 18.7374 |
1990's | 32 (66.67) | 18.2507 |
2000's | 7 (14.58) | 29.6817 |
2010's | 8 (16.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Kaminsky, R; Ngeranwa, J; Zweygarth, E | 1 |
Holmes, PH; Jennings, FW; Osman, AS | 1 |
Kamar, K; Mutugi, M; Njogu, AR; Otsyula, M | 1 |
Adams, JH; Hunter, CA; Jennings, FW; Kennedy, PG; Murray, M | 1 |
Munyua, WK; Mutugi, MW; Njogu, AR; Olaho-Mukani, W; Otsyula, M | 1 |
Jennings, FW | 3 |
Huang, D; Huang, YT; Liang, JX; Lun, ZR; Min, ZP; Yang, XF | 1 |
Baltz, T; Giroud, C; Zhang, ZQ | 2 |
Kaminsky, R; Zweygarth, E | 1 |
Abebe, S; Kassa, B; Zelleke, D | 1 |
Hashimoto, A; Syakalima, M; Yasuda, J | 1 |
Brun, R; Jenni, L; Kaminsky, R; Pospichal, H | 1 |
Abdel-Rahman, AY; Abdoon, AM; Musa, MM; Nasir, BT; Salim, YI; Shommein, AM | 1 |
Boid, R; Jones, TW; Luckins, AG; Partoutomo, S; Payne, RC; Sukanto, IP | 1 |
Kinabo, LD | 1 |
Kaminsky, R; Moloo, SK; Zweygarth, E | 1 |
Jones, TW; Partoutomo, S; Payne, RC; Sukanto, IP | 1 |
Nantulya, VM | 1 |
Berger, BJ; Fairlamb, AH | 1 |
Biswas, RK; Hunter, AG | 1 |
Cunningham, ML; Fairlamb, AH; Zvelebil, MJ | 1 |
Barns, AM; Ross, CA; Sutherland, DV | 1 |
Baltz, T; Barrett, MP; Denise, H; Giroud, C; Zhang, ZQ | 1 |
Scott, AG; Tait, A; Turner, CM | 2 |
Maribei, JM; Nyang'ao, JM; Olaho-Mukani, W; Omuse, JK | 1 |
Barns, AM; Ross, CA | 1 |
Angus, SD; Aslam, N; Turner, CM | 1 |
Atouguia, JM; Jennings, FW; Murray, M | 1 |
Baltz, T; Barrett, MP; Denise, H; Giroud, C | 1 |
Martin, RJ; Ross, CA; Suswam, EA; Taylor, DW | 1 |
Barrett, MP; Brun, R; Burchmore, RJ; de Koning, HP; Enyaru, JC; Geiser, F; Kaminsky, R; Mäser, P; Matovu, E; Seebeck, T; Stewart, ML; Wallace, LJ | 1 |
Martin, RJ; Ross, CA; Suswam, EA | 1 |
Corbera, JA; Doreste, F; Gutierrez, C; Juste, MC; Morales, I | 1 |
Douce, G; Foucher, AL; McIntosh, A; Tait, A; Turner, CM; Wastling, J | 1 |
Bayou, K; Corbera, JA; Gutierrez, C; van Gool, F | 1 |
Aliyu, MM; Ibrahim, UI; Mbaya, AW; Nwosu, CO; Taiwo, VO | 1 |
Alberola, J; Alonso, I; Arroyo, R; Bosch, I; Caballero, C; Gutierrez, C; Jimenez, V; Sirvent, J; Tamarit, A; Zagalá, G | 1 |
Arafa, RK; Boykin, DW; Brun, R; Gillingwater, K; Ismail, MA; Kumar, A; Stephens, CE; Tidwell, RR | 1 |
Alemu, T; Claes, F; Feseha, G; Fikru, R; Goddeeris, BM; Hagos, A; Yacob, HT; Yilkal, K | 1 |
Githua, M; Hassanali, A; Keriko, J; Murilla, G; Ndungu, M; Nyagah, G | 1 |
Kumshe, HA; Mbaya, AW; Nwosu, CO | 1 |
González-Martín, M; Gutiérrez, C; Tamarit, A; Tejedor-Junco, MT | 1 |
Birhanu, H; Büscher, P; Kidane, W; Mekonnen, G; Mohammed, EF; Nesibu, A; Van Reet, N; Yohannes, H | 1 |
Ashenafi, H; Bekana, M; Daba, M; Demissie, T; Duchateau, L; Geldhof, P; Goddeeris, B; Govaere, J; Tola, A; Van Brantegem, L; Van Soom, A; Vercauteren, G; Yasine, A | 1 |
2 review(s) available for melarsomine dihydrochloride and arsenic
Article | Year |
---|---|
Pharmacology of existing drugs for animal trypanosomiasis.
Topics: Animals; Arsenicals; Diminazene; Ethidium; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosomiasis, African | 1993 |
Combination chemotherapy of CNS trypanosomiasis.
Topics: Arsenicals; Central Nervous System Diseases; Drug Therapy, Combination; Humans; Melarsoprol; Nitroimidazoles; Trypanocidal Agents; Trypanosomiasis, African | 1993 |
3 trial(s) available for melarsomine dihydrochloride and arsenic
Article | Year |
---|---|
Preliminary efficacy trial of Cymelarsan, a novel trypanocide, in camels naturally infected with Trypanosoma evansi in Kenya.
Topics: Animals; Arsenicals; Camelus; Dose-Response Relationship, Drug; Injections, Subcutaneous; Kenya; Suramin; Trypanocidal Agents; Trypanosomiasis | 1992 |
Effects of melarsamine hydrochloride (Cymelarsan) and diminazene aceturate (Berenil) on the pathology of experimental Trypanosoma brucei infection in red fronted gazelles (Gazella rufifrons).
Topics: Animals; Antelopes; Arsenicals; Diminazene; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 2009 |
Efficacy of Cymelarsan and Diminasan against Trypanosoma equiperdum infections in mice and horses.
Topics: Animals; Arsenicals; Diminazene; Female; Horse Diseases; Horses; Mice; Parasitemia; Time Factors; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 2010 |
43 other study(ies) available for melarsomine dihydrochloride and arsenic
Article | Year |
---|---|
Preliminary observations on the efficacy of mel Cy (Cymelarsan) in domestic animals infected with stocks of Trypanosoma brucei brucei and T.b. evansi.
Topics: Animals; Arsenicals; Goat Diseases; Goats; Swine; Swine Diseases; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1992 |
The rapid development of drug-resistance by Trypanosoma evansi in immunosuppressed mice.
Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Immunosuppression Therapy; Mice; Phenanthridines; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 1992 |
Subcurative chemotherapy and fatal post-treatment reactive encephalopathies in African trypanosomiasis.
Topics: Adolescent; Adult; Animals; Arsenicals; Brain; Brain Diseases; Child; Child, Preschool; Diminazene; Female; Humans; Male; Mice; Nitroimidazoles; Polymerase Chain Reaction; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1992 |
Trypanosomal antigen and antibody levels in field camels following treatment with two trypanocidal drugs.
Topics: Animals; Antibodies, Protozoan; Antigens, Protozoan; Arsenicals; Camelus; Enzyme-Linked Immunosorbent Assay; Quinolinium Compounds; Trypanocidal Agents; Trypanosoma; Trypanosomiasis, African | 1992 |
Chemotherapy of CNS-trypanosomiasis: the combined use of diminazene aceturate or pentamidine with DL-alpha-difluoromethylornithine (DFMO).
Topics: Animals; Arsenicals; Central Nervous System Diseases; Diminazene; Drug Administration Schedule; Drug Therapy, Combination; Eflornithine; Female; Mice; Pentamidine; Treatment Outcome; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1992 |
Cymelarsan in the treatment of buffaloes naturally infected with Trypanosoma evansi in south China.
Topics: Animals; Arsenicals; Buffaloes; Diminazene; Female; Injections, Intramuscular; Male; Muscles; Necrosis; Recurrence; Skin; Trypanocidal Agents; Trypanosomiasis | 1991 |
In vivo and in vitro sensitivity of Trypanosoma evansi and T. equiperdum to diminazene, suramin, MelCy, quinapyramine and isometamidium.
Topics: Animals; Arsenicals; Diminazene; Female; Mice; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 1991 |
Chemotherapy of CNS-trypanosomiasis: combination chemotherapy with a 5-nitroimidazole (MK 436), an arsenical (Cymelarsan) and suramin.
Topics: Animals; Arsenicals; Brain Diseases; Disease Models, Animal; Drug Therapy, Combination; Female; Mice; Nitroimidazoles; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1991 |
Evaluation of an arsenical compound (RM 110, mel Cy, Cymelarsan) against susceptible and drug-resistant Trypanosoma brucei brucei and T.b. evansi.
Topics: Animals; Arsenicals; Drug Resistance; Female; Humans; Male; Mice; Molecular Structure; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1990 |
Efficacy of RM110, a novel trypanocide, in the treatment of Trypanosoma evansi infections in camels.
Topics: Animals; Arsenicals; Body Weight; Camelus; Female; Hematocrit; Male; Mice; Trypanocidal Agents; Trypanosomiasis, African | 1989 |
Preliminary efficacy trial of Cymelarsan in mice artificially infected with Trypanosoma brucei brucei isolated from a dog in Zambia.
Topics: Animals; Arsenicals; Dog Diseases; Dogs; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred Strains; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African; Zambia | 1995 |
Induction of resistance to melarsenoxide cysteamine (Mel Cy) in Trypanosoma brucei brucei.
Topics: Animals; Arsenicals; Cell Line; Drug Resistance; Immunocompromised Host; Mice; Mice, Inbred ICR; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1994 |
Efficacy of Cymelarsan in the treatment of natural chronic Trypanosoma evansi infection in camels in the Sudan.
Topics: Animals; Arsenicals; Camelus; Sudan; Trypanocidal Agents; Trypanosomiasis, African | 1994 |
Efficacy of Cymelarsan in Friesian Holstein calves infected with Trypanosoma evansi.
Topics: Animals; Antibodies, Protozoan; Antigens, Protozoan; Arsenicals; Cattle; Enzyme-Linked Immunosorbent Assay; Indonesia; Injections, Intramuscular; Injections, Subcutaneous; Trypanocidal Agents; Trypanosoma; Trypanosomiasis, Bovine | 1994 |
Trypanosoma simiae: in vitro studies on drug susceptibility.
Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Eflornithine; Parasitology; Quinolinium Compounds; Species Specificity; Suramin; Trypanocidal Agents; Trypanosoma | 1993 |
Efficacy of Cymelarsan treatment of suramin resistant Trypanosoma evansi in cattle.
Topics: Animals; Arsenicals; Cattle; Drug Resistance; Injections, Subcutaneous; Recurrence; Suramin; Treatment Outcome; Trypanocidal Agents; Trypanosomiasis, Bovine | 1994 |
Suratex: a simple latex agglutination antigen test for diagnosis of Trypanosoma evansi infections (surra).
Topics: Animals; Antibodies, Protozoan; Antigens, Protozoan; Arsenicals; Camelus; Disease Models, Animal; Evaluation Studies as Topic; Latex Fixation Tests; Rabbits; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 1994 |
Properties of melarsamine hydrochloride (Cymelarsan) in aqueous solution.
Topics: Arsenicals; Chromatography, High Pressure Liquid; Drug Stability; Solutions; Trypanocidal Agents | 1994 |
Effect of stage of infection with Trypanosoma evansi on Cymelarsan therapy.
Topics: Animals; Arsenicals; Camelus; Cattle; Horse Diseases; Horses; Mice; Rabbits; Trypanocidal Agents; Trypanosomiasis; Trypanosomiasis, Bovine | 1993 |
Mechanism of inhibition of trypanothione reductase and glutathione reductase by trivalent organic arsenicals.
Topics: Animals; Arsenicals; Binding Sites; Binding, Competitive; Crithidia fasciculata; Disulfides; Erythrocytes; Glutathione; Glutathione Reductase; Humans; Kinetics; Models, Molecular; NADH, NADPH Oxidoreductases; NADP; Structure-Activity Relationship; Trypanocidal Agents | 1994 |
Trypanosoma evansi: in vivo and in vitro determination of trypanocide resistance profiles.
Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma | 1993 |
Trypanosoma evansi: measurement of pyruvate production as an indicator of the drug sensitivity of isolates in vitro.
Topics: Animals; Arsenic Poisoning; Arsenicals; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Pyruvates; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma | 1995 |
A diamidine-resistant Trypanosoma equiperdum clone contains a P2 purine transporter with reduced substrate affinity.
Topics: Adenosine; Animals; Arsenicals; Biological Transport, Active; Carrier Proteins; Diminazene; Drug Resistance; Kinetics; Pentamidine; Receptors, Purinergic P2; Trypanocidal Agents; Trypanosoma | 1995 |
Characterisation of cloned lines of Trypanosoma brucei expressing stable resistance to MelCy and suramin.
Topics: Animals; Arsenicals; Biological Assay; Cells, Cultured; Clone Cells; Drug Resistance; Female; Male; Melarsoprol; Mice; Mice, Inbred BALB C; Phenotype; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei | 1996 |
Evaluation of the efficacy of melarsenoxyde cysteamine (Cymelarsan) in treatment of camels experimentally infected with Trypanosoma evansi using antigen trapping enzyme-linked immunosorbent assay.
Topics: Animals; Antibodies, Protozoan; Antigens, Protozoan; Arsenicals; Camelus; Enzyme-Linked Immunosorbent Assay; Mice; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 1995 |
Alteration to one of three adenosine transporters is associated with resistance to cymelarsan in Trypanosoma evansi.
Topics: Adenosine; Animals; Arsenicals; Trypanosoma | 1996 |
Inhibition of growth of Trypanosoma brucei parasites in chronic infections.
Topics: Animals; Arsenicals; Chronic Disease; Disease Models, Animal; Female; Mice; Mice, Inbred BALB C; Parasitemia; Sheep; Species Specificity; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1996 |
The importance of 2,3-dimercaptopropinol (British anti-lewisite, BAL) in the trypanocidal activity of topical melarsoprol.
Topics: Administration, Topical; Animals; Arsenicals; Dimercaprol; Drug Combinations; Female; Gels; Melarsoprol; Mice; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1996 |
Trypanosoma brucei: lack of cross-resistance to melarsoprol in vitro by cymelarsan-resistant parasites.
Topics: Adenine; Adenosine; Animals; Arsenicals; Diminazene; Dose-Response Relationship, Drug; Drug Resistance; Enzyme Inhibitors; Female; Inosine; Melarsoprol; Mice; Pentamidine; Trypanocidal Agents; Trypanosoma brucei brucei | 1997 |
Affinity chromatography using trypanocidal arsenical drugs identifies a specific interaction between glycerol-3-phosphate dehydrogenase from Trypanosoma brucei and Cymelarsan.
Topics: Animals; Arsenicals; Binding Sites; Chromatography, Affinity; Cloning, Molecular; Cross-Linking Reagents; Cysteine; Escherichia coli; Glycerolphosphate Dehydrogenase; Muscles; Peptides; Polymerase Chain Reaction; Rabbits; Recombinant Proteins; Sequence Analysis; Trypanocidal Agents; Trypanosoma brucei brucei | 1999 |
Changes in properties of adenosine transporters in Trypanosoma evansi and modes of selection of resistance to the melaminophenyl arsenical drug, Mel Cy.
Topics: Adenine; Adenosine; Animals; Arsenicals; Biological Transport; Biomarkers; Carrier Proteins; Diminazene; Dose-Response Relationship, Drug; Drug Resistance; Inosine; Membrane Transport Proteins; Nucleoside Transport Proteins; Parasitic Sensitivity Tests; Trypanocidal Agents; Trypanosoma | 2001 |
Mechanisms of arsenical and diamidine uptake and resistance in Trypanosoma brucei.
Topics: Adenine; Adenosine; Animals; Arsenicals; Benzamidines; Cell Death; Cell Division; Diminazene; Drug Resistance; Female; Gene Silencing; Hypoxanthine; Inhibitory Concentration 50; Inosine; Melarsoprol; Mice; Mutation; Nucleoside Transport Proteins; Pentamidine; Stilbamidines; Trypanosoma brucei brucei | 2003 |
Changes in adenosine transport associated with melaminophenyl arsenical (Mel CY) resistance in Trypanosoma evansi: down-regulation and affinity changes of the P2 transporter.
Topics: Adenine; Adenosine; Animals; Arsenicals; Diminazene; Down-Regulation; Drug Resistance; Inosine; Kinetics; Nucleoside Transport Proteins; Trypanocidal Agents; Trypanosoma | 2003 |
An outbreak of abortions and high neonatal mortality associated with Trypanosoma evansi infection in dromedary camels in the Canary Islands.
Topics: Aborted Fetus; Abortion, Veterinary; Animals; Animals, Newborn; Arsenicals; Atlantic Islands; Camelus; Disease Outbreaks; Female; Parasitemia; Pregnancy; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 2005 |
A proteomic analysis of arsenical drug resistance in Trypanosoma brucei.
Topics: Animals; Arsenicals; Drug Resistance; Electrophoresis, Gel, Two-Dimensional; Mass Spectrometry; Proteome; Trypanocidal Agents; Trypanosoma brucei brucei | 2006 |
Use of cymelarsan in goats chronically infected with Trypanosoma evansi.
Topics: Animals; Arsenicals; Chronic Disease; Female; Goats; Trypanocidal Agents; Trypanosomiasis | 2008 |
Trypanosoma evansi infection in mainland Spain.
Topics: Animals; Antibodies, Protozoan; Arsenicals; Camelus; Disease Outbreaks; DNA, Protozoan; Polymerase Chain Reaction; Seroepidemiologic Studies; Spain; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 2010 |
In vitro activity and preliminary toxicity of various diamidine compounds against Trypanosoma evansi.
Topics: Amidines; Animals; Arsenicals; Cells, Cultured; Diminazene; Drug Resistance; Female; Inhibitory Concentration 50; Mice; Pentamidine; Quinolinium Compounds; Rats; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 2010 |
New antitrypanosomal tetranotriterpenoids from Azadirachta indica.
Topics: Arsenicals; Azadirachta; Chromatography; Humans; Limonins; Plant Extracts; Plants, Medicinal; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosomiasis, African | 2010 |
Genital lesions in male red fronted gazelles (Gazella rufifrons) experimentally infected with Trypanosoma brucei and the effect of melarsamine hydrochloride (Cymelarsan®) and diminazene aceturate (Berenil®) in its treatment.
Topics: Animals; Antelopes; Arsenicals; Body Temperature; Diminazene; Genital Diseases, Male; Hematocrit; Histocytochemistry; Male; Parasitemia; Semen; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 2011 |
Control and eventual eradication of Trypanosoma evansi infection in dromedary camels after an episodic outbreak in mainland Spain: an example in a non-endemic area.
Topics: Animals; Antibodies, Protozoan; Arsenicals; Camelus; Disease Outbreaks; Female; Polymerase Chain Reaction; Pregnancy; Spain; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 2014 |
Isometamidium chloride and homidium chloride fail to cure mice infected with Ethiopian Trypanosoma evansi type A and B.
Topics: Animals; Arsenicals; Diminazene; Disease Models, Animal; Ethiopia; Female; Injections; Mice; Phenanthridines; Recurrence; Treatment Outcome; Trypanocidal Agents; Trypanosoma; Trypanosomiasis | 2018 |
Tissue (re)distribution of Trypanosoma equiperdum in venereal infected and blood transfused horses.
Topics: Animals; Arsenicals; Blood Transfusion; Dourine; Horse Diseases; Horses; Male; Mice; Parasitemia; Peripheral Nerves; Polymerase Chain Reaction; Reproductive Tract Infections; Semen; Spine; Trypanocidal Agents; Trypanosoma | 2019 |