Page last updated: 2024-08-17

lysergic acid diethylamide and ketanserin

lysergic acid diethylamide has been researched along with ketanserin in 65 studies

Research

Studies (65)

Timeframe	Studies, this research(%)	All Research%
pre-1990	22 (33.85)	18.7374
1990's	26 (40.00)	18.2507
2000's	3 (4.62)	29.6817
2010's	9 (13.85)	24.3611
2020's	5 (7.69)	2.80

Authors

Authors	Studies
Andrews, PR; Craik, DJ; Martin, JL	1
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM	1
Glennon, RA	1
Innocent, O; Olufemi, A	1
Cassuto, J; Jodal, M; Lundgren, O; Sjöqvist, A	1
Burris, KD; Sanders-Bush, E	1
Gewecke, M; Roeder, T; Wedemeyer, S	1
Karnovsky, ML; Polanski, M	1
Barker, EL; Burris, KD; Sanders-Bush, E	1
Brazell, C; Campbell, IC; Mitchell, S; Stahl, SM; Twist, EC	1
Himeno, A; Saavedra, JM	2
Buckholtz, NS; Freedman, DX; Potter, WZ; Zhou, DF	1
Appel, NM; De Souza, EB; Garlick, RK; Glennon, RA; Mitchell, WM; Teitler, M	1
Altar, CA; Boyar, WC; Marien, MR	1
Baraban, JM; Glennon, RA; Jan, CR; Leonhardt, S; Lyon, RA; Sadzot, B; Titeler, M	1
Purdy, RE; Xu, Z	1
Elliott, JM; Kent, A	1
Chaudhuri, J; Donahue, MJ	1
Appel, JB; Cunningham, KA; Ginn, SR; Nielsen, EB	1
Godfrey, PP; McClue, SJ; Minchin, MC; Schächter, M; Young, MM	1
Appel, JB; Callahan, PM; Cunningham, KA	1
Hoffmann, D; Wesemann, W	1
Frost, JJ; Hartig, PR; Scheffel, U; Wagner, HN	1
Peroutka, SJ; Pierce, PA	1
Buckholtz, NS; Freedman, DX; Zhou, DF	1
Hartig, PR; Kadan, MJ	1
Mann, JJ; McBride, PA; Polley, MJ; Sweeney, JA; Wiley, AJ	1
Penington, NJ; Reiffenstein, RJ	1
Laduron, PM; Leysen, JE; Van Dun, J; Wouters, W	1
Engel, G; Hoyer, D; Kalkman, HO; Wick, MB	1
Gudelsky, GA; Meltzer, HY; Simonovic, M	1
Affolter, H; Pletscher, A	1
Engel, G; Müller-Schweinitzer, E	1
Heym, J; Jacobs, BL; Rasmussen, K	1
Palacios, JM; Waeber, C	1
Blakely, RD; Davies, P; Pitt, BR; Reynolds, I; Steve, AR; Weng, W	1
Huang, X; Marona-Lewicka, D; Nichols, DE; Pfaff, RC	1
Müller-Oerlinghausen, B; Rüggeberg-Schmidt, K; Steckler, T	1
Ferry, RC; Molinoff, PB; Unsworth, CD	1
Dyer, DC; Zhang, L	1
Fiorella, D; Rabin, RA; Winter, JC	1
Almaula, N; Ballesteros, JA; Ebersole, BJ; Sealfon, SC; Weinstein, H	1
Marona-Lewicka, D; Monte, AP; Nelson, DL; Nichols, DE; Parker, MA; Wainscott, DB	1
Fiorella, D; Helsley, S; Rabin, RA; Winter, JC	1
Austin, RH; Borroni, E; Bourson, A; Monsma, FJ; Sleight, AJ	1
Carey, JE; Chen, C; Elliott, JM; Flanigan, TP; Kumar, C; McDonald, B; Newberry, NR; Newton, RA; Phipps, SL	1
Assié, MB; Kleven, MS; Koek, W	1
Harvey, JA; Hood, H; Romano, AG; Welsh, SE	1
Brunden, K; Doucette, C; Graham, E; Hanniford, D; Harrington, J; Poole, MF; Sherf, B; Song, J; Stricker-Krongrad, A; Ting, A	1
Fernandes, KA; Jha, S; Rajendran, R; Vaidya, VA	1
Aloyo, VJ; Dave, KD; Harvey, JA; Schindler, EA; Smolock, EM	1
Khelashvili, G; Mehler, EL; Mondal, S; Shan, J; Weinstein, H	1
Agnati, LF; Borroto-Escuela, DO; Fuxe, K; Narvaez, M; Oflijan, J; Romero-Fernandez, W	1
Buchborn, T; Dieterich, DC; Grecksch, G; Höllt, V; Schröder, H	1
Herdener, M; Kraehenmann, R; Liechti, ME; Planzer, A; Pokorny, T; Preller, KH; Seifritz, E; Stämpfli, P; Vollenweider, FX	1
Kraehenmann, R; Pokorny, D; Pokorny, T; Preller, KH; Seifritz, E; Vollenweider, FX; Vollenweider, L	1
Barrett, FS; Herdener, M; Janata, P; Preller, KH; Vollenweider, FX	1
Flemming, J; Pokorny, T; Preller, KH; Schilbach, L; Seifritz, E; Vollenweider, FX	1
Bugno, R; Hogendorf, A; Krawczyk, M; Kuziak, A; Nikiforuk, A; Popik, P; Staroń, J	1
Duerler, P; Pokorny, T; Preller, KH; Seifritz, E; Vollenweider, FX	1
Duerler, P; Preller, KH; Schilbach, L; Stämpfli, P; Vollenweider, FX	1
Borgwardt, S; Dolder, P; Duthaler, U; Eckert, A; Holze, F; Ley, L; Liechti, ME; Müller, F; Stocker, M; Varghese, N; Vizeli, P	1
Olbrich, S; Preller, KH; Vollenweider, FX	1
Becker, AM; Duthaler, U; Eckert, A; Holze, F; Istampoulouoglou, I; Klaiber, A; Liechti, ME; Varghese, N	1

Reviews

2 review(s) available for lysergic acid diethylamide and ketanserin

Article	Year
The role of receptor binding in drug discovery. Journal of natural products, 1993, Volume: 56, Issue:4 Topics: Animals; Drug Design; Humans; Receptors, Drug	1993
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7). Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14 Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists	2003

Trials

7 trial(s) available for lysergic acid diethylamide and ketanserin

Article	Year
The Fabric of Meaning and Subjective Effects in LSD-Induced States Depend on Serotonin 2A Receptor Activation. Current biology : CB, 2017, Feb-06, Volume: 27, Issue:3 Topics: Cross-Over Studies; Double-Blind Method; Gene Expression Regulation; Humans; Ketanserin; Lysergic Acid Diethylamide; Music; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Serotonin Receptor Agonists; Task Performance and Analysis	2017
Role of the 5-HT The Journal of neuroscience : the official journal of the Society for Neuroscience, 2018, 04-04, Volume: 38, Issue:14 Topics: Adult; Attention; Brain; Cognition; Eye Movements; Female; Hallucinogens; Humans; Interpersonal Relations; Ketanserin; Lysergic Acid Diethylamide; Magnetic Resonance Imaging; Male; Serotonin Antagonists; Serotonin Receptor Agonists	2018
LSD acutely impairs working memory, executive functions, and cognitive flexibility, but not risk-based decision-making. Psychological medicine, 2020, Volume: 50, Issue:13 Topics: Adult; Cognition; Decision Making; Double-Blind Method; Executive Function; Female; Healthy Volunteers; Humans; Ketanserin; Lysergic Acid Diethylamide; Male; Memory, Short-Term; Neuropsychological Tests; Serotonin Antagonists; Serotonin Receptor Agonists; Young Adult	2020
LSD-induced increases in social adaptation to opinions similar to one's own are associated with stimulation of serotonin receptors. Scientific reports, 2020, 07-22, Volume: 10, Issue:1 Topics: Brain; Double-Blind Method; Female; Healthy Volunteers; Humans; Ketanserin; Lysergic Acid Diethylamide; Magnetic Resonance Imaging; Male; Personality; Placebo Effect; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Social Interaction; Social Norms; Young Adult	2020
Acute dose-dependent effects of lysergic acid diethylamide in a double-blind placebo-controlled study in healthy subjects. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2021, Volume: 46, Issue:3 Topics: Double-Blind Method; Female; Hallucinogens; Healthy Volunteers; Humans; Ketanserin; Lysergic Acid Diethylamide; Male	2021
LSD and ketanserin and their impact on the human autonomic nervous system. Psychophysiology, 2021, Volume: 58, Issue:6 Topics: Adult; Antihypertensive Agents; Autonomic Nervous System; Electrocardiography; Female; Hallucinogens; Healthy Volunteers; Heart Rate; Humans; Ketanserin; Lysergic Acid Diethylamide; Male; Surveys and Questionnaires; Young Adult	2021
Ketanserin Reverses the Acute Response to LSD in a Randomized, Double-Blind, Placebo-Controlled, Crossover Study in Healthy Participants. The international journal of neuropsychopharmacology, 2023, 02-14, Volume: 26, Issue:2 Topics: Brain-Derived Neurotrophic Factor; Cross-Over Studies; Double-Blind Method; Hallucinogens; Healthy Volunteers; Humans; Ketanserin; Lysergic Acid Diethylamide	2023

Other Studies

56 other study(ies) available for lysergic acid diethylamide and ketanserin

Article	Year
Functional group contributions to drug-receptor interactions. Journal of medicinal chemistry, 1984, Volume: 27, Issue:12 Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship	1984
Receptors mediating the actions of 5-hydroxytryptamine on the isolated retractor muscle of the penis preparations from Archachatina marginata (Swainson). Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 101, Issue:2 Topics: Animals; Ergolines; Indoles; Ketanserin; Lysergic Acid Diethylamide; Muscle Contraction; Muscles; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Snails; Tropisetron	1992
Actions of serotonin antagonists on cholera-toxin-induced intestinal fluid secretion. Acta physiologica Scandinavica, 1992, Volume: 145, Issue:3 Topics: Animals; Body Fluids; Cholera Toxin; Female; Granisetron; Imidazoles; Indazoles; Intestinal Mucosa; Ketanserin; Lysergic Acid Diethylamide; Male; Methysergide; Ondansetron; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Zimeldine	1992
Unsurmountable antagonism of brain 5-hydroxytryptamine2 receptors by (+)-lysergic acid diethylamide and bromo-lysergic acid diethylamide. Molecular pharmacology, 1992, Volume: 42, Issue:5 Topics: 3T3 Cells; Animals; Brain; DNA; Ketanserin; Lysergic Acid Diethylamide; Mice; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin Antagonists; Transfection	1992
Pharmacological characterization of a 5-HT receptor in locust nervous tissue. European journal of pharmacology, 1992, Nov-17, Volume: 223, Issue:2-3 Topics: Animals; Antipsychotic Agents; Binding Sites; Brain; Dopamine; Esophagus; Female; Grasshoppers; GTP-Binding Proteins; Ketanserin; Lysergic Acid Diethylamide; Magnesium; Male; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thoracic Nerves	1992
Serotonergic aspects of the response of human platelets to immune-adjuvant muramyl dipeptide. Journal of neuroimmunology, 1992, Volume: 37, Issue:1-2 Topics: Acetylmuramyl-Alanyl-Isoglutamine; Adenosine Diphosphate; Adjuvants, Immunologic; Blood Platelets; Carrier Proteins; Humans; Imipramine; Ketanserin; Lysergic Acid Diethylamide; Paroxetine; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Serotonin; Serotonin Antagonists	1992
Phosphoinositide hydrolysis linked 5-HT2 receptors in fibroblasts from choroid plexus. Brain research, 1991, Jun-28, Volume: 552, Issue:2 Topics: Animals; Cells, Cultured; Choroid Plexus; DOM 2,5-Dimethoxy-4-Methylamphetamine; Fibroblasts; Haloperidol; Hydrolysis; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Phosphatidylinositols; Prazosin; Rabbits; Receptors, Serotonin; Serotonin; Spiperone	1991
5HT2 receptor changes in rat cortex and platelets following chronic ritanserin and clorgyline administration. Biochemical pharmacology, 1990, Jan-01, Volume: 39, Issue:1 Topics: Animals; Blood Platelets; Cerebral Cortex; Clorgyline; Homovanillic Acid; Hydroxyindoleacetic Acid; Ketanserin; Lysergic Acid Diethylamide; Male; Norepinephrine; Piperidines; Propylamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin	1990
Autoradiographic studies of 5HT2 receptors. Advances in experimental medicine and biology, 1991, Volume: 294 Topics: Amphetamines; Animals; Autoradiography; Blood Platelets; Brain Chemistry; Hallucinogens; Humans; Ketanserin; Lysergic Acid Diethylamide; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists	1991
Lysergic acid diethylamide (LSD) administration selectively downregulates serotonin2 receptors in rat brain. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1990, Volume: 3, Issue:2 Topics: Animals; Brain; Cerebral Cortex; Down-Regulation; Ketanserin; Lysergic Acid Diethylamide; Male; Mescaline; Organ Specificity; Psilocybin; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reference Values	1990
Autoradiographic characterization of (+-)-1-(2,5-dimethoxy-4-[125I] iodophenyl)-2-aminopropane ([125I]DOI) binding to 5-HT2 and 5-HT1c receptors in rat brain. The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:2 Topics: Amphetamines; Animals; Autoradiography; Brain; Brain Chemistry; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists	1990
Human platelet [125I]R-DOI binding sites. Characterization by in vitro autoradiography. Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1990, Volume: 3, Issue:1 Topics: Adult; Amphetamines; Autoradiography; Binding, Competitive; Blood Platelets; Cell Membrane; Female; Humans; Iodine Radioisotopes; Ketanserin; Kinetics; Lysergic Acid Diethylamide; Male; Receptors, Serotonin; Stereoisomerism	1990
125I-LSD autoradiography confirms the preferential localization of caudate-putamen S2 receptors to the caudal (peripallidal) region. Brain research, 1986, Apr-30, Volume: 372, Issue:1 Topics: Animals; Autoradiography; Butaclamol; Caudate Nucleus; Frontal Lobe; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Putamen; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin	1986
Hallucinogenic drug interactions at human brain 5-HT2 receptors: implications for treating LSD-induced hallucinogenesis. Psychopharmacology, 1989, Volume: 98, Issue:4 Topics: Animals; Binding, Competitive; Cerebral Cortex; Hallucinations; Hallucinogens; Humans; In Vitro Techniques; Ketanserin; Lysergic Acid Diethylamide; Rats; Receptors, Serotonin	1989
Evidence for allosteric blockade of serotonergic receptors in rabbit thoracic aorta. The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3 Topics: Allosteric Regulation; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; Ketanserin; Lysergic Acid Diethylamide; Male; Rabbits; Receptors, Serotonin; Serotonin; Serotonin Antagonists	1989
Comparison of [125I]iodolysergic acid diethylamide binding in human frontal cortex and platelet tissue. Journal of neurochemistry, 1989, Volume: 53, Issue:1 Topics: Binding, Competitive; Blood Platelets; Cell Membrane; Frontal Lobe; Humans; Iodine Radioisotopes; Ketanserin; Kinetics; Lysergic Acid Diethylamide	1989
Serotonin receptors in the tissues of adult Ascaris suum. Molecular and biochemical parasitology, 1989, Volume: 35, Issue:3 Topics: Animals; Ascaris; Binding Sites; Binding, Competitive; Cell Membrane; Female; Histamine; Intestinal Mucosa; Intestines; Ketanserin; Lysergic Acid Diethylamide; Muscles; Parasympathomimetics; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sympathomimetics	1989
Antagonism of the LSD cue by putative serotonin antagonists: relationship to inhibition of in vivo [3H]spiroperidol binding. Behavioural brain research, 1985, Volume: 16, Issue:2-3 Topics: Animals; Cerebellum; Corpus Striatum; Frontal Lobe; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Pizotyline; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin	1985
Serotonergic agonists stimulate inositol lipid metabolism in rabbit platelets. Life sciences, 1985, Oct-28, Volume: 37, Issue:17 Topics: Animals; Blood Platelets; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Phosphatidylinositols; Piperidines; Quipazine; Rabbits; Receptors, Serotonin; Serotonin	1985
Differentiation between the stimulus effects of l-5-hydroxytryptophan and LSD. European journal of pharmacology, 1985, Jan-22, Volume: 108, Issue:2 Topics: 5-Hydroxytryptophan; Animals; Benserazide; Cues; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains	1985
Characterization of 5-hydroxytryptamine binding sites in the plasma membrane of pig blood platelets. Journal of neural transmission, 1985, Volume: 61, Issue:3-4 Topics: Animals; Binding Sites; Blood Platelets; Brain; Ketanserin; Lysergic Acid Diethylamide; Piperidines; Platelet Aggregation; Serotonin; Sodium; Swine	1985
In vivo binding of 125I-LSD to serotonin 5-HT2 receptors in mouse brain. Life sciences, 1985, Aug-19, Volume: 37, Issue:7 Topics: Animals; Binding, Competitive; Brain; Cinanserin; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Mice; Piperidines; Receptors, Serotonin; Spiperone; Time Factors; Tissue Distribution	1985
Antagonism of 5-hydroxytryptamine2 receptor-mediated phosphatidylinositol turnover by d-lysergic acid diethylamide. The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3 Topics: Amphetamines; Animals; Cerebral Cortex; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Guanosine Triphosphate; In Vitro Techniques; Ketanserin; Lysergic Acid Diethylamide; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Serotonin	1988
Serotonin2 agonist administration down-regulates rat brain serotonin2 receptors. Life sciences, 1988, Volume: 42, Issue:24 Topics: Amphetamines; Animals; Brain; DOM 2,5-Dimethoxy-4-Methylamphetamine; Hallucinogens; Ketanserin; Lysergic Acid Diethylamide; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin	1988
Autoradiographic localization and characterization of [125I]lysergic acid diethylamide binding to serotonin receptors in Aplysia. Neuroscience, 1988, Volume: 24, Issue:3 Topics: Animals; Aplysia; Autoradiography; Binding, Competitive; Ketanserin; Lysergic Acid Diethylamide; Receptors, Serotonin; Serotonin	1988
Assessment of binding indices and physiological responsiveness of the 5-HT2 receptor on human platelets. Life sciences, 1987, May-04, Volume: 40, Issue:18 Topics: Adenosine Diphosphate; Adult; Age Factors; Blood Platelets; Dose-Response Relationship, Drug; Female; Humans; Ketanserin; Lysergic Acid Diethylamide; Male; Middle Aged; Platelet Aggregation; Receptors, Serotonin	1987
Lack of effect of antagonists on serotonin-induced inhibition in rat hippocampus. Canadian journal of physiology and pharmacology, 1986, Volume: 64, Issue:11 Topics: Action Potentials; Animals; Cyproheptadine; Halothane; Hippocampus; Ketanserin; Lysergic Acid Diethylamide; Metergoline; Methysergide; Neural Inhibition; Picrotoxin; Rats; Serotonin; Serotonin Antagonists; Urethane	1986
Photoaffinity probes for serotonin and histamine receptors. Synthesis and characterization of two azide analogues of ketanserin. The Journal of biological chemistry, 1985, Jul-15, Volume: 260, Issue:14 Topics: 4-Aminobenzoic Acid; Affinity Labels; Animals; Azides; Binding, Competitive; Cerebellum; Cerebral Cortex; Guinea Pigs; Histamine Antagonists; Ketanserin; Kinetics; Lysergic Acid Diethylamide; Photochemistry; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Receptors, Serotonin; Serotonin Antagonists; Ultraviolet Rays	1985
Identification of 5HT2-receptors on longitudinal muscle of the guinea pig ileum. Journal of receptor research, 1984, Volume: 4, Issue:1-6 Topics: Animals; Cerebral Cortex; Female; Guinea Pigs; Ileum; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Muscle, Smooth; Piperidines; Rats; Receptors, Serotonin	1984
Effects of pirenperone and ketanserin on rat prolactin secretion in vivo and in vitro. European journal of pharmacology, 1983, Aug-19, Volume: 92, Issue:1-2 Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin Antagonists; Tranquilizing Agents	1983
The 5-hydroxytryptamine receptor of blood platelets. Journal of neural transmission, 1983, Volume: 57, Issue:4 Topics: Animals; Binding, Competitive; Blood Platelets; Brain; Calcium; Cell Membrane; Ketanserin; Kinetics; Lysergic Acid Diethylamide; Models, Neurological; Neurons; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship	1983
Evidence for mediation by 5-HT2 receptors of 5-hydroxytryptamine-induced contraction of canine basilar artery. Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:4 Topics: Animals; Basilar Artery; Cerebral Cortex; Dogs; Female; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium	1983
Some behavioral effects of hallucinogens are mediated by a postsynaptic serotonergic action: evidence from single unit studies in freely moving cats. European journal of pharmacology, 1984, May-18, Volume: 101, Issue:1-2 Topics: Animals; Apomorphine; Behavior, Animal; Cats; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Female; Hallucinogens; Ketanserin; Lisuride; Lysergic Acid Diethylamide; Metergoline; Mianserin; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Synapses	1984
Binding sites for 5-hydroxytryptamine-2 receptor agonists are predominantly located in striosomes in the human basal ganglia. Brain research. Molecular brain research, 1994, Volume: 24, Issue:1-4 Topics: Adult; Aged; Aging; Animals; Basal Ganglia; Binding Sites; Binding, Competitive; Brain; Cats; Cattle; Female; Guinea Pigs; Humans; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Macaca mulatta; Male; Middle Aged; Organ Specificity; Receptors, Serotonin; Serotonin Receptor Agonists; Swine; Tritium	1994
Serotonin increases DNA synthesis in rat proximal and distal pulmonary vascular smooth muscle cells in culture. The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 1 Topics: Animals; Binding, Competitive; Blotting, Northern; Calcium; Cells, Cultured; DNA; Ketanserin; Lung; Lysergic Acid Diethylamide; Mianserin; Muscle, Smooth, Vascular; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA, Messenger; Serotonin; Thymidine	1994
Drug discrimination and receptor binding studies of N-isopropyl lysergamide derivatives. Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Binding, Competitive; Conditioning, Operant; Discrimination, Psychological; Hallucinogens; Iodine Radioisotopes; Ketanserin; Lysergic Acid Diethylamide; Male; Models, Molecular; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reinforcement Schedule	1994
Human platelet 5-HT2 receptor binding sites re-evaluated: a criticism of current techniques [corrected]. Journal of neural transmission. General section, 1993, Volume: 92, Issue:1 Topics: Adult; Blood Platelets; Blood Proteins; Cell Membrane; Evaluation Studies as Topic; Humans; In Vitro Techniques; Ketanserin; Ligands; Lysergic Acid Diethylamide; Male; Receptors, Serotonin	1993
Effects of agonists, partial agonists, and antagonists on the regulation of 5-hydroxytryptamine2 receptors in P11 cells. Molecular pharmacology, 1993, Volume: 43, Issue:5 Topics: Amphetamines; Animals; Down-Regulation; Hydrolysis; Ketanserin; Lysergic Acid Diethylamide; Mianserin; Phosphatidylinositols; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tumor Cells, Cultured	1993
Lysergic acid diethylamide is a partial agonist at 5-HT2 receptors in ovine uterine artery of late pregnancy. European journal of pharmacology, 1993, Jan-05, Volume: 230, Issue:1 Topics: Animals; Arteries; Female; In Vitro Techniques; Ketanserin; Lysergic Acid Diethylamide; Muscle Contraction; Muscle, Smooth, Vascular; Pregnancy; Pregnancy, Animal; Regional Blood Flow; Serotonin; Serotonin Receptor Agonists; Sheep; Uterus	1993
Role of 5-HT2A and 5-HT2C receptors in the stimulus effects of hallucinogenic drugs. II: Reassessment of LSD false positives. Psychopharmacology, 1995, Volume: 121, Issue:3 Topics: Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Hallucinogens; Ketanserin; Lisuride; Lysergic Acid Diethylamide; Male; Rats; Rats, Inbred F344; Receptors, Serotonin	1995
Contribution of a helix 5 locus to selectivity of hallucinogenic and nonhallucinogenic ligands for the human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors: direct and indirect effects on ligand affinity mediated by the same locus. Molecular pharmacology, 1996, Volume: 50, Issue:1 Topics: Amino Acid Sequence; Animals; Binding Sites; Binding, Competitive; Cell Line; Chlorocebus aethiops; Ergolines; Hallucinogens; Humans; Ketanserin; Kinetics; Ligands; Lysergic Acid Diethylamide; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Phosphatidylinositols; Point Mutation; Protein Structure, Secondary; Rats; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Sequence Homology, Amino Acid; Structure-Activity Relationship; Transfection	1996
Dihydrobenzofuran analogues of hallucinogens. 3. Models of 4-substituted (2,5-dimethoxyphenyl)alkylamine derivatives with rigidified methoxy groups. Journal of medicinal chemistry, 1996, Jul-19, Volume: 39, Issue:15 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Benzofurans; Binding, Competitive; Cell Membrane; Cricetinae; Hallucinogens; Hippocampus; Humans; Ketanserin; Lysergic Acid Diethylamide; Male; Mesocricetus; Molecular Conformation; Molecular Structure; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Structure-Activity Relationship; Tritium	1996
5-HT2C receptor-mediated phosphoinositide turnover and the stimulus effects of m-chlorophenylpiperazine. Psychopharmacology, 1995, Volume: 122, Issue:3 Topics: Animals; Choroid Plexus; Conditioning, Operant; DOM 2,5-Dimethoxy-4-Methylamphetamine; Drug Interactions; Ketanserin; Lysergic Acid Diethylamide; Ondansetron; Phosphatidylinositols; Piperazines; Pyrazines; Quipazine; Rats; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists	1995
Effects of altered 5-ht6 expression in the rat: functional studies using antisense oligonucleotides. Behavioural brain research, 1996, Volume: 73, Issue:1-2 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Base Sequence; Behavior, Animal; Binding, Competitive; In Vitro Techniques; Injections, Intraventricular; Ketanserin; Lysergic Acid Diethylamide; Male; Membranes; Molecular Sequence Data; Oligonucleotides, Antisense; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists	1996
Characterisation of human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors expressed in the human neuroblastoma cell line SH-SY5Y: comparative stimulation by hallucinogenic drugs. Journal of neurochemistry, 1996, Volume: 67, Issue:6 Topics: Adrenergic alpha-Agonists; Amphetamines; Antiparkinson Agents; Calcium; Choroid Plexus; Electrophysiology; Ergolines; Ergotamine; Frontal Lobe; Hallucinogens; Humans; Hydrolysis; Ketanserin; Lysergic Acid Diethylamide; Mescaline; Methoxydimethyltryptamines; Neuroblastoma; Phosphatidylinositols; Piperazines; Quipazine; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium; Tumor Cells, Cultured	1996
Pharmacological characterization of in vivo properties of putative mixed 5-HT1A agonist/5-HT(2A/2C) antagonist anxiolytics. II. Drug discrimination and behavioral observation studies in rats. The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:2 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzopyrans; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Nicotinic Acids; Piperazines; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists	1997
Effect of 5-HT2 receptor antagonists on a cranial nerve reflex in the rabbit: evidence for inverse agonism. Psychopharmacology, 1999, Volume: 141, Issue:2 Topics: Animals; Cranial Nerves; Ergolines; Female; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Piperidines; Rabbits; Receptors, Serotonin; Reflex; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists	1999
Development of homogeneous high-affinity agonist binding assays for 5-HT2 receptor subtypes. Assay and drug development technologies, 2005, Volume: 3, Issue:6 Topics: Amphetamines; Binding, Competitive; Calcium Signaling; Cell Line; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Ergolines; Humans; Ketanserin; Lysergic Acid Diethylamide; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Transfection	2005
5-HT2A/2C receptor blockade regulates progenitor cell proliferation in the adult rat hippocampus. Neuroscience letters, 2008, Aug-22, Volume: 441, Issue:2 Topics: Adult Stem Cells; Amphetamines; Animals; Bromodeoxyuridine; Cell Count; Cell Proliferation; Doublecortin Domain Proteins; Drug Administration Schedule; Hippocampus; Ketanserin; Lysergic Acid Diethylamide; Male; Microtubule-Associated Proteins; Neuropeptides; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists	2008
Serotonergic and dopaminergic distinctions in the behavioral pharmacology of (±)-1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane (DOI) and lysergic acid diethylamide (LSD). Pharmacology, biochemistry, and behavior, 2012, Volume: 101, Issue:1 Topics: Amphetamines; Animals; Behavior, Animal; Binding, Competitive; Brain Chemistry; Dopamine; Frontal Lobe; Hallucinogens; Ketanserin; Lysergic Acid Diethylamide; Male; Rabbits; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D1; Ritanserin; Serotonin; Serotonin Agents; Serotonin Antagonists; Temperature	2012
Ligand-dependent conformations and dynamics of the serotonin 5-HT(2A) receptor determine its activation and membrane-driven oligomerization properties. PLoS computational biology, 2012, Volume: 8, Issue:4 Topics: Binding Sites; Cell Membrane; Computer Simulation; Ketanserin; Ligands; Lysergic Acid Diethylamide; Models, Chemical; Models, Molecular; Protein Binding; Protein Conformation; Receptor, Serotonin, 5-HT2A; Serotonin; Structure-Activity Relationship	2012
Hallucinogenic 5-HT2AR agonists LSD and DOI enhance dopamine D2R protomer recognition and signaling of D2-5-HT2A heteroreceptor complexes. Biochemical and biophysical research communications, 2014, Jan-03, Volume: 443, Issue:1 Topics: Amphetamines; Animals; Basal Ganglia; Gene Expression Regulation; Genes, Reporter; Hallucinogens; HEK293 Cells; Humans; Ketanserin; Luciferases; Lysergic Acid Diethylamide; Male; Promoter Regions, Genetic; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists	2014
Tolerance to LSD and DOB induced shaking behaviour: differential adaptations of frontocortical 5-HT(2A) and glutamate receptor binding sites. Behavioural brain research, 2015, Mar-15, Volume: 281 Topics: Animals; Binding Sites; DOM 2,5-Dimethoxy-4-Methylamphetamine; Drug Tolerance; Frontal Lobe; Glutamic Acid; Hallucinogens; Ketanserin; Lysergic Acid Diethylamide; Male; Motor Activity; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Glutamate; Serotonin Antagonists	2015
Dreamlike effects of LSD on waking imagery in humans depend on serotonin 2A receptor activation. Psychopharmacology, 2017, Volume: 234, Issue:13 Topics: Dopamine; Healthy Volunteers; Humans; Ketanserin; Lysergic Acid Diethylamide; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin 5-HT2 Receptor Antagonists	2017
Serotonin 2A Receptor Signaling Underlies LSD-induced Alteration of the Neural Response to Dynamic Changes in Music. Cerebral cortex (New York, N.Y. : 1991), 2018, 11-01, Volume: 28, Issue:11 Topics: Auditory Perception; Brain; Brain Mapping; Double-Blind Method; Emotions; Hallucinogens; Humans; Ketanserin; Lysergic Acid Diethylamide; Magnetic Resonance Imaging; Memory; Music; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists	2018
Serotonin type 5A receptor antagonists inhibit D-lysergic acid diethylamide discriminatory cue in rats. Journal of psychopharmacology (Oxford, England), 2019, Volume: 33, Issue:11 Topics: Animals; Cues; Discrimination Learning; Dose-Response Relationship, Drug; Hallucinogens; Ketanserin; Lysergic Acid Diethylamide; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists	2019