Page last updated: 2024-09-05

melagatran and nafamostat

melagatran has been researched along with nafamostat in 2 studies

Compound Research Comparison

Studies
(melagatran)
Trials
(melagatran)
Recent Studies (post-2010)
(melagatran)
Studies
(nafamostat)
Trials
(nafamostat)
Recent Studies (post-2010) (nafamostat)
185321964054198

Protein Interaction Comparison

ProteinTaxonomymelagatran (IC50)nafamostat (IC50)
Ubiquitin-like modifier activating enzyme 2Homo sapiens (human)7.47
SUMO1 activating enzyme subunit 1Homo sapiens (human)7.47
ubiquitin-like modifier-activating enzyme 1Homo sapiens (human)14
SUMO-conjugating enzyme UBC9Homo sapiens (human)7.47
ubiquitin-conjugating enzyme E2 NHomo sapiens (human)14
ubiquitin-conjugating enzyme E2 variant 1 isoform aHomo sapiens (human)14
ProthrombinHomo sapiens (human)1.9
Complement C1r subcomponentHomo sapiens (human)0.8
PlasminogenHomo sapiens (human)2.9
Cationic trypsinBos taurus (cattle)0.017
Serine protease hepsinHomo sapiens (human)0.005
Trypsin-1Homo sapiens (human)0.017
Complement C1s subcomponentHomo sapiens (human)0.029
Hepatocyte growth factor activatorHomo sapiens (human)0.15

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Abbenante, G; Fairlie, DP; Leung, D1
Pilgram, O; Steinmetzer, T; Wenzel, BM; Wiedemeyer, SJA1

Reviews

1 review(s) available for melagatran and nafamostat

ArticleYear
Protease inhibitors: current status and future prospects.
    Journal of medicinal chemistry, 2000, Feb-10, Volume: 43, Issue:3

    Topics: Animals; Aspartic Acid Endopeptidases; Cysteine Endopeptidases; Cysteine Proteinase Inhibitors; Humans; Metalloendopeptidases; Models, Molecular; Protease Inhibitors; Serine Endopeptidases; Serine Proteinase Inhibitors

2000

Other Studies

1 other study(ies) available for melagatran and nafamostat

ArticleYear
Fibrinolysis Inhibitors: Potential Drugs for the Treatment and Prevention of Bleeding.
    Journal of medicinal chemistry, 2020, 02-27, Volume: 63, Issue:4

    Topics: Animals; Antifibrinolytic Agents; Catalytic Domain; Crystallography, X-Ray; Fibrinolysin; Fibrinolysis; Hemorrhage; Humans; Ligands; Molecular Structure; Plasminogen; Protein Binding; Protein Domains

2020