Page last updated: 2024-08-24

loxiglumide and sincalide

loxiglumide has been researched along with sincalide in 45 studies

Research

Studies (45)

TimeframeStudies, this research(%)All Research%
pre-19904 (8.89)18.7374
1990's36 (80.00)18.2507
2000's5 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bishop, LA; Black, JW; Gerskowitch, VP; Hull, RA; Shankley, NP1
Almegård, B; Bill, A; Stjernschantz, J1
Bennett, A; D'Amato, M; Stamford, IF1
Baba, H; Fujimura, M; Toda, N1
Baba, S; Fujii, M; Fujisawa, T; Koide, M; Nakamura, T; Okabayashi, Y; Otsuki, M; Tani, S2
Bogdal, J; Konturek, JW; Konturek, SJ; Kurek, A; Oleksy, J; Rovati, L1
Beglinger, C; Gyr, K; Hildebrand, P; Köhler, E; Setnikar, I1
Ito, H; Kadowaki, M; Matsuo, M; Nakarai, T; Sato, Y; Sogabe, H; Tokoro, K; Tomoi, M; Yoshida, K1
Kashima, K; Kataoka, K; Kato, M; Kuriyama, K; Mukainaka, T; Ohkuma, S1
Moriyoshi, Y; Shiratori, K; Takeuchi, T; Watanabe, S1
Fölsch, UR; Höcker, M; Hughes, J; Schmidt, WE1
Fujii, K; Haruma, K; Kajiyama, G; Kishimoto, S; Kobayashi, H; Machino, H; Miyoshi, A1
Chey, WY; Imamura, M; Yamauchi, H1
Aufderhaar, U; Bauerfeind, P; Beglinger, C; Burckhardt, B; Delco, F; Ensinck, JW; Gyr, K; Ketterer, S; Meier, R1
Nakano, S; Otsuki, M; Tachibana, I1
Akiyama, T; Otsuki, M1
Beglinger, C1
Bekkering, M; Chua, AS; Keeling, PW; Rovati, LC1
Fukumoto, M; Hayashi, H; Imamura, M; Kawabata, K; Manabe, T; Masai, Y; Morimoto, H; Nio, Y; Tsubono, M1
Funakoshi, A; Miyasaka, K; Nakamura, E; Teraoka, H1
Rakovska, A2
Brotschi, EA; Hilbinger, CL; Kahl, EA; Midis, NA; Vaules, WA1
Arii, S; Funaki, N; Imamura, M; Imamura, T; Kohmoto, M; Ohshio, G; Okada, N; Sasaoki, T; Tanaka, J; Tanaka, T; Wang, ZH; Yoshida, M1
Akiyama, T; Hirohata, Y; Otsuki, M; Shirohara, H; Tachibana, I; Yamamoto, M1
D'Amato, M; Kisfalvi, I; Scarpignato, C; Varga, G1
Endo, T; Nagasaki, M; Taniguchi, H; Yazaki, N1
Beglinger, C; Hartel, M; Niebergall-Roth, E; Riepl, RL; Singer, MV; Teyssen, S; Wetzel, D1
Endo, T; Nagasaki, M; Shikano, T; Taniguchi, H; Yazaki, N; Yomota, E1
Hanada, K; Hirata, M; Itoh, M; Kajiyama, G; Ooishi, H; Tsuchida, A1
Kondo, T; Liu, F; Naruse, S; Ozaki, T; Sazi, T; Toda, Y1
Adler, G; Beckh, K; Dirks, A; Koop, H; Koop, I1
Kihara, Y; Nakano, S; Otsuki, M1
Hayashi, K; Kannbe, M; Kishimoto, S1
Azpiroz, F; Clavé, P; Cussó, X; D'Amato, M; Farré, A; González, A; Lluís, F; López, R; Moreno, A1
Domschke, W; Hengst, K; Konturek, JW; Konturek, SJ; Sito, E; Stachura, J1
Brzozowska, I; Brzozowski, T; Hahn, EG; Konturek, PC; Konturek, SJ; Kwiecién, S; Pajdo, R1
Akiyama, T; Hirohata, Y; Kihara, Y; Otsuki, M; Tashiro, M1
Brzozowski, T; Drozdowicz, D; Hahn, EG; Konturek, PC; Konturek, SJ; Kwiecień, S; Pajdo, R1
Beglinger, C; Drewe, J; Gutzwiller, JP; Hildebrand, P; Ketterer, S; Krautheim, A1
Capellà, G; Clavé, P; Farré, R; González, AA; Monés, J1
Akiyama, T; Fukumitsu, K; Jia, DM; Otani, M; Otsuki, M; Yamamoto, M; Yoshikawa, H1
Mostofsky, DI; Yehuda, S1
Aloj, L; De Luca, S; Lassiani, L; Morelli, G; Saviano, M; Stefanidou, P; Varnavas, A; Yannakopoulou, K1

Reviews

1 review(s) available for loxiglumide and sincalide

ArticleYear
Effect of cholecystokinin on gastric motility in humans.
    Annals of the New York Academy of Sciences, 1994, Mar-23, Volume: 713

    Topics: Benzodiazepinones; Cholecystokinin; Colon; Devazepide; Digestive System; Digestive System Physiological Phenomena; Duodenum; Gastric Emptying; Gastrointestinal Motility; Humans; Ileum; Infusions, Intravenous; Proglumide; Receptors, Cholecystokinin; Sincalide

1994

Trials

4 trial(s) available for loxiglumide and sincalide

ArticleYear
Cholecystokinin is a physiological regulator of gastric acid secretion in man.
    European journal of clinical investigation, 1994, Volume: 24, Issue:6

    Topics: Adult; Cholecystokinin; Dose-Response Relationship, Drug; Drug Interactions; Eating; Gastric Acid; Gastric Mucosa; Gastrins; Homeostasis; Hormones; Humans; Male; Middle Aged; Proglumide; Sincalide; Somatostatin

1994
Clinical efficacy and prokinetic effect of the CCK-A antagonist loxiglumide in nonulcer dyspepsia.
    Annals of the New York Academy of Sciences, 1994, Mar-23, Volume: 713

    Topics: Adult; Analysis of Variance; Double-Blind Method; Dyspepsia; Female; Gastric Emptying; Humans; Male; Middle Aged; Proglumide; Receptors, Cholecystokinin; Sincalide; Time Factors

1994
Physiological role of cholecystokinin in gastroprotection in humans.
    The American journal of gastroenterology, 1998, Volume: 93, Issue:12

    Topics: Adult; Cholecystokinin; Double-Blind Method; Duodenum; Ethanol; Gastric Mucosa; Gastroscopy; Hormone Antagonists; Humans; Injections, Intravenous; Male; Oleic Acid; Proglumide; Sincalide; Somatostatin; Stomach

1998
Interaction between CCK and a preload on reduction of food intake is mediated by CCK-A receptors in humans.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2000, Volume: 279, Issue:1

    Topics: Adult; Cholecystokinin; Cross-Over Studies; Double-Blind Method; Eating; Energy Intake; Humans; Hunger; Infusions, Intravenous; Male; Proglumide; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Satiety Response; Sincalide

2000

Other Studies

40 other study(ies) available for loxiglumide and sincalide

ArticleYear
Combined dose-ratio analysis of cholecystokinin receptor antagonists, devazepide, lorglumide and loxiglumide in the guinea-pig gall bladder.
    British journal of pharmacology, 1992, Volume: 106, Issue:1

    Topics: Analysis of Variance; Animals; Benzodiazepinones; Binding, Competitive; Biological Assay; Cholecystokinin; Devazepide; Dose-Response Relationship, Drug; Gallbladder; Guinea Pigs; Muscle, Smooth; Pentagastrin; Proglumide; Receptors, Cholecystokinin; Sincalide

1992
Cholecystokinin contracts isolated human and monkey iris sphincters; a study with CCK receptor antagonists.
    European journal of pharmacology, 1992, Feb-11, Volume: 211, Issue:2

    Topics: Aged; Aged, 80 and over; Animals; Cholecystokinin; Female; Humans; In Vitro Techniques; Iris; Macaca fascicularis; Male; Middle Aged; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide

1992
Studies of three non-peptide cholecystokinin antagonists (devazepide, lorglumide and loxiglumide) in human isolated alimentary muscle and guinea-pig ileum.
    British journal of pharmacology, 1991, Volume: 102, Issue:2

    Topics: Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Digestive System; Digestive System Physiological Phenomena; Female; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide

1991
Mechanism of inhibitory action of peptide YY on cholecystokinin-induced contractions of isolated dog ileum.
    Regulatory peptides, 1990, Feb-04, Volume: 27, Issue:2

    Topics: Animals; Cholecystokinin; Dogs; Female; Gallbladder; Glutamine; Ileum; Isometric Contraction; Male; Muscle Contraction; Peptide YY; Peptides; Proglumide; Sincalide

1990
Loxiglumide. A new proglumide analog with potent cholecystokinin antagonistic activity in the rat pancreas.
    Digestive diseases and sciences, 1989, Volume: 34, Issue:6

    Topics: Amylases; Animals; Binding, Competitive; Cholecystokinin; Dose-Response Relationship, Drug; Glutamine; Pancreas; Proglumide; Rats; Receptors, Cholecystokinin; Sincalide

1989
[Inhibitory effect of a new proglumide derivative, loxiglumide, on CCK action in isolated rat pancreatic acini].
    Nihon Shokakibyo Gakkai zasshi = The Japanese journal of gastro-enterology, 1989, Volume: 86, Issue:1

    Topics: Amylases; Animals; Cholecystokinin; Glutamine; In Vitro Techniques; Male; Pancreas; Proglumide; Rats; Rats, Inbred Strains; Sincalide

1989
CCK receptor antagonism by loxiglumide and gall bladder contractions in response to cholecystokinin, sham feeding and ordinary feeding in man.
    Gut, 1989, Volume: 30, Issue:8

    Topics: Adolescent; Adult; Cholecystokinin; Food; Gallbladder; Glutamine; Humans; Male; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide

1989
Biological effects of a proglumide derivative as cholecystokinin antagonist in conscious dogs.
    Regulatory peptides, 1987, Aug-17, Volume: 18, Issue:3-4

    Topics: Animals; Cholecystokinin; Dogs; Dose-Response Relationship, Drug; Gastric Acid; Glutamine; Infusions, Intravenous; Pancreatic Juice; Pancreatic Polypeptide; Pentagastrin; Proglumide; Sincalide

1987
Pharmacological profile of FK480, a novel cholecystokinin type-A receptor antagonist: comparison to loxiglumide.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:2

    Topics: Amylases; Animals; Benzodiazepinones; Female; Gastric Emptying; Guinea Pigs; Indoles; Male; Mice; Mice, Inbred ICR; Proglumide; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide

1994
Mechanisms for pancreatic hypertrophy induced by long-term administration of bethanechol.
    European journal of pharmacology, 1994, Nov-01, Volume: 292, Issue:1

    Topics: Amylases; Animals; Atropine; Bethanechol; Cholinergic Agonists; Cholinergic Antagonists; Drug Administration Schedule; Drug Interactions; Gastrins; Hypertrophy; Male; Organ Size; Pancreas; Pentagastrin; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide

1994
Effect of a novel cholecystokinin receptor antagonist, FK480, administered intraduodenally, on pancreatic secretion in rats.
    Pancreas, 1995, Volume: 10, Issue:3

    Topics: Amylases; Animals; Benzodiazepinones; Caseins; Duodenum; Indoles; Male; Pancreas; Pancreatic Juice; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide

1995
PD 135158, a CCKB/gastrin receptor antagonist, stimulates rat pancreatic enzyme secretion as a CCKA receptor agonist.
    European journal of pharmacology, 1993, Sep-21, Volume: 242, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Cholecystokinin; Drug Interactions; Indoles; Lipase; Meglumine; Pancreas; Proglumide; Rats; Sincalide

1993
Inhibitory action of CCK-OP on rat proximal colon.
    Annals of the New York Academy of Sciences, 1994, Mar-23, Volume: 713

    Topics: Acetylcholine; Animals; Atropine; Colon; Fasting; Hexamethonium; Hexamethonium Compounds; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Proglumide; Rats; Receptors, Cholecystokinin; Sincalide

1994
Effect of intraduodenal infusion of tocamphyl on pancreatic exocrine secretion and gastrointestinal hormone release in rats.
    International journal of pancreatology : official journal of the International Association of Pancreatology, 1994, Volume: 15, Issue:3

    Topics: Analysis of Variance; Animals; Atropine; Bile; Camphor; Cholagogues and Choleretics; Cholecystokinin; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Gastrointestinal Hormones; Male; Pancreatic Juice; Proglumide; Radioimmunoassay; Rats; Rats, Wistar; Secretin; Sincalide

1994
Treatment with cholecystokinin receptor antagonist loxiglumide enhances insulin response to intravenous glucose stimulation in postpancreatitic rats.
    Regulatory peptides, 1994, Jul-14, Volume: 52, Issue:2

    Topics: Acute Disease; Animals; Ceruletide; Glucose; Injections, Intravenous; Injections, Subcutaneous; Insulin; Insulin Resistance; Insulin Secretion; Islets of Langerhans; Male; Pancreatitis; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide

1994
Characterization of a new cholecystokinin receptor antagonist FK480 in in vitro isolated rat pancreatic acini.
    Pancreas, 1994, Volume: 9, Issue:3

    Topics: Animals; Benzodiazepinones; Devazepide; In Vitro Techniques; Indoles; Male; Pancreas; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide

1994
Loxiglumide (CR1505), a cholecystokinin antagonist, specifically inhibits the growth of human pancreatic cancer lines xenografted into nude mice.
    Cancer, 1993, Dec-15, Volume: 72, Issue:12

    Topics: Animals; Cell Division; Chloroquine; Cholecystokinin; DNA; Esters; Gabexate; Guanidines; Humans; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplasm Transplantation; Organ Culture Techniques; Pancreatic Neoplasms; Proglumide; Sincalide; Transplantation, Heterologous

1993
Regulation of gene expression of pancreatic secretory trypsin inhibitor-61 and -56 by bile and pancreatic juice in rats.
    Pancreas, 1995, Volume: 11, Issue:3

    Topics: Animals; Base Sequence; Bile; Biliopancreatic Diversion; Ceruletide; Cholecystokinin; Gastrointestinal Agents; Gene Expression; Hormone Antagonists; Infusions, Intravenous; Male; Molecular Sequence Data; Pancreas; Pancreatic Juice; Proglumide; Rats; Rats, Wistar; RNA, Messenger; Sincalide; Trypsin Inhibitor, Kazal Pancreatic

1995
Cholecystokinin [corrected] octapeptide modulates dopamine release in rat striatum.
    Neuroscience letters, 1995, Aug-11, Volume: 195, Issue:3

    Topics: Animals; Anti-Ulcer Agents; Apomorphine; Dopamine; Dopamine Agonists; Electric Stimulation; Hormone Antagonists; Male; Neostriatum; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Tritium

1995
Cholecystokinin-GABA interactions in rat striatum.
    Neuropeptides, 1995, Volume: 29, Issue:5

    Topics: Animals; Calcium; Cholecystokinin; Corpus Striatum; Electric Stimulation; gamma-Aminobutyric Acid; Hormone Antagonists; Indoles; Male; Meglumine; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Tetrodotoxin; Tritium

1995
Luminal cholecystokinin and gastrin cause gallbladder contraction.
    The Journal of surgical research, 1996, Volume: 62, Issue:2

    Topics: Animals; Bile; Cholecystokinin; Female; Gallbladder; Gastrins; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Muscle Contraction; Pentagastrin; Proglumide; Receptors, Cholecystokinin; Sincalide

1996
Effects of cholecystokinin and carbachol on membrane fluidity in pancreatic acini.
    Digestive diseases and sciences, 1996, Volume: 41, Issue:7

    Topics: Animals; Bombesin; Carbachol; Cholecystokinin; Dose-Response Relationship, Drug; Hormone Antagonists; L-Lactate Dehydrogenase; Male; Membrane Fluidity; Pancreas; Pancreatitis; Phosphatidylcholines; Proglumide; Rats; Rats, Wistar; Secretin; Sincalide

1996
Pharmacological profile of TP-680, a new cholecystokininA receptor antagonist.
    British journal of pharmacology, 1996, Volume: 117, Issue:7

    Topics: Amylases; Animals; Benzodiazepinones; Binding, Competitive; Cerebral Cortex; Cysteine; Devazepide; In Vitro Techniques; Intracellular Membranes; Male; Niacin; Pancreas; Proglumide; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide

1996
Effect of dexloxiglumide and spiroglumide, two new CCK-receptor antagonists, on gastric emptying and secretion in the rat: evaluation of their receptor selectivity in vivo.
    Alimentary pharmacology & therapeutics, 1996, Volume: 10, Issue:3

    Topics: Animals; Dose-Response Relationship, Drug; Gastric Acid; Gastric Emptying; Hormone Antagonists; Keto Acids; Male; Pentagastrin; Pentanoic Acids; Proglumide; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide; Spiro Compounds

1996
Pharmacological profile of T-0632, a novel potent and selective CCKA receptor antagonist, in vitro.
    European journal of pharmacology, 1996, May-23, Volume: 304, Issue:1-3

    Topics: Amylases; Animals; Benzodiazepinones; Binding, Competitive; Brain; Cell Membrane; Devazepide; Gallbladder; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Pancreas; Proglumide; Protein Binding; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide

1996
Comparison of the effects of two cholecystokinin-receptor antagonists, loxiglumide and L-364,718, on the pancreatic secretory response to intraduodenal tryptophan in dogs.
    Scandinavian journal of gastroenterology, 1996, Volume: 31, Issue:7

    Topics: Animals; Benzodiazepinones; Bicarbonates; Cholecystokinin; Devazepide; Dogs; Duodenum; Female; Male; Pancreas; Perfusion; Proglumide; Receptors, Cholecystokinin; Secretin; Sincalide; Tryptophan

1996
Pharmacological profile of T-0632, a novel potent and selective CCKA receptor antagonist, in vivo.
    European journal of pharmacology, 1996, Sep-26, Volume: 312, Issue:2

    Topics: Animals; Benzodiazepinones; Ceruletide; Devazepide; Dogs; Female; Gastric Emptying; Indoles; Male; Pancreas; Pancreatitis; Pregnancy; Proglumide; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide

1996
Cholecystokinin receptor antagonist, loxiglumide, inhibits invasiveness of human pancreatic cancer cell lines.
    FEBS letters, 1996, Apr-01, Volume: 383, Issue:3

    Topics: Blotting, Western; Cell Line; Collagenases; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Gelatin; Hormone Antagonists; Humans; Kinetics; Matrix Metalloproteinase 9; Neoplasm Invasiveness; Pancreatic Neoplasms; Proglumide; Sincalide; Tumor Cells, Cultured

1996
Effect of gastrin-releasing peptide (GRP) on guinea pig gallbladder contraction in vitro.
    Journal of gastroenterology, 1995, Volume: 30, Issue:6

    Topics: Acetylcholine; Animals; Atropine; Bombesin; Dose-Response Relationship, Drug; Gallbladder; Gastrin-Releasing Peptide; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Peptides; Proglumide; Sincalide

1995
Impairment of hepatic transport processes in perfused rat liver by the specific CCK receptor antagonist loxiglumide.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1997, Volume: 197, Issue:3

    Topics: Animals; Bile; Biological Transport; Cholagogues and Choleretics; Gastrins; Hormone Antagonists; Indocyanine Green; Leukotriene D4; Liver; Male; Portal Vein; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Taurocholic Acid

1997
CCK administration after CCK receptor blockade accelerates recovery from cerulein-induced acute pancreatitis in rats.
    Pancreas, 1998, Volume: 16, Issue:2

    Topics: Acute Disease; Amylases; Animals; Ceruletide; Cholecystokinin; DNA; Hormone Antagonists; Lipase; Male; Organ Size; Pancreas; Pancreatitis; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Regeneration; Sincalide; Trypsin

1998
Endogenous CCK inhibits colonic contractions in unrestrained conscious rats.
    Regulatory peptides, 1997, Oct-31, Volume: 72, Issue:2-3

    Topics: Animal Feed; Animals; Colon; Dose-Response Relationship, Drug; Duodenum; Eating; Fasting; Gastrointestinal Motility; Hormone Antagonists; Intubation, Gastrointestinal; Male; Muscle Contraction; Muscle, Smooth; Portal Vein; Proglumide; Radioimmunoassay; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Reference Values; Sincalide; Telemetry; Transducers

1997
Endogenous cholecystokinin enhances postprandial gastroesophageal reflux in humans through extrasphincteric receptors.
    Gastroenterology, 1998, Volume: 115, Issue:3

    Topics: Adult; Cholecystokinin; Cholestyramine Resin; Eating; Electric Stimulation; Esophagogastric Junction; Esophagus; Gallbladder; Gastroesophageal Reflux; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Proglumide; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide

1998
Involvement of endogenous cholecystokinin and somatostatin in gastroprotection induced by intraduodenal fat.
    Journal of clinical gastroenterology, 1998, Volume: 27 Suppl 1

    Topics: Animals; Capsaicin; Cholecystokinin; Denervation; Dinoprostone; Dopamine Agents; Enzyme Inhibitors; Gastric Acid; Gastric Mucosa; Hormone Antagonists; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oleic Acid; Pepsin A; Proglumide; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide; Somatostatin; Stomach Ulcer; Vagotomy

1998
Pharmacologic profile of TS-941, a new benzodiazepine derivative cholecystokinin-receptor antagonist, in in vitro isolated rat pancreatic acini.
    Pancreas, 1999, Volume: 18, Issue:2

    Topics: Amylases; Animals; Benzodiazepines; Binding, Competitive; Cell Membrane; Cell Survival; Cells, Cultured; Cerebral Cortex; Devazepide; Dose-Response Relationship, Drug; Hormone Antagonists; Male; Pancreas; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide

1999
Acceleration of ulcer healing by cholecystokinin (CCK): role of CCK-A receptors, somatostatin, nitric oxide and sensory nerves.
    Regulatory peptides, 1999, Jun-30, Volume: 82, Issue:1-3

    Topics: Animals; Cholecystokinin; DNA Replication; Dopamine Agents; Esters; Gabexate; Gastric Mucosa; Gastrins; Guanidines; Hormone Antagonists; Male; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Pancreatin; Proglumide; Protease Inhibitors; Rats; Rats, Wistar; Receptors, Cholecystokinin; Regional Blood Flow; RNA, Messenger; Sensory Receptor Cells; Sincalide; Somatostatin; Stomach; Stomach Ulcer

1999
Pharmacological and molecular characterization of muscular cholecystokinin receptors in the human lower oesophageal sphincter.
    Neurogastroenterology and motility, 2000, Volume: 12, Issue:6

    Topics: Adult; Aged; Benzodiazepines; Benzodiazepinones; Esophagogastric Junction; Female; Gastric Emptying; Gastrins; Gastrointestinal Agents; Gene Expression; Hormone Antagonists; Humans; In Vitro Techniques; Indoleacetic Acids; Male; Middle Aged; Phenylurea Compounds; Proglumide; Receptors, Cholecystokinin; Restriction Mapping; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sincalide; Thiazoles

2000
Differential mechanism and site of action of CCK on the pancreatic secretion and growth in rats.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 285, Issue:4

    Topics: Afferent Pathways; Amylases; Animals; Capsaicin; Cholecystokinin; Duodenum; Eating; Lipase; Male; Organ Size; Pancreas; Proglumide; Rats; Rats, Wistar; Sincalide; Trypsin; Trypsinogen; Vagotomy; Vagus Nerve

2003
The effects of an essential fatty acid compound and a cholecystokinin-8 antagonist on iron deficiency induced anorexia and learning deficits.
    Nutritional neuroscience, 2004, Volume: 7, Issue:2

    Topics: Animal Feed; Animals; Avoidance Learning; Cholecystokinin; Energy Intake; Hormone Antagonists; Iron Deficiencies; Islets of Langerhans; Linoleic Acid; Male; Motor Activity; Peptide Fragments; Proglumide; Rats; Rats, Long-Evans; Swimming; Weight Gain

2004
Anthranilic acid based CCK1 receptor antagonists and CCK-8 have a common step in their "receptor desmodynamic processes".
    Journal of medicinal chemistry, 2006, Apr-20, Volume: 49, Issue:8

    Topics: Animals; Binding, Competitive; Biological Assay; Humans; Indoles; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Structure; ortho-Aminobenzoates; Pancreas; Proglumide; Protein Conformation; Rats; Receptor, Cholecystokinin A; Sincalide; Spectrometry, Fluorescence; Structure-Activity Relationship

2006