Page last updated: 2024-09-05

lu 25-109 and xanomeline

lu 25-109 has been researched along with xanomeline in 3 studies

Compound Research Comparison

Studies
(lu 25-109)
Trials
(lu 25-109)
Recent Studies (post-2010)
(lu 25-109)
Studies
(xanomeline)
Trials
(xanomeline)
Recent Studies (post-2010) (xanomeline)
14211241641

Protein Interaction Comparison

ProteinTaxonomylu 25-109 (IC50)xanomeline (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.1644
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.0251
Muscarinic acetylcholine receptor M1Homo sapiens (human)1.3967

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's1 (33.33)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Allen, JR; Bures, MG; Bymaster, F; Croy, CH; Evans, D; Felder, CC; Hansen, MM; Hitchcock, SA; Hoogestraat, PJ; Jamison, JA; Liu, B; McKinzie, DL; Okha-Mokube, FM; Rao, Z; Stratford, RE; Stuart Gregory, G; Turner, W; Watt, ML1
Bymaster, FP; Calligaro, DO; Carter, PA; DeLapp, N; Fink-Jensen, A; Jeppesen, L; Mitch, CH; Peters, SC; Rimvall, K; Sauerberg, P; Shannon, HE; Sheardown, MJ; Ward, JS; Whitesitt, CA; Zhang, W1
Anderton, BH; Dayanandan, R; Forlenza, OV; Lovestone, S; Olesen, OF; Spink, JM1

Other Studies

3 other study(ies) available for lu 25-109 and xanomeline

ArticleYear
Design and synthesis of N-[6-(Substituted Aminoethylideneamino)-2-Hydroxyindan-1-yl]arylamides as selective and potent muscarinic M₁ agonists.
    Bioorganic & medicinal chemistry letters, 2015, Oct-01, Volume: 25, Issue:19

    Topics: Amides; Animals; Dose-Response Relationship, Drug; Drug Design; Humans; Molecular Structure; Rats; Receptor, Muscarinic M1; Structure-Activity Relationship

2015
Xanomeline compared to other muscarinic agents on stimulation of phosphoinositide hydrolysis in vivo and other cholinomimetic effects.
    Brain research, 1998, Jun-08, Volume: 795, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain Chemistry; Bridged Bicyclo Compounds, Heterocyclic; Cholinergic Agents; Cholinesterase Inhibitors; Dihydropyridines; Dose-Response Relationship, Drug; Hydrolysis; Hypothermia; Imines; Lithium; Male; Mice; Mice, Inbred Strains; Muscarinic Agonists; Oximes; Parasympathomimetics; Phosphatidylinositols; Physostigmine; Pilocarpine; Pyridines; Quinuclidines; Radioligand Assay; Salivation; Tacrine; Tetrazoles; Thiadiazoles; Tremor

1998
Muscarinic agonists reduce tau phosphorylation in non-neuronal cells via GSK-3beta inhibition and in neurons.
    Journal of neural transmission (Vienna, Austria : 1996), 2000, Volume: 107, Issue:10

    Topics: Acetylcholine; Alzheimer Disease; Amyloid beta-Protein Precursor; Animals; Binding Sites; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cells, Cultured; Fetus; Glycogen Synthase Kinase 3; Glycogen Synthase Kinases; Lithium Chloride; Microtubules; Muscarinic Agonists; Neurons; Phosphorylation; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; tau Proteins; Tetrazoles; Thiadiazoles

2000