mecamylamine and a 85380

mecamylamine has been researched along with a 85380 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (40.00)18.2507
2000's3 (30.00)29.6817
2010's3 (30.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dart, MJ; Holladay, MW; Lynch, JK1
Frølund, B; Jensen, AA; Krogsgaard-Larsen, P; Liljefors, T1
Dannals, RF; Finley, PA; Mochizuki, T; Musachio, JL; Scheffel, U; Wagner, HN; Zhan, Y1
Arneric, SP; Bannon, AW; Curzon, P; Decker, MW; Nikkel, AL1
Bottlaender, M; Coulon, C; Crouzel, C; Dollé, F; Fuseau, C; Guenther, I; Hinnen, F; Ottaviani, M; Valette, H1
Decker, MW; Meyer, MD; Rueter, LE1
Briggs, CA; Dubé, GR; Kohlhaas, KL; Meyer, MD; Rueter, LE; Surowy, CS1
Dong, E; Guidotti, A; Kadriu, B; Maloku, E; Pibiri, F; Satta, R; Zhubi, A1
Feng, CS; Liu, Y; Piao, MH; Qiu, JP; Wang, YS1
Meltzer, HY; Miyauchi, M; Neugebauer, NM; Oyamada, Y1

Reviews

2 review(s) available for mecamylamine and a 85380

ArticleYear
Neuronal nicotinic acetylcholine receptors as targets for drug discovery.
    Journal of medicinal chemistry, 1997, Dec-19, Volume: 40, Issue:26

    Topics: Acetylcholine; Animals; Binding Sites; Dopamine; Drug Design; Humans; Molecular Structure; Nervous System; Neurons; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Receptors, Nicotinic; Structure-Activity Relationship

1997
Neuronal nicotinic acetylcholine receptors: structural revelations, target identifications, and therapeutic inspirations.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Allosteric Regulation; Amino Acid Sequence; Animals; Humans; Ligands; Mice; Mice, Knockout; Models, Molecular; Molecular Sequence Data; Nicotinic Agonists; Nicotinic Antagonists; Protein Conformation; Protein Subunits; Receptors, Nicotinic

2005

Other Studies

8 other study(ies) available for mecamylamine and a 85380

ArticleYear
5-[I-125/123]lodo-3(2(S)-azetidinylmethoxy)pyridine, a radioiodinated analog of A-85380 for in vivo studies of central nicotinic acetylcholine receptors.
    Life sciences, 1998, Volume: 62, Issue:22

    Topics: Alkaloids; Animals; Azetidines; Azocines; Binding Sites; Brain; Dose-Response Relationship, Drug; Iodine Radioisotopes; Male; Mecamylamine; Mice; Muscarinic Antagonists; Nicotine; Nicotinic Antagonists; Quinolizines; Radionuclide Imaging; Receptors, Nicotinic; Scopolamine; Tissue Distribution

1998
Differences between the antinociceptive effects of the cholinergic channel activators A-85380 and (+/-)-epibatidine in rats.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:3

    Topics: Analgesics, Non-Narcotic; Anesthetics, Local; Animals; Azetidines; Bridged Bicyclo Compounds, Heterocyclic; Chlorisondamine; Dose-Response Relationship, Drug; Injections, Intraventricular; Lidocaine; Male; Mecamylamine; Nicotinic Agonists; Nicotinic Antagonists; Pain Measurement; Pyridines; Raphe Nuclei; Rats; Rats, Sprague-Dawley

1998
Characterization of the nicotinic ligand 2-[18F]fluoro-3-[2(S)-2-azetidinylmethoxy]pyridine in vivo.
    Life sciences, 1999, Volume: 64, Issue:5

    Topics: Alkaloids; Animals; Azetidines; Azocines; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Fluorine Radioisotopes; Frontal Lobe; Kinetics; Ligands; Male; Mecamylamine; Nicotine; Nicotinic Agonists; Pyridines; Quinolizines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Thalamus; Tissue Distribution

1999
Spinal mechanisms underlying A-85380-induced effects on acute thermal pain.
    Brain research, 2000, Jul-28, Volume: 872, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Animals; Azetidines; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Bungarotoxins; Clonidine; Dose-Response Relationship, Drug; Hot Temperature; Injections, Intraperitoneal; Injections, Spinal; Lumbosacral Region; Male; Mecamylamine; Microdialysis; Muscarinic Antagonists; Nicotinic Agonists; Nicotinic Antagonists; Norepinephrine; Pain; Pain Measurement; Pyridines; Rats; Rats, Sprague-Dawley; Reaction Time; Serotonin; Serotonin Antagonists; Spinal Cord

2000
Loss of functional neuronal nicotinic receptors in dorsal root ganglion neurons in a rat model of neuropathic pain.
    Neuroscience letters, 2005, Mar-07, Volume: 376, Issue:1

    Topics: Acetylcholine; Animals; Azetidines; Cell Count; Cells, Cultured; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Ganglia, Spinal; Ligation; Lumbosacral Region; Male; Mecamylamine; Membrane Potentials; Neurons; Nicotinic Agonists; Nicotinic Antagonists; Pain; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Spinal Cord Injuries

2005
Selective α4β2 nicotinic acetylcholine receptor agonists target epigenetic mechanisms in cortical GABAergic neurons.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2011, Volume: 36, Issue:7

    Topics: Analysis of Variance; Animals; Azetidines; Behavior, Animal; Benzazepines; Cerebral Cortex; Conditioning, Classical; Cues; DNA (Cytosine-5-)-Methyltransferase 1; DNA (Cytosine-5-)-Methyltransferases; Epigenomics; Exploratory Behavior; Fear; Freezing Reaction, Cataleptic; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Male; Mecamylamine; Methyl-CpG-Binding Protein 2; Mice; Neurons; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Promoter Regions, Genetic; Quinoxalines; Receptors, Nicotinic; RNA, Messenger; Varenicline

2011
Volatile anesthetic isoflurane inhibits LTP induction of hippocampal CA1 neurons through α4β2 nAChR subtype-mediated mechanisms.
    Annales francaises d'anesthesie et de reanimation, 2013, Volume: 32, Issue:10

    Topics: Anesthetics, Inhalation; Animals; Azetidines; Bridged Bicyclo Compounds, Heterocyclic; CA1 Region, Hippocampal; Dihydro-beta-Erythroidine; Drug Interactions; Electric Stimulation; In Vitro Techniques; Isoflurane; Long-Term Potentiation; Mecamylamine; Muscarinic Agonists; Neural Pathways; Neurons; Nicotine; Nicotinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic

2013
Nicotinic receptors and lurasidone-mediated reversal of phencyclidine-induced deficit in novel object recognition.
    Behavioural brain research, 2016, Mar-15, Volume: 301

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Azetidines; Benzamides; Bridged Bicyclo Compounds; Cognition Disorders; Disease Models, Animal; Female; Lurasidone Hydrochloride; Mecamylamine; Nicotinic Agonists; Nicotinic Antagonists; Nootropic Agents; Phencyclidine; Random Allocation; Rats, Long-Evans; Receptors, Nicotinic

2016