mefloquine has been researched along with quinacrine in 18 studies
*Quinacrine: An acridine derivative formerly widely used as an antimalarial but superseded by chloroquine in recent years. It has also been used as an anthelmintic and in the treatment of giardiasis and malignant effusions. It is used in cell biological experiments as an inhibitor of phospholipase A2. [MeSH]
*Quinacrine: An acridine derivative formerly widely used as an antimalarial but superseded by chloroquine in recent years. It has also been used as an anthelmintic and in the treatment of giardiasis and malignant effusions. It is used in cell biological experiments as an inhibitor of phospholipase A2. [MeSH]
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (16.67) | 18.7374 |
1990's | 5 (27.78) | 18.2507 |
2000's | 2 (11.11) | 29.6817 |
2010's | 6 (33.33) | 24.3611 |
2020's | 2 (11.11) | 2.80 |
Authors | Studies |
---|---|
Dos Santos, JL; Fernandes, BC; Fernandes, GFDS; Valente, V | 1 |
Bane, CE; Black, C; Butler, K; Caridha, D; Cooper, RA; Dodean, RA; Gaona, H; Gaynor-Ohnstad, L; Huezo, SJ; Kancharla, P; Kelly, JX; Kreishman-Deitrick, M; Leed, SE; Li, Q; Li, Y; Lin, H; Luong, TL; Marcsisin, S; Melendez, V; Nolan, C; Olmeda, R; Potter, B; Pou, S; Rasmussen, SA; Read, L; Riscoe, MK; Roncal, N; Sciotti, RJ; Smilkstein, MJ; Sousa, J; Stephens, MT; Tan, JC; Vesely, B; Vuong, C; Winter, RW; Xie, L; Zeng, Q; Zhang, J; Zhang, P | 1 |
Chellappan, DK; Collet, TA; Dighe, SN; Dua, K; Ekwudu, O; Katavic, PL | 1 |
Bernatchez, JA; Li, J; Li, R; Luan, Y; Siqueira-Neto, JL; Tran, LT | 1 |
Chochillon, C; Favennec, L; Gobert, JG; Magne, D; Meillet, D; Raichvarg, D; Savel, J | 1 |
De Boeck, H; Maguire, PA; Sherman, IW; Zidovetzki, R | 1 |
Atiya, A; De Boeck, H; Sherman, IW; Zidovetzki, R | 1 |
Ferrante, A; Goh, DH | 1 |
Govitrapong, P; Jearnpipatkul, A; Panijpan, B; Wilairat, P; Yuthavong, Y | 1 |
Brault, M; Delling, U; Gros, P; Ruetz, S; Schurr, E | 1 |
Croft, SL; Elueze, EI; Warhurst, DC | 1 |
Weina, PJ | 1 |
Aloisi, GG; Barbafina, A; Canton, M; Dall'Acqua, F; Elisei, F; Facciolo, L; Latterini, L; Viola, G | 1 |
Emerson, LR; Kuchler, K; Skillman, BC; Wirth, DF; Wolfger, H | 1 |
Geng, Y; Klocke, BJ; Kohli, L; Roth, KA | 1 |
Chen, B; Coldham, I; Little, SM; Louth, JC; Thompson, MJ | 1 |
Balasubramanian, A; Bhattacharjee, AK; Kulkarni, AA; Padmanabhan, R; Teramoto, T | 1 |
Bensalem, J; Bryksin, V; Fourrier, C; Hattersley, K; Hein, LK; Sargeant, TJ | 1 |
3 review(s) available for mefloquine and quinacrine
Article | Year |
---|---|
Recent advances in the discovery of small molecules targeting glioblastoma.
Topics: Animals; Central Nervous System Neoplasms; Drug Discovery; Glioblastoma; Humans; Neoplastic Stem Cells | 2019 |
Recent update on anti-dengue drug discovery.
Topics: Animals; Antiviral Agents; Biological Products; Cell Line, Tumor; Dengue Virus; Drug Discovery; Humans; Serine Proteinase Inhibitors; Viral Nonstructural Proteins; Virus Replication | 2019 |
Drugs for the Treatment of Zika Virus Infection.
Topics: Animals; Antiviral Agents; Drug Development; Drug Discovery; Humans; Viral Vaccines; Zika Virus; Zika Virus Infection | 2020 |
15 other study(ies) available for mefloquine and quinacrine
Article | Year |
---|---|
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
Topics: Acridones; Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium; Species Specificity; Structure-Activity Relationship | 2019 |
A new screening assay for antigiardial compounds: effects of various drugs on the adherence of Giardia duodenalis to Caco2 cells.
Topics: Animals; Antiprotozoal Agents; Cell Adhesion; Cell Line; Furazolidone; Giardia; Mefloquine; Metronidazole; Quinacrine | 1992 |
A nuclear magnetic resonance study of the interactions of the antimalarials chloroquine, quinacrine, quinine and mefloquine with lipids extracted from normal human erythrocytes.
Topics: 1,2-Dipalmitoylphosphatidylcholine; Antimalarials; Chloroquine; Deuterium; Erythrocytes; Humans; Magnetic Resonance Spectroscopy; Mefloquine; Membrane Lipids; Phosphatidylethanolamines; Phosphorus Isotopes; Quinacrine; Quinine | 1990 |
A nuclear magnetic resonance study of the interactions of the antimalarials chloroquine, quinacrine, quinine and mefloquine with dipalmitoylphosphatidylcholine bilayers.
Topics: 1,2-Dipalmitoylphosphatidylcholine; Antimalarials; Chloroquine; Lipid Bilayers; Magnetic Resonance Spectroscopy; Mefloquine; Quinacrine; Quinine; Quinolines; Temperature | 1989 |
The effect of anti-malarial drugs on human natural killer cells in vitro.
Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines | 1984 |
Binding of antimalarial drugs to hemozoin from Plasmodium berghei.
Topics: Animals; Antimalarials; Chloroquine; Heme; Hemeproteins; Mefloquine; Methemoglobin; Pigments, Biological; Piperidines; Plasmodium berghei; Protein Binding; Protoporphyrins; Quinacrine; Quinolines; Spectrophotometry | 1980 |
The pfmdr1 gene of Plasmodium falciparum confers cellular resistance to antimalarial drugs in yeast cells.
Topics: Alleles; Animals; Antimalarials; ATP-Binding Cassette Transporters; Dose-Response Relationship, Drug; Drug Resistance; Mefloquine; Mice; Phenanthrenes; Plasmodium falciparum; Polymorphism, Genetic; Protozoan Proteins; Quinacrine; Quinine | 1996 |
Activity of pyronaridine and mepacrine against twelve strains of Plasmodium falciparum in vitro.
Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Mefloquine; Naphthyridines; Plasmodium falciparum; Quinacrine; Quinine | 1996 |
From atabrine in World War II to mefloquine in Somalia: the role of education in preventive medicine.
Topics: Antimalarials; Europe; History, 20th Century; Humans; Malaria; Mefloquine; Military Medicine; Preventive Health Services; Quinacrine; Somalia; United States; Warfare | 1998 |
Photophysical and photobiological behavior of antimalarial drugs in aqueous solutions.
Topics: 3T3 Cells; Animals; Antimalarials; Cell Survival; DNA Damage; Free Radicals; Histidine; Lasers; Mefloquine; Membrane Lipids; Membrane Proteins; Mice; Photobiology; Photochemistry; Photolysis; Quinacrine; Quinine; Spectrometry, Fluorescence; Tryptophan; Ultraviolet Rays | 2004 |
The sensitivities of yeast strains deficient in PDR ABC transporters, to quinoline-ring antimalarial drugs.
Topics: Antimalarials; ATP-Binding Cassette Transporters; Chloroquine; Cycloheximide; Drug Resistance, Multiple, Fungal; Gene Deletion; Genes, Fungal; Mefloquine; Mutation; Quinacrine; Quinidine; Quinine; Saccharomyces cerevisiae; Transcription, Genetic | 2004 |
Chloroquine-induced autophagic vacuole accumulation and cell death in glioma cells is p53 independent.
Topics: Antineoplastic Agents; Autophagy; Blotting, Western; Brain Neoplasms; Cell Line, Tumor; Chloroquine; Glioma; Humans; Immunohistochemistry; Mefloquine; Quinacrine; Tumor Suppressor Protein p53; Vacuoles | 2010 |
2,4-diarylthiazole antiprion compounds as a novel structural class of antimalarial leads.
Topics: Antimalarials; Chloroquine; Mefloquine; Molecular Structure; Plasmodium falciparum; Prions; Quinacrine; Structure-Activity Relationship; Thiazoles | 2011 |
Antiviral activities of selected antimalarials against dengue virus type 2 and Zika virus.
Topics: Amodiaquine; Antimalarials; Antiviral Agents; Autophagy; Computer Simulation; Dengue Virus; Drug Discovery; Humans; Mefloquine; Quinacrine; Replicon; Virus Replication; Zika Virus | 2017 |
Comparison of chloroquine-like molecules for lysosomal inhibition and measurement of autophagic flux in the brain.
Topics: Animals; Autophagy; Brain; Chloroquine; Drug Evaluation, Preclinical; Female; HeLa Cells; Humans; Lysosomes; Macrolides; Male; Mefloquine; Mice, Inbred C57BL; Mice, Transgenic; Microtubule-Associated Proteins; Promazine; Quinacrine; Trifluoperazine | 2021 |