masoprocol and aa 861
masoprocol has been researched along with aa 861 in 35 studies
Research
Studies (35)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 10 (28.57) | 18.7374 |
1990's | 12 (34.29) | 18.2507 |
2000's | 10 (28.57) | 29.6817 |
2010's | 3 (8.57) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Kreft, AF; Musser, JH | 1 |
Bermudez, J; Buckle, DR; Foster, KA; Markwell, RE; Smith, SA; Taylor, JF; Tedder, JM; Thody, VE; Webster, RA | 1 |
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
Lewis, DA; Miller, VM | 1 |
Baba, T; Black, KL; Chio, CC | 1 |
Kanamaru, K; Matsumoto, T; Murata, Y; Sugiyama, Y | 1 |
Ebbesen, MA; Gibel, L; Goodwin, JS; Harford, AM; Shopp, GM; Smith, AY; Sterling, WA | 1 |
Kurachi, Y; Nakajima, T; Sugimoto, T | 1 |
Jarvis, WD; Judd, AM; MacLeod, RM; Spangelo, BL | 1 |
Chand, N; Diamantis, W; Nolan, K; Pillar, J; Sofia, RD | 1 |
Kreofsky, T; Rohrbach, MS; Rolstad, RA; Russell, JA | 1 |
Bonta, IL; Elliott, GR; van Hilten, JA | 2 |
Behrens, TW; Goodwin, JS; Lianos, EA; Lum, LG | 1 |
Niwa, Y; Ohashi, T; Ozaki, Y | 1 |
Aizu, E; Kato, R; Nakadate, T; Yamamoto, S | 2 |
Goldin, E; Harel, S; Magal, E; Yavin, E | 1 |
Fujimoto, K; Kobayashi, T; Kubo, K; Matsuzawa, Y; Okada, K; Shinozaki, S; Sugane, K | 1 |
Higuchi, K; Kominami, S; Takemori, S; Yamazaki, T | 1 |
Armacost, LM; Cobb, RR; Felts, KA; Lee, S; Parry, GC | 1 |
Ghosh, J; Myers, CE | 1 |
Izumi, T; Koyama, S; Kubo, K; Nagai, S; Nomura, H; Sato, E | 1 |
Haniuda, M; Izumi, T; Koyama, S; Kubo, K; Nagai, S; Nomura, H; Sato, E | 1 |
Catalano, A; Claria, J; Crescenzi, C; D'Urbano, E; Davi, G; Libner, R; Nutini, M; Procopio, A; Romano, M | 1 |
Loscalzo, J; Walker, JL; Zhang, YY | 1 |
Jhamandas, K; Quirion, R; Sutak, M; Trang, T | 1 |
Jhamandas, K; McNaull, B; Quirion, R; Trang, T | 1 |
Cao, YB; Chen, XS; Cheng, MH; Li, J; Wang, Y; Yin, M; Zhou, B | 1 |
Artemenko, IP; Jefcoate, CR | 1 |
Goda, AE; Horinaka, M; Miki, T; Mizutani, Y; Nakata, S; Nishikawa, A; Sakai, T; Shiraishi, T; Wakada, M; Yasuda, T; Yoshida, T | 1 |
Challis, JR; Chisaka, H; Okamura, K; Sato, K | 1 |
Choi, YS; Hah, YS; Hwang, EM; Jeong, YS; Lee, SH; Ok, SH; Park, JY; Shin, IW; Sohn, JT | 1 |
Kim, BJ; Kim, SJ; Nam, JH | 1 |
Czapski, GA; Czubowicz, K; Strosznajder, RP | 1 |
Reviews
1 review(s) available for masoprocol and aa 861
Article | Year |
---|---|
5-lipoxygenase: properties, pharmacology, and the quinolinyl(bridged)aryl class of inhibitors.
Topics: Animals; Arachidonate 5-Lipoxygenase; Asthma; Eosinophils; Humans; Inflammation; Leukotriene Antagonists; Lipoxygenase Inhibitors; Lung Diseases; Neutrophils; Quinolines | 1992 |
Other Studies
34 other study(ies) available for masoprocol and aa 861
Article | Year |
---|---|
Novel 1H-benzimidazol-4-ols with potent 5-lipoxygenase inhibitory activity.
Topics: Animals; Arachidonate Lipoxygenases; Benzimidazoles; Female; Lipoxygenase Inhibitors; Rats; Rats, Inbred Strains; SRS-A; Structure-Activity Relationship | 1987 |
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
Role of lipoxygenase and cytochrome P-450 in production of endothelium-derived relaxing factors in canine femoral veins.
Topics: Animals; Arachidonate 5-Lipoxygenase; Arachidonic Acid; Arginine; Benzoquinones; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Dogs; Femoral Vein; In Vitro Techniques; Lipoxygenase Inhibitors; Masoprocol; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; omega-N-Methylarginine; Piperidines; Proadifen | 1992 |
The effect of 5-lipoxygenase inhibition on blood-brain barrier permeability in experimental brain tumors.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Analysis of Variance; Animals; Autoradiography; Benzoquinones; Blood-Brain Barrier; Brain Neoplasms; Carcinoma 256, Walker; Female; gamma-Glutamyltransferase; Leukotrienes; Lipoxygenase Inhibitors; Masoprocol; Rats; Rats, Inbred Strains | 1992 |
Endothelium-derived relaxation of the pregnant and nonpregnant canine uterine artery.
Topics: Acetylcholine; Animals; Benzoquinones; Calcimycin; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Evaluation Studies as Topic; Female; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Nitric Oxide; Pregnancy; Pregnancy, Animal; Uterus; Vasoconstriction | 1992 |
Murine thymocyte lysis by inhibitors of arachidonic acid metabolism.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Adrenal Cortex Hormones; Animals; Arachidonic Acid; Arachidonic Acids; Benzoquinones; Caffeic Acids; Cells, Cultured; Dexamethasone; Dinoprostone; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Mice; Mice, Inbred C57BL; Spleen; Thymus Gland | 1991 |
Platelet-activating factor activates cardiac GK via arachidonic acid metabolites.
Topics: Animals; Arachidonic Acids; Benzoquinones; Cells, Cultured; Flavanones; Flavonoids; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guinea Pigs; Heart; Heart Atria; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Membrane Potentials; Myocardium; Platelet Activating Factor; Potassium Channels; Virulence Factors, Bordetella | 1991 |
Induction of interleukin-6 release by interleukin-1 in rat anterior pituitary cells in vitro: evidence for an eicosanoid-dependent mechanism.
Topics: Animals; Arachidonic Acid; Aristolochic Acids; Benzoquinones; Cells, Cultured; Cyclooxygenase Inhibitors; Eicosanoids; Ethacrynic Acid; Female; Glycerylphosphorylcholine; Interleukin-1; Interleukin-6; Lipoxygenase Inhibitors; Masoprocol; Organic Chemicals; Phenanthrenes; Phospholipases A; Phospholipases A2; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Signal Transduction | 1991 |
Inhibition of allergic and nonallergic leukotriene C4 formation and histamine secretion by azelastine: implication for its mechanism of action.
Topics: Animals; Benzhydryl Compounds; Benzoquinones; Guinea Pigs; Histamine Release; Immunosuppressive Agents; Male; Masoprocol; Mast Cells; Phthalazines; Pyridazines; Quinones; Rats; Rats, Inbred Strains; Respiratory Hypersensitivity; SRS-A; Terfenadine | 1989 |
Tannin-mediated secretion of a neutrophil chemotactic factor from alveolar macrophages. Potential contribution to the acute pulmonary inflammatory reaction associated with byssinosis.
Topics: Animals; Benzoquinones; Byssinosis; Cells, Cultured; Chemotactic Factors; Cycloheximide; Dust; Endotoxins; Enterobacter; Gossypium; Humans; Interleukin-8; Lipoxygenase Inhibitors; Lung; Macrophages; Masoprocol; Pulmonary Alveoli; Quinones; Rabbits; Tannins | 1989 |
Endogenous lipoxygenase metabolites mediate A23187 induced macrophage cytostasis towards P815 tumor cells in vitro.
Topics: Animals; Antineoplastic Agents; Benzoquinones; Calcimycin; Lipoxygenase; Lipoxygenase Inhibitors; Macrophage Activation; Masoprocol; Mice; Quinones; Tumor Cells, Cultured | 1989 |
Lipoxygenase inhibitors enhance the proliferation of human B cells.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Adjuvants, Immunologic; Adult; B-Lymphocytes; Benzoquinones; Cell Differentiation; Child; Cyclooxygenase Inhibitors; Dose-Response Relationship, Immunologic; Humans; Immunoglobulins; Indomethacin; Interleukin-4; Interleukins; Kinetics; Lipoxygenase Inhibitors; Lymphocyte Activation; Masoprocol; Palatine Tonsil; Pyrazoles; Quinones; Staphylococcal Protein A | 1989 |
A comparative study on the effects of inhibitors of the lipoxygenase pathway on neutrophil function. Inhibitory effects on neutrophil function may not be attributed to inhibition of the lipoxygenase pathway.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Benzoquinones; Calcimycin; Chemotaxis, Leukocyte; Epoprostenol; Humans; Hydroxides; Hydroxyl Radical; Leukotriene B4; Lipoxygenase Inhibitors; Masoprocol; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phospholipases A; Phospholipases A2; Platelet Activating Factor; Quinones; Tetradecanoylphorbol Acetate; Umbelliferones | 1986 |
Inhibition of 12-O-tetradecanoylphorbol-13-acetate-mediated epidermal ornithine decarboxylase induction and skin tumor promotion by new lipoxygenase inhibitors lacking protein kinase C inhibitory effects.
Topics: Animals; Benzoquinones; Chalcone; Chalcones; Enzyme Induction; Female; Lipoxygenase Inhibitors; Masoprocol; Mice; Ornithine Decarboxylase; Propiophenones; Protein Kinase C; Quercetin; Quinones; Skin; Skin Neoplasms; Tetradecanoylphorbol Acetate | 1986 |
Acute uteroplacental ischemic embryo: lactic acid accumulation and prostaglandin production in the fetal rat brain.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Benzoquinones; Brain; Cyclooxygenase Inhibitors; Dinoprost; Dinoprostone; Female; Indomethacin; Ischemia; Lactates; Lactic Acid; Lipoxygenase Inhibitors; Masoprocol; Placenta; Pregnancy; Prostaglandins; Prostaglandins E; Prostaglandins F; Pyrazoles; Quinones; Rats; Uterus | 1988 |
Specific lipoxygenase inhibition reverses macrophage cytotasis towards P815 tumor cells in vitro induced by the calcium ionophore A23187.
Topics: Animals; Arachidonate Lipoxygenases; Benzoquinones; Calcimycin; Cytotoxicity, Immunologic; Female; Lipoxygenase Inhibitors; Macrophages; Masoprocol; Mice; Mice, Inbred BALB C; Neoplasms, Experimental; Quinones | 1988 |
Inhibition of 12-O-tetradecanoylphorbol-13-acetate-induced increase in vascular permeability in mouse skin by lipoxygenase inhibitors.
Topics: Animals; Benzoquinones; Capillary Permeability; Catechols; Female; Indomethacin; Lipoxygenase; Lipoxygenase Inhibitors; Masoprocol; Mice; Mice, Inbred Strains; Ornithine Decarboxylase; Phorbols; Prostaglandin-Endoperoxide Synthases; Quercetin; Quinones; Skin; Tetradecanoylphorbol Acetate | 1985 |
Neutrophil elastase inhibitor reduces asthmatic responses in allergic sheep.
Topics: Airway Resistance; Animals; Antigens; Asthma; Benzoquinones; Bronchial Hyperreactivity; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Calcimycin; Glycine; Heterocyclic Compounds; Leukocyte Elastase; Leukocytes; Leukotriene B4; Masoprocol; Methacholine Chloride; Pancreatic Elastase; Polycyclic Compounds; Sheep; Sulfonamides; Thromboxane B2 | 1995 |
15-lipoxygenase metabolite(s) of arachidonic acid mediates adrenocorticotropin action in bovine adrenal steroidogenesis.
Topics: Animals; Arachidonate 15-Lipoxygenase; Arachidonic Acids; Benzoquinones; Bucladesine; Cattle; Cells, Cultured; Cosyntropin; Cyclic AMP; Dihydrotestosterone; Enzyme Inhibitors; Indomethacin; Isoquinolines; Kinetics; Leukotrienes; Lipid Peroxides; Lipoxygenase Inhibitors; Masoprocol; Pregnenolone; Sulfonamides; Tetrahydronaphthalenes; Zona Fasciculata; Zona Reticularis | 1996 |
Inhibition of 5-lipoxygenase blocks IL-1 beta-induced vascular adhesion molecule-1 gene expression in human endothelial cells.
Topics: Benzoquinones; Biological Transport; Cell Nucleus; Cells, Cultured; Endothelium, Vascular; Gene Expression Regulation; Humans; Interleukin-1; Lipoxygenase Inhibitors; Masoprocol; NF-kappa B; Phosphorylation; Promoter Regions, Genetic; Transcription, Genetic; Vascular Cell Adhesion Molecule-1 | 1997 |
Arachidonic acid stimulates prostate cancer cell growth: critical role of 5-lipoxygenase.
Topics: Arachidonate 5-Lipoxygenase; Arachidonic Acid; Arachidonic Acids; Benzoquinones; Cell Division; Cyclooxygenase Inhibitors; Eicosanoids; Enzyme Inhibitors; Flavanones; Flavonoids; Humans; Hydroxyeicosatetraenoic Acids; Ibuprofen; Indoles; Lipoxygenase Inhibitors; Male; Masoprocol; Proadifen; Prostatic Neoplasms; Tumor Cells, Cultured | 1997 |
Acetylcholine and substance P stimulate bronchial epithelial cells to release eosinophil chemotactic activity.
Topics: Acetylcholine; Animals; Benzoquinones; Bronchi; Cattle; Cells, Cultured; Chemokines; Chemotaxis; Cycloheximide; Cyclooxygenase Inhibitors; Diethylcarbamazine; Eosinophils; Leukotriene B4; Lipoxygenase Inhibitors; Lung; Masoprocol; Substance P | 1998 |
Histamine stimulates alveolar macrophages to release neutrophil and monocyte chemotactic activity.
Topics: Acetates; Animals; Benzoquinones; Cattle; Cells, Cultured; Chemotactic Factors; Chromatography, Gel; Diethylcarbamazine; Histamine; Hot Temperature; Leukotriene B4; Macrophages, Alveolar; Masoprocol; Monocytes; Neutrophils; Platelet Membrane Glycoproteins; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Serotonin; Trypsin | 2001 |
5-lipoxygenase regulates malignant mesothelial cell survival: involvement of vascular endothelial growth factor.
Topics: Apoptosis; Arachidonate 5-Lipoxygenase; Arachidonic Acid; Benzoquinones; Cell Division; Cell Line; Cell Survival; DNA, Antisense; Endothelial Growth Factors; Gene Expression Regulation; Gene Expression Regulation, Enzymologic; Green Fluorescent Proteins; Humans; Lipoxygenase Inhibitors; Luminescent Proteins; Lymphokines; Masoprocol; Mesothelioma; Mutation; Promoter Regions, Genetic; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA; Thymidine; Time Factors; Transcription, Genetic; Transfection; Tritium; Tumor Cells, Cultured; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2001 |
5-Lipoxygenase and human pulmonary artery endothelial cell proliferation.
Topics: Apoptosis; Arachidonate 5-Lipoxygenase; Benzoquinones; Cell Division; Cells, Cultured; Comet Assay; Cyclooxygenase Inhibitors; Endothelium, Vascular; Growth Substances; Humans; Indoles; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Oligonucleotides, Antisense; Pulmonary Artery; S Phase; Thymidine; Transfection; Tritium | 2002 |
Spinal administration of lipoxygenase inhibitors suppresses behavioural and neurochemical manifestations of naloxone-precipitated opioid withdrawal.
Topics: Animals; Benzoquinones; Calcitonin Gene-Related Peptide; Dose-Response Relationship, Drug; Flavanones; Flavonoids; Immunohistochemistry; Injections, Spinal; Lipoxygenase Inhibitors; Male; Masoprocol; Morphine; Morphine Dependence; Naloxone; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Spinal Cord; Substance Withdrawal Syndrome | 2003 |
Involvement of spinal lipoxygenase metabolites in hyperalgesia and opioid tolerance.
Topics: Analgesics, Opioid; Animals; Benzoquinones; Dose-Response Relationship, Drug; Drug Tolerance; Flavanones; Formaldehyde; Hindlimb; Hyperalgesia; Injections, Spinal; Leukotriene B4; Leukotrienes; Lipid Peroxides; Lipoxygenase; Lipoxygenase Inhibitors; Male; Masoprocol; Morphine; Pain; Pain Measurement; Rats; Rats, Sprague-Dawley; Spinal Cord; Time Factors | 2004 |
Inhibitors of 5-lipoxygenase inhibit expression of intercellular adhesion molecule-1 in human melanoma cells.
Topics: Benzoquinones; Cell Adhesion; Cells, Cultured; Endothelial Cells; Humans; Indoles; Intercellular Adhesion Molecule-1; Lipoxygenase Inhibitors; Masoprocol; Melanoma; RNA, Messenger; Tumor Cells, Cultured; Umbilical Veins | 2004 |
Multiple contributions from long-chain fatty acid metabolism in Y-1 and MA-10 cells.
Topics: Animals; Arachidonic Acid; Benzoquinones; Cell Line; Fatty Acids; Linoleic Acid; Lipoxygenase Inhibitors; Masoprocol; Mice; Oleic Acid; Phosphoproteins; Steroids | 2004 |
Lipoxygenase inhibitors induce death receptor 5/TRAIL-R2 expression and sensitize malignant tumor cells to TRAIL-induced apoptosis.
Topics: Apoptosis; Apoptosis Regulatory Proteins; Benzoquinones; Cell Line, Tumor; Down-Regulation; Drug Synergism; Humans; Immunoglobulin Fc Fragments; Jurkat Cells; Leukemia, T-Cell; Lipoxygenase Inhibitors; Masoprocol; Mutant Chimeric Proteins; Receptors, TNF-Related Apoptosis-Inducing Ligand; TNF-Related Apoptosis-Inducing Ligand; Up-Regulation | 2007 |
Effect of the interaction between lipoxygenase pathway and progesterone on the regulation of hydroxysteroid 11-Beta dehydrogenase 2 in cultured human term placental trophoblasts.
Topics: 11-beta-Hydroxysteroid Dehydrogenase Type 2; Benzoquinones; Cells, Cultured; Enzyme Activation; Female; Flavanones; Gene Expression Regulation, Enzymologic; Gestational Age; Humans; Lipoxygenase; Lipoxygenase Inhibitors; Masoprocol; Models, Biological; Placenta; Pregnancy; Progesterone; RNA, Messenger; Signal Transduction; Trophoblasts | 2008 |
The direct effect of levobupivacaine in isolated rat aorta involves lipoxygenase pathway activation and endothelial nitric oxide release.
Topics: Anesthetics, Local; Animals; Aorta, Thoracic; Benzoquinones; Bupivacaine; Calcium; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; In Vitro Techniques; Levobupivacaine; Lipoxygenase; Lipoxygenase Inhibitors; Male; Masoprocol; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Potassium Chloride; Quinacrine; Rats; Rats, Sprague-Dawley; Verapamil | 2010 |
Effects of transient receptor potential channel blockers on pacemaker activity in interstitial cells of Cajal from mouse small intestine.
Topics: Animals; Arachidonate 5-Lipoxygenase; Benzoquinones; Biological Clocks; Calcium Channel Blockers; Cell Line; Gastrointestinal Motility; Humans; Interstitial Cells of Cajal; Intestine, Small; Lipoxygenase Inhibitors; Masoprocol; Mice; Mice, Inbred BALB C; Patch-Clamp Techniques | 2011 |
Evaluation of the antioxidative properties of lipoxygenase inhibitors.
Topics: Animals; Antioxidants; Benzoquinones; Flavanones; Lipoxygenase Inhibitors; Male; Masoprocol; Rats; Rats, Wistar | 2012 |