Page last updated: 2024-08-22

lutetium and triazoles

lutetium has been researched along with triazoles in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (14.29)29.6817
2010's5 (71.43)24.3611
2020's1 (14.29)2.80

Authors

AuthorsStudies
Banerjee, S; Chakraborty, S; Das, T; Kagiya, VT; Mukherjee, A; Nair, CK; Samuel, G; Sarma, HD; Venkatesh, M1
Adam, MJ; Bailey, GA; Boros, E; Ferreira, CL; Lacasse, MJ; Lewis, JS; Orvig, C; Patrick, BO; Price, EW; Zeglis, BM1
Huxol, E; Mindt, TL; Valverde, IE1
Fischer, CA; Mascarin, A; Mindt, TL; Valverde, IE; Vomstein, S1
Mascarin, A; Mindt, TL; Valverde, IE; Vomstein, S1
Almobarak, B; Altiparmak, G; Arvidsson, Y; Elf, AK; Elias, E; Forssell-Aronsson, E; Hofving, T; Johanson, V; Kristiansson, E; Nilsson, O; Sandblom, V; Shubbar, E; Swanpalmer, J1
Behe, M; Grob, NM; Mindt, TL; Schibli, R; Schmid, S1

Other Studies

7 other study(ies) available for lutetium and triazoles

ArticleYear
Preparation and preliminary biological evaluation of a 177Lu labeled sanazole derivative for possible use in targeting tumor hypoxia.
    Bioorganic & medicinal chemistry, 2004, Dec-01, Volume: 12, Issue:23

    Topics: Animals; Antineoplastic Agents; Drug Delivery Systems; Fibrosarcoma; Hypoxia; Lutetium; Mice; Neoplasms; Radioisotopes; Radiopharmaceuticals; Tissue Distribution; Triazoles

2004
H(2)azapa: a versatile acyclic multifunctional chelator for (67)Ga, (64)Cu, (111)In, and (177)Lu.
    Inorganic chemistry, 2012, Nov-19, Volume: 51, Issue:22

    Topics: Animals; Aza Compounds; Chelating Agents; Coordination Complexes; Copper Radioisotopes; Crystallography, X-Ray; Female; Gallium Radioisotopes; Heterocyclic Compounds, 1-Ring; Humans; Indium Radioisotopes; Lutetium; Mice; Mice, Nude; Models, Molecular; Molecular Structure; Positron-Emission Tomography; Radioisotopes; Radiopharmaceuticals; Tissue Distribution; Triazoles

2012
Radiolabeled antagonistic bombesin peptidomimetics for tumor targeting.
    Journal of labelled compounds & radiopharmaceuticals, 2014, Volume: 57, Issue:4

    Topics: Amino Acid Sequence; Bombesin; Cell Line, Tumor; Heterocyclic Compounds, 1-Ring; Humans; Isotope Labeling; Lutetium; Male; Peptide Fragments; Peptidomimetics; Prostatic Neoplasms; Proteolysis; Radioisotopes; Tomography, Emission-Computed, Single-Photon; Triazoles

2014
Probing the Backbone Function of Tumor Targeting Peptides by an Amide-to-Triazole Substitution Strategy.
    Journal of medicinal chemistry, 2015, Sep-24, Volume: 58, Issue:18

    Topics: Amides; Animals; Bombesin; Cell Line, Tumor; Heterografts; Humans; Lutetium; Mice, Nude; Neoplasm Transplantation; Peptide Fragments; Peptidomimetics; Proteolysis; Radiopharmaceuticals; Receptors, Bombesin; Structure-Activity Relationship; Tissue Distribution; Triazoles

2015
1,2,3-Triazole Stabilized Neurotensin-Based Radiopeptidomimetics for Improved Tumor Targeting.
    Bioconjugate chemistry, 2015, Oct-21, Volume: 26, Issue:10

    Topics: Animals; Antineoplastic Agents; Chemistry Techniques, Synthetic; Cycloaddition Reaction; Female; Half-Life; HT29 Cells; Humans; Isotope Labeling; Lutetium; Mice, Nude; Molecular Targeted Therapy; Neurotensin; Peptide Fragments; Peptidomimetics; Radioisotopes; Receptors, Neurotensin; Structure-Activity Relationship; Tissue Distribution; Triazoles; Xenograft Model Antitumor Assays

2015
177Lu-octreotate therapy for neuroendocrine tumours is enhanced by Hsp90 inhibition.
    Endocrine-related cancer, 2019, 04-01, Volume: 26, Issue:4

    Topics: Adult; Aged; Aged, 80 and over; Animals; Antineoplastic Agents; Female; HSP90 Heat-Shock Proteins; Humans; Lutetium; Male; Mice, Inbred BALB C; Mice, Nude; Middle Aged; Neuroendocrine Tumors; Octreotide; Radiopharmaceuticals; Triazoles; Tumor Cells, Cultured

2019
Design of Radiolabeled Analogs of Minigastrin by Multiple Amide-to-Triazole Substitutions.
    Journal of medicinal chemistry, 2020, 05-14, Volume: 63, Issue:9

    Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Drug Design; Gastrins; Humans; Lutetium; Mice; Neoplasms; Peptidomimetics; Protein Binding; Radioisotopes; Radiopharmaceuticals; Receptor, Cholecystokinin B; Triazoles

2020
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