melagatran has been researched along with sulpiride in 2 studies
Studies (melagatran) | Trials (melagatran) | Recent Studies (post-2010) (melagatran) | Studies (sulpiride) | Trials (sulpiride) | Recent Studies (post-2010) (sulpiride) |
---|---|---|---|---|---|
185 | 32 | 19 | 4,152 | 427 | 635 |
Protein | Taxonomy | melagatran (IC50) | sulpiride (IC50) |
---|---|---|---|
Carbonic anhydrase 1 | Homo sapiens (human) | 1.2 | |
Carbonic anhydrase 2 | Homo sapiens (human) | 0.04 | |
Alpha-2A adrenergic receptor | Homo sapiens (human) | 2.019 | |
D(2) dopamine receptor | Homo sapiens (human) | 0.0858 | |
D(3) dopamine receptor | Homo sapiens (human) | 0.2651 | |
D(2) dopamine receptor | Rattus norvegicus (Norway rat) | 0.2215 | |
Carbonic anhydrase 4 | Bos taurus (cattle) | 0.62 | |
D(2) dopamine receptor | Canis lupus familiaris (dog) | 0.2 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
2 other study(ies) available for melagatran and sulpiride
Article | Year |
---|---|
Physicochemical determinants of human renal clearance.
Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight | 2009 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |