Page last updated: 2024-08-17

lysine and osimertinib

lysine has been researched along with osimertinib in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's3 (100.00)2.80

Authors

AuthorsStudies
Cui, Y; Feng, D; Liu, X; Zheng, M; Zhong, D1
Campos, S; Evans, JP; Fournier, JCL; Patel, VK; Thomas, DA; Tomkinson, NCO; White, GV; Zappacosta, F1
Chen, J; Chen, L; Diao, X; He, Q; Wu, Y; Xue, H; Zhong, D1

Other Studies

3 other study(ies) available for lysine and osimertinib

ArticleYear
Characterization of covalent binding of tyrosine kinase inhibitors to plasma proteins.
    Drug metabolism and pharmacokinetics, 2020, Volume: 35, Issue:5

    Topics: Acrylamides; Adenine; Aminoquinolines; Aniline Compounds; Animals; Binding Sites; Dogs; Haplorhini; Humans; Indoles; Lysine; Mice; Molecular Docking Simulation; Molecular Structure; Piperidines; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Quinolines; Rabbits; Rats; Serum Albumin, Human

2020
Acetylation of the Catalytic Lysine Inhibits Kinase Activity in PI3Kδ.
    ACS chemical biology, 2021, 09-17, Volume: 16, Issue:9

    Topics: Acetylation; Acrylamides; Adenine; Afatinib; Amino Acid Sequence; Aniline Compounds; Catalysis; Catalytic Domain; Class I Phosphatidylinositol 3-Kinases; Humans; Lysine; Mass Spectrometry; Molecular Docking Simulation; Phosphoinositide-3 Kinase Inhibitors; Piperidines; Protein Binding; Protein Conformation; Substrate Specificity

2021
Covalent Binding Mechanism of Furmonertinib and Osimertinib With Human Serum Albumin.
    Drug metabolism and disposition: the biological fate of chemicals, 2023, Volume: 51, Issue:1

    Topics: Carcinoma, Non-Small-Cell Lung; Humans; Lung Neoplasms; Lysine; Serum Albumin; Serum Albumin, Human

2023