Page last updated: 2024-09-03

ly 274614 and enkephalin, d-penicillamine (2,5)-

ly 274614 has been researched along with enkephalin, d-penicillamine (2,5)- in 3 studies

Compound Research Comparison

Studies
(ly 274614)
Trials
(ly 274614)
Recent Studies (post-2010)
(ly 274614)
Studies
(enkephalin, d-penicillamine (2,5)-)
Trials
(enkephalin, d-penicillamine (2,5)-)
Recent Studies (post-2010) (enkephalin, d-penicillamine (2,5)-)
960151,314073

Protein Interaction Comparison

ProteinTaxonomyly 274614 (IC50)enkephalin, d-penicillamine (2,5)- (IC50)
Mu-type opioid receptorHomo sapiens (human)0.0016
Delta-type opioid receptorHomo sapiens (human)0.0011

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bhargava, HN; Zhao, GM1
Bharagava, HN; Zhao, GM1
Bhargava, HN; Bian, JT; Cao, YJ1

Other Studies

3 other study(ies) available for ly 274614 and enkephalin, d-penicillamine (2,5)-

ArticleYear
Effect of antagonism of the NMDA receptor on tolerance to [D-Pen2,D-Pen5]enkephalin, a delta 1-opioid receptor agonist.
    Peptides, 1996, Volume: 17, Issue:2

    Topics: Analgesics; Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Tolerance; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Isoquinolines; Male; Mice; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, delta

1996
Effects of competitive and noncompetitive antagonists of the N-methyl-D-aspartate receptor on the analgesic action of delta 1- and delta 2-opioid receptor agonists in mice.
    British journal of pharmacology, 1996, Volume: 119, Issue:8

    Topics: Analgesics, Opioid; Animals; Antiparkinson Agents; Binding, Competitive; Dizocilpine Maleate; Dose-Response Relationship, Drug; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Excitatory Amino Acid Antagonists; Injections, Intraventricular; Isoquinolines; Male; Membranes; Mice; Oligopeptides; Pain Measurement; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, delta

1996
Effects of NMDA receptor antagonists on delta1- and delta2-opioid receptor agonists-induced changes in the mouse brain [3H]DPDPE binding.
    European journal of pharmacology, 1997, Sep-24, Volume: 335, Issue:2-3

    Topics: Animals; Brain; Dizocilpine Maleate; Down-Regulation; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Excitatory Amino Acid Antagonists; Isoquinolines; Male; Membranes; Mice; Oligopeptides; Protein Binding; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, delta

1997