lisuride has been researched along with dironyl in 136 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 46 (33.82) | 18.7374 |
1990's | 45 (33.09) | 18.2507 |
2000's | 31 (22.79) | 29.6817 |
2010's | 14 (10.29) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Audinot, V; Boutin, JA; Cussac, D; Maiofiss, L; Millan, MJ; Newman-Tancredi, A | 1 |
Bowie, M; Boyar, RM; Budinger, JM; Hellman, L; Mountain, IM; Rosenberg, BJ; Stock, CC; Teller, MN | 1 |
Filip, V; Hálková, E; Karen, P; Marsálek, M | 1 |
Horowski, R; Jähnig, P; Jenner, P; Lange, KW; Löschmann, PA; Marsden, CD; Wachtel, H | 1 |
Baronti, F; Brughitta, G; Chase, TN; Conant, KE; Giuffra, M; Mouradian, MM | 1 |
Judd, AM; MacLeod, RM | 1 |
Ahlenius, S; Hillegaart, V; Wijkström, A | 1 |
Carlsson, A; Kujacic, M; Löfberg, L; Svensson, K | 1 |
Olbrich, R; Schanz, H | 2 |
Carlsson, A; Ekman, A; Hoffmann, WE; Lum, JT; Piercey, MF; Svensson, K | 1 |
Agnoli, A; Baronti, F; Horowski, R; Lucarelli, C; Ruggieri, S; Stocchi, F; Viselli, F | 1 |
Clark, D; Ericsson, M; Furmidge, LJ; Johnson, D; Petry, N; Tong, ZY | 1 |
Krause, W; Kühne, G; Seifert, W | 1 |
Carratù, MR; DeSerio, A; Federico, F; Mitolo-Chieppa, D | 1 |
Clark, D; Galloway, MP; Salah, RS | 1 |
Carratù, MR; Conte-Camerino, D; De Serio, A; Ferrari, E; Lagioia, R; Mitolo-Chieppa, D | 1 |
Krecek, J; Rasková, H; Sladkovský, J; Treu, M; Urbanová, Z | 1 |
Brest'ák, M; Danĕk, J; Hasanová, M; Lidický, J; Mares, J | 1 |
Fingerová, H; Gazárek, F; Pohanka, J; Talas, M; Vĕtr, M | 1 |
Horowski, R; Schmelzle, A; Scholz, A; Wüster, C; Ziegler, R | 1 |
Genitrini, S; Giovannini, P; Girotti, F; Piccolo, I; Scigliano, G; Suchy, I; Testa, D | 1 |
Dorow, R; Gräf, KJ; Krause, W; Kühne, G; Sauerbrey, N; Träger, H | 1 |
Dlabac, A; Dobrovský, K; Valchár, M | 1 |
Agnoli, A; Antonini, A; Argenta, M; Berardelli, A; Carta, A; Formica, A; Stocchi, F | 1 |
Cepický, P; Vido, I | 1 |
Dlabac, A; Dobrovský, K; Krejcí, I; Valchár, M | 1 |
Al-Sereiti, MR; Turner, P | 1 |
Gieschen, H; Hümpel, M; Labitzky, C; Sostarek, D | 1 |
Carlsson, M; Eriksson, E | 1 |
Carlsson, A; Clark, D; Hjorth, S | 2 |
Celeda, L; Elis, J; Krecek, J; Krejcí, I; Lavický, J; Príborská, Z; Rasková, H; Urbanová, Z; Vanĕcek, J | 1 |
Albizzati, MG; Bassi, S; Corsini, GU; Frattola, L; Piolti, R; Suchy, I; Trabucchi, M | 1 |
Krejcí, I; Vĕtr, M | 1 |
Talas, M; Vĕtr, M | 1 |
Konecný, V; Vĕtr, M | 1 |
König, A; Losa, M; Müller, OA; Schopohl, J; Stalla, GK; von Werder, K | 1 |
Dĕdicová, A; Jakoubek, B; Kosar, E; Sumová, A | 1 |
Filip, V; Filipová, M; Kás, S; Krejcová, H; Krivka, J; Macek, Z; Marková, J; Müllerová, S; Votavová, M; Zizková, B | 1 |
Badino, G; De Cecco, L; Fasce, V; Ferreri, C; Horowski, R; Rainer, E; Scholz, A; Valenzano, M; Venturini, PL | 1 |
Dorow, R; Gräf, KJ; Horowski, R; Köhler, D | 1 |
Lidický, J; Pícha, J; Píchová, D; Sedláková, J | 1 |
Rinne, UK | 1 |
Besser, M; Ciccarelli, E; Grossman, A; Touzel, R | 1 |
Bankiewicz, K; Brücke, T; Harvey-White, J; Kopin, I | 1 |
Dlabac, A; Krejcí, I; Valchár, M; Vrsecká, M | 1 |
Rinne, UK; Suchy, I; Wachtel, H | 1 |
Herbster, G; Koller, WC | 1 |
Suchy, I; Ulrich, G | 1 |
Hoffmann, WE; Piercey, MF; Travis, M; Vogelsang, GD | 1 |
Carlsson, A; Carlsson, M; Eriksson, E | 1 |
Costantini, S; De Cecco, L; Fasce, V; Gorlero, F; Horowski, R; Rainer, E; Valenzano, M; Venturini, PL | 1 |
Franc, Z; Lapka, R; Marek, J; Rejholec, V | 1 |
Chiodini, P; Cozzi, R; Dallabonzana, D; Dorow, R; Horowski, R; Liuzzi, A; Oppizzi, G; Rainer, E; Verde, G | 1 |
Critchley, P; Parkes, D | 1 |
Brücke, T; Danielczyk, W; Riederer, P; Simányi, M; Sofic, E | 1 |
Bauer, J; Hána, V; Marek, J; Srámková, J | 1 |
Jahodová, J; Schreiber, V | 1 |
Chiodini, PG; Dallabonzana, D; Dorow, R; Horowski, R; Liuzzi, A; Oppizzi, G; Verde, G | 1 |
Bonuccelli, U; Corsini, GU; Del Zompo, M; Rainer, E | 1 |
Felt, V; Nedvídková, J | 1 |
Ausková, M; Rezábek, K; Semonský, M; Zikán, V | 1 |
Kehr, W | 1 |
Dorow, R; Hasan, SH; Krause, W; Nieuweboer, B | 1 |
Franc, Z; Lapka, R; Smolík, S | 1 |
Dorow, R; Wachtel, H | 1 |
Bone, RG; Villar, HO | 1 |
Spealman, RD | 1 |
Cvak, L; Golda, V | 1 |
Akai, T; Kuno, S; Mizuta, E; Ozawa, M; Yamaguchi, M | 1 |
Klimes, J; Sochor, J; Srumová, M | 1 |
Brown, D; Factor, SA; Molho, ES; Podskalny, GD | 1 |
Aufdembrinke, B; Bruggi, P; Godi, L; Martignoni, E; Miltenburger, C; Nappi, G; Pacchetti, C; Voet, B | 1 |
Akai, T; Hasan, S; Mizokawa, T; Nakada, Y; Nakagawa, H; Rettig, KJ; Wachtel, H; Yamaguchi, M | 1 |
Akai, T; Kuno, S; Mizuta, E; Yamaguchi, M | 1 |
Gerlach, J; Peacock, L | 1 |
Ferrarese, C; Piolti, R; Pozzi, C | 1 |
Akai, T; Hara, K; Ikoma, Y; Nakata, Y; Wachtel, H; Yamaguchi, M | 1 |
Gieschen, H; Hildebrand, M; Husemann, M; Rauschenbach, R; Salomon, B | 1 |
Attanasio, R; Costa, A; Cozzi, R; Dallabonzana, D; Horowski, R; Liuzzi, A; Martignoni, E; Nappi, G; Rainer, E | 1 |
Golda, V; Hilgertová, J | 4 |
Kokunai, T; Tamaki, N; Yonezawa, K | 1 |
Haluzík, M; Hána, V; Schreiber, V | 1 |
Golda, V | 1 |
Balducci, C; Koob, GF; Piercy, M; Pulvirenti, L | 1 |
Ichihara, K; Kamei, H; Mizukoshi, K; Nagasaka, M; Okumura, K | 1 |
Golda, V; Hilgertová, J; Zórad, S | 1 |
Golda, V; Jurcovicová, J | 1 |
Hána, V; Justová, V; Krsek, M; Lacinová, Z; Marek, J | 1 |
Asano, S; Kirino, T; Suzuki, I; Ueki, K | 1 |
Ficková, M; Golda, V; Jurcovicová, J; Macho, L; Pinterova, L; Zórad, S | 2 |
Izzo, E; Koob, GF; Orsini, C; Pulvirenti, L | 1 |
Koob, GF; Orsini, C; Pulvirenti, L | 1 |
Fiserová, A; Halada, P; Kren, V; Pospísil, M; Prikrylová, V; Sedmera, P; Stibor, I; Weignerová, L | 1 |
Ishiguro, T; Iwai, Y; Komiyama, M; Matsuzaka, Y; Morikawa, T; Yamanaka, K; Yasui, T | 1 |
Platt, DM; Rodefer, JS; Rowlett, JK; Spealman, RD | 1 |
Hashimoto, S; Midorikawa, S; Sanada, H; Watanabe, T; Yatabe, J | 1 |
Iga, T; Irizuki, N; Sawada, Y; Takayanagi, R; Yamada, Y; Yamamoto, K | 1 |
Calda, P; Pavlista, D; Zivný, J | 1 |
Krall, CM; Matea, PJ; McDougall, SA; Sibole, JM | 1 |
Kranda, K; Pretl, M; Sonka, K | 1 |
Eich, E; Kren, V; Pertz, HH | 1 |
Cador, M; Koob, GF; Stinus, L; Zorrilla, EP | 1 |
Golda, V; Kudlackova, Z | 1 |
Farley, CM; Hernandez, RM; McDougall, SA; Reichel, CM | 1 |
Burris, KD; Kikuchi, T; Miwa, T; Mori, T; Stark, A; Tadori, Y; Tottori, K | 1 |
Cvak, J; Flieger, M; Honzátko, A; Vaingátová, S | 1 |
Baella, SA; Crawford, CA; McDougall, SA; Stuebner, NM; Yoshida, ST | 1 |
Farley, CM; McDougall, SA; Reichel, CM; Wacan, JJ | 1 |
Hoefer, ME; Koob, GF; Pulvirenti, L; Voskanian, SJ | 1 |
Feenstra, RW; Glennon, JC; Hesselink, MB; Long, SK; McCreary, AC; Reinders, JH; Ronken, E; Van Der Neut, M; Van Scharrenburg, G | 1 |
Chen, R; Johnson, JL; Jordan, S; Kambayashi, J; Kikuchi, T; Kitagawa, H; McQuade, R; Regardie, K; Tadori, Y | 1 |
Gustafsson, BI; Hauso, Ø; Loennechen, JP; Nordrum, I; Stunes, AK; Waldum, HL | 1 |
Cortez, AM; Crawford, CA; Iñiguez, SD; McDougall, SA | 1 |
Hayashi, S; Inoue, Y; Matsumoto, Y; Okawara, M; Okawara, S; Yamaguchi, H | 1 |
Gustafsson, BI; Hauso, O; Nordrum, IS; Waldum, HL | 1 |
Chen, JF; Herm, L; Kalda, A; Rinken, A; Zharkovsky, A | 1 |
Bendszus, M; Distler, O; Dokoupilova, E; Dvorak, Z; Eich, W; Fleck, M; Gaubitz, M; Hechler, M; Jansen, JP; Krause, A; Müller-Ladner, U; Pache, L; Reiter, R | 1 |
Amarie, OV; Dumitrascu, R; Eickelberg, O; Grimminger, F; Königshoff, M; Reiter, R; Schermuly, RT; Seeger, W; Udalov, S | 1 |
Chen, H; Hao, W; Su, Q; Wang, X; Xiang, X; Zhang, D; Zhang, J | 1 |
Dumitrascu, R; Eickelberg, O; Ghofrani, HA; Grimminger, F; Königshoff, M; Kouri, F; Kulcke, C; Morrell, N; Pullamsetti, SS; Reiter, R; Schermuly, RT; Seeger, W; Weissmann, N; Yang, X | 1 |
Glusa, E; Görnemann, T; Jantschak, F; Kekewska, A; Pertz, HH | 1 |
Morrell, N; Sitbon, O | 1 |
Brosda, J; Fink, H; Franke, RT; Gmeiner, P; Hübner, H; Jantschak, F; Möller, D; Pertz, HH | 1 |
Gong, Q; Huang, C; Huang, J; Li, G | 1 |
Amodeo, LR; Crawford, CA; Der-Ghazarian, T; Gonzalez, AE; Gutierrez, A; Humphrey, DE; McDougall, SA; Valentine, JM; Widarma, CB | 1 |
Attard, M; Ghataorhe, P; Lythgoe, MP; Rhodes, CJ; Wharton, J; Wilkins, MR | 1 |
Allanore, Y; Bruni, C; Distler, O; Gabrielli, A; Iannone, F; Matucci-Cerinic, M; Praino, E | 1 |
Makary, S; Tawfik, MK | 1 |
Distler, JHW; Ensminger, SM; Gocht, A; Heim, C; Ramsperger-Gleixner, M; Spriewald, B; Weyand, M | 1 |
Agarwal, V; Chaturvedi, S; Misra, DP; Prasad, N; Rai, MK; Rastogi, K; Singh, H | 1 |
8 review(s) available for lisuride and dironyl
Article | Year |
---|---|
Comparative effects of a series of prolactin inhibitors, 17beta-estradiol and 2alpha-methyldihydrotestosterone propionate, on growth of 7,12-dimethylbenz(a)anthracene-induced rat mammary carcinomas.
Topics: 9,10-Dimethyl-1,2-benzanthracene; Acetonitriles; Androstanols; Animals; Breast Neoplasms; Bromocriptine; Drug Evaluation, Preclinical; Ergolines; Ergot Alkaloids; Estradiol; Female; Humans; Lisuride; Mammary Neoplasms, Experimental; Prolactin; Rats; Urea | 1977 |
Dopamine receptor agonists: mechanisms underlying autoreceptor selectivity. II. Theoretical considerations.
Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Corpus Striatum; Cyclic AMP; Dextroamphetamine; Dopamine; Humans; Isomerism; Lisuride; Models, Neurological; Molecular Conformation; Motor Activity; Nucleus Accumbens; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Dopamine; Substantia Nigra; Synaptosomes | 1985 |
Dopamine-receptor agonists: mechanisms underlying autoreceptor selectivity. I. Review of the evidence.
Topics: Acetylcholine; Adenylyl Cyclases; Animals; Behavior, Animal; Brain; Caudate Nucleus; Deoxyglucose; Dopamine; Humans; Lisuride; Models, Biological; Nerve Tissue Proteins; Phenanthrenes; Piperidines; Rats; Receptors, Dopamine; Stereoisomerism; Substantia Nigra; Synaptosomes; Tegmentum Mesencephali | 1985 |
Parkinson's disease: drug-induced psychiatric states.
Topics: Aged; Anxiety; Bipolar Disorder; Clozapine; Depression; Electroconvulsive Therapy; Humans; Levodopa; Lisuride; Male; Ondansetron; Parkinson Disease; Psychoses, Substance-Induced; Sexual Dysfunctions, Psychological | 1995 |
Pathways in pulmonary arterial hypertension: the future is here.
Topics: Acetamides; Animals; Antihypertensive Agents; Benzamides; Clinical Trials as Topic; Drugs, Investigational; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Epoprostenol; Guanylate Cyclase; Humans; Hypertension, Pulmonary; Imatinib Mesylate; Lisuride; Nitric Oxide; Phosphodiesterase 5 Inhibitors; Piperazines; Protein Kinase Inhibitors; Pyrazines; Pyrazoles; Pyrimidines; Serotonin Antagonists; Sulfonamides | 2012 |
Relationships between serotoninergic system and skin fibrotic.
Topics: Animals; Cell Growth Processes; Dopamine Agonists; Fibrosis; Humans; Lisuride; Precision Medicine; Receptor, Serotonin, 5-HT1A; Scleroderma, Systemic; Selective Serotonin Reuptake Inhibitors; Serotonin; Skin | 2014 |
Why drugs fail in clinical trials in pulmonary arterial hypertension, and strategies to succeed in the future.
Topics: Animals; Biomarkers; Clinical Studies as Topic; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Combinations; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypertension, Pulmonary; Lisuride; Phenotype; Phentolamine; Protein-Tyrosine Kinases; Vasoactive Intestinal Peptide | 2016 |
Use of biologics and other novel therapies for the treatment of systemic sclerosis.
Topics: Abatacept; Acetamides; Antibodies, Monoclonal, Humanized; Biological Products; Clinical Trials as Topic; Fibrinolytic Agents; Fibrosis; Humans; Hypertension, Pulmonary; Indoles; Inflammation; Joints; Lisuride; Lung; PubMed; Pyrazines; Pyrazoles; Pyrimidines; Scleroderma, Systemic; Skin | 2017 |
17 trial(s) available for lisuride and dironyl
Article | Year |
---|---|
Treatment of extrapyramidal side effects with terguride.
Topics: Administration, Oral; Adult; Antipsychotic Agents; Dopamine Agents; Dyskinesia, Drug-Induced; Female; Humans; Lisuride; Male; Middle Aged; Neurologic Examination; Parkinson Disease, Secondary; Psychotic Disorders; Schizophrenia; Schizophrenic Psychology | 1992 |
An evaluation of the partial dopamine agonist terguride regarding positive symptoms reduction in schizophrenics.
Topics: Adolescent; Adult; Antipsychotic Agents; Drug Evaluation; Female; Humans; Lisuride; Psychological Tests; Receptors, Dopamine; Schizophrenia; Schizophrenia, Paranoid | 1991 |
Antagonist effect of terguride in Parkinson's disease.
Topics: Adult; Aged; Dopamine Agents; Humans; Levodopa; Lisuride; Middle Aged; Parkinson Disease | 1991 |
[Terguride in hyperprolactinemia--experiences with 5 patients].
Topics: Adult; Clinical Trials as Topic; Dose-Response Relationship, Drug; Ergolines; Female; Follow-Up Studies; Humans; Hyperprolactinemia; Lisuride; Male; Middle Aged; Pituitary Neoplasms; Prolactin; Prolactinoma; Prospective Studies | 1990 |
Pharmacokinetics and endocrine effects of terguride in healthy subjects.
Topics: Adult; Affect; Double-Blind Method; Electrocardiography; Enzyme Induction; Ergolines; Female; Half-Life; Humans; Hydrocortisone; Injections, Intravenous; Lisuride; Male; Pituitary Gland, Anterior; Pituitary Hormones; Prolactin; Psychomotor Performance; Reference Values; Sex Factors | 1990 |
Effects of terguride in patients with Huntington's disease.
Topics: Adult; Affect; Aged; Awareness; Clinical Trials as Topic; Dopamine Agents; Double-Blind Method; Ergolines; Female; Humans; Huntington Disease; Lisuride; Male; Middle Aged | 1989 |
The effects of lisuride, terguride and bromocriptine on intraocular pressure (IOP).
Topics: Adult; Bromocriptine; Double-Blind Method; Ergolines; Humans; Intraocular Pressure; Lisuride; Random Allocation | 1989 |
Therapeutic experience with transdihydrolisuride in Huntington's disease.
Topics: Adolescent; Adult; Clinical Trials as Topic; Double-Blind Method; Ergolines; Female; Humans; Huntington Disease; Lisuride; Male; Mental Processes; Middle Aged; Movement Disorders; Neuropsychological Tests; Random Allocation; Receptors, Dopamine; Time Factors | 1986 |
Terguride in parkinsonism. A multicenter trial.
Topics: Adult; Aged; Aged, 80 and over; Clinical Trials as Topic; Ergolines; Female; Humans; Lisuride; Male; Middle Aged; Motor Skills; Neurologic Examination; Parkinson Disease | 1988 |
Suppression of puerperal lactation by terguride. A double-blind study.
Topics: Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Ergolines; Female; Humans; Lactation; Lisuride; Postpartum Period; Pregnancy; Prolactin | 1988 |
Terguride--a new dopamine agonist drug: a comparison of its neuroendocrine and side effect profile with bromocriptine.
Topics: Adult; Blood Pressure; Bromocriptine; Double-Blind Method; Drug Evaluation; Ergolines; Follicle Stimulating Hormone; Growth Hormone; Humans; Hydrocortisone; Lisuride; Male; Prolactin; Pulse; Random Allocation; Thyrotropin | 1988 |
Evaluation of terguride in patients with Parkinson's disease.
Topics: Adult; Aged; Brain; Clinical Trials as Topic; Disability Evaluation; Ergolines; Female; Humans; Lisuride; Male; Middle Aged; Motor Skills; Parkinson Disease; Receptors, Dopamine | 1987 |
[The effect of terguride on the dynamics and mean level of vigilance. A controlled electroencephalographic study with elderly subjects].
Topics: Aged; Alpha Rhythm; Arousal; Double-Blind Method; Electroencephalography; Ergolines; Humans; Lisuride; Middle Aged | 1987 |
Effects of terguride on anterior pituitary function in parkinsonian patients treated with L-dopa: a double-blind study versus placebo.
Topics: Aged; Antiparkinson Agents; Dopamine Agonists; Double-Blind Method; Female; Humans; Hyperprolactinemia; Levodopa; Lisuride; Male; Middle Aged; Parkinson Disease; Pituitary Function Tests; Pituitary Gland, Anterior; Pituitary Hormones, Anterior | 1996 |
[Arrest of lactation after 2nd trimester abortion with a single dose of cabergoline in comparison with 10-day administration of teguride].
Topics: Abortion, Induced; Adolescent; Adult; Cabergoline; Drug Administration Schedule; Ergolines; Female; Humans; Lactation; Lisuride; Pregnancy; Pregnancy Trimester, Second; Prospective Studies | 2003 |
Management of restless legs syndrome by the partial D2-agonist terguride.
Topics: Adult; Aged; Dopamine Agonists; Female; Humans; Lisuride; Male; Middle Aged; Receptors, Dopamine D2; Restless Legs Syndrome; Self-Assessment; Sleep; Sleep Stages; Treatment Outcome | 2003 |
Evaluation of the efficacy and safety of terguride in patients with fibromyalgia syndrome: results of a twelve-week, multicenter, randomized, double-blind, placebo-controlled, parallel-group study.
Topics: Adult; Cervical Vertebrae; Depression; Dopamine Agonists; Double-Blind Method; Female; Fibromyalgia; Humans; Lisuride; Male; Middle Aged; Pain; Pain Measurement; Psychiatric Status Rating Scales; Sickness Impact Profile; Spinal Stenosis; Surveys and Questionnaires; Treatment Outcome | 2010 |
111 other study(ies) available for lisuride and dironyl
Article | Year |
---|---|
Differential actions of antiparkinson agents at multiple classes of monoaminergic receptor. I. A multivariate analysis of the binding profiles of 14 drugs at 21 native and cloned human receptor subtypes.
Topics: Animals; Antiparkinson Agents; Binding Sites; Binding, Competitive; Cholinergic Antagonists; Cloning, Molecular; Cluster Analysis; Dopamine Agonists; Humans; Rats; Receptor, Muscarinic M1; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Histamine H1; Receptors, Muscarinic; Receptors, Neurotransmitter; Receptors, Serotonin | 2002 |
Terguride stimulates locomotor activity at 2 months but not 10 months after 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine treatment of common marmosets.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Antiparkinson Agents; Callithrix; Disease Models, Animal; Dopamine Agents; Female; Lisuride; Male; Motor Activity; Parkinson Disease, Secondary; Time Factors | 1992 |
Partial dopamine agonist therapy of levodopa-induced dyskinesias.
Topics: Adult; Aged; Dopamine Agents; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Humans; Levodopa; Lisuride; Middle Aged; Movement | 1992 |
Dopamine receptor and adrenoceptor agonists inhibit prolactin release from MMQ cells.
Topics: Adrenergic Agonists; Cyclic AMP; Depression, Chemical; Dopamine; Humans; Lisuride; Marine Toxins; Oxocins; Pituitary Neoplasms; Prolactin; Receptors, Dopamine; Tumor Cells, Cultured | 1991 |
Quinpirole--a 5-HT receptor antagonist?
Topics: Animals; Brain; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agents; Ergolines; Hydrazines; Lisuride; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reference Values; Reserpine; Serotonin | 1991 |
Dopamine receptors, controlling dopamine levels in rat adrenal glands-comparison with central dopaminergic autoreceptors.
Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenal Medulla; Animals; Apomorphine; Azepines; Diencephalon; Domperidone; Dopamine; Dopamine Agents; Epinephrine; Ergolines; Lisuride; Male; Norepinephrine; Phenanthrenes; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Telencephalon | 1991 |
Effects of the partial dopamine receptor agonists SDZ 208-911, SDZ 208-912 and terguride on central monoamine receptors. A behavioral, biochemical and electrophysiological study.
Topics: 4-Butyrolactone; Animals; Behavior, Animal; Brain; Dopamine; Dopamine Agents; Ergolines; Lisuride; Male; Motor Activity; Neurons; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Reserpine; Serotonin; Substantia Nigra; Time Factors | 1991 |
Behavioural profile of partial D2 dopamine receptor agonists. 1. Atypical inhibition of d-amphetamine-induced locomotor hyperactivity and stereotypy.
Topics: Animals; Dextroamphetamine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Lisuride; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Stereotyped Behavior | 1991 |
Pharmacokinetics of 3H-terguride in elderly volunteers.
Topics: Aged; Biotransformation; Computer Simulation; Feces; Humans; Intestinal Absorption; Lisuride; Male; Middle Aged; Radioimmunoassay; Reference Values; Tissue Distribution | 1991 |
Comparative evaluation of lisuride and terguride, ergot alkaloid derivatives, on the field-stimulated vas deferens of mouse.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Ergolines; Lisuride; Male; Mice; Molecular Structure; Muscle Contraction; Muscle, Smooth; Quinpirole; Receptors, Dopamine; Structure-Activity Relationship; Vas Deferens | 1991 |
Differential agonist profile of the enantiomers of 3-PPP at striatal dopamine autoreceptors: dependence on extracellular dopamine.
Topics: Animals; Biogenic Monoamines; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Electrochemistry; Ergolines; In Vitro Techniques; Lisuride; Male; Nerve Tissue Proteins; Nucleus Accumbens; Piperidines; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism | 1991 |
[Effects of the partial dopamine receptor agonist, terguride, on the field-stimulated vas deferens in the mouse].
Topics: Animals; Dopamine Agents; Electric Stimulation; Ergolines; In Vitro Techniques; Lisuride; Male; Mice; Muscle, Smooth; Vas Deferens | 1990 |
Metipranolol and tergurid induced enhancement of delayed hypersensitivity and sedative effect in stressed calves.
Topics: Animals; Cattle; Hypersensitivity, Delayed; Hypnotics and Sedatives; Lisuride; Metipranolol; Stress, Physiological | 1990 |
[The effect of terguride on contractility of rat uterine strips].
Topics: Animals; Female; In Vitro Techniques; Lisuride; Rats; Rats, Inbred Strains; Uterine Contraction | 1990 |
Terguride in the treatment of hyperprolactinemia.
Topics: Adolescent; Adult; Female; Humans; Hyperprolactinemia; Lisuride; Prolactin | 1990 |
Terguride in the treatment of Parkinson disease: preliminary experience.
Topics: Dyskinesia, Drug-Induced; Humans; Levodopa; Lisuride; Male; Middle Aged; Parkinson Disease | 1990 |
The binding characteristics of 3H-terguride in various brain areas.
Topics: Animals; Brain; Cattle; Ergolines; Ergotamines; Lisuride; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Species Specificity; Swine | 1989 |
[Pharmacologic arrest of lactation. Comparison of Deprenon, lisuride, terguride and mestranol].
Topics: Adult; Ergolines; Female; Humans; Lactation; Lisuride; Mestranol; Pregnancy; Prolactin | 1989 |
Comparison of (3H)-terguride and (3H)-spiperone binding to dopamine receptors in the rat striatum.
Topics: Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Ergolines; Ergotamines; Lisuride; Male; Rats; Receptors, Dopamine; Spiperone | 1989 |
Studies on the biotransformation of lonazolac, bromerguride, lisuride and terguride in laboratory animals and their hepatocytes.
Topics: Animals; Biotransformation; Dogs; Female; Guinea Pigs; In Vitro Techniques; Lisuride; Liver; Macaca fascicularis; Models, Biological; Molecular Structure; Perfusion; Pyrazoles; Rats; Rats, Inbred Strains; Species Specificity; Xenobiotics | 1989 |
The enhanced responsiveness of hypophyseal DA receptors in female rats induced by repeated reserpine treatment is not due to decreased oestrogen secretion.
Topics: Animals; Estradiol; Estrogens; Female; Lisuride; Ovariectomy; Piperidines; Pituitary Gland, Posterior; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine | 1989 |
Pharmacologic interventions to antagonize stress-induced immune consequences.
Topics: Animals; Blindness; Cattle; Cattle Diseases; Ergolines; Hypersensitivity, Delayed; Leukocyte Count; Lisuride; Metipranolol; Mice; Organ Size; Propanolamines; Respiratory Tract Diseases; Spleen; Stress, Physiological; Thymus Gland; Vibration | 1987 |
The effect of the partial dopamine agonist terguride on negative symptoms in schizophrenics.
Topics: Adult; Dopamine Agents; Ergolines; Humans; Lisuride; Male; Middle Aged; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenic Psychology | 1988 |
Suppression of lactation with Terguride.
Topics: Ergolines; Female; Humans; Lactation; Lisuride; Pregnancy | 1988 |
Terguride in the treatment of prolactin-induced luteal insufficiency.
Topics: Adolescent; Adult; Corpus Luteum; Ergolines; Female; Humans; Hyperprolactinemia; Infertility, Female; Lisuride; Menstruation Disturbances | 1988 |
Lactation-inhibiting and prolactin-lowering effect of lisuride and transdihydrolisuride. A comparative study.
Topics: Ergolines; Female; Humans; Lactation; Lisuride; Pregnancy; Prolactin | 1988 |
Combined pituitary function-test with four hypothalamic releasing hormones.
Topics: Adrenocorticotropic Hormone; Adult; Corticotropin-Releasing Hormone; Female; Follicle Stimulating Hormone; Growth Hormone; Growth Hormone-Releasing Hormone; Humans; Hydrocortisone; Lisuride; Luteinizing Hormone; Male; Pituitary Function Tests; Pituitary Gland, Anterior; Pituitary Hormone-Releasing Hormones; Premedication; Prolactin; Radioimmunoassay; Thyrotropin; Thyrotropin-Releasing Hormone | 1986 |
Effects of ergot alkaloids on stress-induced analgesia.
Topics: Animals; Dihydroergotoxine; Endorphins; Ergot Alkaloids; Lisuride; Male; Pain; Rats; Receptors, Opioid; Stress, Physiological | 1986 |
Rapid regression of macroprolactinomas by the new dopamine partial agonist terguride.
Topics: Adenoma; Adult; Ergolines; Female; Follow-Up Studies; Humans; Lisuride; Pituitary Neoplasms; Prolactin; Receptors, Dopamine; Thyrotropin-Releasing Hormone; Tomography, X-Ray Computed | 1986 |
[The effect of ovarian steroids on the pharmacokinetics of Terguride in the rat uterus].
Topics: Age Factors; Animals; Ergolines; Estradiol; Female; Kinetics; Lisuride; Organ Size; Ovariectomy; Progesterone; Rats; Rats, Inbred Strains; Uterus | 1986 |
Dopamine agonists as primary treatment in Parkinson's disease.
Topics: Antiparkinson Agents; Bromocriptine; Disability Evaluation; Drug Therapy, Combination; Ergolines; Humans; Levodopa; Lisuride; Long-Term Care; Parkinson Disease; Pergolide; Receptors, Dopamine | 1987 |
The partial dopamine receptor agonist terguride in the MPTP-induced hemiparkinsonian monkey model.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Disease Models, Animal; Ergolines; Female; Lisuride; Macaca fascicularis; Parkinson Disease, Secondary; Pyridines; Receptors, Dopamine | 1988 |
Binding characteristics of the dopamine agonist/antagonist [3H]terguride (transdihydrolisuride) in the rat striatum.
Topics: Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Kinetics; Lisuride; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1987 |
Terguride, a mixed dopamine agonist-antagonist, in animal models of Parkinson's disease.
Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; Brain; Disease Models, Animal; Ergolines; Levodopa; Lisuride; Male; Motor Activity; Parkinson Disease; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior | 1987 |
Electrophysiological evaluation of a partial agonist of dopamine receptors.
Topics: Amphetamine; Animals; Apomorphine; Clozapine; Dose-Response Relationship, Drug; Electric Stimulation; Ergolines; Haloperidol; Lisuride; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra | 1987 |
The intrinsic activities of the partial dopamine receptor agonists (-)-3-PPP and TDHL on pituitary dopamine receptors are lower in female than in male rats.
Topics: Animals; Antiparkinson Agents; Ergolines; Female; In Vitro Techniques; Lisuride; Male; Piperidines; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sex Factors; Stereoisomerism | 1987 |
Effect of terguride on prolactin levels in normal, puerperal and hyperprolactinaemic women.
Topics: Adult; Dose-Response Relationship, Drug; Ergolines; Female; Humans; Hyperprolactinemia; Lactation; Lisuride; Postpartum Period; Pregnancy; Prolactin; Time Factors | 1986 |
Pharmacokinetics of oral terguride in patients with a prolactinoma.
Topics: Acromegaly; Adult; Ergolines; Female; Half-Life; Humans; Kinetics; Lisuride; Male; Middle Aged; Pituitary Neoplasms; Prolactin | 1986 |
Chronic treatment of pathological hyperprolactinemia and acromegaly with the new ergot derivative terguride.
Topics: Acromegaly; Adenoma; Adolescent; Adult; Ergolines; Female; Humans; Hyperprolactinemia; Lisuride; Male; Menstruation; Middle Aged; Pituitary Neoplasms | 1986 |
Transdihydrolisuride in parkinsonism.
Topics: Aged; Blood Pressure; Ergolines; Female; Humans; Levodopa; Lisuride; Male; Middle Aged; Movement Disorders; Nausea; Parkinson Disease; Psychoses, Substance-Induced | 1987 |
Terguride: partial dopamine agonist in the treatment of Parkinson's disease.
Topics: Aged; Aged, 80 and over; Ergolines; Female; Humans; Lisuride; Male; Motor Skills; Parkinson Disease | 1987 |
[Terguride in the treatment of hyperprolactinemia and acromegaly].
Topics: Acromegaly; Adolescent; Adult; Aged; Ergolines; Female; Humans; Hyperprolactinemia; Lisuride; Male; Middle Aged; Pregnancy | 1986 |
[Comparison of the dopaminergic activity of the new Czechoslovak ergoline derivate transdihydrolisuride (Tergurid Spofa) with lisuride].
Topics: Animals; Dopamine; Ergolines; Estradiol; Hypertrophy; Lisuride; Male; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains | 1986 |
Effect of the new ergot derivative terguride on plasma PRL and GH levels in patients with pathological hyperprolactinemia or acromegaly.
Topics: Acromegaly; Adolescent; Adult; Bromocriptine; Ergolines; Female; Growth Hormone; Humans; Lisuride; Male; Middle Aged; Prolactin; Time Factors | 1985 |
Therapeutic efficacy of a partial dopamine agonist in drug-free parkinsonian patients.
Topics: Aged; Disability Evaluation; Dopamine; Drug Evaluation; Ergolines; Female; Humans; Lisuride; Male; Middle Aged; Nervous System; Parkinson Disease | 1985 |
[Use of dironyl in the treatment of acromegaly and hyperprolactinemia].
Topics: Acromegaly; Adult; Aged; Ergolines; Female; Growth Hormone; Humans; Hyperprolactinemia; Lisuride; Male; Middle Aged; Prolactin | 1985 |
[Inhibition of lactation by N-(D-6-methyl-8-isoergolin-1-yl)-N',N'-diethylurea (VUFB-6638)].
Topics: Administration, Oral; Animals; Body Weight; Drug Synergism; Ergolines; Female; Lactation; Lethal Dose 50; Lisuride; Oxytocin; Pregnancy; Prolactin; Urea | 1974 |
Transdihydrolisuride, a partial dopamine receptor antagonist: effects on monoamine metabolism.
Topics: 3,4-Dihydroxyphenylacetic Acid; 5-Hydroxytryptophan; Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Brain; Catecholamines; Dihydroxyphenylalanine; Ergolines; Lisuride; Male; Methyltyrosines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1984 |
Pharmacokinetics and pharmacodynamics of the ergot derivative, transdihydrolisuride, in man.
Topics: Adult; Biological Availability; Ergolines; Humans; Kidney; Kinetics; Lisuride; Male; Prolactin; Radioimmunoassay | 1984 |
Radioreceptor assay for ergot derivatives, transdihydrolisuride and lisuride, in biological fluids.
Topics: Animals; Antibody Specificity; Ergolines; Female; Hydrogen-Ion Concentration; Kinetics; Lisuride; Radioligand Assay; Rats; Rats, Inbred Strains | 1984 |
Dual action on central dopamine function of transdihydrolisuride, a 9, 10-dihydrogenated analogue of the ergot dopamine agonist lisuride.
Topics: Adult; Animals; Apomorphine; Behavior, Animal; Body Temperature; Catalepsy; Ergolines; Female; Haloperidol; Humans; Lisuride; Male; Mice; Motor Activity; Prolactin; Rats; Rats, Inbred Strains | 1983 |
Discriminating D1 and D2 agonists with a hydrophobic similarity index.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Apomorphine; Benzazepines; Chemical Phenomena; Chemistry, Physical; Chromans; Dopamine Agonists; Drug Design; Ergolines; Indoles; Ligands; Lisuride; Models, Molecular; Phenanthridines; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1995 |
Discriminative stimulus effects of cocaine in squirrel monkeys: lack of antagonism by the dopamine D2 partial agonists terguride, SDZ 208-911, and SDZ 208-912.
Topics: Animals; Cocaine; Discrimination, Psychological; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Lisuride; Male; Receptors, Dopamine D2; Saimiri | 1995 |
Terguride but not bromocriptine alleviated glucose tolerance abnormalities and hyperlipidaemia in obese and lean genetically hypertensive Koletsky rats.
Topics: Animals; Blood Pressure; Body Weight; Bromocriptine; Disease Models, Animal; Female; Glucose Intolerance; Hyperlipidemias; Hypertension; Insulin; Lipids; Lisuride; Male; Obesity; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Rats, Wistar; Sex Factors | 1994 |
Combination treatment of the partial D2 agonist terguride with the D1 agonist SKF 82958 in 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine-lesioned parkinsonian cynomolgus monkeys.
Topics: Animals; Benzazepines; Dopamine Agonists; Drug Therapy, Combination; Lisuride; Macaca fascicularis; MPTP Poisoning; Parkinson Disease; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1995 |
High-performance liquid chromatographic determination of terguride in solid dosage forms and plasma.
Topics: Animals; Chromatography, High Pressure Liquid; Dopamine Agonists; Ergot Alkaloids; Lisuride; Rats; Tablets | 1995 |
Terguride in fluctuating parkinsonian patients: a double-blind study versus placebo.
Topics: Adult; Aged; Dopamine; Dopamine Agents; Double-Blind Method; Drug Therapy, Combination; Drug Tolerance; Female; Humans; Levodopa; Lisuride; Male; Middle Aged; Parkinson Disease; Placebos | 1993 |
Terguride as a new anti-hyperprolactinemic agent: characterization in rats and dogs in comparison with bromocriptine.
Topics: Animals; Bromocriptine; Dogs; Dopamine Agents; Estradiol; Female; Glutathione; Hyperprolactinemia; Lactation; Lisuride; Luteinizing Hormone; Male; Motor Activity; Pituitary Neoplasms; Prolactinoma; Rats; Rats, Wistar; Receptors, Dopamine D2; Reserpine; Stereotyped Behavior; Vomiting | 1993 |
Effects of terguride, a partial D2 agonist, on MPTP-lesioned parkinsonian cynomolgus monkeys.
Topics: Aggression; Analysis of Variance; Animals; Apomorphine; Behavior, Animal; Dopamine Agents; Haloperidol; Lisuride; Macaca fascicularis; Motor Activity; MPTP Poisoning; Parkinson Disease, Secondary; Receptors, Dopamine D2; Time Factors | 1993 |
Effects of several partial dopamine D2 receptor agonists in Cebus apella monkeys previously treated with haloperidol.
Topics: Administration, Oral; Amphetamine; Animals; Antipsychotic Agents; Behavior, Animal; Benzothiazoles; Cebus; Disease Models, Animal; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dyskinesia, Drug-Induced; Dystonia; Ergolines; Female; Haloperidol; Lisuride; Male; Piperidines; Pramipexole; Quinpirole; Raclopride; Salicylamides; Thiazoles | 1993 |
Terguride for dyskinesias.
Topics: Dopamine Agents; Humans; Levodopa; Lisuride; Parkinson Disease | 1993 |
[Effects of terguride, an ergot alkaloid derivative, on the central nervous system: biochemical and behavioral studies].
Topics: Animals; Catalepsy; Ergot Alkaloids; Female; Guinea Pigs; Lisuride; Male; Mice; Motor Activity; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Dopamine; Receptors, Serotonin; Stereotyped Behavior; Yawning | 1993 |
Stable expression of human cytochrome P450 3A4 in V79 cells and its application for metabolic profiling of ergot derivatives.
Topics: Animals; Cell Line; Cells, Cultured; Cloning, Molecular; Cricetinae; Cricetulus; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Dopamine Agonists; Fibroblasts; Gene Expression Regulation, Enzymologic; Genetic Vectors; Humans; Lisuride; Liver; Mixed Function Oxygenases; Plasmids; Polymerase Chain Reaction; Testosterone; Transcription, Genetic; Transfection | 1995 |
Multiple regression analysis of parameters of lipid and glycide metabolism in obese and lean genetically hypertensive Koletsky rats under long lasting terguride treatment.
Topics: Animals; Dopamine Agonists; Female; Glucose; Glucose Tolerance Test; Hypertension; Insulin; Lisuride; Male; Obesity; Rats; Rats, Inbred SHR; Regression Analysis; Triglycerides | 1996 |
Glucose intolerance induced by oligemic brain hypoxia: the effect of terguride.
Topics: Animals; Blood Glucose; Body Water; Brain Chemistry; Brain Edema; Dopamine Agonists; Female; Glucose Intolerance; Hypoxia, Brain; Insulin; Lisuride; Rats; Rats, Inbred SHR; Rats, Wistar | 1997 |
Effects of bromocriptine and terguride on cell proliferation and apoptosis in the estrogen-stimulated anterior pituitary gland of the rat.
Topics: Animals; Apoptosis; Bromocriptine; Cell Division; Cell Migration Inhibition; Dopamine Agonists; Estradiol; Female; Hormone Antagonists; Lisuride; Neoplastic Cells, Circulating; Pituitary Gland; Pituitary Neoplasms; Prolactinoma; Proliferating Cell Nuclear Antigen; Rats; Rats, Wistar | 1997 |
Effect of long lasting terguride treatment on mutual relationship between glycide and lipid parameters in SHR/N-cp Koletsky rats.
Topics: Animals; Blood Glucose; Dopamine Agonists; Erythrocytes; Female; Glucose Tolerance Test; Hypertension; Insulin; Lisuride; Male; Obesity; Rats; Rats, Inbred SHR; Triglycerides | 1998 |
Independence of estrogen-induced pituitary proliferation on local IGF-I mRNA and EGF mRNA expression. Modifying effects of tamoxifen and terguride.
Topics: Animals; Dopamine Agonists; Epidermal Growth Factor; Estradiol; Estrogen Antagonists; Gene Expression Regulation; Hyperplasia; Insulin-Like Growth Factor I; Lisuride; Male; Organ Size; Pituitary Gland; Rats; Rats, Wistar; RNA, Messenger; Tamoxifen | 1998 |
Ambivalent effect of long lasting terguride treatment on genetically based glycide and lipid metabolism abnormalities in SHR/N-cp Koletsky rats.
Topics: Animals; Blood Glucose; Dopamine Agonists; Female; Hypertension; Insulin; Lipids; Lisuride; Male; Obesity; Rats; Rats, Inbred SHR; Rats, Inbred Strains | 1998 |
Effect of terguride on insulin binding, insulinaemia, glucose tolerance and hyperlipaemia in lean SHR Koletsky rats.
Topics: Animals; Body Weight; Dopamine Agonists; Eating; Erythrocytes; Female; Glucose Tolerance Test; Hyperlipidemias; Insulin; Lisuride; Male; Rats; Rats, Inbred SHR | 1997 |
Characterization of the effects of the partial dopamine agonist terguride on cocaine self-administration in the rat.
Topics: Animals; Cocaine; Dopamine Agonists; Dose-Response Relationship, Drug; Lisuride; Male; Rats; Rats, Wistar; Reinforcement, Psychology; Self Administration | 1998 |
Pharmacological effects of BAM-1120, a novel ergoline derivative, on central dopaminergic functions in rats.
Topics: Animals; Bromocriptine; Dopamine; Dopamine Agents; Dopamine Agonists; Ergolines; Estradiol; Female; Hyperprolactinemia; Lisuride; Male; Rats; Rats, Wistar; Reserpine; Rotation; Stereotyped Behavior; Sympathectomy, Chemical; Sympatholytics | 1998 |
Muscle GLUT-4 and insulin binding to erythrocytes and to adipose, liver and muscle tissue in genetically hypertensive obese rats and in their lean siblings: effect of long lasting terguride treatment.
Topics: Adipose Tissue; Animals; Erythrocytes; Female; Glucose Transporter Type 4; Hypertension; Insulin; Lisuride; Liver; Male; Monosaccharide Transport Proteins; Muscle Proteins; Muscle, Skeletal; Obesity; Rats; Rats, Inbred SHR | 1998 |
Hyperprolactinemia in obese as well as in lean females of Koletsky rats: effect of long lasting terguride treatment.
Topics: Animals; Body Weight; Dopamine Agonists; Female; Hyperprolactinemia; Hypertension; Insulin; Lipids; Lisuride; Male; Obesity; Prolactin; Rats; Rats, Inbred SHR; Rats, Wistar | 1998 |
[Combined therapy of acromegaly with a combination of lanreotide and terguride].
Topics: Acromegaly; Adult; Carrier Proteins; Dopamine Agonists; Drug Therapy, Combination; Female; Growth Hormone; Humans; Insulin-Like Growth Factor Binding Protein 3; Insulin-Like Growth Factor I; Lisuride; Male; Middle Aged; Peptides, Cyclic; Somatostatin | 2000 |
Clinical features and medical treatment of male prolactinomas.
Topics: Adult; Bromocriptine; Decompression, Surgical; Dopamine Agonists; Hormone Antagonists; Humans; Libido; Lisuride; Male; Middle Aged; Optic Chiasm; Pituitary Neoplasms; Prolactinoma; Retrospective Studies; Treatment Outcome; Visual Fields | 2001 |
Terguride attenuates prolactin levels and ameliorates insulin sensitivity and insulin binding in obese spontaneously hypertensive rats.
Topics: Adipose Tissue; Animals; Blood Glucose; Dopamine Agonists; Female; Hypertension; Insulin; Insulin Resistance; Lisuride; Male; Obesity; Prolactin; Rats; Rats, Inbred SHR | 2001 |
A dopamine partial agonist and antagonist block amphetamine self-administration in a progressive ratio schedule.
Topics: Amphetamine; Animals; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Infusions, Intravenous; Lisuride; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Reinforcement Schedule; Salicylamides; Self Administration | 2001 |
Dopamine partial agonist reverses amphetamine withdrawal in rats.
Topics: Amphetamine; Animals; Conditioning, Operant; Dopamine Agonists; Dopamine Uptake Inhibitors; Lisuride; Male; Motivation; Rats; Rats, Wistar; Substance Withdrawal Syndrome | 2001 |
Clustered ergot alkaloids modulate cell-mediated cytotoxicity.
Topics: Adjuvants, Immunologic; Animals; Carbamates; Dimerization; Drug Evaluation, Preclinical; Ergolines; Female; Humans; Immunosuppressive Agents; Killer Cells, Natural; Lisuride; Mice; Mice, Inbred BALB C; Spleen; Structure-Activity Relationship; Tumor Cells, Cultured | 2002 |
Terguride treatment attenuated prolactin release and enhanced insulin receptor affinity and GLUT 4 content in obese spontaneously hypertensive female, but not male rats.
Topics: Animals; Female; Glucose Transporter Type 4; Insulin; Lisuride; Male; Monosaccharide Transport Proteins; Muscle Proteins; Obesity; Prolactin; Protein Binding; Rats; Rats, Inbred SHR; Receptor, Insulin; Sex Factors | 2002 |
[Results of treatment for male prolactinomas].
Topics: Adult; Bromocriptine; Dopamine Agonists; Humans; Lisuride; Magnetic Resonance Imaging; Male; Middle Aged; Pituitary Apoplexy; Pituitary Neoplasms; Prolactin; Prolactinoma | 2002 |
Suppression of cocaine- and food-maintained behavior by the D2-like receptor partial agonist terguride in squirrel monkeys.
Topics: Animals; Behavior, Animal; Benzamides; Cocaine; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Food; Injections, Intravenous; Lisuride; Male; Motor Activity; Muscle Rigidity; Quinpirole; Receptors, Dopamine D2; Reinforcement Schedule; Reward; Saimiri | 2003 |
Inhibition of growth hormone excess reduces insulin resistance and ovarian dysfunction in a lean case of polycystic ovary syndrome with a growth-hormone-producing pituitary adenoma.
Topics: Acanthosis Nigricans; Acromegaly; Adenoma; Adult; Bromocriptine; Dopamine Agents; Female; Glucose Tolerance Test; Human Growth Hormone; Humans; Insulin; Insulin Resistance; Insulin-Like Growth Factor I; Lisuride; Magnetic Resonance Imaging; Menstrual Cycle; Ovary; Pancreatic Function Tests; Pituitary Function Tests; Pituitary Neoplasms; Polycystic Ovary Syndrome; Theca Cells | 2003 |
[Pharmacokinetic/pharmacodynamic analysis of anti-hyperprolactinemic effect of terguride based on dopamine D2 receptor occupancy].
Topics: Administration, Oral; Drug Administration Schedule; Humans; Hyperprolactinemia; Lisuride; Models, Biological; Pituitary Gland; Receptors, Dopamine D2; Retrospective Studies | 2003 |
Effects of a partial dopamine D2-like agonist on the cocaine-induced behavioral sensitization of preweanling rats.
Topics: Animals; Animals, Newborn; Cocaine; Dopamine Agonists; Dose-Response Relationship, Drug; Female; Lisuride; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Weaning | 2003 |
Pergolide, terguride and N,N'-spacer-linked oligomers of both interact with 5-HT2A receptors of rat tail artery.
Topics: Animals; Arteries; Dimerization; Dopamine Agonists; Dose-Response Relationship, Drug; Lisuride; Male; Peptide Fragments; Pergolide; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Serotonin; Tail; Vasoconstriction | 2004 |
Buprenorphine and a CRF1 antagonist block the acquisition of opiate withdrawal-induced conditioned place aversion in rats.
Topics: Acamprosate; Analgesics, Opioid; Animals; Antidepressive Agents, Second-Generation; Avoidance Learning; Buprenorphine; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Implants; Fluoxetine; Lisuride; Male; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome; Taurine | 2005 |
Effects of terguride treatment on glucose abnormalities induced by ischemic brain damage in SHR/N-cp lean Koletsky strain and in rats of Wistar strain.
Topics: Animals; Area Under Curve; Brain Ischemia; Dopamine Agonists; Female; Glucose; Glucose Tolerance Test; Lisuride; Male; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Rats, Wistar | 2004 |
The partial D2-like dopamine receptor agonist terguride acts as a functional antagonist in states of high and low dopaminergic tone: evidence from preweanling rats.
Topics: Animals; Animals, Newborn; Apomorphine; Body Weight; Corpus Striatum; Dextroamphetamine; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Hyperkinesis; Lisuride; Methyltyrosines; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Substance Withdrawal Syndrome; Tyrosine 3-Monooxygenase | 2005 |
Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic.
Topics: Animals; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; DNA, Complementary; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Humans; Lisuride; Piperazines; Piperidines; Quinolones; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Risperidone; Transfection; Tritium | 2005 |
Influence of steric hindrance on enantioseparation of Dns-amino acids and pesticides on terguride based chiral selectors in capillary electrophoresis.
Topics: Amino Acids; Electrophoresis, Capillary; Lisuride; Mandelic Acids; Molecular Structure; Optical Rotation; Pesticides; Stereoisomerism | 2005 |
Effects of a partial D2-like receptor agonist on striatal dopamine autoreceptor functioning in preweanling rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Animals, Newborn; Autoreceptors; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Enzyme Inhibitors; Haloperidol; Hydrazines; Lisuride; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reserpine | 2006 |
The partial dopamine D2-like receptor agonist terguride functions as an agonist in preweanling rats after a 5-day reserpine regimen.
Topics: alpha-Methyltyrosine; Animals; Behavior, Animal; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enzyme Inhibitors; Lisuride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reserpine | 2006 |
Effects of terguride, ropinirole, and acetyl-L-carnitine on methamphetamine withdrawal in the rat.
Topics: Acetylcarnitine; Animals; Antidepressive Agents; Conditioning, Operant; Dopamine Agonists; Indoles; Lisuride; Male; Methamphetamine; Motivation; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Sweetening Agents | 2006 |
In vitro characterization of SLV308 (7-[4-methyl-1-piperazinyl]-2(3H)-benzoxazolone, monohydrochloride): a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist.
Topics: Animals; Benzoxazoles; Binding, Competitive; Brain; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Lisuride; Male; Molecular Structure; Parkinson Disease; Piperazines; Quinpirole; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Fusion Proteins; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists | 2006 |
In vitro functional characteristics of dopamine D2 receptor partial agonists in second and third messenger-based assays of cloned human dopamine D2Long receptor signalling.
Topics: Animals; Antipsychotic Agents; Aripiprazole; Calcium Signaling; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Immunoblotting; Lisuride; MAP Kinase Signaling System; Microscopy, Confocal; Mitogen-Activated Protein Kinase 1; Phosphorylation; Piperazines; Piperidines; Quinolones; Raclopride; Receptors, Dopamine D2; Schizophrenia; Time Factors; Transfection | 2007 |
Long-term serotonin effects in the rat are prevented by terguride.
Topics: 3T3 Cells; Animals; Carcinoid Heart Disease; Cell Proliferation; Echocardiography; Epidermis; Female; Heart; Injections, Subcutaneous; Lisuride; Mice; Myocardium; Organ Size; Rats; Rats, Sprague-Dawley; Serotonin; Skin; Stomach | 2007 |
Effects of aripiprazole and terguride on dopamine synthesis in the dorsal striatum and medial prefrontal cortex of preweanling rats.
Topics: Animals; Animals, Newborn; Aripiprazole; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Dopamine Agonists; Lisuride; Piperazines; Prefrontal Cortex; Quinolones; Rats; Rats, Sprague-Dawley | 2008 |
[A case of ruptured internal carotid artery aneurysm mimicking pituitary apoplexy].
Topics: Carotid Artery Diseases; Carotid Artery, Internal; Cerebral Hemorrhage; Diagnosis, Differential; Embolization, Therapeutic; Female; Humans; Intracranial Aneurysm; Lisuride; Middle Aged; Pituitary Apoplexy; Pituitary Neoplasms; Rupture, Spontaneous | 2007 |
The effect of terguride in carbon tetrachloride-induced liver fibrosis in rat.
Topics: Actins; Animals; Blood Chemical Analysis; Carbon Tetrachloride; Female; Immunohistochemistry; Lisuride; Liver; Liver Cirrhosis, Experimental; Organ Size; Rats; Rats, Sprague-Dawley; Serotonin Antagonists | 2008 |
Co-administration of the partial dopamine D2 agonist terguride with L-dopa attenuates L-dopa-induced locomotor sensitization in hemiparkinsonian mice.
Topics: Adenosine A2 Receptor Antagonists; Animals; Antiparkinson Agents; Benzazepines; Caffeine; Corpus Striatum; Dopamine Agonists; Drug Therapy, Combination; Guanosine 5'-O-(3-Thiotriphosphate); Levodopa; Lisuride; Male; Mice; Mice, Inbred C57BL; Motor Activity; Oxidopamine; Parkinson Disease, Secondary; Random Allocation; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulfur Radioisotopes | 2009 |
Increased expression of 5-hydroxytryptamine2A/B receptors in idiopathic pulmonary fibrosis: a rationale for therapeutic intervention.
Topics: Animals; Bleomycin; Disease Models, Animal; Drug Evaluation, Preclinical; Female; Humans; Lisuride; Lung; Male; Mice; Mice, Inbred C57BL; Pulmonary Fibrosis; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Serotonin 5-HT2 Receptor Antagonists; Serotonin Plasma Membrane Transport Proteins | 2010 |
The dopamine D(2) partial agonist and antagonist terguride decreases heroin self-administration on fixed- and progressive-ratio schedules.
Topics: Animals; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Heroin Dependence; Lisuride; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reinforcement Schedule; Self Administration; Substance Abuse, Intravenous; Sucrose | 2010 |
Terguride ameliorates monocrotaline-induced pulmonary hypertension in rats.
Topics: Adult; Animals; Cell Proliferation; Cells, Cultured; Dopamine Agonists; Female; Humans; Hypertension, Pulmonary; Lisuride; Lung; Lung Transplantation; Male; Monocrotaline; Muscle, Smooth, Vascular; Pulmonary Artery; Rats; Serotonin 5-HT2 Receptor Antagonists | 2011 |
Antiserotonergic properties of terguride in blood vessels, platelets, and valvular interstitial cells.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenosine Diphosphate; Animals; Aortic Valve; Blood Vessels; Cells, Cultured; Collagen; Coronary Vessels; Dose-Response Relationship, Drug; Heart Valves; Humans; In Vitro Techniques; Inhibitory Concentration 50; Ketanserin; Kinetics; Lisuride; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitral Valve; Phosphorylation; Platelet Aggregation; Pulmonary Artery; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Sus scrofa; Vasoconstriction; Vasodilation | 2012 |
Pharmacological profile of 2-bromoterguride at human dopamine D2, porcine serotonin 5-hydroxytryptamine 2A, and α2C-adrenergic receptors, and its antipsychotic-like effects in rats.
Topics: Animals; Antipsychotic Agents; CHO Cells; Coronary Vessels; Cricetinae; Cricetulus; Dopamine Agonists; HEK293 Cells; Humans; Lisuride; Male; Motor Activity; Organ Culture Techniques; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Dopamine D2; Swine | 2013 |
Behavioral effects of dopamine receptor inactivation in the caudate-putamen of preweanling rats: role of the D2 receptor.
Topics: Aging; Alkylating Agents; Animals; Apomorphine; Benzazepines; Caudate Nucleus; Dimethyl Sulfoxide; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Lisuride; Male; Motor Activity; Putamen; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Weaning | 2014 |
5-HT7 receptor antagonism (SB-269970) attenuates bleomycin-induced pulmonary fibrosis in rats via downregulating oxidative burden and inflammatory cascades and ameliorating collagen deposition: Comparison to terguride.
Topics: Animals; Bleomycin; Collagen; Down-Regulation; Inflammation; Interleukin-6; Lisuride; Lung; Male; Oxidative Stress; Phenols; Pulmonary Fibrosis; Rats; Receptors, Serotonin; Sulfonamides; Tumor Necrosis Factor-alpha; Water | 2017 |
Effects of different serotonin receptor subtype antagonists on the development of cardiac allograft vasculopathy in murine aortic allografts.
Topics: Animals; Aorta; Cell Proliferation; Female; Graft Rejection; Heart Transplantation; Humans; Indoles; Lisuride; Male; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Models, Animal; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Succinates; Transendothelial and Transepithelial Migration; Transplantation, Homologous; Urea | 2018 |
5-HT
Topics: Adult; Cells, Cultured; Extracellular Matrix Proteins; Extracellular Signal-Regulated MAP Kinases; Female; Fibroblasts; Fibrosis; Gene Expression Regulation; Humans; Indoles; Lisuride; Phenotype; Phosphorylation; Receptor, Serotonin, 5-HT2B; Scleroderma, Systemic; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Signal Transduction; Skin; STAT3 Transcription Factor; Transforming Growth Factor beta1; Urea | 2018 |