Page last updated: 2024-09-03

ly 255283 and mocetinostat

ly 255283 has been researched along with mocetinostat in 3 studies

Compound Research Comparison

Studies
(ly 255283)
Trials
(ly 255283)
Recent Studies (post-2010)
(ly 255283)
Studies
(mocetinostat)
Trials
(mocetinostat)
Recent Studies (post-2010) (mocetinostat)
5401521,7353908,606

Protein Interaction Comparison

ProteinTaxonomyly 255283 (IC50)mocetinostat (IC50)
Histone deacetylase 3Homo sapiens (human)0.7851
Nuclear receptor corepressor 1Homo sapiens (human)0.022
Cytochrome P450 3A4Homo sapiens (human)0.57
Cytochrome P450 2D6Homo sapiens (human)0.102
Cytochrome P450 2C19Homo sapiens (human)0.102
Histone deacetylase 4Homo sapiens (human)0.5717
Histone deacetylase 1Homo sapiens (human)0.3433
Histone deacetylase 7Homo sapiens (human)0.6725
Histone deacetylase 2Homo sapiens (human)0.3537
Histone deacetylase 11 Homo sapiens (human)0.6386
Histone deacetylase 8Homo sapiens (human)0.6725
Histone deacetylase 6Homo sapiens (human)0.5717
Histone deacetylase 5Homo sapiens (human)0.6725
Nuclear receptor corepressor 2Homo sapiens (human)0.045

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Guo, JP; Karasawa, A; Lefer, AM; Ma, XL; Tsao, PS1
Fink, MP; Fleisch, JH; Menconi, MJ; O'Sullivan, BP; Wang, H; Wollert, PS; Youssef, ME1
Cara, DC; Coutinho, SF; Silveira, MR; Souza, DG; Teixeira, MM1

Other Studies

3 other study(ies) available for ly 255283 and mocetinostat

ArticleYear
Protective actions of a leukotriene B4 antagonist in splanchnic ischemia and reperfusion in rats.
    The American journal of physiology, 1991, Volume: 261, Issue:2 Pt 1

    Topics: Animals; Arteries; Blood Pressure; Cathepsin D; Constriction; Endothelium, Vascular; Ileum; Ischemia; Leukotriene B4; Male; Neutrophils; Peroxidase; Rats; Rats, Inbred Strains; Reperfusion; Splanchnic Circulation; Tetrazoles

1991
A novel leukotriene B4-receptor antagonist in endotoxin shock: a prospective, controlled trial in a porcine model.
    Critical care medicine, 1993, Volume: 21, Issue:12

    Topics: 6-Ketoprostaglandin F1 alpha; Animals; Bronchoalveolar Lavage Fluid; Disease Models, Animal; Drug Evaluation, Preclinical; Escherichia coli Infections; Extravascular Lung Water; Hemodynamics; Leukotriene B4; Male; Peroxidase; Proteins; Random Allocation; Respiratory Distress Syndrome; Shock, Septic; Swine; Tetrazoles; Thromboxane B2

1993
Effects of a BLT receptor antagonist on local and remote reperfusion injuries after transient ischemia of the superior mesenteric artery in rats.
    European journal of pharmacology, 2000, Sep-01, Volume: 403, Issue:1-2

    Topics: Animals; Antibodies, Monoclonal; Benzopyrans; Capillary Permeability; Carboxylic Acids; CD18 Antigens; Disease Models, Animal; Dose-Response Relationship, Drug; Evans Blue; Intestinal Mucosa; Intestines; Leukotriene Antagonists; Lung; Male; Mesenteric Artery, Superior; Mesentery; Neutrophils; Peroxidase; Polysaccharides; Rats; Rats, Wistar; Receptors, Leukotriene B4; Reperfusion Injury; Tetrazoles

2000