Page last updated: 2024-09-05

ly 300164 and gyki 53655

ly 300164 has been researched along with gyki 53655 in 4 studies

Compound Research Comparison

Studies
(ly 300164)
Trials
(ly 300164)
Recent Studies (post-2010)
(ly 300164)
Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010) (gyki 53655)
73712111022

Protein Interaction Comparison

ProteinTaxonomyly 300164 (IC50)gyki 53655 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)1
Glutamate receptor 2Rattus norvegicus (Norway rat)1
Glutamate receptor 3Rattus norvegicus (Norway rat)1
Glutamate receptor 4Rattus norvegicus (Norway rat)1

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (50.00)18.2507
2000's2 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ballyk, BA; Bath, CP; Bleakman, D; Bufton, HR; Kamboj, RK; Lodge, D; Palmer, AJ; Schoepp, DD; Sharpe, EF; Tarnawa, I; Woolley, ML1
Cotton, JL; Partin, KM1
Gacsályi, I; Gigler, G; Gyertyán, I; Lévay, G; Szabados, T2

Other Studies

4 other study(ies) available for ly 300164 and gyki 53655

ArticleYear
Activity of 2,3-benzodiazepines at native rat and recombinant human glutamate receptors in vitro: stereospecificity and selectivity profiles.
    Neuropharmacology, 1996, Volume: 35, Issue:12

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Cell Line; Cerebellum; Cerebral Cortex; Excitatory Amino Acid Antagonists; Ganglia, Spinal; Humans; Kidney; Membrane Potentials; Molecular Structure; Neurons; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Recombinant Proteins; Spinal Cord; Structure-Activity Relationship; Transfection

1996
The contributions of GluR2 to allosteric modulation of AMPA receptors.
    Neuropharmacology, 2000, Volume: 39, Issue:1

    Topics: Allosteric Regulation; Amino Acid Substitution; Animals; Benzodiazepines; Benzothiadiazines; Cell Membrane; Excitatory Amino Acid Antagonists; Membrane Potentials; Oocytes; Receptors, AMPA; Recombinant Proteins; Xenopus laevis

2000
Duration of action of GYKI 52466 and its analogues in antiepileptic, anti-ischaemic and muscle relaxant tests.
    Neurobiology (Budapest, Hungary), 1999, Volume: 7, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Brain Ischemia; Epilepsy; Excitatory Amino Acid Antagonists; Mice; Muscle Relaxants, Central

1999
Comparison of anticonvulsive and acute neuroprotective activity of three 2,3-benzodiazepine compounds, GYKI 52466, GYKI 53405, and GYKI 53655.
    Brain research bulletin, 2001, Volume: 55, Issue:3

    Topics: Acoustic Stimulation; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Brain Ischemia; Dose-Response Relationship, Drug; Electroshock; Magnesium Chloride; Male; Mice; Mice, Inbred Strains; Neuroprotective Agents; Seizures; Survival Analysis; Time Factors

2001