lu 25-109 has been researched along with arecoline in 1 studies
Studies (lu 25-109) | Trials (lu 25-109) | Recent Studies (post-2010) (lu 25-109) | Studies (arecoline) | Trials (arecoline) | Recent Studies (post-2010) (arecoline) |
---|---|---|---|---|---|
14 | 2 | 1 | 1,110 | 20 | 271 |
Protein | Taxonomy | lu 25-109 (IC50) | arecoline (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | 3.6 | |
Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | 1.011 | |
Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | 0.963 | |
Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | 0.963 | |
Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | 0.963 | |
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 0.9163 | |
Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | 0.115 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bøgesø, KP; Frederiksen, K; Løve Lembøl, H; Meier, E; Moltzen, EK; Pedersen, H; Sánchez, C | 1 |
1 other study(ies) available for lu 25-109 and arecoline
Article | Year |
---|---|
Bioisosteres of arecoline: 1,2,3,6-tetrahydro-5-pyridyl-substituted and 3-piperidyl-substituted derivatives of tetrazoles and 1,2,3-triazoles. Synthesis and muscarinic activity.
Topics: Animals; Arecoline; Female; Guinea Pigs; Male; Mice; Rats; Rats, Wistar; Structure-Activity Relationship; Tetrazoles; Triazoles | 1994 |