mdl-201112 has been researched along with adenosine in 3 studies
Studies (mdl-201112) | Trials (mdl-201112) | Recent Studies (post-2010) (mdl-201112) | Studies (adenosine) | Trials (adenosine) | Recent Studies (post-2010) (adenosine) |
---|---|---|---|---|---|
10 | 0 | 0 | 32,536 | 1,075 | 8,930 |
Protein | Taxonomy | mdl-201112 (IC50) | adenosine (IC50) |
---|---|---|---|
high affinity choline transporter 1 isoform a | Homo sapiens (human) | 0.3851 | |
Sodium/nucleoside cotransporter 1 | Homo sapiens (human) | 5.5 | |
Sodium/nucleoside cotransporter 2 | Homo sapiens (human) | 5.5 | |
Adenosine receptor A3 | Homo sapiens (human) | 0.0011 | |
Adenosine receptor A1 | Homo sapiens (human) | 0.0023 | |
Equilibrative nucleoside transporter 1 | Homo sapiens (human) | 63 | |
Solute carrier family 28 member 3 | Homo sapiens (human) | 3.3 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Borcherding, DR; Bowlin, TL; Edwards, CK; Hoffman, PF; Munson, HR; Peet, NP; Zhang, H | 1 |
Borcherding, DR; Edwards, CK; Linnik, MD; Long, RE; Parmely, MJ; Watts, LM | 1 |
Borcherding, DR; Edwards, CK; Morrison, DC; Parmely, MJ; Silverstein, R; Zhou, WW | 1 |
3 other study(ies) available for mdl-201112 and adenosine
Article | Year |
---|---|
Carbocyclic nucleosides as inhibitors of human tumor necrosis factor-alpha production: effects of the stereoisomers of (3-hydroxycyclopentyl)adenines.
Topics: Adenine; Adenosine; Animals; Cyclopentanes; Galactosamine; Humans; Interleukin-1; Interleukin-6; Lipopolysaccharides; Macrophages; Magnetic Resonance Spectroscopy; Mice; Molecular Structure; Stereoisomerism; Tumor Necrosis Factor-alpha | 1996 |
Effect of the carbocyclic nucleoside analogue MDL 201,112 on inhibition of interferon-gamma-induced priming of Lewis (LEW/N) rat macrophages for enhanced respiratory burst and MHC class II Ia+ antigen expression.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Animals; Bordetella pertussis; Brain; Dipyridamole; Down-Regulation; Female; Histocompatibility Antigens Class II; Interferon-gamma; Kinetics; Lipopolysaccharides; Macrophage Activation; Macrophages, Peritoneal; Mycobacterium tuberculosis; Rats; Rats, Inbred Lew; Receptors, Purinergic P1; Receptors, Purinergic P2; Recombinant Proteins; Respiratory Burst; Stimulation, Chemical; Superoxides; Tumor Necrosis Factor-alpha; Zymosan | 1994 |
Adenosine and a related carbocyclic nucleoside analogue selectively inhibit tumor necrosis factor-alpha production and protect mice against endotoxin challenge.
Topics: Adenine; Adenosine; Animals; Cytokines; Endotoxins; Female; Interleukin-1; Macrophage Activation; Macrophages; Mice; Tumor Necrosis Factor-alpha | 1993 |