loe 908 has been researched along with thapsigargin in 7 studies
Studies (loe 908) | Trials (loe 908) | Recent Studies (post-2010) (loe 908) | Studies (thapsigargin) | Trials (thapsigargin) | Recent Studies (post-2010) (thapsigargin) |
---|---|---|---|---|---|
50 | 0 | 5 | 5,234 | 3 | 918 |
Protein | Taxonomy | loe 908 (IC50) | thapsigargin (IC50) |
---|---|---|---|
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | 0.002 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (28.57) | 18.2507 |
2000's | 4 (57.14) | 29.6817 |
2010's | 1 (14.29) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Birke, FW; Encabo, A; Groschner, K; Kukovetz, WR; Romanin, C | 1 |
Enoki, T; Furutani, H; Hasegawa, H; Hashimoto, N; Ishikawa, M; Iwamuro, Y; Masaki, T; Minowa, T; Miwa, S; Okamoto, Y; Okazawa, M; Zhang, XF | 1 |
Igarashi, T; Imai, T; Otsuka, K; Shigenobu, K; Takayanagi, K; Tanaka, H; Tanaka, Y; Yamaki, F | 1 |
Iwamuro, Y; Lee, K; Miwa, S; Morita, H; Okamoto, Y; Zhang, XF | 1 |
Enoki, T; Hashimoto, N; Kawanabe, Y; Masaki, T; Okamoto, Y | 1 |
Bootman, MD; Holmes, AM; McDonald, F; Roderick, HL | 1 |
Ambily, A; Authi, KS; Chamberlain, EV; Gibbins, JM; Jones, CI; Kaiser, WJ; Kassouf, N; Li, Z; Pierro, C | 1 |
7 other study(ies) available for loe 908 and thapsigargin
Article | Year |
---|---|
Inhibition of a store-operated Ca2+ entry pathway in human endothelial cells by the isoquinoline derivative LOE 908.
Topics: Acetamides; Calcium; Calcium Channels; Cells, Cultured; Endothelium, Vascular; Humans; Ionomycin; Isoquinolines; Membrane Potentials; Thapsigargin | 1996 |
Activation of three types of voltage-independent Ca2+ channel in A7r5 cells by endothelin-1 as revealed by a novel Ca2+ channel blocker LOE 908.
Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cations; Cells, Cultured; Drug Interactions; Endothelin-1; Imidazoles; Ionomycin; Isoquinolines; Patch-Clamp Techniques; Rats; Thapsigargin | 1999 |
Comparison of the Ca2+ entry channels responsible for mechanical responses of guinea-pig aorta to noradrenaline and thapsigargin using SK&F 96365 and LOE 908.
Topics: Acetamides; Animals; Aorta, Thoracic; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Cytoplasm; Enzyme Inhibitors; Extracellular Space; Female; Guinea Pigs; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Thapsigargin; Type C Phospholipases | 2000 |
Failure of endothelin-1 to activate store-operated Ca2+ channels by lack of mobilization from intracellular Ca2+ stores in cultured bovine adrenal chromaffin cells.
Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cattle; Cells, Cultured; Chromaffin Cells; Endothelin-1; Enzyme Inhibitors; Imidazoles; Ion Channels; Isoquinolines; Thapsigargin | 2001 |
Ca(2+) channels activated by endothelin-1 in CHO cells expressing endothelin-A or endothelin-B receptors.
Topics: Acetamides; Adenosine Triphosphatases; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; CHO Cells; Cricetinae; Electrophysiology; Endothelin-1; Enzyme Inhibitors; Imidazoles; Inositol Phosphates; Isoquinolines; Patch-Clamp Techniques; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Thapsigargin | 2001 |
Interaction between store-operated and arachidonate-activated calcium entry.
Topics: Acetamides; Arachidonic Acid; Calcium Channels; Calcium Signaling; Cell Line; Cytosol; Humans; Imidazoles; Isoquinolines; Nitric Oxide; Thapsigargin | 2007 |
The role of plasma membrane STIM1 and Ca(2+)entry in platelet aggregation. STIM1 binds to novel proteins in human platelets.
Topics: Acetamides; Actins; Anilides; Antibodies; Blood Platelets; Calcium; Calcium Signaling; Collagen; Endoplasmic Reticulum; Enzyme Inhibitors; Guanine Nucleotide Exchange Factors; Humans; Ion Channels; Isoquinolines; Membrane Proteins; Myosins; Neoplasm Proteins; Platelet Activation; Platelet Aggregation; Protein Binding; Stromal Interaction Molecule 1; Thapsigargin; Thiadiazoles; Thrombosis; Thrombospondin 1 | 2014 |