mazindol and benztropine

mazindol has been researched along with benztropine in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19904 (36.36)18.7374
1990's4 (36.36)18.2507
2000's3 (27.27)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chilco, PJ; Donnan, GA; Kaczmarczyk, SJ; Kalnins, RM; Mendelsohn, FA; Paxinos, G; Woodhouse, DG1
Rothman, RB1
Kruk, ZL; Millar, J; Stamford, JA1
Brooks, JD; DeLanney, LE; Irwin, I; Langston, JW; Ricaurte, GA1
McKearney, JW1
Kalix, P1
Meiergerd, SM; Schenk, JO1
Hattori, T; Sugimoto, T; Takada, M1
Berfield, JL; Ferrer, JV; Javitch, JA; Reith, ME; Wang, LC1
Bondi, CD; Kozikowski, AP; Kulkarni, SS; Newman, AH; Pan, S; Surratt, CK; Ukairo, OT1
Ramanujapuram, S; Surratt, CK; Ukairo, OT1

Other Studies

11 other study(ies) available for mazindol and benztropine

ArticleYear
Distribution of catecholamine uptake sites in human brain as determined by quantitative [3H] mazindol autoradiography.
    The Journal of comparative neurology, 1991, Feb-15, Volume: 304, Issue:3

    Topics: Aged; Benztropine; Binding, Competitive; Biological Transport; Brain Chemistry; Brain Mapping; Caudate Nucleus; Citalopram; Clomipramine; Corpus Striatum; Desipramine; Dopamine; Humans; Locus Coeruleus; Mazindol; Medulla Oblongata; Mianserin; Middle Aged; Norepinephrine; Piperazines; Pons; Substantia Nigra

1991
High affinity dopamine reuptake inhibitors as potential cocaine antagonists: a strategy for drug development.
    Life sciences, 1990, Volume: 46, Issue:20

    Topics: Benztropine; Bupropion; Cocaine; Dopamine; Drug Evaluation, Preclinical; Humans; Mazindol; Nomifensine; Propiophenones; Substance-Related Disorders

1990
In vivo voltammetric characterization of low affinity striatal dopamine uptake: drug inhibition profile and relation to dopaminergic innervation density.
    Brain research, 1986, May-14, Volume: 373, Issue:1-2

    Topics: Animals; Benztropine; Corpus Striatum; Dextroamphetamine; Dopamine; Electric Stimulation; Male; Mazindol; Medial Forebrain Bundle; Methylphenidate; Nalidixic Acid; Naphthyridines; Neural Pathways; Nomifensine; Rats; Rats, Inbred Strains

1986
Dopamine uptake blockers protect against the dopamine depleting effect of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine (MPTP) in the mouse striatum.
    Neuroscience letters, 1985, Sep-06, Volume: 59, Issue:3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Benztropine; Bupropion; Corpus Striatum; Dopamine; Male; Mazindol; Mice; Mice, Inbred C57BL; Nalidixic Acid; Naphthyridines; Parasympatholytics; Propiophenones; Pyridines; Receptors, Dopamine

1985
Effects of dopamine uptake inhibitors on schedule-controlled behavior in the squirrel monkey.
    Psychopharmacology, 1982, Volume: 78, Issue:4

    Topics: Animals; Behavior, Animal; Benztropine; Bupropion; Conditioning, Operant; Dopamine; Electroshock; Male; Mazindol; Nomifensine; Propiophenones; Psychotropic Drugs; Reinforcement Schedule; Saimiri

1982
The amphetamine-like releasing effect of the alkaloid (-)cathinone on rat nucleus accumbens and rabbit caudate nucleus.
    Progress in neuro-psychopharmacology & biological psychiatry, 1982, Volume: 6, Issue:1

    Topics: Alkaloids; Animals; Benztropine; Caudate Nucleus; Dextroamphetamine; Dopamine; Dose-Response Relationship, Drug; Mazindol; Neural Inhibition; Nomifensine; Nucleus Accumbens; Rabbits; Septal Nuclei

1982
Kinetic evaluation of the commonality between the site(s) of action of cocaine and some other structurally similar and dissimilar inhibitors of the striatal transporter for dopamine.
    Journal of neurochemistry, 1994, Volume: 63, Issue:5

    Topics: Animals; Benztropine; Biological Transport; Cocaine; Corpus Striatum; Dopamine; Male; Mazindol; Models, Biological; Neurotransmitter Uptake Inhibitors; Nomifensine; Piperazines; Rats; Rats, Sprague-Dawley

1994
MPTP neurotoxicity to cerebellar Purkinje cells in mice.
    Neuroscience letters, 1993, Feb-05, Volume: 150, Issue:1

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Benztropine; Dose-Response Relationship, Drug; Male; Mazindol; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; MPTP Poisoning; Neurotoxins; Pargyline; Purkinje Cells; Selegiline

1993
The uptake inhibitors cocaine and benztropine differentially alter the conformation of the human dopamine transporter.
    The Journal of biological chemistry, 2001, Aug-03, Volume: 276, Issue:31

    Topics: Benztropine; Binding Sites; Binding, Competitive; Carrier Proteins; Cell Membrane; Cocaine; Cysteine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Humans; Indicators and Reagents; Kinetics; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Mesylates; Models, Molecular; Nerve Tissue Proteins; Protein Conformation

2001
Recognition of benztropine by the dopamine transporter (DAT) differs from that of the classical dopamine uptake inhibitors cocaine, methylphenidate, and mazindol as a function of a DAT transmembrane 1 aspartic acid residue.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:2

    Topics: Amino Acid Substitution; Animals; Aspartic Acid; Benztropine; Binding, Competitive; CHO Cells; Cocaine; Cricetinae; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Humans; Immunohistochemistry; Kinetics; Ligands; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Methylphenidate; Microscopy, Confocal; Models, Molecular; Mutagenesis, Site-Directed; Nerve Tissue Proteins; Transfection

2005
Fluctuation of the dopamine uptake inhibition potency of cocaine, but not amphetamine, at mammalian cells expressing the dopamine transporter.
    Brain research, 2007, Feb-02, Volume: 1131, Issue:1

    Topics: Amphetamine; Amphetamine-Related Disorders; Animals; Benztropine; Binding, Competitive; Brain; Brain Chemistry; Cell Line, Tumor; Chlorocebus aethiops; CHO Cells; Cocaine; Cocaine-Related Disorders; COS Cells; Cricetinae; Cricetulus; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Mazindol; Methylphenidate; Neurons; Radioligand Assay

2007