Page last updated: 2024-09-05

ly 300164 and ly 293558

ly 300164 has been researched along with ly 293558 in 3 studies

Compound Research Comparison

Studies
(ly 300164)
Trials
(ly 300164)
Recent Studies (post-2010)
(ly 300164)
Studies
(ly 293558)
Trials
(ly 293558)
Recent Studies (post-2010) (ly 293558)
73712103418

Protein Interaction Comparison

ProteinTaxonomyly 300164 (IC50)ly 293558 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)2.7869
Glutamate receptor 2Rattus norvegicus (Norway rat)2.7869
Glutamate receptor 3Rattus norvegicus (Norway rat)2.7869
Glutamate receptor 4Rattus norvegicus (Norway rat)2.7869
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.23
Glutamate receptor ionotropic, kainate 1Homo sapiens (human)0.5
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.23
Glutamate receptor 1Homo sapiens (human)3.075
Glutamate receptor 2Homo sapiens (human)3.075
Glutamate receptor 3Homo sapiens (human)3.075
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.23
Glutamate receptor 4Homo sapiens (human)3.075
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.23
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.23

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carcache, D; Kalkman, HO; Koller, M; Mattes, H1
Deverill, M; Hoo, KH; Iyengar, S; Li, DL; Ornstein, PL; Simmons, RM1
Vanover, KE1

Other Studies

3 other study(ies) available for ly 300164 and ly 293558

ArticleYear
alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) antagonists: from bench to bedside.
    Journal of medicinal chemistry, 2010, Aug-12, Volume: 53, Issue:15

    Topics: Analgesics; Animals; Anticonvulsants; Antipsychotic Agents; Clinical Trials as Topic; Drug Evaluation, Preclinical; Humans; Neuroprotective Agents; Protein Subunits; Receptors, AMPA

2010
Kainate GluR5 receptor subtype mediates the nociceptive response to formalin in the rat.
    Neuropharmacology, 1998, Volume: 37, Issue:1

    Topics: Animals; Benzodiazepines; Excitatory Amino Acid Antagonists; Formaldehyde; Humans; Isoquinolines; Male; Pain Threshold; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Kainic Acid; Tetrazoles

1998
Interaction of ethanol with excitatory amino acid receptor antagonists in mice.
    European journal of pharmacology, 1999, Mar-05, Volume: 368, Issue:2-3

    Topics: Animals; Ataxia; Behavior, Animal; Benzodiazepines; Central Nervous System Depressants; Chlordiazepoxide; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Excitatory Amino Acid Antagonists; Hypnotics and Sedatives; Isoquinolines; Male; Mice; Muscle Relaxation; Pentobarbital; Piperazines; Pregnanolone; Psychomotor Performance; Quinoxalines; Receptors, Glutamate; Tetrazoles

1999