Page last updated: 2024-09-05

lurasidone and aripiprazole

lurasidone has been researched along with aripiprazole in 3 studies

Compound Research Comparison

Studies
(lurasidone)
Trials
(lurasidone)
Recent Studies (post-2010)
(lurasidone)
Studies
(aripiprazole)
Trials
(aripiprazole)
Recent Studies (post-2010) (aripiprazole)
6032,9895091,788

Protein Interaction Comparison

ProteinTaxonomylurasidone (IC50)aripiprazole (IC50)
ATP-dependent translocase ABCB1Homo sapiens (human)0.78
D(2) dopamine receptorHomo sapiens (human)0.0158
5-hydroxytryptamine receptor 2AHomo sapiens (human)1.945
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.38
Alpha-1A adrenergic receptorHomo sapiens (human)0.17
Histamine H1 receptorHomo sapiens (human)0.42
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.8572

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's2 (66.67)2.80

Authors

AuthorsStudies
Azmanova, M; Barry, NPE; Pitto-Barry, A1
Altamura, C; Arzuaga, A; Ciranna, L; Costa, L; Desaphy, JF; Lacivita, E; Leopoldo, M; Niso, M; Ragozzino, ME; Stama, ML1
Ablordeppey, SY; Bloom, SH; Bricker, B; Eshleman, AJ; Gonela, UM; Janowsky, AJ; Ofori, E; Onyameh, EK; Schmachtenberg, JL; Swanson, TL; Voshavar, C1

Reviews

1 review(s) available for lurasidone and aripiprazole

ArticleYear
Schizophrenia: synthetic strategies and recent advances in drug design.
    MedChemComm, 2018, May-01, Volume: 9, Issue:5

    Topics:

2018

Other Studies

2 other study(ies) available for lurasidone and aripiprazole

ArticleYear
Privileged scaffold-based design to identify a novel drug-like 5-HT
    European journal of medicinal chemistry, 2020, Aug-01, Volume: 199

    Topics: Dose-Response Relationship, Drug; Drug Design; Fragile X Syndrome; HEK293 Cells; Humans; Molecular Structure; Piperazines; Receptors, Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship

2020
New dual 5-HT1A and 5-HT7 receptor ligands derived from SYA16263.
    European journal of medicinal chemistry, 2021, Mar-15, Volume: 214

    Topics: Dose-Response Relationship, Drug; Humans; Ligands; Molecular Structure; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Structure-Activity Relationship

2021