Page last updated: 2024-08-23

mefloquine and rifampin

mefloquine has been researched along with rifampin in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (11.11)29.6817
2010's7 (77.78)24.3611
2020's1 (11.11)2.80

Authors

AuthorsStudies
Chibale, K; Franzblau, SG; Gut, J; Little, S; Rosenthal, PJ; Tukulula, M; Wan, B1
Bowornwiriyapan, K; Daengrot, C; Phongpaichit, S; Rukachaisirikul, V; Sakayaroj, J; Tansakul, C; Thongpanchang, T1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Bowornwiriyapan, K; Duangjai, A; Muanprasat, C; Phainuphong, P; Phongpaichit, S; Rukachaisirikul, V; Saithong, S; Sakayaroj, J; Srimaroeng, C1
Delabio, LC; Dutra, JP; Hembecker, M; Kita, DH; Moure, VR; Pereira, GDS; Scheiffer, G; Valdameri, G; Zattoni, IF1
Chaipol, P; Mahatthanatrakul, W; Ridtitid, W; Sunbhanich, M; Wongnawa, M1
Babrak, L; Bermudez, LE; Burrows, G; Chinison, JJJ; Danelishvili, L; Hu, J; Morgun, A; Shulzhenko, N1
Cleary, Y; Johnson, TN; Parrott, N; Reigner, B; Smith, JR; Toovey, S1
Chounna Ndongmo, WP; Enyong, P; Esum, ME; Fombad, FF; Gandjui, NVT; Hoerauf, A; Kien, CA; Layland, LE; Njiokou, F; Njouendou, AJ; Pfarr, K; Ritter, M; Turner, J; Wanji, S1

Reviews

2 review(s) available for mefloquine and rifampin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Targeting breast cancer resistance protein (BCRP/ABCG2): Functional inhibitors and expression modulators.
    European journal of medicinal chemistry, 2022, Jul-05, Volume: 237

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Breast Neoplasms; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Neoplasm Proteins; Neoplastic Stem Cells

2022

Other Studies

7 other study(ies) available for mefloquine and rifampin

ArticleYear
The design, synthesis, in silico ADME profiling, antiplasmodial and antimycobacterial evaluation of new arylamino quinoline derivatives.
    European journal of medicinal chemistry, 2012, Volume: 57

    Topics: Aminoquinolines; Antiprotozoal Agents; Antitubercular Agents; Biological Assay; Blood-Brain Barrier; Computer Simulation; Drug Design; Erythrocytes; Humans; Inhibitory Concentration 50; Mefloquine; Microbial Sensitivity Tests; Models, Biological; Mycobacterium tuberculosis; Plasmodium falciparum; Quinine; Structure-Activity Relationship; Tetrazoles

2012
Eremophilane Sesquiterpenes and Diphenyl Thioethers from the Soil Fungus Penicillium copticola PSU-RSPG138.
    Journal of natural products, 2015, Apr-24, Volume: 78, Issue:4

    Topics: Animals; Antimalarials; Antineoplastic Agents; Biphenyl Compounds; Chlorocebus aethiops; Drug Screening Assays, Antitumor; Humans; Inhibitory Concentration 50; Molecular Structure; Penicillium; Plasmodium falciparum; Sesquiterpenes; Soil Microbiology; Sulfides; Thailand; Vero Cells

2015
Lovastatin Analogues from the Soil-Derived Fungus Aspergillus sclerotiorum PSU-RSPG178.
    Journal of natural products, 2016, 06-24, Volume: 79, Issue:6

    Topics: Animals; Aspergillus; Chlorocebus aethiops; Crystallography, X-Ray; Drug Screening Assays, Antitumor; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Inhibitory Concentration 50; KB Cells; Lovastatin; Microbial Sensitivity Tests; Molecular Conformation; Mycobacterium scrofulaceum; Nuclear Magnetic Resonance, Biomolecular; Plasmodium falciparum; Soil Microbiology; Thailand; Vero Cells

2016
Effect of rifampin on plasma concentrations of mefloquine in healthy volunteers.
    The Journal of pharmacy and pharmacology, 2000, Volume: 52, Issue:10

    Topics: Adult; Analysis of Variance; Antimalarials; Area Under Curve; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Drug Interactions; Enzyme Inhibitors; Humans; Male; Mefloquine; Mixed Function Oxygenases; Rifampin

2000
Mycobacterium tuberculosis Proteome Response to Antituberculosis Compounds Reveals Metabolic "Escape" Pathways That Prolong Bacterial Survival.
    Antimicrobial agents and chemotherapy, 2017, Volume: 61, Issue:7

    Topics: Antitubercular Agents; Diarylquinolines; Fluoroquinolones; Isoniazid; Mefloquine; Moxifloxacin; Mycobacterium tuberculosis; Proteome; Proteomics; Rifampin

2017
Development of a physiologically based pharmacokinetic model for mefloquine and its application alongside a clinical effectiveness model to select an optimal dose for prevention of malaria in young Caucasian children.
    British journal of clinical pharmacology, 2019, Volume: 85, Issue:1

    Topics: Adult; Age Factors; Antimalarials; Child; Child, Preschool; Drug Dosage Calculations; Drug Interactions; Female; Humans; Infant; Ketoconazole; Malaria; Mefloquine; Middle Aged; Models, Biological; Rifampin; Treatment Outcome; White People; Young Adult

2019
In vitro maintenance of Mansonella perstans microfilariae and its relevance for drug screening.
    Experimental parasitology, 2019, Volume: 206

    Topics: Amodiaquine; Animals; Antimalarials; Antinematodal Agents; Area Under Curve; Artesunate; Cattle; Cell Line; Culture Media; Filaricides; Haplorhini; Ivermectin; Mansonella; Mefloquine; Microfilariae; Movement; Rifampin

2019