Page last updated: 2024-08-23

mefloquine and artemisinin

mefloquine has been researched along with artemisinin in 124 studies

Research

Studies (124)

TimeframeStudies, this research(%)All Research%
pre-199013 (10.48)18.7374
1990's25 (20.16)18.2507
2000's28 (22.58)29.6817
2010's52 (41.94)24.3611
2020's6 (4.84)2.80

Authors

AuthorsStudies
Bogyo, M; Charman, SA; Fontaine, SD; Gut, J; Katneni, K; Lauterwasser, EM; Li, H; Renslo, AR; Rosenthal, PJ1
Albuquerque, IS; Burojević, J; D'Alessandro, S; Djurković-Djaković, O; Konstantinović, J; Machado, M; Pecic, S; Prudêncio, M; Sciotti, RJ; Šolaja, BA; Srbljanović, J; Štajner, T; Taramelli, D; Terzić, N; Tot, M; Verbić, T; Zlatović, M1
Feng, LS; Gao, C; Hu, YQ; Wu, X; Xu, L; Xu, Z; Zhang, S; Zhao, F1
Chu, XM; Gong, KK; Liang, LL; Liu, W; Sun, KL; Wang, C; Wang, WL1
Baum, J; Bridgford, JL; Charman, SA; Churchyard, A; Crespo, B; Deni, I; Fidock, DA; Gahalawat, S; Gamo, FJ; Laleu, B; Lawong, A; Mittal, N; Mok, S; Niederstrasser, H; Okombo, J; Palmer, MJ; Phillips, MA; Posner, B; Ready, JM; Striepen, J; Winzeler, E; Wittlin, S; Yeo, T; Zhou, A1
Augereau, JM; Benoit-Vical, F; Deraeve, C; Jimenez, T; Mustière, R; Nguyen, M; Ouji, M1
Chu, YH; Shao, BR; Ye, XY2
Than, M; Thwe, Y; Win, K1
Trigg, PI1
Bourdeau, EF; Childs, GE; Milhous, WK; Pang, L; Wimonwattratee, T1
Coulaud, JP; Ngo Van, P1
Newbold, CI; Pasvol, G; Peto, TE1
Arnold, K1
Walter, RD1
Druilhe, P; Gentilini, M; Stahel, E1
Coleman, RE; Do Rosario, VE; Hayes, DO; Hollingdale, MR; Vaughan, JA1
Wagner, WH1
Peters, W1
Li, GD1
Warhurst, DC1
Arnold, K; Guo, XB; Jiang, JB; Kong, YC; Li, GQ1
Arnold, K; Fu, LC; Guo, XB; Jian, HX; Li, GQ1
Chiodini, PL; Ellis, CJ1
Nosten, F; Price, RN1
Chen, PQ; Guo, XB; Li, GQ1
Baric, RS; Bright, P; Handy, J; Peel, SA; Yount, B1
Basco, LK; Le Bras, J2
Holfels, E; Mack, D; McAuley, J; McLeod, R; Milhous, WK1
Alin, MH; Ashton, M; Bjorkman, A; Bwijo, BA; Kihamia, CM; Mtey, GJ; Premji, Z1
Alin, MH; Ashton, M; Björkman, A; Kihamia, CM; Mtey, GJ1
Burgmann, H; Graninger, W; Looareesuwan, S; Vanijanonta, S; Viravan, C; Vorbach, H; Zedwitz-Liebenstein, K1
Heppner, DG; Kawamoto, F; Nguyen, TD; Sookto, P; Trieu, NT; Wimonwattrawatee, T; Wongsrichanalai, C1
Alin, MH1
Abbas, N; Alin, MH; Björkman, A; Bwijo, B; Wernsdorfer, W1
Arnold, K; Dung, NT; Hien, TT; HoaiTam, DT; Hung, NT; Mai, PP; Phung, MQ; Toan, LM; Vinh, NN; VinhChau, NV1
Kremsner, PG; Philipps, J; Radloff, PD; Wernsdorfer, W1
Le Bras, J1
Hien, TT; Nosten, F; White, NJ1
McIntosh, HM; Olliaro, P1
White, N1
Chongsuphajaisiddhi, T; Luxemburger, C; Nosten, F; Phaipun, L; Price, R; Simpson, JA; ter Kuile, F; van Vugt, M; White, NJ1
Duraisingh, MT; Jones, P; Pinder, M; Sambou, I; von Seidlein, L; Warhurst, DC2
Burgmann, H; Chullawichit, S; Daxböck, F; El-Menyawi, I; Graninger, W; Looareesuwan, S; Stoiser, B; Thalhammer, F1
Caruana, SR; Cowman, AF; Kirk, K; Reed, MB; Saliba, KJ1
Duraisingh, MT; Roper, C; Walliker, D; Warhurst, DC1
Bloland, PB; Ettling, M; Meek, S1
Faiz, MA; Kawamoto, F; Laoboonchai, A; Lin, K; Noedl, H; Pang, LW; Wimonwattrawatee, T; Wongsrichanalai, C1
Kollaritsch, H; Krudsood, S; Looareesuwan, S; Noedl, H; Viriyavejakul, P; Wernsdorfer, WH; Wiedermann, G; Wilairatana, P1
Björkman, A; Gupta, S; Thapar, MM; Wernsdorfer, WH1
Alin, H; Ashton, M; Bergqvist, Y; Karlsson, MO; Svensson, US1
Fidock, DA; Sidhu, AB; Verdier-Pinard, D1
Dagan, A; Flescher, E; Gatt, S; Gold, D; Pankova-Kholmyansky, I; Skutelsky, E; Zaslavsky, Z1
Brown, ML; Geyer, JA; Terrell, JC; Trotta, RF1
Egan, J; Hoppe, HC; Meredith, SA; van Schalkwyk, DA; Weber, BW; Wiehart, UI1
Majori, G1
Day, NP; Dondorp, AM; Farrar, JJ; Green, MD; Hien, TT; Johnson, A; Looareesuwan, S; Lynam, AJ; Mayxay, M; McGready, R; Newton, PN; Petit, A; Smithuis, FM; Van Damme, W; White, NJ; Yeung, S1
Adams, B; Elandalloussi, LM; Smith, PJ1
Fidock, DA; Sidhu, AB; Valderramos, SG1
Krishna, S; Woodrow, CJ1
Ashley, E; Aye, KZ; Barends, M; Htet, L; Kyaw, MK; Lindegardh, N; Lwin, S; Phe, O; Singtoroj, T; Smithuis, F; Stepniewska, K; White, NJ1
Fidock, DA; Krishna, S; Sidhu, AB; Uhlemann, AC; Valderramos, JC; Valderramos, SG1
Congpuong, K; Na-Bangchang, K1
Congpuong, K; Rojanawatsirivet, C; Sirichaisinthop, J; Wernsdorfer, G; Wernsdorfer, WH; Woitsch, B1
Mills, A; Socheat, D; Van Damme, W; White, NJ; Yeung, S1
Anova, L; Opsenica, DM; Smith, KS; Smith, PL; Solaja, BA; Terzić, N; Yang, Y1
Brittenham, GM; Kano, S; Krudsood, S; Li, G; Looareesuwan, S; Pengruksa, C; Phophak, N; Tangpukdee, N; Thanachartwet, V; Wilairatana, P1
Chen, X; Hergenrother, PJ; Liu, JO; Posner, GH; Rosenthal, AS; Shapiro, TA; West, DC1
Co, EM; Dennull, RA; Johnson, JD; Reinbold, DD; Waters, NC1
Donegan, S; Garner, P; Olliaro, P; Sinclair, D; Zani, B1
Chavchich, M; Chen, N; Cheng, Q; Gerena, L; Kyle, DE; Peters, J1
Alvarez, G; Blair, S; Piñeros, JG; Ríos, A; Tobón, A1
Alvarez, M; Benoit-Vical, F; Berry, A; Iriart, X; Magnaval, JF; Marchou, B; Menard, S; Naneix-Laroche, V; Soh, PN; Witkowski, B1
Duthaler, U; Keiser, J; Utzinger, J1
Björkman, A; Ferreira, PE; Gil, JP; Ribacke, U; Schmidt, BA; Tichopad, A; Veiga, MI1
Ashley, E; Aung, PP; Imwong, M; Kyaw, MK; Lee, SJ; Myint, NZ; Naing, AL; Nyo, MY; Oo, AP; Phe, O; Smithuis, F; White, NJ; Win, T1
Chen, N; Cheng, Q; Gatton, ML; Kyle, DE; Peters, J; Teuscher, F1
Congpuong, K; Kerschbaumer, G; Sirichaisinthop, J; Wernsdorfer, G; Wernsdorfer, WH; Wiedermann, U1
Congpuong, K; Hüttinger, F; Satimai, W; Wernsdorfer, G; Wernsdorfer, WH; Wiedermann, U1
Moon, DK; Parkin, S; Posner, GH; Siegler, MA; Sullivan, D; Tripathi, A1
Carvalho, LJ; Clemmer, L; Frangos, JA; Martins, YC; Zanini, GM1
Björkman, A; Ferreira, PE; Gil, JP; Jörnhagen, L; Kone, A; Malmberg, M; Nosten, F; Petzold, M; Schmidt, BA; Veiga, MI1
Borges, S; Cravo, P; Creasey, A; Fawcett, R; Hunt, P; Martinelli, A; Modrzynska, K; Rodrigues, L1
Congpuong, K; Sirichaisinthop, J; Treiber, M; Wernsdorfer, G; Wernsdorfer, WH; Wiedermann, U1
Ensom, MH; Wilby, KJ1
Kittikool, D; Sibmooh, N; Srihirun, S; Tangnitipong, S; Thaptimthong, T; Udomsangpetch, R; Unchern, S1
Arango, EM; Carmona-Fonseca, J; Upegui, YA1
Al-Farsi, HM; Al-Hashami, ZS; Al-Qahtani, A; Al-Sheikh, AA; Babiker, HA; Bin Dajem, SM1
Jacobine, AM; Mazzone, JR; Posner, GH; Slack, RD; Sullivan, DJ; Tripathi, AK1
Delacollette, C; Kaewkungwal, J; Khamsiriwatchara, A; Lawpoolsri, S; Potithavoranan, T; Sangvichean, A; Satimai, W; Sawang, S; Singhasivanon, P; Sudathip, P; Vijaykadga, S1
Amaratunga, C; Anderson, JM; Anderson, TJ; Dondorp, AM; Duong, S; Fairhurst, RM; Fay, MP; Jiang, H; Lim, P; Lindegardh, N; Mao, S; Mu, J; Phelps, ES; Song, J; Sreng, S; Stepniewska, K; Su, XZ; Suon, S; White, NJ; Zhou, C1
Garner, P; Gelband, H; Graves, PM3
Ariey, F; Beck, HP; Csajka, C; Decosterd, LA; Duong, S; Genton, B; Guidi, M; Kabanywanyi, AM; Olliaro, P; Staehli Hodel, EM1
Beeson, JG; Goodman, CD; Langer, C; McFadden, GI; Wilson, DW1
Ashley, E; Boel, M; Carrara, VI; Chu, C; Lwin, KM; McGready, R; Nosten, F; Phyo, AP; Proux, S; Rijken, M; Singhasivanon, P; Sriprawat, K; White, N; Wiladphaingern, J1
Alcantara, LM; Ayong, LS; Franco, CH; Franzoi, KD; Freitas-Junior, LH; Kim, J; Lee, S; Moraes, CB1
Cooksey, R; Dahlström, S; Fairhurst, RM; Flegg, JA; Guerin, PJ; Johnson, JD; Le Bras, J; Le Nagard, H; Lim, P; Ménard, D; Mentré, F; Murillo, C; Musset, L; Noedl, H; Nosten, F; Nsobya, SL; Pradines, B; Quashie, NB; Sibley, CH; Sinou, V; Sriprawat, K; Woodrow, CJ1
Dondorp, AM; Faiz, MA; Hien, TT; Mokuolu, OA; Pukrittayakamee, S; White, NJ1
Aubouy, A; Dahlström, S; Deloron, P; Ezinmègnon, S; Faucher, JF; Houzé, P; Houzé, S; Kendjo, E; Le Bras, J; Maïga-Ascofaré, O; Massougbodji, A; Wakpo, A1
Cremers, S; Fidock, DA; Henrich, PP; Kyle, DE; O'Brien, C; Sáenz, FE1
Conyers, RC; Mazzone, JR; Mott, BT; Posner, GH; Siegler, MA; Sullivan, DJ; Tripathi, AK1
Bukirwa, H; Kramer, CV; Nair, S; Sinclair, D; Tharyan, P; Unnikrishnan, B1
Dahlstrom, S; Ferreira, PE; Franzén, O; Gil, JP; Lum, JK; Nosten, F; Osório, NS; Veiga, MI1
Buathong, N; Chanarat, N; Chann, S; Chaorattanakawee, S; Chuor, CM; Gosi, P; Heng, TK; Jacob, C; Kong, N; Kuntawunginn, W; Lanteri, CA; Lin, JT; Lon, C; Plowe, C; Prom, S; Saingam, P; Saunders, DL; Se, Y; Sea, D; Sriwichai, S; Sundrakes, S; Takala-Harrison, S; Tangthongchaiwiriya, K; Teja-Isavadharm, P; Tyner, SD; Yingyuen, K; Yom, Y1
Bouth, DM; Char, MC; Domergue, A; Duru, V; Khim, N; Kim, S; Leang, R; Menard, D; Ringwald, P; Song, L; Tarning, J; Taylor, WR; Witkowski, B1
Akala, HM; Auschwitz, JM; Cheruiyot, AC; Gaona, HW; Hickman, MR; Johnson, JD; Kamau, E; Lee, PJ; Leed, SE; Murthy, T; Okello, CO; Talwar, M; Yeda, RA1
Bhardwaj, J; Goyal, M; Prakash, K; Puri, SK; Siddiqui, AJ; Soni, A1
Maxmen, A1
Cabral, L; Cristiano, ML; Lobo, L; Nogueira, F; Sousa, Bd1
Ackermann, I; Aubin, F; Carn, G; Gesase, S; Lusingu, JPA; Mnkande, E; Mrango, Z; Mtoro, A; Ngocho, JS; Ogutu, B; Onyango, KO; Ouedraogo, A; Sirima, SB; Strub, N; Vanraes, J; Yaro, JB1
Liu, XJ; Peng, HJ; Wei, HX; Xia, J; Zhou, LJ1
Bailey, JA; Barnett, EJ; Brazeau, NF; Chaorattanakawee, S; Gosi, P; Juliano, JJ; Lanteri, CA; Lin, JT; Lon, C; Meshnick, SR; Norris, LD; Parobek, CM; Parr, JB; Saunders, DL; Spring, MD1
Chaijaroenkul, W; Na-Bangchang, K; Phompradit, P1
Cao, P; Dini, S; Fowkes, FJI; McCaw, JM; Price, RN; Simpson, JA; van der Pluijm, RW; Zaloumis, S1
Buffet, P; Chambrion, C; Chartrel, N; Mouri, O; Ndour, PA; Roussel, C; Smith, B; Smith, P; Thellier, M; Wojnarski, M1
Chy, S; Felger, I; Hastings, I; Hodel, EM; Jones, S; Kay, K; Mbituyumuremyi, A; Menard, D; Uwimana, A1
Amaratunga, C; Amato, R; Anvikar, AR; Ashley, E; Baidya, S; Behera, PK; Callery, JJ; Chau, NH; Cheah, PY; Chotivanich, K; Chutasmit, K; Day, NPJ; Dhorda, M; Dondorp, AM; Fairhurst, RM; Faiz, A; Fanello, C; Gantait, K; Ghosh, T; Gonçalves, S; Grobusch, MP; Hanboonkunupakarn, B; Heaton, J; Hien, TT; Hlaing, TM; Hoa, NT; Hoglund, RM; Huy, R; Imwong, M; Jacob, CG; Jittamala, P; Kaewmok, W; Kwiatkowski, DP; Lek, D; Lin, K; Mao, S; Maude, RJ; Mayxay, M; Miotto, O; Mohanty, AK; Mukaka, M; Newton, PN; Onyamboko, M; Oun, S; Pearson, RD; Peto, TJ; Pukrittayakamee, S; Pyae Phyo, A; Runcharern, R; Saelow, C; Satpathi, P; Satpathi, S; Smithuis, F; Sovann, Y; Sreng, S; Suon, S; Tarning, J; Thanh, NV; Thant, M; Thuy-Nhien, NT; Tripura, A; Tripura, R; Ul Islam, A; Valecha, N; van der Pluijm, RW; van Vugt, M; von Seidlein, L; Waithira, N; White, NJ; Winterberg, M; Woodrow, CJ; Yen, S1
Anywar, DA; Auma, MA; Balikagala, B; Emoto, S; Fukuda, N; Hashimoto, M; Hirai, M; Horii, T; Ikeda, M; Kataoka, M; Katuro, OT; Kimura, E; Mita, T; Mori, T; Obwoya, PS; Odongo-Aginya, EI; Ogwang, M; Opio, W; Palacpac, NMQ; Sakurai-Yatsushiro, M; Sekihara, M; Tachibana, SI; Yamauchi, M; Yatsushiro, S1
Barale, JC; Bouillon, A; Chy, S; Eam, R; Kauy, C; Ke, S; Khean, C; Khim, N; Kim, S; Kloeung, N; Kul, C; Leang, R; Mairet-Khedim, M; Ringwald, P; Roesch, C; Srun, S; Witkowski, B1
Chiheb, D; Erhart, A; Guetens, P; Hong, NV; Imamura, H; Kattenberg, JH; Monsieurs, P; Phuc, BQ; Rosanas-Urgell, A; Rovira-Vallbona, E; Xa, NX1

Reviews

21 review(s) available for mefloquine and artemisinin

ArticleYear
Quinoline hybrids and their antiplasmodial and antimalarial activities.
    European journal of medicinal chemistry, 2017, Oct-20, Volume: 139

    Topics: Antimalarials; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines

2017
Triazole derivatives and their antiplasmodial and antimalarial activities.
    European journal of medicinal chemistry, 2019, Mar-15, Volume: 166

    Topics: Animals; Antimalarials; Humans; Parasitic Sensitivity Tests; Plasmodium; Triazoles

2019
The problem of drug resistance in malaria.
    Parasitology, 1985, Volume: 90 ( Pt 4)

    Topics: Africa; Animals; Antimalarials; Artemisinins; Chemical Phenomena; Chemistry; Chloroquine; Clinical Trials as Topic; Dapsone; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance, Microbial; Humans; India; Malaria; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Sesquiterpenes; Sulfadoxine

1985
New drugs and their potential use against drug-resistant malaria.
    Annali dell'Istituto superiore di sanita, 1985, Volume: 21, Issue:3

    Topics: Aminoquinolines; Animals; Antimalarials; Artemisinins; Drug Resistance, Microbial; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Mice; Naphthoquinones; Plasmodium falciparum; Pyrimethamine; Quinolines; Sesquiterpenes; Sulfadoxine

1985
New antimalarials. A risk-benefit analysis.
    Drug safety, 1995, Volume: 12, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; Dose-Response Relationship, Drug; Drug Resistance; Drug Synergism; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Pregnancy; Risk Assessment; Sesquiterpenes

1995
Management of multiple drug-resistant malaria in Viet Nam.
    Annals of the Academy of Medicine, Singapore, 1997, Volume: 26, Issue:5

    Topics: Antimalarials; Artemisinins; Clinical Trials as Topic; Drug Resistance, Multiple; Humans; Malaria; Mefloquine; Sesquiterpenes; Vietnam

1997
Use of artemisinin derivatives for the control of malaria.
    Medecine tropicale : revue du Corps de sante colonial, 1998, Volume: 58, Issue:3 Suppl

    Topics: Antimalarials; Artemisinins; Drug Resistance; Drug Therapy, Combination; Humans; Incidence; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Prospective Studies; Refugees; Risk Factors; Seasons; Sesquiterpenes; Thailand; Treatment Outcome; Vietnam

1998
Treatment of uncomplicated malaria with artemisinin derivatives. A systematic review of randomised controlled trials.
    Medecine tropicale : revue du Corps de sante colonial, 1998, Volume: 58, Issue:3 Suppl

    Topics: Adult; Antimalarials; Artemisinins; Child; Dose-Response Relationship, Drug; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Randomized Controlled Trials as Topic; Research Design; Sesquiterpenes; Time Factors; Treatment Outcome

1998
Combination therapy for malaria in Africa: hype or hope?
    Bulletin of the World Health Organization, 2000, Volume: 78, Issue:12

    Topics: Africa; Antimalarials; Artemisinins; Artesunate; Asia, Southeastern; Chloroquine; Cross-Cultural Comparison; Half-Life; Humans; Insecticide Resistance; Malaria; Mefloquine; Pyrimethamine; Self Medication; Sesquiterpenes; Sulfadoxine; Thailand

2000
[Combined antimalarial therapy using artemisinin].
    Parassitologia, 2004, Volume: 46, Issue:1-2

    Topics: Amodiaquine; Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Chloroquine; Doxycycline; Drug Resistance; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Plasmodium; Pyrimethamine; Quinine; Sesquiterpenes; Sulfadoxine

2004
Antimalarial drugs: recent advances in molecular determinants of resistance and their clinical significance.
    Cellular and molecular life sciences : CMLS, 2006, Volume: 63, Issue:14

    Topics: Africa; Amino Alcohols; Animals; Antimalarials; Artemisinins; Asia, Southeastern; Biological Transport; Calcium-Transporting ATPases; Chloroquine; Drug Resistance; Drug Resistance, Multiple; Drug Therapy, Combination; Gene Amplification; Humans; Malaria, Falciparum; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Models, Biological; Multidrug Resistance-Associated Proteins; Mutation; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Quinine; Sesquiterpenes

2006
Current malaria status and distribution of drug resistance in East and Southeast Asia with special focus to Thailand.
    The Tohoku journal of experimental medicine, 2007, Volume: 211, Issue:2

    Topics: Age Factors; Animals; Antimalarials; Artemisinins; Asia, Southeastern; Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine; Plasmodium; Quinine; Sesquiterpenes; Sex Factors; Sulfadoxine

2007
Artemisinin-based combination therapy for treating uncomplicated malaria.
    The Cochrane database of systematic reviews, 2009, Jul-08, Issue:3

    Topics: Antimalarials; Artemisinins; Artesunate; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Fluorenes; Humans; Lumefantrine; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Parasitemia; Pyrimethamine; Quinolines; Randomized Controlled Trials as Topic; Sulfadoxine

2009
Update on the diagnosis and treatment of food-borne trematode infections.
    Current opinion in infectious diseases, 2010, Volume: 23, Issue:5

    Topics: Animals; Anthelmintics; Artemisinins; Benzimidazoles; Foodborne Diseases; Humans; Immunoassay; Mefloquine; Molecular Diagnostic Techniques; Phenylenediamines; Praziquantel; Sensitivity and Specificity; Trematode Infections; Triclabendazole

2010
Pharmacokinetics of antimalarials in pregnancy: a systematic review.
    Clinical pharmacokinetics, 2011, Nov-01, Volume: 50, Issue:11

    Topics: Anti-Bacterial Agents; Antimalarials; Artemisinins; Atovaquone; Chloroquine; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria; Mefloquine; Pregnancy; Pregnancy Complications, Parasitic; Proguanil; Pyrimethamine; Quinine; Sulfadoxine

2011
Primaquine for reducing Plasmodium falciparum transmission.
    The Cochrane database of systematic reviews, 2012, Sep-12, Issue:9

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2012
Malaria.
    Lancet (London, England), 2014, Feb-22, Volume: 383, Issue:9918

    Topics: Africa South of the Sahara; Amodiaquine; Animals; Anopheles; Antimalarials; Artemisinins; Artesunate; Asia, Southeastern; Chloroquine; Drug Administration Schedule; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Female; Humans; Insecticide-Treated Bednets; Insecticides; Malaria; Malaria Vaccines; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Pregnancy; Pregnancy Complications, Infectious; Primary Prevention; Pyrimethamine; Quinine; Quinolines; Seasons; Sulfadoxine

2014
Artesunate plus pyronaridine for treating uncomplicated Plasmodium falciparum malaria.
    The Cochrane database of systematic reviews, 2014, Mar-04, Issue:3

    Topics: Adult; Antimalarials; Artemisinins; Artesunate; Child; Drug Therapy, Combination; Ethanolamines; Fluorenes; Humans; Liver; Lumefantrine; Malaria, Falciparum; Mefloquine; Naphthyridines; Randomized Controlled Trials as Topic

2014
Primaquine or other 8-aminoquinoline for reducing P. falciparum transmission.
    The Cochrane database of systematic reviews, 2014, Jun-30, Issue:6

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2014
Primaquine or other 8-aminoquinoline for reducing Plasmodium falciparum transmission.
    The Cochrane database of systematic reviews, 2015, Feb-19, Issue:2

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2015
Risk of drug resistance in Plasmodium falciparum malaria therapy-a systematic review and meta-analysis.
    Parasitology research, 2017, Volume: 116, Issue:2

    Topics: Amodiaquine; Antimalarials; Artemisinins; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinolines; Risk; Sulfadoxine

2017

Trials

17 trial(s) available for mefloquine and artemisinin

ArticleYear
Comparison of combinations of parenteral artemisinin derivatives plus oral mefloquine with intravenous quinine plus oral tetracycline for treating cerebral malaria.
    Bulletin of the World Health Organization, 1992, Volume: 70, Issue:6

    Topics: Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Artesunate; Humans; Malaria, Cerebral; Mefloquine; Middle Aged; Prospective Studies; Quinine; Sesquiterpenes; Tetracycline

1992
The problem of drug resistance in malaria.
    Parasitology, 1985, Volume: 90 ( Pt 4)

    Topics: Africa; Animals; Antimalarials; Artemisinins; Chemical Phenomena; Chemistry; Chloroquine; Clinical Trials as Topic; Dapsone; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance, Microbial; Humans; India; Malaria; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Sesquiterpenes; Sulfadoxine

1985
Antimalarial activity of mefloquine and qinghaosu.
    Lancet (London, England), 1982, Aug-07, Volume: 2, Issue:8293

    Topics: Administration, Oral; Adolescent; Adult; Antimalarials; Artemisinins; Child; China; Female; Humans; Injections, Intramuscular; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Quinolines; Sesquiterpenes; Time Factors

1982
Randomised comparative study of mefloquine, qinghaosu, and pyrimethamine-sulfadoxine in patients with falciparum malaria.
    Lancet (London, England), 1984, Dec-15, Volume: 2, Issue:8416

    Topics: Adolescent; Adult; Antimalarials; Artemisinins; Child; China; Clinical Trials as Topic; Drug Combinations; Drug Therapy, Combination; Female; Humans; Malaria; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Prospective Studies; Pyrimethamine; Quinolines; Random Allocation; Sesquiterpenes; Sulfadoxine; Sulfanilamides

1984
[The infectivity of gametocytes of Plasmodium falciparum from patients treated with artemisinine].
    Zhonghua yi xue za zhi, 1994, Volume: 74, Issue:4

    Topics: Animals; Anopheles; Antimalarials; Artemisinins; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Sesquiterpenes

1994
Efficacy of oral and intravenous artesunate in male Tanzanian adults with Plasmodium falciparum malaria and in vitro susceptibility to artemisinin, chloroquine, and mefloquine.
    The American journal of tropical medicine and hygiene, 1995, Volume: 53, Issue:6

    Topics: Administration, Oral; Adolescent; Adult; Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Drugs, Chinese Herbal; Erythrocytes; Humans; Injections, Intravenous; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Parasitemia; Plasmodium falciparum; Recurrence; Sesquiterpenes; Tanzania

1995
Clinical efficacy and pharmacokinetics of artemisinin monotherapy and in combination with mefloquine in patients with falciparum malaria.
    British journal of clinical pharmacology, 1996, Volume: 41, Issue:6

    Topics: Administration, Oral; Adult; Animals; Antimalarials; Artemisinins; Drug Therapy, Combination; Female; Half-Life; Humans; Malaria, Falciparum; Male; Mefloquine; Sesquiterpenes

1996
In vivo-in vitro model for the assessment of clinically relevant antimalarial cross-resistance.
    The American journal of tropical medicine and hygiene, 2001, Volume: 65, Issue:6

    Topics: Adult; Animals; Antimalarials; Artemisinins; Chloroquine; Cross Reactions; Drug Resistance; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Models, Biological; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine; Recurrence; Sesquiterpenes

2001
Population pharmacokinetic and pharmacodynamic modelling of artemisinin and mefloquine enantiomers in patients with falciparum malaria.
    European journal of clinical pharmacology, 2002, Volume: 58, Issue:5

    Topics: Adolescent; Adult; Antimalarials; Artemisinins; Drug Interactions; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Middle Aged; Models, Biological; Sesquiterpenes; Stereoisomerism; Structure-Activity Relationship

2002
Efficacy and effectiveness of dihydroartemisinin-piperaquine versus artesunate-mefloquine in falciparum malaria: an open-label randomised comparison.
    Lancet (London, England), 2006, 06-24, Volume: 367, Issue:9528

    Topics: Adolescent; Animals; Antimalarials; Artemisinins; Artesunate; Child; Child, Preschool; Drug Therapy, Combination; Female; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Myanmar; Plasmodium falciparum; Quinolines; Recurrence; Sesquiterpenes; Treatment Outcome

2006
Efficacy of Artequick versus artesunate-mefloquine in the treatment of acute uncomplicated falciparum malaria in Thailand.
    The Southeast Asian journal of tropical medicine and public health, 2008, Volume: 39, Issue:1

    Topics: Acute Disease; Adolescent; Adult; Antimalarials; Artemisinins; Artesunate; Drug Combinations; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Primaquine; Prospective Studies; Quinolines; Thailand; Treatment Outcome

2008
Effectiveness of five artemisinin combination regimens with or without primaquine in uncomplicated falciparum malaria: an open-label randomised trial.
    The Lancet. Infectious diseases, 2010, Volume: 10, Issue:10

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antimalarials; Artemisinins; Child; Child, Preschool; Drug Therapy, Combination; Female; Humans; Infant; Malaria, Falciparum; Malaria, Vivax; Male; Mefloquine; Middle Aged; Myanmar; Plasmodium falciparum; Primaquine; Treatment Outcome; Young Adult

2010
Efficacy of different primaquine-based antimalarial regimens against Plasmodium falciparum gametocytemia.
    Acta tropica, 2012, Volume: 122, Issue:2

    Topics: Adolescent; Adult; Aged; Amodiaquine; Antimalarials; Artemisinins; Artesunate; Child; Child, Preschool; Colombia; Drug Combinations; Drug Therapy, Combination; Female; Follow-Up Studies; Germ Cells; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Parasitemia; Plasmodium falciparum; Primaquine; Pyrimethamine; Sulfadoxine; Treatment Outcome; Young Adult

2012
Artemisinin-resistant Plasmodium falciparum in Pursat province, western Cambodia: a parasite clearance rate study.
    The Lancet. Infectious diseases, 2012, Volume: 12, Issue:11

    Topics: Adolescent; Adult; Animals; Antimalarials; Artemisinins; Cambodia; Drug Resistance; Female; Genotype; Glucosephosphate Dehydrogenase; Humans; Malaria, Falciparum; Male; Mefloquine; Microsatellite Repeats; Plasmodium falciparum; Treatment Outcome; Young Adult

2012
Evidence of Plasmodium falciparum Malaria Multidrug Resistance to Artemisinin and Piperaquine in Western Cambodia: Dihydroartemisinin-Piperaquine Open-Label Multicenter Clinical Assessment.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:8

    Topics: Adolescent; Adult; Antigens, Bacterial; Antigens, Surface; Antimalarials; Artemisinins; Cambodia; Child; Child, Preschool; Drug Resistance, Multiple; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Quinolines; Treatment Failure; Young Adult

2015
Comparison of artesunate-mefloquine and artemether-lumefantrine fixed-dose combinations for treatment of uncomplicated Plasmodium falciparum malaria in children younger than 5 years in sub-Saharan Africa: a randomised, multicentre, phase 4 trial.
    The Lancet. Infectious diseases, 2016, Volume: 16, Issue:10

    Topics: Africa South of the Sahara; Antimalarials; Artemether; Artemisinins; Artesunate; Child, Preschool; Ethanolamines; Female; Fluorenes; Humans; Infant; Lumefantrine; Malaria, Falciparum; Male; Mefloquine; Patient Safety; Polymerase Chain Reaction

2016
Triple artemisinin-based combination therapies versus artemisinin-based combination therapies for uncomplicated Plasmodium falciparum malaria: a multicentre, open-label, randomised clinical trial.
    Lancet (London, England), 2020, 04-25, Volume: 395, Issue:10233

    Topics: Adolescent; Adult; Amodiaquine; Anthraquinones; Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Drug Resistance; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Plasmodium falciparum; Polymerase Chain Reaction; Quinolines; Treatment Outcome; Young Adult

2020

Other Studies

87 other study(ies) available for mefloquine and artemisinin

ArticleYear
Trioxolane-Mediated Delivery of Mefloquine Limits Brain Exposure in a Mouse Model of Malaria.
    ACS medicinal chemistry letters, 2015, Nov-12, Volume: 6, Issue:11

    Topics:

2015
Reinvestigating Old Pharmacophores: Are 4-Aminoquinolines and Tetraoxanes Potential Two-Stage Antimalarials?
    Journal of medicinal chemistry, 2016, Jan-14, Volume: 59, Issue:1

    Topics: Aminoquinolines; Animals; Antimalarials; Drug Evaluation, Preclinical; Ether-A-Go-Go Potassium Channels; Hemin; Hepatocytes; Humans; In Vitro Techniques; Liver; Mice; Microsomes, Liver; Parasite Load; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship; Tetraoxanes

2016
Novel Antimalarial Tetrazoles and Amides Active against the Hemoglobin Degradation Pathway in
    Journal of medicinal chemistry, 2021, 03-11, Volume: 64, Issue:5

    Topics: Amides; Antimalarials; Drug Resistance, Microbial; Hemeproteins; Hemoglobins; Hep G2 Cells; Humans; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Small Molecule Libraries; Structure-Activity Relationship; Tetrazoles

2021
Novel molecule combinations and corresponding hybrids targeting artemisinin-resistant Plasmodium falciparum parasites.
    Bioorganic & medicinal chemistry letters, 2021, 05-01, Volume: 39

    Topics: Antimalarials; Artemisinins; Atovaquone; Dose-Response Relationship, Drug; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Triclosan

2021
[The blood schizontocidal effects of pyronaridine, amodiaquine, mefloquine and qinghaosu on mice infected with Plasmodium berghei].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 1992, Volume: 10, Issue:2

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Drug Resistance; Female; Malaria; Male; Mefloquine; Mice; Naphthyridines; Plasmodium berghei; Sesquiterpenes

1992
Comparison of effects of pyronaridine, amodiaquine, mefloquine and qinghaosu on rodent malaria.
    The Southeast Asian journal of tropical medicine and public health, 1992, Volume: 23, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Drug Administration Schedule; Drug Evaluation, Preclinical; Drug Resistance; Female; Malaria; Male; Mefloquine; Mice; Naphthyridines; Plasmodium berghei; Sesquiterpenes

1992
Drug use and design in the nineties.
    Acta Leidensia, 1991, Volume: 60, Issue:1

    Topics: Aminoquinolines; Amodiaquine; Antimalarials; Artemisinins; Calcium Channel Blockers; Chloroquine; Humans; Malaria; Mefloquine; Naphthoquinones; Phenanthrenes; Primaquine; Quinine; Sesquiterpenes; Sulfadoxine

1991
In vitro and clinical correlates of mefloquine resistance of Plasmodium falciparum in eastern Thailand.
    The American journal of tropical medicine and hygiene, 1991, Volume: 44, Issue:5

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Butylated Hydroxytoluene; Chloroquine; Drug Resistance; Drugs, Chinese Herbal; Mefloquine; Molecular Structure; Phenanthrenes; Plasmodium falciparum; Pyridines; Pyrimethamine; Quinine; Sesquiterpenes; Thailand

1991
[New antiparasitic drugs].
    Annales de dermatologie et de venereologie, 1988, Volume: 115, Issue:4

    Topics: Amebicides; Anthelmintics; Antifungal Agents; Antimalarials; Artemisinins; Fluconazole; Humans; Itraconazole; Ketoconazole; Mefloquine; Phenanthrenes; Quinolines; Sesquiterpenes; Triazoles

1988
Qinghaosu, mefloquine, and pyrimethamine-sulfadoxine in falciparum malaria.
    Lancet (London, England), 1985, Jan-26, Volume: 1, Issue:8422

    Topics: Antimalarials; Artemisinins; Drug Combinations; Humans; Malaria; Mefloquine; Pyrimethamine; Quinolines; Sesquiterpenes; Sulfadoxine

1985
Qinghaosu, mefloquine, and pyrimethamine-sulfadoxine in falciparum malaria.
    Lancet (London, England), 1985, Mar-23, Volume: 1, Issue:8430

    Topics: Artemisinins; Drug Combinations; Drug Resistance, Microbial; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Pyrimethamine; Quinolines; Sesquiterpenes; Sulfadoxine; Sulfanilamides

1985
Plasmodium falciparum: inhibition of dolichol kinase by mefloquine.
    Experimental parasitology, 1986, Volume: 62, Issue:3

    Topics: Animals; Artemisinins; Cations, Divalent; Chloroquine; Cytidine Triphosphate; Detergents; Dolichols; Egtazic Acid; Erythrocytes; Hydrogen-Ion Concentration; Kinetics; Mefloquine; Microsomes; Nucleotides; Phosphotransferases; Phosphotransferases (Alcohol Group Acceptor); Plasmodium falciparum; Quinolines; Sesquiterpenes; Trifluoperazine

1986
Antagonism of chloroquine with other antimalarials.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1988, Volume: 82, Issue:2

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Chloroquine; Drug Combinations; Drug Interactions; Drug Resistance; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Sesquiterpenes; Sulfadoxine

1988
Effect of mefloquine and artemisinin on the sporogonic cycle of Plasmodium berghei ANKA in Anopheles stephensi mosquitoes.
    Acta Leidensia, 1988, Volume: 57, Issue:1

    Topics: Animals; Anopheles; Antimalarials; Artemisinins; Female; Insect Vectors; Malaria; Mefloquine; Mice; Plasmodium berghei; Quinolines; Sesquiterpenes

1988
[Control of malaria--chemotherapy and immunoprophylaxis. 1. Chemotherapy].
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:1

    Topics: Antimalarials; Artemisinins; Drug Combinations; Drug Resistance; Humans; In Vitro Techniques; Malaria; Mefloquine; Plasmodium; Quinolines; Sesquiterpenes; Vaccination

1986
[Development of a piperaquine-resistant line of Plasmodium berghei K 173 strain].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1985, Volume: 20, Issue:6

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Resistance; Malaria; Male; Mefloquine; Mice; Plasmodium berghei; Quinolines; Sesquiterpenes

1985
The treatment of falciparum malaria.
    The Journal of antimicrobial chemotherapy, 1984, Volume: 13, Issue:4

    Topics: Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Humans; Malaria; Mefloquine; Plasmodium falciparum; Quinidine; Quinine; Quinolines; Sesquiterpenes

1984
A strong association between mefloquine and halofantrine resistance and amplification, overexpression, and mutation in the P-glycoprotein gene homolog (pfmdr) of Plasmodium falciparum in vitro.
    The American journal of tropical medicine and hygiene, 1994, Volume: 51, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Base Sequence; Blotting, Northern; Blotting, Southern; Chloroquine; DNA Primers; DNA, Protozoan; Drug Resistance; Gene Amplification; Gene Expression; Genes, Protozoan; Mefloquine; Molecular Sequence Data; Phenanthrenes; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Quinine; RNA, Messenger; Selection, Genetic; Sequence Homology, Nucleic Acid; Sesquiterpenes

1994
In vitro susceptibility of Cambodian isolates of Plasmodium falciparum to halofantrine, pyronaridine and artemisinin derivatives.
    Annals of tropical medicine and parasitology, 1994, Volume: 88, Issue:2

    Topics: Adult; Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Humans; In Vitro Techniques; Mefloquine; Naphthyridines; Phenanthrenes; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinine; Sesquiterpenes; Triazines

1994
In vitro effects of artemisinin ether, cycloguanil hydrochloride (alone and in combination with sulfadiazine), quinine sulfate, mefloquine, primaquine phosphate, trifluoperazine hydrochloride, and verapamil on Toxoplasma gondii.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:6

    Topics: Animals; Artemisinins; Female; Mefloquine; Mice; Primaquine; Proguanil; Quinine; Sesquiterpenes; Sulfadiazine; Toxoplasma; Triazines; Trifluoperazine; Uracil; Verapamil

1994
In vitro activity of artemisinin derivatives against African isolates and clones of Plasmodium falciparum.
    The American journal of tropical medicine and hygiene, 1993, Volume: 49, Issue:3

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Chloroquine; Drug Resistance; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes

1993
Serum laminin and basic fibroblast growth factor concentrations in patients with complicated Plasmodium falciparum malaria.
    Journal of clinical immunology, 1996, Volume: 16, Issue:5

    Topics: Adolescent; Adult; Aged; Antimalarials; Artemisinins; Artesunate; Fibroblast Growth Factor 2; Humans; Kinetics; Laminin; Malaria, Falciparum; Mefloquine; Middle Aged; Sesquiterpenes

1996
In vitro susceptibility of Plasmodium falciparum isolates in Vietnam to artemisinin derivatives and other antimalarials.
    Acta tropica, 1997, Volume: 63, Issue:2-3

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Mefloquine; Microbial Sensitivity Tests; Plasmodium falciparum; Quinine; Sesquiterpenes; Vietnam

1997
In vitro susceptibility of Tanzanian wild isolates of Plasmodium falciparum to artemisinin, chloroquine, sulfadoxine/pyrimethamine and mefloquine.
    Parasitology, 1997, Volume: 114 ( Pt 6)

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Humans; Mefloquine; Plasmodium falciparum; Pyrimethamine; Sesquiterpenes; Sulfadoxine; Tanzania

1997
Efficacy of artemisinin and mefloquine combinations against Plasmodium falciparum. In vitro simulation of in vivo pharmacokinetics.
    Tropical medicine & international health : TM & IH, 1997, Volume: 2, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Drug Synergism; Mefloquine; Plasmodium falciparum; Sesquiterpenes

1997
Follow-up of the susceptibility of Plasmodium falciparum to antimalarials in Gabon.
    The American journal of tropical medicine and hygiene, 1998, Volume: 58, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Dose-Response Relationship, Drug; Drug Resistance; Follow-Up Studies; Gabon; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Quinine; Sesquiterpenes; Sulfadoxine

1998
In vitro susceptibility of African Plasmodium falciparum isolates to dihydroartemisinin and the risk factors for resistance to qinghaosu.
    Medecine tropicale : revue du Corps de sante colonial, 1998, Volume: 58, Issue:3 Suppl

    Topics: Africa; Animals; Antimalarials; Artemisinins; Chloroquine; Cross Reactions; Drug Evaluation, Preclinical; Drug Resistance; France; Humans; Malaria, Falciparum; Mefloquine; Phenanthrenes; Plasmodium falciparum; Sesquiterpenes; Travel

1998
Antimalarial drug resistance and combination chemotherapy.
    Philosophical transactions of the Royal Society of London. Series B, Biological sciences, 1999, Apr-29, Volume: 354, Issue:1384

    Topics: Animals; Antimalarials; Artemisinins; Atovaquone; Chloroquine; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Naphthoquinones; Plasmodium falciparum; Sesquiterpenes

1999
Risk factors for gametocyte carriage in uncomplicated falciparum malaria.
    The American journal of tropical medicine and hygiene, 1999, Volume: 60, Issue:6

    Topics: Adolescent; Adult; Animals; Antimalarials; Artemisinins; Carrier State; Child; Child, Preschool; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Multivariate Analysis; Parasitemia; Phenanthrenes; Plasmodium falciparum; Prospective Studies; Quinine; Regression Analysis; Risk Factors; Seroepidemiologic Studies; Sesquiterpenes; Thailand

1999
Inoculum effect leads to overestimation of in vitro resistance for artemisinin derivatives and standard antimalarials: a Gambian field study.
    Parasitology, 1999, Volume: 119 ( Pt 5)

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Gambia; Hematocrit; Humans; Malaria, Falciparum; Mefloquine; Parasitemia; Phenanthrenes; Plasmodium falciparum; Quinine; Scintillation Counting; Sensitivity and Specificity; Sesquiterpenes

1999
Serum concentrations of granulocyte-colony stimulating factor in complicated Plasmodium falciparum malaria.
    European cytokine network, 2000, Volume: 11, Issue:1

    Topics: Adolescent; Adult; Animals; Antimalarials; Artemisinins; Artesunate; Calcitonin; Calcitonin Gene-Related Peptide; Chemokine CCL4; Child; Enzyme-Linked Immunosorbent Assay; Erythrocytes; Erythropoietin; Female; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Macrophage Inflammatory Proteins; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Nitrates; Plasmodium falciparum; Protein Precursors; Reference Values; Sesquiterpenes; Stem Cell Factor

2000
Pgh1 modulates sensitivity and resistance to multiple antimalarials in Plasmodium falciparum.
    Nature, 2000, Feb-24, Volume: 403, Issue:6772

    Topics: Amino Acid Substitution; Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; Chloroquine; Cloning, Molecular; Drug Resistance; Mefloquine; Mutation; Phenanthrenes; Plasmodium falciparum; Protozoan Proteins; Quinine; Sesquiterpenes; Verapamil

2000
The tyrosine-86 allele of the pfmdr1 gene of Plasmodium falciparum is associated with increased sensitivity to the anti-malarials mefloquine and artemisinin.
    Molecular and biochemical parasitology, 2000, Apr-30, Volume: 108, Issue:1

    Topics: Alleles; Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Polymerase Chain Reaction; Polymorphism, Genetic; Polymorphism, Restriction Fragment Length; Protozoan Proteins; Sesquiterpenes; Tetrahydrofolate Dehydrogenase; Tyrosine

2000
Increased sensitivity to the antimalarials mefloquine and artemisinin is conferred by mutations in the pfmdr1 gene of Plasmodium falciparum.
    Molecular microbiology, 2000, Volume: 36, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; Cells, Cultured; Humans; Mefloquine; Mutagenesis; Plasmodium falciparum; Protozoan Proteins; Sesquiterpenes

2000
In vitro susceptibility of Plasmodium falciparum isolates from Myanmar to antimalarial drugs.
    The American journal of tropical medicine and hygiene, 2001, Volume: 65, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Sesquiterpenes

2001
In vitro interactions of artemisinin with atovaquone, quinine, and mefloquine against Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2002, Volume: 46, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Atovaquone; Drug Synergism; Humans; Mefloquine; Naphthoquinones; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine; Sesquiterpenes

2002
Chloroquine resistance in Plasmodium falciparum malaria parasites conferred by pfcrt mutations.
    Science (New York, N.Y.), 2002, Oct-04, Volume: 298, Issue:5591

    Topics: Alleles; Amodiaquine; Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; Chloroquine; Cloning, Molecular; Drug Resistance; Genes, Protozoan; Haplotypes; Mefloquine; Membrane Proteins; Membrane Transport Proteins; Parasitic Sensitivity Tests; Phenotype; Plasmodium falciparum; Point Mutation; Protozoan Proteins; Quinine; Sesquiterpenes; Transfection; Verapamil

2002
Ceramide mediates growth inhibition of the Plasmodium falciparum parasite.
    Cellular and molecular life sciences : CMLS, 2003, Volume: 60, Issue:3

    Topics: Animals; Antiprotozoal Agents; Apoptosis; Artemisinins; Ceramides; Glutathione; Growth Inhibitors; Lysophospholipids; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Sesquiterpenes; Sphingomyelin Phosphodiesterase; Sphingosine

2003
Defective DNA repair as a potential mechanism for the rapid development of drug resistance in Plasmodium falciparum.
    Biochemistry, 2004, May-04, Volume: 43, Issue:17

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; DNA Damage; DNA Repair; Drug Resistance; Drug Resistance, Multiple; Humans; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Pyrimethamine; Quinine; Sesquiterpenes; Sulfanilamide; Sulfanilamides; Ultraviolet Rays

2004
Antimalarial quinolines and artemisinin inhibit endocytosis in Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2004, Volume: 48, Issue:7

    Topics: Ammonium Chloride; Animals; Antimalarials; Artemisinins; Biotin; Blotting, Western; Chloroquine; Dextrans; Endocytosis; Fluorescein-5-isothiocyanate; Fluorescent Antibody Technique; Fluorescent Dyes; Hemoglobins; Mefloquine; Microscopy, Electron; Microscopy, Fluorescence; Monensin; Plasmodium falciparum; Quinolones; Sesquiterpenes; Transport Vesicles; Vacuoles

2004
Fake antimalarials in Southeast Asia are a major impediment to malaria control: multinational cross-sectional survey on the prevalence of fake antimalarials.
    Tropical medicine & international health : TM & IH, 2004, Volume: 9, Issue:12

    Topics: Antimalarials; Artemisinins; Artesunate; Asia, Southeastern; Cross-Sectional Studies; Drug Labeling; Fraud; Humans; Malaria; Mefloquine; Self Medication; Sesquiterpenes

2004
ATPase activity of purified plasma membranes and digestive vacuoles from Plasmodium falciparum.
    Molecular and biochemical parasitology, 2005, Volume: 141, Issue:1

    Topics: Adenosine Triphosphatases; Animals; Antimalarials; Artemisinins; Cell Membrane; Chloroquine; Drug Resistance; Mefloquine; Plasmodium falciparum; Quinine; Sesquiterpenes; Subcellular Fractions; Vacuoles

2005
pfmdr1 mutations contribute to quinine resistance and enhance mefloquine and artemisinin sensitivity in Plasmodium falciparum.
    Molecular microbiology, 2005, Volume: 57, Issue:4

    Topics: Alleles; Animals; Antimalarials; Artemisinins; Asparagine; Aspartic Acid; ATP-Binding Cassette Transporters; Drug Resistance; Mefloquine; Phenanthrenes; Plasmodium falciparum; Point Mutation; Protozoan Proteins; Quinine; Sesquiterpenes

2005
Decreasing pfmdr1 copy number in plasmodium falciparum malaria heightens susceptibility to mefloquine, lumefantrine, halofantrine, quinine, and artemisinin.
    The Journal of infectious diseases, 2006, Aug-15, Volume: 194, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; DNA, Protozoan; Drug Resistance, Multiple; Ethanolamines; Fluorenes; Genes, MDR; Inhibitory Concentration 50; Lumefantrine; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Phenanthrenes; Plasmodium falciparum; Polymerase Chain Reaction; Protozoan Proteins; Quinine; Sesquiterpenes

2006
Susceptibility to chloroquine, mefloquine and artemisinin of Plasmodium vivax in northwestern Thailand.
    Wiener klinische Wochenschrift, 2007, Volume: 119, Issue:19-20 Supp

    Topics: Antimalarials; Artemisinins; Chloroquine; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Humans; Lethal Dose 50; Malaria, Vivax; Mefloquine; Plasmodium vivax; Survival Rate; Thailand; Treatment Outcome

2007
Cost of increasing access to artemisinin combination therapy: the Cambodian experience.
    Malaria journal, 2008, May-20, Volume: 7

    Topics: Animals; Antimalarials; Artemisinins; Cambodia; Costs and Cost Analysis; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine

2008
Mixed tetraoxanes containing the acetone subunit as antimalarials.
    Bioorganic & medicinal chemistry, 2008, Jul-15, Volume: 16, Issue:14

    Topics: Acetone; Animals; Antimalarials; Artemisinins; Drug Evaluation, Preclinical; Drug Resistance, Multiple; Mefloquine; Mice; Plasmodium falciparum; Tetraoxanes

2008
Malaria-infected mice are cured by a single oral dose of new dimeric trioxane sulfones which are also selectively and powerfully cytotoxic to cancer cells.
    Journal of medicinal chemistry, 2009, Feb-26, Volume: 52, Issue:4

    Topics: Administration, Oral; Animals; Antimalarials; Antineoplastic Agents; Artemisinins; Cell Line, Tumor; Drug Screening Assays, Antitumor; Drug Stability; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Mice; Sulfones

2009
Assessment of malaria in vitro drug combination screening and mixed-strain infections using the malaria Sybr green I-based fluorescence assay.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:6

    Topics: Animals; Antimalarials; Artemisinins; Benzothiazoles; Chloroquine; Diamines; Drug Combinations; Drug Evaluation, Preclinical; Drug Interactions; Fluorescent Dyes; Hypoxanthine; Mefloquine; Organic Chemicals; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines

2009
Role of pfmdr1 amplification and expression in induction of resistance to artemisinin derivatives in Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:6

    Topics: Alleles; Animals; Antimalarials; Artemisinins; Drug Resistance; Gene Amplification; Gene Dosage; Gene Expression; Genes, Protozoan; Humans; In Vitro Techniques; Malaria, Falciparum; Mefloquine; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; RNA, Messenger; RNA, Protozoan

2010
Dynamics of Plasmodium falciparum parasitemia regarding combined treatment regimens for acute uncomplicated malaria, Antioquia, Colombia.
    The American journal of tropical medicine and hygiene, 2010, Volume: 83, Issue:1

    Topics: Administration, Oral; Animals; Antimalarials; Artemisinins; Artesunate; Clinical Protocols; Colombia; Drug Therapy, Combination; Female; Humans; Malaria; Malaria, Falciparum; Male; Mefloquine; Parasitemia; Patient Compliance; Plasmodium falciparum; Primaquine; Treatment Outcome

2010
pfmdr1 amplification associated with clinical resistance to mefloquine in West Africa: implications for efficacy of artemisinin combination therapies.
    Journal of clinical microbiology, 2010, Volume: 48, Issue:10

    Topics: Adult; Africa, Western; Artemisinins; Drug Resistance; Drug Therapy, Combination; Gene Dosage; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Male; Mefloquine; Multidrug Resistance-Associated Proteins; Treatment Failure

2010
Antimalarial exposure delays Plasmodium falciparum intra-erythrocytic cycle and drives drug transporter genes expression.
    PloS one, 2010, Aug-25, Volume: 5, Issue:8

    Topics: Antimalarials; Artemisinins; Cell Cycle; Drug Therapy, Combination; Erythrocytes; Gene Expression Regulation; Mefloquine; Membrane Transport Proteins; Plasmodium falciparum; Protozoan Proteins; RNA, Messenger

2010
Artemisinin‐induced dormancy in plasmodium falciparum: duration, recovery rates, and implications in treatment failure.
    The Journal of infectious diseases, 2010, Nov-01, Volume: 202, Issue:9

    Topics: Antimalarials; Artemisinins; Mefloquine; Microbial Viability; Plasmodium falciparum; Time Factors

2010
Synergism between mefloquine and artemisinin and its enhancement by retinol in Plasmodium falciparum in vitro.
    Wiener klinische Wochenschrift, 2010, Volume: 122 Suppl 3

    Topics: Antimalarials; Artemisinins; Dose-Response Relationship, Drug; Drug Synergism; Lethal Dose 50; Mefloquine; Plasmodium falciparum; Thailand; Vitamin A

2010
Sensitivity to artemisinin, mefloquine and quinine of Plasmodium falciparum in northwestern Thailand.
    Wiener klinische Wochenschrift, 2010, Volume: 122 Suppl 3

    Topics: Antimalarials; Artemisinins; Dose-Response Relationship, Drug; Lethal Dose 50; Mefloquine; Plasmodium falciparum; Quinine; Thailand

2010
A single, low, oral dose of a 5-carbon-linked trioxane dimer orthoester plus mefloquine cures malaria-infected mice.
    Bioorganic & medicinal chemistry letters, 2011, May-01, Volume: 21, Issue:9

    Topics: Administration, Oral; Animals; Antimalarials; Artemisinins; Crystallography, X-Ray; Drug Therapy, Combination; Esters; Heterocyclic Compounds; Heterocyclic Compounds, 4 or More Rings; Malaria; Mefloquine; Mice; Molecular Structure; Plasmodium berghei

2011
Artemether and artesunate show the highest efficacies in rescuing mice with late-stage cerebral malaria and rapidly decrease leukocyte accumulation in the brain.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:4

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Brain; Leukocytes; Malaria, Cerebral; Mefloquine; Mice; Parasitemia; Plasmodium berghei; Quinine

2011
Novel polymorphisms in Plasmodium falciparum ABC transporter genes are associated with major ACT antimalarial drug resistance.
    PloS one, 2011, Volume: 6, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; ATP-Binding Cassette Transporters; Base Sequence; Drug Resistance; Ethanolamines; Fluorenes; Gene Frequency; Genotype; Haplotypes; Humans; Inhibitory Concentration 50; Lumefantrine; Malaria, Falciparum; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins

2011
Genomewide scan reveals amplification of mdr1 as a common denominator of resistance to mefloquine, lumefantrine, and artemisinin in Plasmodium chabaudi malaria parasites.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:10

    Topics: Antimalarials; Artemisinins; Base Sequence; Chromosome Mapping; Drug Resistance, Multiple; Ethanolamines; Fluorenes; Genetic Linkage; Genome, Protozoan; Lumefantrine; Malaria; Mefloquine; Multidrug Resistance-Associated Proteins; Plasmodium chabaudi; Sequence Analysis, DNA

2011
Sensitivity of Plasmodium vivax to chloroquine, mefloquine, artemisinin and atovaquone in north-western Thailand.
    Wiener klinische Wochenschrift, 2011, Volume: 123 Suppl 1

    Topics: Animals; Antimalarials; Artemisinins; Atovaquone; Chloroquine; Dose-Response Relationship, Drug; Lethal Dose 50; Mefloquine; Plasmodium vivax; Thailand

2011
Extracellular heme enhances the antimalarial activity of artemisinin.
    Biological & pharmaceutical bulletin, 2012, Volume: 35, Issue:1

    Topics: Antimalarials; Antioxidants; Artemisia; Artemisinins; Chloroquine; Cholesterol, LDL; Fluorescence; Heme; Hemin; Humans; Lipid Peroxidation; Mefloquine; Oxidants; Oxidation-Reduction; Plasmodium falciparum; Quinine; Tryptophan; Vitamin E

2012
Distribution of drug resistance genotypes in Plasmodium falciparum in an area of limited parasite diversity in Saudi Arabia.
    The American journal of tropical medicine and hygiene, 2012, Volume: 86, Issue:5

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antimalarials; Artemisinins; Child; Child, Preschool; Chloroquine; Drug Combinations; Drug Resistance; Female; Genotype; Humans; Infant; Male; Mefloquine; Membrane Transport Proteins; Middle Aged; Multidrug Resistance-Associated Proteins; Mutation; Phenanthrenes; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Pyrimethamine; Saudi Arabia; Sulfadoxine; Tetrahydrofolate Dehydrogenase; Young Adult

2012
Malaria-infected mice live until at least day 30 after a new artemisinin-derived thioacetal thiocarbonate combined with mefloquine are administered together in a single, low, oral dose.
    Journal of medicinal chemistry, 2012, Sep-13, Volume: 55, Issue:17

    Topics: Acetals; Administration, Oral; Animals; Antimalarials; Artemisinins; Magnetic Resonance Spectroscopy; Malaria; Mefloquine; Mice; Mice, Inbred C57BL; Spectrometry, Mass, Fast Atom Bombardment

2012
Artemisinin resistance containment project in Thailand. II: Responses to mefloquine-artesunate combination therapy among falciparum malaria patients in provinces bordering Cambodia.
    Malaria journal, 2012, Aug-28, Volume: 11

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antimalarials; Artemisinins; Artesunate; Cambodia; Child; Child, Preschool; Drug Resistance; Drug Therapy, Combination; Epidemiological Monitoring; Female; Humans; Infant; Infant, Newborn; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Thailand; Treatment Outcome; Young Adult

2012
Effect of single nucleotide polymorphisms in cytochrome P450 isoenzyme and N-acetyltransferase 2 genes on the metabolism of artemisinin-based combination therapies in malaria patients from Cambodia and Tanzania.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:2

    Topics: Alleles; Antimalarials; Artemether, Lumefantrine Drug Combination; Artemisinins; Artesunate; Arylamine N-Acetyltransferase; Base Sequence; Cambodia; Cytochrome P-450 Enzyme System; Drug Combinations; Ethanolamines; Fluorenes; Gene Frequency; Humans; Isoenzymes; Malaria; Mefloquine; Pharmacogenetics; Polymorphism, Single Nucleotide; Quinolines; Sequence Analysis, DNA; Tanzania

2013
Defining the timing of action of antimalarial drugs against Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:3

    Topics: Amodiaquine; Antimalarials; Artemisinins; Artesunate; Chloroquine; Erythrocytes; Flow Cytometry; High-Throughput Screening Assays; Hydroxamic Acids; Inhibitory Concentration 50; Mefloquine; Merozoites; Plasmodium falciparum; Quinine; Quinolines; Schizonts; Time Factors

2013
Malaria burden and artemisinin resistance in the mobile and migrant population on the Thai-Myanmar border, 1999-2011: an observational study.
    PLoS medicine, 2013, Volume: 10, Issue:3

    Topics: Antimalarials; Artemisinins; Artesunate; Climate; Community Health Workers; Cross-Sectional Studies; Drug Resistance; Female; Geography; Hospitalization; Humans; Malaria; Mefloquine; Myanmar; Plasmodium falciparum; Plasmodium vivax; Pregnancy; Pregnancy Complications, Parasitic; Prevalence; Rain; Reproducibility of Results; Temperature; Thailand; Transients and Migrants

2013
Chemosensitization potential of P-glycoprotein inhibitors in malaria parasites.
    Experimental parasitology, 2013, Volume: 134, Issue:2

    Topics: Antimalarials; Artemisinins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzamides; Boron Compounds; Chloroquine; Chlorpheniramine; Dibenzocycloheptenes; Drug Interactions; Drug Resistance, Multiple; Erythrocytes; Fluorescent Dyes; Gefitinib; Humans; Imatinib Mesylate; Mefloquine; Piperazines; Plasmodium falciparum; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Quinolines

2013
High-throughput analysis of antimalarial susceptibility data by the WorldWide Antimalarial Resistance Network (WWARN) in vitro analysis and reporting tool.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:7

    Topics: Amodiaquine; Antimalarials; Artemisinins; Automation, Laboratory; Chloroquine; Drug Resistance; Drug Therapy, Combination; High-Throughput Screening Assays; Internet; Malaria, Falciparum; Mefloquine; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinine

2013
Plasmodium falciparum Polymorphisms associated with ex vivo drug susceptibility and clinical effectiveness of artemisinin-based combination therapies in Benin.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:1

    Topics: Amodiaquine; Antimalarials; Artemisinins; Drug Combinations; Ethanolamines; Female; Fluorenes; Humans; Inhibitory Concentration 50; Lumefantrine; Male; Mefloquine; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Pyrimethamine; Quinine; Sulfadoxine

2014
Evidence for pyronaridine as a highly effective partner drug for treatment of artemisinin-resistant malaria in a rodent model.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Artesunate; Drug Combinations; Drug Resistance; Female; Flow Cytometry; Malaria, Falciparum; Mefloquine; Mice; Naphthyridines

2014
The survival times of malaria-infected mice are prolonged more by several new two-carbon-linked artemisinin-derived dimer carbamates than by the trioxane antimalarial drug artemether.
    Bioorganic & medicinal chemistry letters, 2014, Mar-01, Volume: 24, Issue:5

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Carbamates; Carbon; Crystallography, X-Ray; Dimerization; Drug Therapy, Combination; Malaria; Mefloquine; Mice; Molecular Conformation; Plasmodium berghei; Structure-Activity Relationship; Survival Analysis

2014
Complex polymorphisms in the Plasmodium falciparum multidrug resistance protein 2 gene and its contribution to antimalarial response.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:12

    Topics: Amino Acid Sequence; Antimalarials; Artemisinins; Biological Transport; Chloroquine; Chromosomes; Drug Resistance, Multiple; Erythrocytes; Humans; INDEL Mutation; Malaria, Falciparum; Mefloquine; Molecular Sequence Data; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Single Nucleotide; Quinolines; Thailand

2014
Ex Vivo Drug Susceptibility Testing and Molecular Profiling of Clinical Plasmodium falciparum Isolates from Cambodia from 2008 to 2013 Suggest Emerging Piperaquine Resistance.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:8

    Topics: Adolescent; Adult; Aged; Antimalarials; Artemisinins; Cambodia; Chloroquine; Drug Resistance; Female; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Male; Mefloquine; Membrane Transport Proteins; Middle Aged; Multidrug Resistance-Associated Proteins; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Young Adult

2015
Assessment of the Worldwide Antimalarial Resistance Network Standardized Procedure for In Vitro Malaria Drug Sensitivity Testing Using SYBR Green Assay for Field Samples with Various Initial Parasitemia Levels.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:4

    Topics: Antimalarials; Artemisinins; Atovaquone; Benzothiazoles; Biological Assay; Chloroquine; Diamines; DNA, Protozoan; Drug Resistance; Erythrocytes; Fluorescent Dyes; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Organic Chemicals; Parasitemia; Plasmodium falciparum; Public Health Surveillance; Quinolines; Reproducibility of Results; Sensitivity and Specificity

2016
Repetitive live sporozoites inoculation under arteether chemoprophylaxis confers protection against subsequent sporozoite challenge in rodent malaria model.
    Acta tropica, 2016, Volume: 158

    Topics: Animals; Antimalarials; Artemisinins; Chemoprevention; Chloroquine; Female; Immunization; Malaria; Mefloquine; Mice; Parasite Load; Plasmodium yoelii; Primaquine; Sporozoites; Vaccination

2016
Back on TRAC: New trial launched in bid to outpace multidrug-resistant malaria.
    Nature medicine, 2016, Volume: 22, Issue:3

    Topics: Antimalarials; Artemisinins; Asia, Southeastern; Drug Resistance, Multiple; Drug Therapy, Combination; Humans; India; Malaria; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Quinolines

2016
Highly active ozonides selected against drug resistant malaria.
    Memorias do Instituto Oswaldo Cruz, 2016, Jun-07, Volume: 0

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Disease Models, Animal; Female; Humans; Malaria, Falciparum; Mefloquine; Mice; Parasitemia; Plasmodium falciparum

2016
Partner-Drug Resistance and Population Substructuring of Artemisinin-Resistant Plasmodium falciparum in Cambodia.
    Genome biology and evolution, 2017, 06-01, Volume: 9, Issue:6

    Topics: Adult; Antipruritics; Artemisinins; Cambodia; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Phylogeny; Plasmodium falciparum; Protozoan Proteins; Quinolines; Treatment Failure

2017
Cellular mechanisms of action and resistance of Plasmodium falciparum to artemisinin.
    Parasitology research, 2017, Volume: 116, Issue:12

    Topics: Antimalarials; Antioxidants; Artemisinins; Artesunate; Drug Resistance; Hemeproteins; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Polymorphism, Genetic; Thailand

2017
Investigating the Efficacy of Triple Artemisinin-Based Combination Therapies for Treating Plasmodium falciparum Malaria Patients Using Mathematical Modeling.
    Antimicrobial agents and chemotherapy, 2018, Volume: 62, Issue:11

    Topics: Antimalarials; Artemisinins; Asia, Southeastern; Drug Therapy, Combination; Humans; Malaria, Falciparum; Mefloquine; Models, Theoretical; Plasmodium falciparum; Quinolines

2018
Plasmodium falciparum Clearance Is Pitting-Dependent With Artemisinin-Based Drugs but Pitting-Independent With Atovaquone-Proguanil or Mefloquine.
    The Journal of infectious diseases, 2019, 07-02, Volume: 220, Issue:3

    Topics: Adolescent; Adult; Antimalarials; Artemisinins; Artesunate; Atovaquone; Child; Drug Combinations; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Proguanil; Young Adult

2019
Improving Methods for Analyzing Antimalarial Drug Efficacy Trials: Molecular Correction Based on Length-Polymorphic Markers
    Antimicrobial agents and chemotherapy, 2019, Volume: 63, Issue:9

    Topics: Algorithms; Antigens, Protozoan; Antimalarials; Artemisinins; Biomarkers; Clinical Trials as Topic; Gene Expression; Humans; Lumefantrine; Malaria, Falciparum; Mefloquine; Merozoite Surface Protein 1; Models, Statistical; Parasitic Sensitivity Tests; Plasmodium falciparum; Polymorphism, Restriction Fragment Length; Protozoan Proteins; Quinolines; Time Factors; Treatment Outcome

2019
Ex vivo susceptibility of Plasmodium falciparum to antimalarial drugs in Northern Uganda.
    Parasitology international, 2021, Volume: 81

    Topics: Amodiaquine; Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Lumefantrine; Mefloquine; Plasmodium falciparum; Quinine; Uganda

2021
Prevalence and characterization of piperaquine, mefloquine and artemisinin derivatives triple-resistant Plasmodium falciparum in Cambodia.
    The Journal of antimicrobial chemotherapy, 2023, 02-01, Volume: 78, Issue:2

    Topics: Antimalarials; Artemisinins; Artesunate; Cambodia; Drug Resistance; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Prevalence; Quinolines

2023
Molecular surveillance of Plasmodium falciparum drug-resistance markers in Vietnam using multiplex amplicon sequencing (2000-2016).
    Scientific reports, 2023, 08-25, Volume: 13, Issue:1

    Topics: Artemisinins; Genotype; Mefloquine; Plasmodium falciparum; Vietnam

2023