Page last updated: 2024-09-03

loe 908 and endothelin-1

loe 908 has been researched along with endothelin-1 in 21 studies

Compound Research Comparison

Studies
(loe 908)
Trials
(loe 908)
Recent Studies (post-2010)
(loe 908)
Studies
(endothelin-1)
Trials
(endothelin-1)
Recent Studies (post-2010) (endothelin-1)
500512,7406323,394

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (28.57)18.2507
2000's15 (71.43)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Enoki, T; Furutani, H; Hasegawa, H; Hashimoto, N; Ishikawa, M; Iwamuro, Y; Masaki, T; Minowa, T; Miwa, S; Okamoto, Y; Okazawa, M; Zhang, XF1
Enoki, T; Furutani, H; Hasegawa, H; Iwamuro, Y; Komuro, T; Lee, K; Masaki, T; Minowa, T; Miwa, S; Okamoto, Y; Okazawa, M; Zhang, XF1
Inoki, T; Iwamuro, Y; Masaki, T; Miwa, S; Okamoto, Y; Okazawa, M; Zhang, XF1
Furutani, H; Hasegawa, H; Iwamuro, Y; Lee, K; Masaki, T; Miwa, S; Morita, H; Nakagawa, T; Okamoto, Y; Zhang, XF1
Iwamuro, Y; Masaki, T; Miwa, S; Okamoto, Y; Zhang, XF2
Iwamuro, Y; Kawanabe, Y; Masaki, T; Miwa, S; Okamoto, Y; Zhang, XF1
Furutani, H; Iwamuro, Y; Masaki, T; Miwa, S; Okamoto, Y; Zhang, XF1
Hashimoto, N; Kawanabe, Y; Masaki, T; Okamoto, Y1
Iwamuro, Y; Lee, K; Miwa, S; Morita, H; Okamoto, Y; Zhang, XF1
Hashimoto, N; Kawanabe, Y; Masaki, T10
Enoki, T; Hashimoto, N; Kawanabe, Y; Masaki, T; Okamoto, Y1

Reviews

1 review(s) available for loe 908 and endothelin-1

ArticleYear
Ca2+ entry channels in rat thoracic aortic smooth muscle cells activated by endothelin-1.
    Japanese journal of pharmacology, 1999, Volume: 80, Issue:4

    Topics: Acetamides; Animals; Aorta, Thoracic; Calcium Channel Blockers; Calcium Channels; Endothelin-1; Imidazoles; Isoquinolines; Muscle, Smooth, Vascular; Rats

1999

Other Studies

20 other study(ies) available for loe 908 and endothelin-1

ArticleYear
Activation of three types of voltage-independent Ca2+ channel in A7r5 cells by endothelin-1 as revealed by a novel Ca2+ channel blocker LOE 908.
    British journal of pharmacology, 1999, Volume: 126, Issue:5

    Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cations; Cells, Cultured; Drug Interactions; Endothelin-1; Imidazoles; Ionomycin; Isoquinolines; Patch-Clamp Techniques; Rats; Thapsigargin

1999
Pharmacological characterization of Ca2+ entry channels in endothelin-1-induced contraction of rat aorta using LOE 908 and SK&F 96365.
    British journal of pharmacology, 1999, Volume: 127, Issue:6

    Topics: Acetamides; Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Dose-Response Relationship, Drug; Endothelin-1; Imidazoles; Isoquinolines; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rats; Rats, Wistar

1999
Pharmacological characterization of receptor-mediated Ca2+ entry in endothelin-1-induced catecholamine release from cultured bovine adrenal chromaffin cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:6

    Topics: Acetamides; Adrenal Glands; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Cattle; Cells, Cultured; Chromaffin Cells; Dose-Response Relationship, Drug; Endothelin-1; Epinephrine; Imidazoles; Inhibitory Concentration 50; Ion Channels; Isoquinolines; Linear Models; Nifedipine; Norepinephrine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Receptor, Endothelin A; Receptors, Endothelin; Signal Transduction

1999
[Characterization of voltage-independent Ca2+ channels activated by endothelin-1].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114 Suppl 1

    Topics: Acetamides; Animals; Calcium Channel Blockers; Calcium Channels; Cell Line; Endothelin-1; Imidazoles; Isoquinolines; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Rats

1999
[Analysis of Ca2+ entry channels in endothelin-1-induced contraction of rat aorta using new blockers].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114 Suppl 1

    Topics: Acetamides; Animals; Aorta, Thoracic; Calcium Channel Blockers; Calcium Channels; Endothelin-1; Imidazoles; In Vitro Techniques; Isoquinolines; Nifedipine; Rats; Vasoconstriction

1999
Endothelin-1-induced contraction of rat thoracic aorta depends on calcium entry through three types of calcium channel.
    Journal of cardiovascular pharmacology, 2000, Volume: 36, Issue:5 Suppl 1

    Topics: Acetamides; Animals; Aorta, Thoracic; Calcium; Calcium Channels; Endothelin-1; Imidazoles; In Vitro Techniques; Isoquinolines; Rats; Vasoconstriction

2000
Pharmacological properties of calcium entry channels in A7r5 cells activated by endothelin-1.
    Journal of cardiovascular pharmacology, 2000, Volume: 36, Issue:5 Suppl 1

    Topics: Acetamides; Calcium; Calcium Channels; Cell Line; Endothelin-1; Imidazoles; Isoquinolines

2000
Characterization of Ca(2+) channels involved in endothelin-1-induced mitogenic responses in vascular smooth muscle cells.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Count; Cell Division; Cell Line; DNA; Dose-Response Relationship, Drug; Endothelin-1; Imidazoles; Isoquinolines; Muscle, Smooth, Vascular; Nifedipine; Time Factors

2001
Failure of endothelin-1 to activate store-operated Ca2+ channels by lack of mobilization from intracellular Ca2+ stores in cultured bovine adrenal chromaffin cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 364, Issue:1

    Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cattle; Cells, Cultured; Chromaffin Cells; Endothelin-1; Enzyme Inhibitors; Imidazoles; Ion Channels; Isoquinolines; Thapsigargin

2001
Ca(2+) influx through nonselective cation channels plays an essential role in endothelin-1-induced mitogenesis in C6 glioma cells.
    Neuropharmacology, 2001, Volume: 41, Issue:3

    Topics: Acetamides; Animals; Brain Neoplasms; Calcium; Cell Division; Cell Line; Electrophysiology; Endothelin-1; Glioma; Imidazoles; Ion Channels; Isoquinolines; Mitosis; Patch-Clamp Techniques; Rats; Tumor Cells, Cultured

2001
Ca(2+) channels activated by endothelin-1 in CHO cells expressing endothelin-A or endothelin-B receptors.
    American journal of physiology. Cell physiology, 2001, Volume: 281, Issue:5

    Topics: Acetamides; Adenosine Triphosphatases; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; CHO Cells; Cricetinae; Electrophysiology; Endothelin-1; Enzyme Inhibitors; Imidazoles; Inositol Phosphates; Isoquinolines; Patch-Clamp Techniques; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Thapsigargin

2001
Ca(2+) channels involved in endothelin-induced mitogenic response in carotid artery vascular smooth muscle cells.
    American journal of physiology. Cell physiology, 2002, Volume: 282, Issue:2

    Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Carotid Arteries; Electric Conductivity; Endothelin-1; Imidazoles; Intracellular Membranes; Isoquinolines; Male; Mitosis; Muscle, Smooth, Vascular; Osmolar Concentration; Patch-Clamp Techniques; Rabbits

2002
Effects of extracellular Ca2+ influx on endothelin-1-induced intracellular mitogenic cascades in C6 glioma cells.
    European journal of pharmacology, 2002, Jan-25, Volume: 435, Issue:2-3

    Topics: Acetamides; Animals; Brain Neoplasms; Calcium; Calcium Channel Blockers; Calcium Channels; DNA; Drug Interactions; Endothelin-1; Enzyme Inhibitors; Flavonoids; Glioma; Imidazoles; Isoquinolines; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Mitogens; Rats; Thymidine; Tritium; Tumor Cells, Cultured

2002
Extracellular Ca2+ influx and endothelin-1-induced intracellular mitogenic cascades in rabbit internal carotid artery vascular smooth muscle cells.
    Journal of cardiovascular pharmacology, 2002, Volume: 40, Issue:2

    Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Carotid Arteries; Cells, Cultured; Drug Interactions; Endothelin-1; Isoquinolines; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Nifedipine; Rabbits

2002
Effects of phosphoinositide 3-kinase on the endothelin-1-induced activation of voltage-independent Ca(2+) channels and mitogenesis in Chinese hamster ovary cells stably expressing endothelin(a) receptor.
    Molecular pharmacology, 2002, Volume: 62, Issue:3

    Topics: Acetamides; Androstadienes; Animals; Calcium; Calcium Channels; CHO Cells; Chromones; Cricetinae; Drug Interactions; Endothelin-1; Enzyme Inhibitors; Imidazoles; Isoquinolines; Morpholines; Phosphatidylinositol 3-Kinases; Receptor, Endothelin A; Receptors, Endothelin; Transfection; Wortmannin

2002
Characterization of Ca2+ channels involved in ET-1-induced transactivation of EGF receptors.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 283, Issue:6

    Topics: Acetamides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Carotid Artery, Internal; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; ErbB Receptors; Extracellular Space; Imidazoles; Isoquinolines; Male; Muscle, Smooth, Vascular; Phosphorylation; Rabbits; Transcriptional Activation

2002
Role of phosphoinositide 3-kinase in the nonselective cation channel activation by endothelin-1/endothelinB receptor.
    American journal of physiology. Cell physiology, 2003, Volume: 284, Issue:2

    Topics: Acetamides; Androstadienes; Animals; Calcium; Calcium Channel Blockers; Calcium Signaling; Cell Membrane; CHO Cells; Chromones; Cricetinae; Endothelin-1; Endothelium, Vascular; Enzyme Inhibitors; Imidazoles; Ion Channels; Isoquinolines; Morpholines; Phosphatidylinositol 3-Kinases; Receptor, Endothelin B; Receptors, Endothelin; Signal Transduction; Up-Regulation; Wortmannin

2003
Involvements of voltage-independent Ca2+ channels and phosphoinositide 3-kinase in endothelin-1-induced PYK2 tyrosine phosphorylation.
    Molecular pharmacology, 2003, Volume: 63, Issue:4

    Topics: Acetamides; Androstadienes; Animals; Calcium; Calcium Channels; Cells, Cultured; Chromones; Drug Interactions; Endothelin-1; Enzyme Inhibitors; Focal Adhesion Kinase 2; Imidazoles; Isoquinolines; Morpholines; Muscle, Smooth, Vascular; Nifedipine; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein-Tyrosine Kinases; Rabbits; Tyrosine; Wortmannin

2003
Molecular mechanisms for the activation of Ca2+-permeable nonselective cation channels by endothelin-1 in C6 glioma cells.
    Biochemical pharmacology, 2003, May-01, Volume: 65, Issue:9

    Topics: Acetamides; Animals; Calcium; Calcium Channels; Cation Transport Proteins; Endothelin-1; Estrenes; Glioma; GTP-Binding Protein alpha Subunits, G12-G13; GTP-Binding Proteins; Heterotrimeric GTP-Binding Proteins; Imidazoles; Isoquinolines; Pertussis Toxin; Pyrrolidinones; Rats; Tumor Cells, Cultured

2003
Effects of phosphoinositide 3-kinase on endothelin-1-induced activation of voltage-independent Ca2+ channels and vasoconstriction.
    Biochemical pharmacology, 2004, Jul-15, Volume: 68, Issue:2

    Topics: Acetamides; Androstadienes; Animals; Basilar Artery; Calcium; Calcium Channels; Chromones; Drug Interactions; Endothelin-1; Endothelium, Vascular; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Isoquinolines; Morpholines; Muscle, Smooth, Vascular; Phosphatidylinositol 3-Kinases; Rabbits; Vasoconstriction; Wortmannin

2004