Page last updated: 2024-09-03

marimastat and ro 31-9790

marimastat has been researched along with ro 31-9790 in 2 studies

Compound Research Comparison

Studies
(marimastat)
Trials
(marimastat)
Recent Studies (post-2010)
(marimastat)
Studies
(ro 31-9790)
Trials
(ro 31-9790)
Recent Studies (post-2010) (ro 31-9790)
21528532800

Protein Interaction Comparison

ProteinTaxonomymarimastat (IC50)ro 31-9790 (IC50)
Interstitial collagenaseHomo sapiens (human)0.0058
72 kDa type IV collagenaseHomo sapiens (human)0.0074
Stromelysin-1Homo sapiens (human)0.47
Matrix metalloproteinase-9Homo sapiens (human)0.012
Matrix metalloproteinase-14Homo sapiens (human)0.0019

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hori, N; Ikeda, S; Inoue, S; Ohishi, Y; Okada, Y; Tsujishita, H; Yamamoto, M1
Barlaam, B; Bird, TG; Campbell, D; Foster, SJ; Lambert-Van Der Brempt, C; Maciewicz, R1

Other Studies

2 other study(ies) available for marimastat and ro 31-9790

ArticleYear
Inhibition of membrane-type 1 matrix metalloproteinase by hydroxamate inhibitors: an examination of the subsite pocket.
    Journal of medicinal chemistry, 1998, Apr-09, Volume: 41, Issue:8

    Topics: Amino Acid Sequence; Dipeptides; Humans; Hydroxamic Acids; Ligands; Matrix Metalloproteinases, Membrane-Associated; Metalloendopeptidases; Models, Molecular; Mutation; Phenylalanine; Protease Inhibitors; Protein Conformation; Structure-Activity Relationship; Thiophenes

1998
New alpha-substituted succinate-based hydroxamic acids as TNFalpha convertase inhibitors.
    Journal of medicinal chemistry, 1999, Nov-18, Volume: 42, Issue:23

    Topics: ADAM Proteins; ADAM17 Protein; Administration, Oral; Animals; Callithrix; Humans; Hydroxamic Acids; Metalloendopeptidases; Protease Inhibitors; Quinazolines; Succinates; Tumor Necrosis Factor-alpha

1999