Page last updated: 2024-09-03

marimastat and tosedostat

marimastat has been researched along with tosedostat in 1 studies

Compound Research Comparison

Studies
(marimastat)
Trials
(marimastat)
Recent Studies (post-2010)
(marimastat)
Studies
(tosedostat)
Trials
(tosedostat)
Recent Studies (post-2010) (tosedostat)
215285333727

Protein Interaction Comparison

ProteinTaxonomymarimastat (IC50)tosedostat (IC50)
72 kDa type IV collagenaseHomo sapiens (human)0.19
Matrix metalloproteinase-9Homo sapiens (human)1.5
Aminopeptidase NHomo sapiens (human)0.68
Puromycin-sensitive aminopeptidaseHomo sapiens (human)0.26

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Butler, GS; Charman, SA; Drinkwater, N; Gazdik, M; Grin, PM; Kannan Sivaraman, K; Lee, J; McGowan, S; Overall, CM; Scammells, PJ; Schembri, LS; Vinh, NB; Yang, W1

Other Studies

1 other study(ies) available for marimastat and tosedostat

ArticleYear
Novel Human Aminopeptidase N Inhibitors: Discovery and Optimization of Subsite Binding Interactions.
    Journal of medicinal chemistry, 2019, 08-08, Volume: 62, Issue:15

    Topics: Animals; Binding Sites; CD13 Antigens; Drug Discovery; Enzyme Inhibitors; Humans; Male; Mice; Protein Binding; Protein Structure, Tertiary

2019