lomerizine and flunarizine

lomerizine has been researched along with flunarizine in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19902 (11.11)18.7374
1990's10 (55.56)18.2507
2000's5 (27.78)29.6817
2010's0 (0.00)24.3611
2020's1 (5.56)2.80

Authors

AuthorsStudies
Anger, T; Madge, DJ; Mulla, M; Riddall, D1
Birch, PJ; Earnshaw, CG; Fiumana, A; Gilbert, J; Hobbs, CJ; James, IF; Knutsen, LJ; Mellor, SL; Radford, F; Russell Burley, J; Smith, NJ; Ward, SD1
Belardetti, F; Ding, Y; Dolphin, D; Feng, ZP; Mitscher, LA; Pajouhesh, H; Snutch, TP; Zamponi, GW; Zhang, L1
Hara, H; Ikegami, A; Ito, K; Ozaki, A; Sukamoto, T; Yamashita, A1
Ikegami, A; Ito, K; Yamamoto, N; Yamashita, A; Yokota, K1
Iwamoto, T; Morita, T; Sukamoto, T1
Handa, J; Kidooka, M; Shiino, A1
Ando, S; Kon, K; Tanaka, Y; Waki, H1
Ando, S; Waki, H1
Ito, K; Iwamoto, T; Kanazawa, T; Morita, T; Ohtaka, H1
Akaike, N; Hara, H; Ishibashi, H; Oyama, Y; Ueha, T1
Hara, H; Shimazawa, M; Sukamoto, T; Watano, T1
Liou, SY; Takagi, H; Takashima, M1
Hara, H; Hashimoto, M; Shimazawa, M; Sukamoto, T1
Hara, H; Hashimoto, M; Iwakura, Y; Maeda, Y; Sakai, T; Sasaoka, M; Shimazawa, M; Sukamoto, T; Yamada, C; Yamaguchi, T1
Akaike, A; Hara, H; Honda, Y; Kashii, S; Shimazawa, M; Toriu, N; Yasuyoshi, H; Zhang, S1
Negoro, K1
Chu, MK; Wang, SJ1

Reviews

3 review(s) available for lomerizine and flunarizine

ArticleYear
Medicinal chemistry of neuronal voltage-gated sodium channel blockers.
    Journal of medicinal chemistry, 2001, Jan-18, Volume: 44, Issue:2

    Topics: Amyotrophic Lateral Sclerosis; Analgesics; Anticonvulsants; Epilepsy; Humans; Ion Channel Gating; Models, Molecular; Mutation; Nerve Tissue Proteins; Neuroprotective Agents; Protein Binding; Sodium Channel Blockers; Sodium Channels; Stroke

2001
[Ca antagonists in neurosurgical practice].
    No to shinkei = Brain and nerve, 1990, Volume: 42, Issue:1

    Topics: Animals; Anticonvulsants; Brain; Calcium Channel Blockers; Cerebral Infarction; Disease Models, Animal; Fatty Acids, Nonesterified; Flunarizine; Humans; Intracranial Aneurysm; Ischemic Attack, Transient; Nimodipine; Piperazines; Verapamil

1990
[Calcium antagonists in the prophylactic treatment of migraine].
    Brain and nerve = Shinkei kenkyu no shinpo, 2009, Volume: 61, Issue:10

    Topics: Calcium Channel Blockers; Calcium Channels; Drug Administration Schedule; Flunarizine; Humans; Hypoxia, Brain; Migraine Disorders; Neurotransmitter Agents; Piperazines; Premedication; Vasodilation

2009

Other Studies

15 other study(ies) available for lomerizine and flunarizine

ArticleYear
Synthesis and SAR of novel 2-arylthiazolidinones as selective analgesic N-type calcium channel blockers.
    Bioorganic & medicinal chemistry letters, 2007, Feb-01, Volume: 17, Issue:3

    Topics: Analgesics; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, N-Type; Cell Line, Tumor; Chromatography, High Pressure Liquid; Drug Evaluation, Preclinical; Humans; Indicators and Reagents; Spectrophotometry, Ultraviolet; Structure-Activity Relationship; Thiazolidinediones

2007
Scaffold-based design and synthesis of potent N-type calcium channel blockers.
    Bioorganic & medicinal chemistry letters, 2009, Nov-15, Volume: 19, Issue:22

    Topics: Analgesics; Animals; Binding Sites; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, N-Type; Calcium Channels, T-Type; Disease Models, Animal; Drug Design; Pain; Pain Measurement; Pain Threshold; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship

2009
Neurochemical investigation on the effects of a new diphenylpiperazine calcium antagonist, KB-2796, on the central dopaminergic system of rats.
    Japanese journal of pharmacology, 1992, Volume: 58, Issue:4

    Topics: Animals; Calcium Channel Blockers; Chlorpromazine; Corpus Striatum; Dopamine; Flunarizine; In Vitro Techniques; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Tritium

1992
[Hemorheological effect of KB-2796, a new Ca2+ antagonist].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1992, Volume: 100, Issue:2

    Topics: Animals; Blood Viscosity; Calcium Channel Blockers; Cerebrovascular Disorders; Erythrocyte Deformability; Flunarizine; Guinea Pigs; In Vitro Techniques; Male; Micropore Filters; Pentoxifylline; Piperazines; Rabbits

1992
Calcium antagonism by KB-2796, a new diphenylpiperazine analogue, in dog vascular smooth muscle.
    The Journal of pharmacy and pharmacology, 1991, Volume: 43, Issue:8

    Topics: Animals; Binding Sites; Calcium; Calcium Channel Blockers; Cinnarizine; Dogs; Drug Interactions; Female; Flunarizine; Male; Muscle, Smooth, Vascular; Nitrendipine; Piperazines

1991
Age-related changes in the uptake of calcium channel blockers by brain capillary endothelial cells and synaptosomal fractions.
    Neuroscience letters, 1990, Aug-24, Volume: 116, Issue:3

    Topics: Aging; Animals; Brain; Calcium Channel Blockers; Capillaries; Cerebrovascular Circulation; Endothelium, Vascular; Female; Flunarizine; Male; Osmolar Concentration; Piperazines; Rats; Rats, Inbred F344; Synaptosomes

1990
Column liquid chromatography of calcium channel blockers.
    Journal of chromatography, 1989, Sep-29, Volume: 494

    Topics: Animals; Blood-Brain Barrier; Brain Chemistry; Calcium Channel Blockers; Chromatography, High Pressure Liquid; Cinnarizine; Female; Flunarizine; Piperazines; Rats; Rats, Inbred F344; Subcellular Fractions

1989
Effects of KB-2796, a new calcium antagonist, and other diphenylpiperazines on [3H]nitrendipine binding.
    Japanese journal of pharmacology, 1988, Volume: 48, Issue:2

    Topics: Animals; Binding Sites; Calcium Channel Blockers; Calcium Channels; Cerebral Cortex; Flunarizine; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Nitrendipine; Piperazines; Synaptosomes; Vasodilation

1988
Effect of KB-2796, a new diphenylpiperazine Ca2+ antagonist, on voltage-dependent Ca2+ currents and oxidative metabolism in dissociated mammalian CNS neurons.
    Brain research, 1993, Aug-13, Volume: 619, Issue:1-2

    Topics: Animals; Brain; Calcium Channel Blockers; Calcium Channels; Cerebellum; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; Flow Cytometry; Flunarizine; Fluoresceins; Fluorescent Dyes; Hippocampus; In Vitro Techniques; Membrane Potentials; Neurons; Nystatin; Oxidation-Reduction; Piperazines; Pyramidal Tracts; Rats; Rats, Wistar

1993
Effects of Ca2+ channel blockers on cortical hypoperfusion and expression of c-Fos-like immunoreactivity after cortical spreading depression in rats.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Animals; Blood Pressure; Brain; Calcium Channel Blockers; Cerebrovascular Circulation; Cortical Spreading Depression; Flunarizine; Heart Rate; Histamine H1 Antagonists; Laser-Doppler Flowmetry; Male; Oncogene Proteins v-fos; Phenothiazines; Piperazines; Potassium Chloride; Rats; Rats, Wistar

1995
[Effect of KB-2796, a novel calcium channel blocker, on spreading depression in rat hippocampal slices].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1998, Volume: 111, Issue:5

    Topics: Animals; Calcium Channel Blockers; Cortical Spreading Depression; Flunarizine; Hippocampus; Histamine H1 Antagonists; Humans; In Vitro Techniques; Infant, Newborn; Male; Migraine Disorders; Phenothiazines; Piperazines; Rats; Rats, Sprague-Dawley; Sumatriptan

1998
[Anti-migraine effects of lomerizine].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1998, Volume: 112 Suppl 1

    Topics: Animals; Calcium Channel Blockers; Cerebrovascular Circulation; Cortical Spreading Depression; Flunarizine; Hippocampus; In Vitro Techniques; Migraine Disorders; Piperazines; Proto-Oncogene Proteins c-fos; Rats

1998
Selective effects of lomerizine, a novel diphenylmethylpiperazine Ca2+ channel blocker, on cerebral blood flow in rats and dogs.
    Clinical and experimental pharmacology & physiology, 1999, Volume: 26, Issue:11

    Topics: Animals; Blood Pressure; Calcium Channel Blockers; Cerebral Cortex; Cerebrovascular Circulation; Dogs; Dose-Response Relationship, Drug; Flunarizine; Heart Rate; Laser-Doppler Flowmetry; Male; Piperazines; Rats; Rats, Wistar; Spine

1999
Lomerizine, a Ca2+ channel blocker, reduces glutamate-induced neurotoxicity and ischemia/reperfusion damage in rat retina.
    Experimental eye research, 2000, Volume: 70, Issue:4

    Topics: Animals; Calcium Channel Blockers; Cells, Cultured; Dizocilpine Maleate; Dose-Response Relationship, Drug; Flunarizine; Glutamic Acid; Male; Neuroprotective Agents; Neurotoxicity Syndromes; Piperazines; Rats; Rats, Sprague-Dawley; Reperfusion Injury

2000
Nomenclature for flunarizine, cinnarizine, and lomerizine.
    Cephalalgia : an international journal of headache, 2020, Volume: 40, Issue:3

    Topics: Calcium Channel Blockers; Cinnarizine; Flunarizine; Humans; Migraine Disorders; Piperazines; Terminology as Topic

2020