losartan has been researched along with pd 123177 in 111 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 104 (93.69) | 18.2507 |
2000's | 6 (5.41) | 29.6817 |
2010's | 1 (0.90) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Benfield, P; Chiu, AT; Herblin, WF; Smith, RD; Timmermans, PB; Wong, PC | 1 |
Achard, JM; Gardin, JP; Houillier, P; Lazar, G; Paillard, M; Poggioli, J | 1 |
Ambühl, P; Felix, D; Ferrario, CM; Imboden, H; Khosla, MC | 1 |
Aguilera, G | 1 |
Fujimoto, M; Itazaki, K; Mihara, S; Shigeri, Y | 1 |
Chang, RS; Chiu, AT; Leung, KH; Lotti, VJ; Roscoe, WA; Smith, RD; Timmermans, PB | 1 |
Abdelrahman, A; Pang, CC | 1 |
Christ, DD; Timmermans, PB; Wong, PC | 1 |
Bennett, T; Gardiner, SM; Kemp, PA; Widdop, RE | 2 |
Phillips, MI; Renaud, LP; Yang, CR | 1 |
Kang, J; Posner, P; Sumners, C | 1 |
Gonzales, N; Hornsby, PJ; Nadler, J; Natarajan, R | 1 |
García-Sáinz, JA; González-Espinosa, C | 1 |
Hogarty, DC; Phillips, MI; Puig, V; Speakman, EA | 1 |
Chiu, AT; Herblin, WF; Smith, RD; Timmermans, PB; Wong, PC | 2 |
Grady, EF; Griffin, CA; Kalinyak, JE; Schambelan, M; Sechi, LA | 2 |
Allen, AM; Mendelsohn, FA; Paxinos, G; Song, K | 1 |
Rowe, BP; Saylor, DL; Speth, RC | 1 |
Bernard, R; Timmermans, PB; Wong, PC | 1 |
Christ, DD; Duncia, JV; Pierce, SK; Reilly, TM; Timmermans, PB | 1 |
Saavedra, JM; Strömberg, C; Tsutsumi, K; Viswanathan, M | 1 |
Bunting, PB; Cartwright, ME; Frank, JD; Gibson, RE; Schorn, TW; Siegl, PK; Thorpe, HH | 1 |
Chappell, MC; Diz, DI; Ferrario, CM; Jaiswal, N; Khosla, MC | 1 |
Jackson, EK; Pong, AS; Tofovic, SP | 1 |
Duncia, JV; Hart, SD; Timmermans, PB; Wong, PC | 1 |
Barber, PC; Barnes, JM; Barnes, NM | 1 |
Carter, MR; Cook, VI; Grove, KL; Harding, JW; McMenamin, KM; Speth, RC | 1 |
Chiu, AT; McCall, DE; Roscoe, WA; Timmermans, PB | 1 |
Raizada, MK; Sumners, C; Tang, W; Zelezna, B | 1 |
Cogan, MG; Liu, FY; Timmermans, PB; Wong, PC | 1 |
Saavedra, JM; Tsutsumi, K | 1 |
Bauer, PH; Chiu, AT; Garrison, JC | 1 |
Hart, SD; Timmermans, PB; Wong, PC | 1 |
Grove, KL; Rowe, BP; Saylor, DL; Speth, RC | 1 |
Chiu, AT; Leung, KH; Smith, RD; Timmermans, BM | 1 |
García-Sáinz, JA; Macías-Silva, M | 1 |
Ardecky, RJ; Chiu, AT; Hart, SD; Smith, RD; Timmermans, PB; Wong, PC; Zaspel, AM | 1 |
Alburges, ME; Herblin, WF; Hunt, M; Wamsley, JK | 1 |
Kunert-Radek, J; Mucha, S; Pawlikowski, M; Pisarek, H; Sepien, H; Stawowy, A | 1 |
Pfaffendorf, M; van Zwieten, PA; Zhang, J | 3 |
Kunihara, M; Kushida, H; Morita, O | 1 |
Bornkessel, B | 1 |
Aguilera, G; Burns, RC; Cahill, PA; Sitzmann, JV; Wu, Y | 1 |
Ahmed, A; Barnes, NM; Gregory, J; Li, XF; Newton, JR; Rollason, T; Shams, M | 1 |
Baker, KM; Dostal, DE; Du, J; Motel, TJ; Thekkumkara, TJ; Thomas, WG | 1 |
Baldi, E; Catalioto, RM; Cioni, A; Finetti, G; Maggi, M; Mancina, R; Renzetti, AR; Serio, M | 1 |
Beyer, C; Höhle, S; Nagy, E; Rohmeiss, P; Strauch, M; Tschöpe, C; Unger, T | 1 |
de Gasparo, M; Levens, NR | 1 |
Grove, KL; Lu, XY; Speth, RC; Zhang, W | 1 |
Culman, J; Höhle, S; Rascher, W; Spitznagel, H; Unger, T | 1 |
Allen, AM; MacGregor, DP; Mendelsohn, FA; Murone, C; Paxinos, G; Song, K | 1 |
Smith, RD; Timmermans, PB | 1 |
Bottari, SP; Metzger, R; Paul, M; Steckelings, UM; Stoll, M; Unger, T | 1 |
Hamilton, TA; Harding, JW; Wright, JW | 1 |
Griffin, CA; Schambelan, M; Sechi, LA | 1 |
Chiu, AT; Duncia, JV; Santella, JB; Smith, RD; Timmermans, PB; Wexler, RR; Wong, PC | 1 |
Chiyotani, A; Isono, K; Konno, K; Sugimoto, F; Tagaya, E; Tamaoki, J | 1 |
Haruno, A; Hoshino, T; Inabe, K; Kimura, R; Matsuura, N; Nozawa, Y; Oda, N; Suzuki, H; Yamada, S; Yamasaki, Y | 1 |
Bihoreau, C; Clauser, E; Conchon, S; Corvol, P; Monnot, C; Sirieix, ME | 1 |
Pfaffendorf, M; Van Zwieten, PA; Zhang, J; Zhang, JS | 1 |
Heemskerk, FM; Michels, KM; Saavedra, JM | 1 |
Bartoli, E; De Carli, S; Griffin, CA; Schambelan, M; Sechi, G; Sechi, LA | 2 |
Lu, D; Raizada, MK; Rydzewski, B; Sumners, C | 1 |
Brown, JA; Cobb, CS | 1 |
Cazaubon, C; Chatelain, P; Delisée, C; Schaeffer, P | 1 |
Bensoussan, M; Mitchell, T; Reilly, T; Ronco, PM; Timmermans, PB; Verroust, PJ | 1 |
Gonzales, N; Lanting, L; Nadler, J; Natarajan, R | 1 |
Griffin, CA; Schambelan, M; Sechi, LA; Valentin, JP | 1 |
Barnes, JC; Clark, SA; Marshall, FH; Michel, AD | 1 |
Benfield, P; Carini, DJ; Chiu, AT; Herblin, WF; Lee, RJ; Saye, JA; Smith, RD; Timmermans, PB; Wexler, RR; Wong, PC | 1 |
Couch, SJ; Pals, DT | 1 |
Dagenais, P; Escher, E | 1 |
Barber, PC; Barnes, JM; Barnes, NM; Steward, LJ | 1 |
Dickinson, KE; Michel, I; Monshizadegan, H; Moreland, S; Murphy, TJ; Seiler, SM; Serafino, R; Webb, ML | 1 |
Baubonis, W; Benfield, P; Chiu, AT; Dunscomb, JH; McCall, DE; Sauer, B | 1 |
Aguilera, G; Feuillan, PP; Millan, MA | 1 |
Ball, AE; Felgenhauer, GP; Hall, KL; Hanesworth, JM; Harding, JW; Hosick, HL | 1 |
Barnes, JC; Hawcock, AB | 1 |
Clarke, DE; Hegde, SS | 1 |
Liu, YJ | 1 |
Catalioto, RM; Criscuoli, M; Giachetti, A; Porchia, R; Renzetti, AR; Subissi, A | 1 |
Coviello, A; Peral de Bruno, M | 1 |
Bing, C; Broughton Pipkin, F; Johnson, IR | 1 |
Böhm, M; Flesch, M; Kilter, H; Kuhn-Regnier, F; La Rosée, K; Lenz, O; Schmid, B; Südkamp, M | 1 |
Bill, DJ; Dourish, CT; Grewal, SS; McLenachan, A; Shepherd, J; Stanhope, KJ | 1 |
Ardaillou, R; Chansel, D; Czekalski, S; Ronco, P; Vandermeersch, S | 1 |
Chan, HC; Fu, LX; Law, SH; Leung, PS; Wong, PY | 1 |
Harding, JW; Kramár, EA; Wright, JW | 1 |
Eijsman, L; Feenstra, M; Li, Q; Pfaffendorf, M; van Zwieten, PA | 1 |
García-Sáinz, JA; Macías-Silva, M; Olivares-Reyes, JA | 1 |
García-Sáinz, JA; González-Espinosa, C; Martínez-Alfaro, M; Romero-Avila, MT | 1 |
Ganjam, VK; Ramires, FJ; Sun, Y; Weber, KT; Zhou, G | 1 |
Naitoh, T; Shikada, K; Tanaka, S; Yotsumoto, T | 1 |
Bai, D; Renaud, LP | 1 |
Barbera, F; Diamond, S; Gibson, RE; Herblin, WF; Timmermans, P | 1 |
Campbell, SE; Dhalla, AK; Kandala, JC; Katwa, LC; Sun, Y; Tyagi, SC; Weber, KT | 1 |
Ardaillou, R | 1 |
Jung, YS; Lee, BH; Lee, SH; Shin, HS; Yoo, SE; Yun, SI | 1 |
Hori, K; Kohzuki, M; Sato, T; Suzuki, M; Tanda, S; Yoshida, K | 1 |
Li, Q; Pfaffendorf, M; van Zwieten, PA | 1 |
Fischer, JW; Hahn, AW; Stoll, M; Unger, T | 1 |
Chen, Y; Dong, X; Lam, SY; Leung, PS | 1 |
Dobrucki, LW; Heitsch, H; Louka, FR; Malinski, T; Wiemer, G | 1 |
Cappugi, P; Cresci, B; Giannini, S; Magg, E; Maggi, E; Manuelli, C; Mavilia, C; Pala, L; Rotella, CM | 1 |
Bild, W; Ciobica, A; Hritcu, L; Stefanescu, C | 1 |
8 review(s) available for losartan and pd 123177
Article | Year |
---|---|
Angiotensin II receptors and functional correlates.
Topics: Acrylates; Angiotensin Receptor Antagonists; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Humans; Hypertension; Imidazoles; Losartan; Pyridines; Receptors, Angiotensin; Renin-Angiotensin System; Tetrazoles; Thiophenes | 1992 |
Angiotensin II receptor subtypes.
Topics: Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Binding Sites; Biphenyl Compounds; Drug Resistance; Humans; Imidazoles; Losartan; Oligopeptides; Pyridines; Receptors, Angiotensin; Terminology as Topic; Tetrazoles; Tissue Distribution | 1992 |
[Angiotensin II receptor antagonists].
Topics: Amino Acid Sequence; Angiotensin II; Angiotensin Receptor Antagonists; Antihypertensive Agents; Biphenyl Compounds; Hemodynamics; Humans; Hypertension; Imidazoles; Losartan; Molecular Sequence Data; Pyridines; Receptors, Angiotensin; Renin-Angiotensin System; Saralasin; Tetrazoles | 1995 |
Pharmacology of angiotensin II receptors in the kidney.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Humans; Imidazoles; Kidney; Losartan; Oligopeptides; Pyridines; Rats; Receptors, Angiotensin; Species Specificity; Tetrazoles; Tissue Distribution | 1994 |
Human angiotensin receptor subtypes.
Topics: Angiotensin I; Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; DNA, Complementary; Gene Library; Humans; Imidazoles; Losartan; Oligopeptides; Pyridines; Receptors, Angiotensin; Tetrazoles | 1994 |
New perspectives in angiotensin system control.
Topics: Amino Acid Sequence; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Pressure; Cardiomegaly; Hemodynamics; Humans; Imidazoles; Losartan; Molecular Sequence Data; Pyridines; Renin-Angiotensin System; Tetrazoles | 1993 |
Angiotensin II receptors and angiotensin II receptor antagonists.
Topics: Amino Acid Sequence; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Cloning, Molecular; Hemodynamics; Humans; Hypertension; Imidazoles; Kidney; Losartan; Molecular Sequence Data; Pyridines; Receptors, Angiotensin; Tetrazoles | 1993 |
Angiotensin II receptors.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Benzimidazoles; Biphenyl Compounds; Endothelium; Humans; Imidazoles; Kidney; Losartan; Peptide Fragments; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Tetrazoles | 1999 |
103 other study(ies) available for losartan and pd 123177
Article | Year |
---|---|
Effects of angiotensin II and nonpeptide receptor antagonists on transduction pathways in rat proximal tubule.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Calcium; Cyclic AMP; Imidazoles; Inositol Phosphates; Kidney Tubules, Proximal; Losartan; Male; Osmolar Concentration; Pyridines; Rats; Rats, Sprague-Dawley; Signal Transduction; Tetrazoles | 1992 |
Effects of angiotensin II and its selective antagonists on inferior olivary neurones.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Biphenyl Compounds; Imidazoles; Losartan; Neurons; Oligopeptides; Olivary Nucleus; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Synaptic Transmission; Tetrazoles | 1992 |
Role of angiotensin II receptor subtypes on the regulation of aldosterone secretion in the adrenal glomerulosa zone in the rat.
Topics: Aldosterone; Angiotensin II; Animals; Biphenyl Compounds; Cells, Cultured; Cyclic AMP; Dithiothreitol; Imidazoles; Inositol Phosphates; Losartan; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Secretory Rate; Signal Transduction; Sodium, Dietary; Tetrazoles; Zona Glomerulosa | 1992 |
Possible implication of peptidase activity in different potency of angiotensins II and III for displacing [125I]angiotensin II binding in pig aorta.
Topics: Aminopeptidases; Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Aorta; Binding, Competitive; Biphenyl Compounds; Calcium; Cells, Cultured; Endopeptidases; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Losartan; Membranes; Muscle, Smooth, Vascular; Pyridines; Swine; Tetrazoles | 1992 |
AT1 receptors mediate the release of prostaglandins in porcine smooth muscle cells and rat astrocytes.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Arachidonic Acids; Astrocytes; Biphenyl Compounds; Calcimycin; Cattle; Cells, Cultured; Dinoprost; Dose-Response Relationship, Drug; Endothelium, Vascular; Epoprostenol; Glioma; Imidazoles; Iodine Radioisotopes; Losartan; Macrophages; Male; Muscle, Smooth, Vascular; Prostaglandins; Pyridines; Radioimmunoassay; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Swine; Tetrazoles; Thromboxanes; Tumor Cells, Cultured | 1992 |
Competitive antagonism of pressor responses to angiotensin II and angiotensin III by the angiotensin II-1 receptor ligand losartan.
Topics: Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Pressure; Dose-Response Relationship, Drug; Imidazoles; Losartan; Male; Pyridines; Rats; Rats, Sprague-Dawley; Tetrazoles | 1992 |
Enhancement of losartan (DuP 753)-induced angiotensin II receptor antagonism by PD123177 in rats.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Pressure; Decerebrate State; Hypertension, Renal; Imidazoles; Losartan; Male; Pyridines; Rats; Rats, Sprague-Dawley; Renin-Angiotensin System; Tetrazoles | 1992 |
Inhibition of the haemodynamic effects of angiotensin II in conscious rats by AT2-receptor antagonists given after the AT1-receptor antagonist, EXP 3174.
Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hemodynamics; Imidazoles; Losartan; Male; Pyridines; Rats; Regional Blood Flow; Tetrazoles | 1992 |
Angiotensin II receptor activation depolarizes rat supraoptic neurons in vitro.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Culture Media; Electrophysiology; Imidazoles; Losartan; Male; Neurons; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Supraoptic Nucleus; Tetrazoles; Tetrodotoxin | 1992 |
Modulation of net outward current in cultured neurons by angiotensin II: involvement of AT1 and AT2 receptors.
Topics: Action Potentials; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Brain Stem; Cells, Cultured; Hypothalamus; Imidazoles; Losartan; Membrane Potentials; Neurons; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1992 |
Mechanism of angiotensin II-induced proliferation in bovine adrenocortical cells.
Topics: 12-Hydroxy-5,8,10,14-eicosatetraenoic Acid; Adrenal Cortex; Angiotensin II; Angiotensin Receptor Antagonists; Biphenyl Compounds; Cell Division; Cells, Cultured; DNA Replication; Dose-Response Relationship, Drug; Flavanones; Flavonoids; Humans; Hydroxyeicosatetraenoic Acids; Imidazoles; Losartan; Protein Kinase C; Pyrazoles; Pyridines; Pyrimidine Nucleosides; Tetrazoles; Thymidine | 1992 |
Angiotensin II and active phorbol esters induce proto-oncogene expression in isolated rat hepatocytes.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Cycloheximide; Dactinomycin; Female; Gene Expression Regulation; Imidazoles; Liver; Losartan; Phorbol Esters; Proto-Oncogene Proteins c-fos; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1992 |
The role of angiotensin, AT1 and AT2 receptors in the pressor, drinking and vasopressin responses to central angiotensin.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Arginine Vasopressin; Biphenyl Compounds; Blood Pressure; Cerebral Ventricles; Drinking Behavior; Imidazoles; Injections, Intraventricular; Losartan; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1992 |
Distribution of angiotensin II receptor subtypes in rat and human kidney.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Binding, Competitive; Biphenyl Compounds; Humans; Imidazoles; Kidney; Losartan; Male; Pyridines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles; Tissue Distribution | 1992 |
Mapping of angiotensin II receptor subtype heterogeneity in rat brain.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Binding, Competitive; Biphenyl Compounds; Brain; Brain Mapping; Dithiothreitol; Imidazoles; Iodine Radioisotopes; Losartan; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1992 |
Analysis of angiotensin II receptor subtypes in individual rat brain nuclei.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Binding, Competitive; Biphenyl Compounds; Brain Chemistry; Imidazoles; Losartan; Male; Mercaptoethanol; Pituitary Gland, Anterior; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1992 |
Effect of blocking angiotensin II receptor subtype on rat sympathetic nerve function.
Topics: Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Pressure; Cardiac Output; Decerebrate State; Electric Stimulation; Heart Rate; Imidazoles; Losartan; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Spinal Cord; Sympathetic Nervous System; Tetrazoles; Vascular Resistance | 1992 |
Monoclonal antibodies to the nonpeptide angiotensin II receptor antagonist, losartan.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies, Monoclonal; Antibody Specificity; Biphenyl Compounds; Cross Reactions; Enzyme-Linked Immunosorbent Assay; Imidazoles; Losartan; Mice; Mice, Inbred BALB C; Pyridines; Saralasin; Structure-Activity Relationship; Tetrazoles | 1992 |
Angiotensin-II receptor subtypes in fetal tissue of the rat: autoradiography, guanine nucleotide sensitivity, and association with phosphoinositide hydrolysis.
Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Binding, Competitive; Fetus; Gestational Age; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Hydrolysis; Imidazoles; Losartan; Oligopeptides; Phosphatidylinositols; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles; Tissue Distribution | 1991 |
Angiotensin II receptor subtypes in renal cortex of rats and rhesus monkeys.
Topics: Aldosterone; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Binding, Competitive; Biphenyl Compounds; Blood Pressure; Enalaprilat; Heart Rate; Imidazoles; Iodine Radioisotopes; Kidney Cortex; Losartan; Macaca mulatta; Male; Pyridines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Renin; Tetrazoles | 1991 |
Stimulation of endothelial cell prostaglandin production by angiotensin peptides. Characterization of receptors.
Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Cells, Cultured; Dinoprostone; Endothelium, Vascular; Epoprostenol; Imidazoles; Losartan; Oligopeptides; Prostaglandins; Pyridines; Receptors, Angiotensin; Tetrazoles | 1992 |
Effects of angiotensin subtype 1 and subtype 2 receptor antagonists in normotensive versus hypertensive rats.
Topics: Aldosterone; Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Pressure; Dose-Response Relationship, Drug; Hypertension; Imidazoles; Infusions, Intravenous; Losartan; Mesentery; Pyridines; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Angiotensin; Tetrazoles; Vasoconstriction | 1991 |
Nonpeptide angiotensin II receptor antagonists. Studies with DuP 753 and EXP3174 in dogs.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Captopril; Dogs; Female; Furosemide; Imidazoles; Kidney; Kidney Function Tests; Losartan; Male; Pyridines; Radioimmunoassay; Renin-Angiotensin System; Tetrazoles | 1991 |
Identification of angiotensin II receptor subtypes in human brain.
Topics: Aged; Angiotensin II; Angiotensin Receptor Antagonists; Autoradiography; Binding, Competitive; Biphenyl Compounds; Cerebellum; Female; Humans; Imidazoles; Iodine Radioisotopes; Losartan; Male; Pyridines; Receptors, Angiotensin; Tetrazoles | 1991 |
The AT2 angiotensin receptor subtype predominates in the 18 day gestation fetal rat brain.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Binding Sites; Biphenyl Compounds; Brain; Densitometry; Fetus; Imidazoles; Losartan; Pyridines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Angiotensin; Tetrazoles | 1991 |
Characterization of angiotensin II receptor subtypes in the rat kidney and heart using the non-peptide antagonists DuP 753 and PD 123 177.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Imidazoles; Kidney; Losartan; Male; Myocardium; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1991 |
Angiotensin II-1 receptors mediate both vasoconstrictor and hypertrophic responses in rat aortic smooth muscle cells.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Aorta, Thoracic; Biphenyl Compounds; Cells, Cultured; DNA; Fluorescent Dyes; Fura-2; Hypertrophy; Imidazoles; Losartan; Male; Muscle Proteins; Muscle, Smooth, Vascular; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Tetrazoles; Vasoconstriction | 1991 |
Angiotensin II receptor subtypes are coupled with distinct signal-transduction mechanisms in neurons and astrocytes from rat brain.
Topics: Angiotensin II; Animals; Animals, Newborn; Astrocytes; Binding, Competitive; Biphenyl Compounds; Brain; Cells, Cultured; Imidazoles; Kinetics; Ligands; Losartan; Neurons; Oligopeptides; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Signal Transduction; Tetrazoles | 1991 |
Comparison of inhibitory potency by nonpeptide angiotensin II receptor antagonists PD123177 and DuP 753 on proximal nephron and renal transport.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biological Transport; Biphenyl Compounds; Electrolytes; Glomerular Filtration Rate; Imidazoles; Kidney; Kidney Tubules, Distal; Kidney Tubules, Proximal; Losartan; Male; Nephrons; Perfusion; Pyridines; Rats; Rats, Inbred Strains; Tetrazoles | 1991 |
Angiotensin-II receptor subtypes in median eminence and basal forebrain areas involved in regulation of pituitary function.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Binding, Competitive; Biphenyl Compounds; Cerebral Arteries; Dithiothreitol; Imidazoles; Losartan; Male; Median Eminence; Oligopeptides; Pituitary Gland; Prosencephalon; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1991 |
DuP 753 can antagonize the effects of angiotensin II in rat liver.
Topics: Adenylyl Cyclase Inhibitors; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Calcium; Imidazoles; Inositol Phosphates; Iodine Radioisotopes; Liver; Losartan; Male; Membranes; Pyridines; Rats; Rats, Inbred Strains; Second Messenger Systems; Tetrazoles | 1991 |
Effect of angiotensin II antagonism on canine renal sympathetic nerve function.
Topics: Angiotensin II; Animals; Blood Pressure; Captopril; Dogs; Electric Stimulation; Female; Imidazoles; Kidney; Losartan; Male; Norepinephrine; Pyridines; Saralasin; Sympathetic Nervous System; Tetrazoles; Vascular Resistance; Vasoconstriction | 1991 |
Discrimination of angiotensin II receptor subtype distribution in the rat brain using non-peptidic receptor antagonists.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Binding, Competitive; Brain; Brain Chemistry; Cell Nucleus; Imidazoles; Losartan; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1991 |
Regional distribution of the two subtypes of angiotensin II receptor in rat brain using selective nonpeptide antagonists.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Binding, Competitive; Brain; Cell Membrane; Imidazoles; Kinetics; Losartan; Male; Organ Specificity; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1991 |
Angiotensin II stimulates phosphoinositide turnover and phosphorylase through AII-1 receptors in isolated rat hepatocytes.
Topics: Angiotensin II; Animals; Antihypertensive Agents; Cells, Cultured; Female; Imidazoles; Inositol Phosphates; Kinetics; Losartan; Phosphatidylinositols; Phosphorylase a; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles | 1990 |
Functional studies of nonpeptide angiotensin II receptor subtype-specific ligands: DuP 753 (AII-1) and PD123177 (AII-2).
Topics: Aldosterone; Angiotensin II; Animals; Blood Pressure; Dose-Response Relationship, Drug; Drinking; Epinephrine; Heart Rate; Imidazoles; Losartan; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Angiotensin; Tetrazoles; Vasoconstriction | 1990 |
Evidence for the presence of angiotensin II-type 1 receptors in brain.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Brain Chemistry; Imidazoles; Iodine Radioisotopes; Losartan; Male; Pyridines; Rats; Receptors, Angiotensin; Tetrazoles | 1990 |
Is estrogen-induced pituitary hyperplasia and hyperprolactinaemia mediated by angiotensin II?
Topics: Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Biphenyl Compounds; Cell Division; Diethylstilbestrol; Enalapril; Enalaprilat; Estrogens; Estrogens, Non-Steroidal; Humans; Hyperpituitarism; Hyperplasia; Hyperprolactinemia; Imidazoles; Losartan; Prolactin; Pyridines; Rats; Rats, Inbred F344; Rats, Wistar; Tetrazoles; Tumor Cells, Cultured | 1995 |
Effect of various angiotensin receptor antagonists on cardiovascular responses to angiotensin II in pithed rats.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Benzimidazoles; Biphenyl Compounds; Blood Pressure; Cardiac Output; Cardiovascular Physiological Phenomena; Cardiovascular System; Heart Rate; Imidazoles; Losartan; Male; Methylurea Compounds; Propranolol; Pyridines; Rats; Rats, Wistar; Receptors, Angiotensin; Tetrazoles | 1994 |
Effects of U-97018 on pressor responses to intracerebroventricularly administered angiotensin II in conscious normotensive rats.
Topics: Administration, Oral; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Disease Models, Animal; Dose-Response Relationship, Drug; Hypertension; Imidazoles; Injections, Intravenous; Injections, Intraventricular; Losartan; Male; Pyridazines; Pyridines; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Saralasin; Tetrazoles | 1995 |
Hemodynamic effects of angiotensin II and the influence of angiotensin receptor antagonists in pithed rabbits.
Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Benzimidazoles; Biphenyl Compounds; Blood Pressure; Decerebrate State; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Losartan; Male; Methylurea Compounds; Propranolol; Pyridines; Rabbits; Tetrazoles; Ventricular Function, Left | 1995 |
Loss of angiotensin-II receptors in portal hypertensive rabbits.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Biphenyl Compounds; Hypertension, Portal; Imidazoles; Ligation; Losartan; Male; Mesenteric Arteries; Portal Vein; Pyridines; Rabbits; Receptors, Angiotensin; Tetrazoles | 1995 |
Localization of the angiotensin II and its receptor subtype expression in human endometrium and identification of a novel high-affinity angiotensin II binding site.
Topics: Adult; Angiotensin II; Arterioles; Biphenyl Compounds; Endometrium; Endothelium; Endothelium, Vascular; Female; Gene Expression Regulation; Humans; Imidazoles; In Situ Hybridization; Losartan; Menstrual Cycle; Pyridines; Receptors, Angiotensin; RNA, Messenger; Tetrazoles | 1995 |
Stable expression of a functional rat angiotensin II (AT1A) receptor in CHO-K1 cells: rapid desensitization by angiotensin II.
Topics: Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Base Sequence; Calcium; Cell Membrane; CHO Cells; Concanavalin A; Cricetinae; Gene Expression; Guanosine Triphosphate; Imidazoles; Losartan; Membrane Potentials; Molecular Sequence Data; Pyridines; Rats; Receptors, Angiotensin; Tetradecanoylphorbol Acetate; Tetrazoles; Transfection; Verapamil | 1995 |
Identification and characterization of functional angiotensin II receptors in human neuroblastoma cells.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Binding, Competitive; Biphenyl Compounds; Calcium; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Imidazoles; Kinetics; Losartan; Neuroblastoma; Oligopeptides; Pyridines; Receptors, Angiotensin; Tetrazoles; Tumor Cells, Cultured; Vasoactive Intestinal Peptide | 1995 |
NaCl injections in brain induce natriuresis and blood pressure responses sensitive to ANG II AT1 receptors.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Pressure; Brain; Imidazoles; Injections; Losartan; Male; Natriuresis; Pyridines; Rats; Rats, Wistar; Receptors, Angiotensin; Saline Solution, Hypertonic; Sodium Chloride; Tetrazoles | 1995 |
Influence of tissue freezing on the binding of 125I-sarcosine1, isoleucine8 angiotensin II to angiotensin II receptor subtypes in the rat.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Adrenal Glands; Animals; Binding Sites; Binding, Competitive; Biphenyl Compounds; Brain; Epididymis; Freezing; Imidazoles; In Vitro Techniques; Liver; Losartan; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Tetrazoles | 1995 |
Angiotensin AT1 receptor-mediated vasopressin release and drinking are potentiated by an AT2 receptor antagonist.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Drinking; Imidazoles; Losartan; Male; Pyridines; Rats; Rats, Wistar; Receptors, Angiotensin; Tetrazoles; Vasopressins | 1995 |
Angiotensin II receptor subtypes in the human central nervous system.
Topics: Aged; Aged, 80 and over; Angiotensin II; Angiotensin Receptor Antagonists; Autoradiography; Biphenyl Compounds; Brain; Central Nervous System; Female; Humans; Imidazoles; Losartan; Male; Pyridines; Radioligand Assay; Receptors, Angiotensin; Spinal Cord; Tetrazoles | 1995 |
The angiotensin AT2-receptor mediates inhibition of cell proliferation in coronary endothelial cells.
Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Aorta; Base Sequence; Binding, Competitive; Biphenyl Compounds; Cell Division; Cells, Cultured; Coronary Vessels; DNA; DNA Primers; Dose-Response Relationship, Drug; Endothelium, Vascular; Gene Expression; Imidazoles; Kinetics; Losartan; Molecular Sequence Data; Muscle, Smooth, Vascular; Oligopeptides; Polymerase Chain Reaction; Pyridines; Rats; Receptors, Angiotensin; RNA, Messenger; Tetrazoles; Thymidine | 1995 |
Anomalous effects of losartan on aminopeptidase-induced reductions of blood pressure in SHR.
Topics: Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Pressure; CD13 Antigens; Hypertension; Imidazoles; Injections, Intraventricular; Losartan; Male; Pyridines; Rats; Rats, Inbred SHR; Tetrazoles | 1995 |
The cardiac renin-angiotensin system in STZ-induced diabetes.
Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Diabetes Mellitus, Experimental; Gene Expression; Hyperglycemia; Imidazoles; Insulin; Kinetics; Losartan; Male; Myocardium; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Reference Values; Renin-Angiotensin System; RNA, Messenger; Tetrazoles | 1994 |
EXP597, a nonpeptide angiotensin II receptor antagonist with high affinities for the angiotensin AT1 and AT2 receptor subtypes.
Topics: Administration, Oral; Adrenal Cortex; Adrenal Medulla; Angiotensin Receptor Antagonists; Animals; Aorta; Binding, Competitive; Biphenyl Compounds; Disease Models, Animal; Dose-Response Relationship, Drug; Hypertension, Renal; Imidazoles; In Vitro Techniques; Injections, Intravenous; Losartan; Male; Pyridines; Rabbits; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Receptors, Angiotensin; Renin-Angiotensin System; Sulfonamides; Tetrazoles | 1994 |
Angiotensin II 1 receptor-mediated contraction of pulmonary artery and its modulation by prolylcarboxypeptidase.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Arginine; Biphenyl Compounds; Carboxypeptidases; Dogs; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Isometric Contraction; Losartan; Male; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Protease Inhibitors; Pulmonary Artery; Pyridines; Receptors, Angiotensin; Tetrazoles | 1994 |
Angiotensin II receptor subtypes in bovine and human ventricular myocardium.
Topics: Aged; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Cattle; Dithiothreitol; Heart Ventricles; Humans; Imidazoles; Iodine Radioisotopes; Losartan; Male; Myocardium; Pyridines; Radioligand Assay; Receptors, Angiotensin; Tetrazoles | 1994 |
Positive inotropic action of angiotensin II in the pithed rat.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Pressure; Decerebrate State; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Losartan; Male; Myocardial Contraction; Pyridines; Rats; Rats, Wistar; Stimulation, Chemical; Tetrazoles | 1993 |
Synthetic cDNA encoding the rat AT1a receptor: a useful tool for structure-function relationship analysis.
Topics: Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Base Sequence; Biphenyl Compounds; CHO Cells; Codon; Cricetinae; DNA, Complementary; Imidazoles; Kinetics; Losartan; Molecular Sequence Data; Mutagenesis, Site-Directed; Oligodeoxyribonucleotides; Oligopeptides; Open Reading Frames; Pyridines; Rats; Receptors, Angiotensin; Restriction Mapping; Saralasin; Signal Transduction; Structure-Activity Relationship; Tetrazoles; Transfection | 1994 |
A non-competitive type of angiotensin-receptor antagonism by losartan in renal artery preparations.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Losartan; Muscle Contraction; Muscle, Smooth, Vascular; Pyridines; Rabbits; Renal Artery; Tetrazoles; Vasoconstriction | 1994 |
Selective changes in angiotensin II AT1 and AT2 receptor subtypes in the rat superior colliculus following eye enucleation.
Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Biphenyl Compounds; Eye Enucleation; Geniculate Bodies; Imidazoles; Iodine Radioisotopes; Losartan; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Retina; Saralasin; Subcellular Fractions; Superior Colliculi; Suprachiasmatic Nucleus; Synapses; Tetrazoles; Visual Pathways | 1994 |
[Angiotensin receptors in the rat myocardium during pre- and postnatal development].
Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Biphenyl Compounds; Heart; Imidazoles; Ligands; Losartan; Male; Myocardium; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Tetrazoles | 1993 |
Angiotensin II type 1 receptor-mediated stimulation of c-fos gene expression in astroglial cultures.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Astrocytes; Biphenyl Compounds; Dose-Response Relationship, Drug; Gene Expression; Genes, fos; Imidazoles; Losartan; Pyridines; Rats; Receptors, Angiotensin; RNA, Messenger; Tetrazoles | 1993 |
Characterization of putative glomerular receptors for angiotensin II in the rainbow trout Oncorhynchus mykiss using the antagonists Losartan, PD 123177, and saralasin.
Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Imidazoles; Iodine Radioisotopes; Kidney Glomerulus; Kinetics; Losartan; Oncorhynchus mykiss; Pyridines; Receptors, Angiotensin; Saralasin; Tetrazoles | 1993 |
Characterization of cardiac angiotensin AT1 receptors by [3H]SR 47436.
Topics: Angiotensin I; Angiotensin Receptor Antagonists; Animals; Animals, Newborn; Biphenyl Compounds; Calcium; Cells, Cultured; Heart; Homeostasis; Imidazoles; Irbesartan; Kinetics; Losartan; Myocardium; Pyridines; Rats; Rats, Wistar; Receptors, Angiotensin; Tetrazoles | 1993 |
Immunological reactivity of angiotensin II receptor antagonists: possible implications for receptor binding sites.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies, Monoclonal; Antihypertensive Agents; Biphenyl Compounds; Imidazoles; In Vitro Techniques; Indicators and Reagents; Iodine Radioisotopes; Losartan; Molecular Conformation; Oligopeptides; Pyridines; Rats; Receptors, Angiotensin; Saralasin; Tetrazoles | 1993 |
Role of the lipoxygenase pathway in angiotensin II-induced vascular smooth muscle cell hypertrophy.
Topics: 12-Hydroxy-5,8,10,14-eicosatetraenoic Acid; Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Aorta; Arachidonate 12-Lipoxygenase; Arachidonate 15-Lipoxygenase; Biphenyl Compounds; Cells, Cultured; Dose-Response Relationship, Drug; Fibronectins; Flavanones; Flavonoids; Hydroxyeicosatetraenoic Acids; Hypertrophy; Ibuprofen; Imidazoles; Lipoxygenase Inhibitors; Losartan; Muscle, Smooth, Vascular; Pyridines; Swine; Tetrazoles | 1994 |
[The role of G-regulatory proteins in the intracellular mechanism of cardiac angiotensin-II receptors].
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Binding, Competitive; Biphenyl Compounds; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Heart; Imidazoles; Losartan; Male; Myocardium; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Tetrazoles | 1993 |
Autoradiographic characterization of angiotensin II receptor subtypes in rat intestine.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Biphenyl Compounds; Imidazoles; Intestinal Mucosa; Losartan; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Tetrazoles; Tissue Distribution | 1993 |
Differential blockade of central effects of angiotensin II by AT2-receptor antagonists.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Brain; Cardiovascular System; Imidazoles; Injections, Intraventricular; Losartan; Male; Pyridines; Rats; Tetrazoles | 1993 |
Binding of angiotensin antagonists to rat liver and brain membranes measured ex vivo.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Binding, Competitive; Biphenyl Compounds; Blood-Brain Barrier; Brain; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Liver; Losartan; Male; Membranes; Nicotinic Acids; Pyridines; Rats; Receptors, Angiotensin; Saralasin; Tetrazoles | 1993 |
Renin release induced by losartan (DuP 753), an angiotensin II receptor antagonist.
Topics: Angiotensin Receptor Antagonists; Animals; Atenolol; Biphenyl Compounds; Dose-Response Relationship, Drug; Feedback; Imidazoles; Indomethacin; Injections, Intravenous; Losartan; Male; Meclofenamic Acid; Propranolol; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Angiotensin; Renin; Sympathetic Nervous System; Tetrazoles | 1993 |
Anti-angiotensin antibodies cross-reactive with nonpeptide angiotensin antagonists as angiotensin receptor model.
Topics: Adrenocorticotropic Hormone; Amino Acid Sequence; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies; Biphenyl Compounds; Cross Reactions; Enzyme-Linked Immunosorbent Assay; Imidazoles; Losartan; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Naloxone; Pyridines; Saralasin; Structure-Activity Relationship; Tetrazoles | 1993 |
Identification and characterisation of angiotensin II receptor subtypes in human brain.
Topics: Aged; Angiotensin II; Angiotensin Receptor Antagonists; Autoradiography; Binding, Competitive; Biphenyl Compounds; Brain Chemistry; Female; Humans; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Losartan; Male; Middle Aged; Pyridines; Radioligand Assay; Receptors, Angiotensin; Saralasin; Tetrazoles | 1993 |
Binding and signal transduction of the cloned vascular angiotensin II (AT1a) receptor cDNA stably expressed in Chinese hamster ovary cells.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Adenylyl Cyclases; Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Binding Sites; Biphenyl Compounds; Calcium; CHO Cells; Cloning, Molecular; Cricetinae; DNA; Imidazoles; Losartan; Pyridines; Radioligand Assay; Receptors, Angiotensin; Signal Transduction; Tetrazoles; Transfection | 1993 |
Characterization of angiotensin AT1A receptor isoform by its ligand binding signature.
Topics: Adrenal Cortex; Angiotensin I; Angiotensin III; Animals; Base Sequence; Binding, Competitive; Biphenyl Compounds; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Imidazoles; Losartan; Molecular Sequence Data; Muscle, Smooth, Vascular; Nicotinic Acids; Pyridines; Rats; Receptors, Angiotensin; Recombinant Proteins; Saralasin; Tetrazoles; Transfection | 1993 |
Angiotensin II binding sites in the rat fetus: characterization of receptor subtypes and interaction with guanyl nucleotides.
Topics: Adrenal Glands; Animals; Autoradiography; Binding Sites; Biphenyl Compounds; Dithiothreitol; Fetus; Guanosine 5'-O-(3-Thiotriphosphate); Image Processing, Computer-Assisted; Imidazoles; Liver; Losartan; Muscles; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Skin; Tetrazoles | 1993 |
Identification and characterization of a novel angiotensin binding site in cultured vascular smooth muscle cells that is specific for the hexapeptide (3-8) fragment of angiotensin II, angiotensin IV.
Topics: Amino Acid Sequence; Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Aorta; Binding, Competitive; Biphenyl Compounds; Cattle; Cells, Cultured; Guanosine 5'-O-(3-Thiotriphosphate); Imidazoles; Losartan; Molecular Sequence Data; Muscle, Smooth, Vascular; Pyridines; Radioligand Assay; Receptors, Angiotensin; Tetrazoles | 1993 |
Pharmacological characterization of the contractile responses to angiotensin analogues in guinea-pig isolated longitudinal muscle of small intestine.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Atropine; Biphenyl Compounds; Guinea Pigs; Hypnotics and Sedatives; Imidazoles; In Vitro Techniques; Intestine, Small; Losartan; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Tetrazoles; Tetrodotoxin | 1993 |
Characterization of angiotensin receptors mediating the neuromodulatory effects of angiotensin in the vas deferens of the rabbit.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Drug Interactions; Electric Stimulation; Imidazoles; Losartan; Male; Muscle Contraction; Pyridines; Rabbits; Receptors, Angiotensin; Tetrazoles; Vas Deferens | 1993 |
Evidence that [Sar1]angiotensin II behaves differently from angiotensin II at angiotensin AT1 receptors in rabbit aorta.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Aorta; Binding Sites; Biphenyl Compounds; Drug Interactions; Imidazoles; In Vitro Techniques; Losartan; Male; Muscle Contraction; Muscle, Smooth, Vascular; Pyridines; Rabbits; Receptors, Angiotensin; Tetrazoles | 1993 |
Angiotensin II-induced responses in vascular smooth muscle cells: inhibition by non-peptide receptor antagonists.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Aorta, Thoracic; Biphenyl Compounds; Cells, Cultured; Dinoprostone; DNA; Epoprostenol; Imidazoles; Inositol 1,4,5-Trisphosphate; Leucine; Losartan; Male; Muscle, Smooth, Vascular; Protein Biosynthesis; Pyridines; Pyrimidinones; Rats; Rats, Sprague-Dawley; Tetrazoles; Thiophenes; Thymidine | 1995 |
Effects of angiotensin II antagonists on the contractile and hydrosmotic effect of AT II and AT III in the toad (Bufo arenarum).
Topics: Analysis of Variance; Angiotensin II; Angiotensin III; Animals; Antihypertensive Agents; Aorta; Biphenyl Compounds; Bufo arenarum; Dose-Response Relationship, Drug; Drug Interactions; Female; Imidazoles; Losartan; Male; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Osmolar Concentration; Osmosis; Pyridines; Skin; Tetrazoles; Vasoconstrictor Agents | 1996 |
Angiotensin receptors in myometrium and myometrial vessels from uteri of women during the follicular and luteal phases of the menstrual cycle and in late pregnancy.
Topics: Adult; Angiotensin II; Angiotensin Receptor Antagonists; Biphenyl Compounds; Blood Vessels; Cell Membrane; Female; Follicular Phase; Humans; Imidazoles; Losartan; Luteal Phase; Myometrium; Pregnancy; Pregnancy Trimester, Third; Pyridines; Receptors, Angiotensin; Tetrazoles | 1996 |
Effects of angiotensin II and angiotensin-converting enzyme inhibitors on human myocardium.
Topics: Adolescent; Adult; Aged; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Biphenyl Compounds; Electric Stimulation; Female; Heart; Heart Atria; Heart Ventricles; Humans; Imidazoles; In Vitro Techniques; Isometric Contraction; Losartan; Male; Middle Aged; Myocardial Contraction; Papillary Muscles; Pyridines; Receptors, Angiotensin; Tetrazoles; Vasoconstrictor Agents | 1995 |
Effects of the selective angiotensin II receptor antagonists losartan and PD123177 in animal models of anxiety and memory.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Anti-Anxiety Agents; Anxiety; Biphenyl Compounds; Diazepam; Dose-Response Relationship, Drug; Imidazoles; Losartan; Male; Memory; Motor Activity; Pyridines; Rats; Rats, Sprague-Dawley; Scopolamine; Tetrazoles | 1996 |
Evidence for angiotensin IV receptors in human collecting duct cells.
Topics: Aminopeptidases; Angiotensin II; Angiotensin Receptor Antagonists; Binding, Competitive; Biphenyl Compounds; Blotting, Northern; Calcium; CD13 Antigens; Cells, Cultured; Dose-Response Relationship, Drug; Humans; Imidazoles; Kidney Tubules, Collecting; Leucine; Losartan; Pyridines; Receptors, Angiotensin; RNA, Messenger; Tetrazoles | 1996 |
Angiotensin II receptor type I-regulated anion secretion in cystic fibrosis pancreatic duct cells.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Angiotensin II; Angiotensin Receptor Antagonists; Antiporters; Bicarbonates; Biological Transport, Active; Biphenyl Compounds; Calcium; Cell Polarity; Cells, Cultured; Chloride-Bicarbonate Antiporters; Chlorides; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Humans; Imidazoles; Intracellular Fluid; Ion Transport; Losartan; Microscopy, Confocal; Nystatin; Pancreatic Ducts; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Secretory Rate; Tetrazoles | 1997 |
Angiotensin II- and IV-induced changes in cerebral blood flow. Roles of AT1, AT2, and AT4 receptor subtypes.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Blood Flow Velocity; Blood Pressure; Cerebrovascular Circulation; Female; Imidazoles; Laser-Doppler Flowmetry; Losartan; Male; Microcirculation; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Tetrazoles | 1997 |
Comparative vasoconstrictor effects of angiotensin II, III, and IV in human isolated saphenous vein.
Topics: Aged; Aged, 80 and over; Aminopeptidases; Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Anti-Bacterial Agents; Antihypertensive Agents; Biphenyl Compounds; Dose-Response Relationship, Drug; Drug Synergism; Female; Glutamyl Aminopeptidase; Humans; Imidazoles; In Vitro Techniques; Losartan; Male; Metalloendopeptidases; Methionyl Aminopeptidases; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Peptides; Protease Inhibitors; Pyridines; Saphenous Vein; Tachyphylaxis; Tetrazoles; Vasoconstrictor Agents | 1997 |
Atypical angiotensin II receptors coupled to phosphoinositide turnover/calcium signalling in catfish hepatocytes.
Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Binding, Competitive; Biphenyl Compounds; Calcium; Cell Membrane; Egtazic Acid; Humans; Ictaluridae; Imidazoles; Liver; Losartan; Phosphatidylinositols; Pyridines; Receptors, Angiotensin; Signal Transduction; Tetrazoles | 1997 |
Characterization of the AT1 angiotensin II receptor expressed in guinea pig liver.
Topics: Angiotensin I; Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Binding, Competitive; Biphenyl Compounds; Enzyme Activation; Guinea Pigs; Imidazoles; Irbesartan; Liver; Losartan; Male; Polymerase Chain Reaction; Pyridines; Receptors, Angiotensin; RNA, Messenger; Tetrazoles | 1997 |
Fibrous tissue and angiotensin II.
Topics: Actins; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Collagen; Connective Tissue; Croton Oil; Fibroblasts; Granuloma; Hydroxyproline; Imidazoles; Lisinopril; Losartan; Macrophages; Male; Peptidyl-Dipeptidase A; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Wound Healing | 1997 |
Effects of specific antagonists of angiotensin II receptors and captopril on diabetic nephropathy in mice.
Topics: Albuminuria; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Captopril; Creatinine; Diabetes Mellitus, Experimental; Diabetic Nephropathies; Disease Models, Animal; Hypertrophy; Imidazoles; Kidney Diseases; Losartan; Male; Mice; Mice, Inbred Strains; Pyridines; Receptors, Angiotensin; Streptozocin | 1997 |
ANG II AT1 receptors induce depolarization and inward current in rat median preoptic neurons in vitro.
Topics: Action Potentials; Angiotensin II; Animals; Fluorescent Dyes; Imidazoles; In Vitro Techniques; Isoquinolines; Losartan; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Preoptic Area; Pyridines; Rats; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Tetrodotoxin | 1998 |
A novel angiotensin II binding site in murine tissues.
Topics: Amino Acid Sequence; Angiotensin II; Animals; Autoradiography; Binding Sites; Humans; Imidazoles; Losartan; Mice; Mice, Inbred C57BL; Mice, Nude; Pyridines; Saralasin; Tumor Cells, Cultured | 1998 |
Pouch tissue and angiotensin peptide generation.
Topics: Angiotensin I; Angiotensin II; Angiotensinogen; Angiotensins; Animals; Aspartic Acid Endopeptidases; Cathepsin D; Collagen; Gene Expression; Imidazoles; Lisinopril; Losartan; Myocardium; Peptide Biosynthesis; Peptides; Peptidyl-Dipeptidase A; Pyridines; Rats; Renin; Transforming Growth Factor beta | 1998 |
Characterization of angiotensin II antagonism displayed by SK-1080, a novel nonpeptide AT1-receptor antagonist.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Aorta, Thoracic; Binding, Competitive; Blood Pressure; Decerebrate State; Diastole; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; In Vitro Techniques; Losartan; Male; Muscle Contraction; Pyridines; Rabbits; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Sensitivity and Specificity; Tetrazoles | 1999 |
Decreased binding sites of angiotensin II in rat LY-80 and AH109A tumour and human gastric cancer using quantitative in vitro autoradiography.
Topics: Aged; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Angiotensin II Type 2 Receptor Blockers; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Autoradiography; Binding Sites; Biomarkers, Tumor; Blood Flow Velocity; Carcinoma; Humans; Imidazoles; Losartan; Male; Middle Aged; Neoplasm Transplantation; Neoplasms, Experimental; Pyridines; Rats; Rats, Nude; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Skin Neoplasms; Stomach Neoplasms; Tumor Cells, Cultured | 2000 |
Different types of antagonism by losartan and irbesartan on the effects of angiotensin II and its degradation products in rabbit arteries.
Topics: Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Anti-Bacterial Agents; Antihypertensive Agents; Biphenyl Compounds; Endothelium, Vascular; Femoral Artery; Imidazoles; In Vitro Techniques; Irbesartan; Leucine; Losartan; Male; Peptides; Protease Inhibitors; Pyridines; Rabbits; Receptor, Angiotensin, Type 1; Renal Artery; Tetrazoles; Vasoconstrictor Agents | 2001 |
Differential regulation of thrombospondin-1 and fibronectin by angiotensin II receptor subtypes in cultured endothelial cells.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Aorta; Arteriosclerosis; Blotting, Northern; Cattle; Cell Division; Cells, Cultured; DNA; Dose-Response Relationship, Drug; Endothelium, Vascular; Fibronectins; Imidazoles; Losartan; Male; Oligopeptides; Pyridines; Rats; Rats, Wistar; Receptors, Angiotensin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thrombospondin 1 | 2001 |
Postnatal hypoxemia increases angiotensin II sensitivity and up-regulates AT1a angiotensin receptors in rat carotid body chemoreceptors.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Animals, Newborn; Calcium; Carotid Body; Dose-Response Relationship, Drug; Hypoxia; Imidazoles; Losartan; Models, Animal; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Reverse Transcriptase Polymerase Chain Reaction; Spectrometry, Fluorescence | 2002 |
AVE 0991, a nonpeptide mimic of the effects of angiotensin-(1-7) on the endothelium.
Topics: Angiotensin I; Animals; Binding, Competitive; Cattle; Cells, Cultured; Cricetinae; Electrochemistry; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Humans; Imidazoles; Losartan; Molecular Mimicry; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Peptide Fragments; Pyridines; Radioligand Assay; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Substrate Specificity; Superoxides; Tetrazoles | 2002 |
AT1 and AT2 receptors in human glomerular endothelial cells at different passages.
Topics: Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Angiotensin II Type 2 Receptor Blockers; Antihypertensive Agents; Blotting, Western; Cell Culture Techniques; Cell Division; Dose-Response Relationship, Drug; Endothelial Cells; Humans; Imidazoles; Kidney Glomerulus; Kinetics; Losartan; Platelet-Derived Growth Factor; Protein Binding; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Reverse Transcriptase Polymerase Chain Reaction; Thymidine; Time Factors | 2003 |
Inhibition of central angiotensin II enhances memory function and reduces oxidative stress status in rat hippocampus.
Topics: Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Angiotensin II Type 2 Receptor Blockers; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Avoidance Learning; Behavior, Animal; Captopril; Glutathione Peroxidase; Hippocampus; Imidazoles; Lipid Peroxidation; Losartan; Male; Malondialdehyde; Maze Learning; Memory; Memory, Short-Term; Oxidative Stress; Psychomotor Performance; Pyridines; Rats; Rats, Wistar; Superoxide Dismutase | 2013 |