mecamylamine and lobeline

mecamylamine has been researched along with lobeline in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19903 (14.29)18.7374
1990's10 (47.62)18.2507
2000's5 (23.81)29.6817
2010's3 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hernandez, J; Hook, R; Martin, WR; Sloan, JW1
Bourlaud, I; Patte, F; Perault, MC; Underner, M1
Grabowski, J; Hall, SM1
Brase, DA; Loh, HH; Tseng, LF; Way, EL1
Holley, LA; Sarter, M; Turchi, J1
Curzon, P; Decker, MW; Kim, DJ1
Khan, IM; Taylor, P; Yaksh, TL1
Buccafusco, JJ; Decker, MW; Evans-Martin, FF; Jackson, WJ; Terry, AV; Zagrodnik, S1
Crooks, PA; Dwoskin, LP; Sonsalla, PK; Teng, L1
Baranyi, M; Lajtha, A; Lendvai, B; Santha, E; Sershen, H; Vizi, ES1
Imoto, M; Ohno, T; Saito, K; Tani, Y1
Buerkle, H; Khan, IM; Taylor, P; Yaksh, TL1
Arneric, SP; Briggs, CA; Gopalakrishnan, M; McKenna, DG; Monteggia, LM; Roch, JM; Sullivan, JP; Touma, E1
Costa, E; Javaid, JI; Lecca, D; Shim, I1
Crooks, PA; Dwoskin, LP; Miller, DK1
Clemente Jiménez, M; Pérez Trullén, A1
Cunningham, CS; Jany, JR; Miller, DK; Polston, JE; Segert, IL1
Baskett, JA; Kracke, GR; Lever, JR; Miller, DK; Rodvelt, KR; Will, MJ1
Dwivedi, C; Rahman, S; Sajja, RK1
Rahman, S; Roni, MA1
Buoli, M; Cahn, W; Serati, M1

Reviews

4 review(s) available for mecamylamine and lobeline

ArticleYear
[Pharmacology of nicotine].
    Revue des maladies respiratoires, 1992, Volume: 9, Issue:4

    Topics: Cardiovascular System; Humans; Lobeline; Mecamylamine; Metabolism; Nervous System; Nicotine; Respiration; Smoking Prevention

1992
Tobacco use, treatment strategies, and pharmacological adjuncts: an overview.
    NIDA research monograph, 1985, Volume: 53

    Topics: Bicarbonates; Humans; Legislation, Medical; Lobeline; Mecamylamine; Nicotine; Psychotropic Drugs; Reinforcement, Psychology; Self-Help Groups; Smoking Prevention; Sodium; Sodium Bicarbonate; Taxes; United States

1985
[Current and future drug therapies for smoking cessation].
    Archivos de bronconeumologia, 2001, Volume: 37, Issue:4

    Topics: Administration, Cutaneous; Administration, Oral; Anti-Anxiety Agents; Antidepressive Agents; Central Nervous System Stimulants; Chewing Gum; Clinical Protocols; Clonidine; Delayed-Action Preparations; Humans; Lobeline; Mecamylamine; Nebulizers and Vaporizers; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Polymethacrylic Acids; Polyvinyls; Smoking; Tobacco Use Cessation Devices

2001
Alternative pharmacological strategies for adult ADHD treatment: a systematic review.
    Expert review of neurotherapeutics, 2016, Volume: 16, Issue:2

    Topics: Adrenergic alpha-Agonists; Adult; Amphetamines; Antidepressive Agents; Attention Deficit Disorder with Hyperactivity; Benzhydryl Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bupropion; Central Nervous System Stimulants; Desipramine; Dopamine Agents; Droxidopa; Drug Combinations; Duloxetine Hydrochloride; Guanfacine; Histamine Agents; Humans; Lisdexamfetamine Dimesylate; Lithium Compounds; Lobeline; Mecamylamine; Memantine; Modafinil; Morpholines; Nicotinic Agonists; Nicotinic Antagonists; Nomifensine; Paroxetine; Pyridines; Pyridoxine; Pyrrolidonecarboxylic Acid; Quinazolinones; Reboxetine; Venlafaxine Hydrochloride; Wakefulness-Promoting Agents

2016

Trials

1 trial(s) available for mecamylamine and lobeline

ArticleYear
[Pharmacology of nicotine].
    Revue des maladies respiratoires, 1992, Volume: 9, Issue:4

    Topics: Cardiovascular System; Humans; Lobeline; Mecamylamine; Metabolism; Nervous System; Nicotine; Respiration; Smoking Prevention

1992

Other Studies

17 other study(ies) available for mecamylamine and lobeline

ArticleYear
Structure-activity relationships of some pyridine, piperidine, and pyrrolidine analogues for enhancing and inhibiting the binding of (+/-)-[3H]nicotine to the rat brain P2 preparation.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:9

    Topics: Acetylcholine; Animals; Binding Sites; Brain; Female; Nicotine; Piperidines; Pyridines; Pyrrolidines; Rats; Structure-Activity Relationship

1985
Cholinergic modification of naloxone-induced jumping in morphine dependent mice.
    European journal of pharmacology, 1974, Volume: 26, Issue:1

    Topics: Animals; Arecoline; Atropine; Behavior, Animal; Benztropine; Brain Chemistry; Dimethylphenylpiperazinium Iodide; Humans; Lobeline; Male; Mecamylamine; Mice; Mice, Inbred ICR; Morphine Dependence; Naloxone; Nicotine; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pempidine; Physostigmine; Pilocarpine; Tremorine; Tritium

1974
Effects of nicotinic acetylcholine receptor ligands on behavioral vigilance in rats.
    Psychopharmacology, 1995, Volume: 118, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Arousal; Attention; Behavior, Animal; Isoxazoles; Ligands; Lobeline; Mecamylamine; Nicotine; Pyrrolidines; Rats; Receptors, Nicotinic; Time Factors

1995
Effect of nicotine, lobeline, and mecamylamine on sensory gating in the rat.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:4

    Topics: Acoustic Stimulation; Animals; Dose-Response Relationship, Drug; Lobeline; Male; Mecamylamine; Nicotine; Rats; Reflex, Startle

1994
Cardiovascular and behavioral responses to nicotinic agents administered intrathecally.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:1

    Topics: Aconitine; Alkaloids; Animals; Atropine; Azocines; Behavior, Animal; Blood Pressure; Bungarotoxins; Cardiovascular System; Dihydro-beta-Erythroidine; Ganglionic Stimulants; Heart Rate; Injections, Spinal; Lobeline; Male; Mecamylamine; Nicotine; Nicotinic Antagonists; Nociceptors; Quinolizines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Sensitivity and Specificity; Spinal Cord; Trimethaphan

1994
Effects of stimulation or blockade of central nicotinic-cholinergic receptors on performance of a novel version of the rat stimulus discrimination task.
    Psychopharmacology, 1996, Volume: 123, Issue:2

    Topics: Animals; Discrimination, Psychological; Dose-Response Relationship, Drug; Lobeline; Male; Mecamylamine; Nicotine; Rats; Rats, Wistar; Receptors, Nicotinic; Task Performance and Analysis

1996
Lobeline and nicotine evoke [3H]overflow from rat striatal slices preloaded with [3H]dopamine: differential inhibition of synaptosomal and vesicular [3H]dopamine uptake.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Calcium; Corpus Striatum; Dopamine; In Vitro Techniques; Lobeline; Male; Mecamylamine; Nicotine; Rats; Rats, Sprague-Dawley; Synaptic Vesicles; Synaptosomes; Tritium

1997
Differential mechanisms involved in the effect of nicotinic agonists DMPP and lobeline to release [3H]5-HT from rat hippocampal slices.
    Neuropharmacology, 1996, Volume: 35, Issue:12

    Topics: Alkaloids; Animals; Azocines; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Hippocampus; In Vitro Techniques; Kinetics; Lobeline; Male; Mecamylamine; Nicotine; Nicotinic Agonists; Pyridines; Quinolizines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Serotonin; Tritium; Tubocurarine

1996
Pharmacological characterization of nicotinic receptor-mediated acetylcholine release in rat brain--an in vivo microdialysis study.
    European journal of pharmacology, 1998, Jun-19, Volume: 351, Issue:2

    Topics: Acetylcholine; Alkaloids; Animals; Azocines; Brain; Cotinine; Hippocampus; Injections, Intraperitoneal; Ligands; Lobeline; Male; Mecamylamine; Microdialysis; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Prefrontal Cortex; Quinolizines; Rats; Rats, Inbred F344; Receptors, Nicotinic; Visual Cortex

1998
Nociceptive and antinociceptive responses to intrathecally administered nicotinic agonists.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: Alkaloids; Analgesia; Animals; Azocines; Bridged Bicyclo Compounds, Heterocyclic; Escape Reaction; Hindlimb; Hot Temperature; Injections, Spinal; Lobeline; Male; Mecamylamine; Microinjections; Nicotine; Nicotinic Agonists; Pain; Pyridines; Quinolizines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Valine; Vocalization, Animal

1998
Gain of function mutation of the alpha7 nicotinic receptor: distinct pharmacology of the human alpha7V274T variant.
    European journal of pharmacology, 1999, Feb-05, Volume: 366, Issue:2-3

    Topics: Acetylcholine; Aconitine; alpha7 Nicotinic Acetylcholine Receptor; Amino Acid Substitution; Animals; Atropine; Choline; Dihydro-beta-Erythroidine; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Genetic Variation; Humans; Lobeline; Mecamylamine; Membrane Potentials; Muscarinic Antagonists; Mutation; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Pyridines; Pyrrolidines; Receptors, Nicotinic; Threonine; Tubocurarine; Valine; Xenopus

1999
Striatal application of nicotine, but not of lobeline, attenuates dopamine release in freely moving rats.
    Neuropharmacology, 2000, Volume: 39, Issue:1

    Topics: Aconitine; Animals; Cocaine; Corpus Striatum; Dopamine; Kinetics; Lobeline; Male; Mecamylamine; Microdialysis; Nerve Endings; Nicotine; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic

2000
Lobeline inhibits nicotine-evoked [(3)H]dopamine overflow from rat striatal slices and nicotine-evoked (86)Rb(+) efflux from thalamic synaptosomes.
    Neuropharmacology, 2000, Volume: 39, Issue:13

    Topics: Animals; Dopamine; In Vitro Techniques; Lobeline; Male; Mecamylamine; Neostriatum; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Rubidium Radioisotopes; Stereoisomerism; Synaptosomes; Thalamus

2000
Interaction of lobeline and nicotinic receptor ligands with the discriminative stimulus properties of cocaine and amphetamine.
    Drug and alcohol dependence, 2006, Oct-01, Volume: 84, Issue:3

    Topics: Amphetamine; Animals; Cocaine; Discrimination, Psychological; Hexamethonium; Ligands; Lobeline; Male; Mecamylamine; Narcotics; Nicotinic Agonists; Nicotinic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Reinforcement, Psychology

2006
Lobeline, a potential pharmacotherapy for drug addiction, binds to mu opioid receptors and diminishes the effects of opioid receptor agonists.
    Drug and alcohol dependence, 2007, Jul-10, Volume: 89, Issue:2-3

    Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Dopamine; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Guinea Pigs; In Vitro Techniques; Lobeline; Mecamylamine; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Nicotine; Oocytes; Radioligand Assay; Receptors, Opioid; Receptors, Opioid, mu; Xenopus laevis

2007
Nicotinic ligands modulate ethanol-induced dopamine function in mice.
    Pharmacology, 2010, Volume: 86, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Alkaloids; Animals; Azocines; Basal Ganglia; Dopamine; Dose-Response Relationship, Drug; Ethanol; Ligands; Lobeline; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Nicotinic Agonists; Nicotinic Antagonists; Quinolizines; Receptors, Nicotinic

2010
Neuronal nicotinic receptor antagonist reduces anxiety-like behavior in mice.
    Neuroscience letters, 2011, Oct-31, Volume: 504, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Blood-Brain Barrier; Brain; Exploratory Behavior; Hexamethonium; Lobeline; Mecamylamine; Mice; Mice, Inbred C57BL; Nicotinic Agonists; Nicotinic Antagonists; Receptors, Nicotinic

2011