Page last updated: 2024-09-03

mci 154 and carbachol

mci 154 has been researched along with carbachol in 2 studies

Compound Research Comparison

Studies
(mci 154)
Trials
(mci 154)
Recent Studies (post-2010)
(mci 154)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
651013,91881968

Protein Interaction Comparison

ProteinTaxonomymci 154 (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gwathmey, JK; Kihara, Y; Morgan, JP; Pesaturo, J; Phillips, P; Warren, SE1
Endoh, M; Kitada, Y; Narimatsu, A; Suzuki, R; Taira, N1

Other Studies

2 other study(ies) available for mci 154 and carbachol

ArticleYear
Inotropic and lusitropic effects of MCI-154 (6-[4-(4- pyridyl)aminophenyl]-4,5-dihydro-3(2H)-pyridazinone) on human myocardium.
    Journal of molecular and cellular cardiology, 1989, Volume: 21, Issue:10

    Topics: Aequorin; Carbachol; Cardiotonic Agents; Cyclic AMP; Heart; Heart Ventricles; Humans; Muscle Relaxation; Myocardial Contraction; Pyridazines

1989
Does the positive inotropic action of a novel cardiotonic agent, MCI-154, involve mechanisms other than cyclic AMP?
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:2

    Topics: Animals; Carbachol; Cardiotonic Agents; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Phosphoric Diester Hydrolases; Pindolol; Pyridazines; Reserpine; Stimulation, Chemical; Tetrodotoxin

1987