Compounds > levocabastine
Page last updated: 2024-08-23

levocabastine and sr 48692

levocabastine has been researched along with sr 48692 in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (31.25)18.2507
2000's6 (37.50)29.6817
2010's5 (31.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Botto, JM; Chabry, J; Mazella, J; Sarret, P; Vincent, JP1
Barroso, S; Kitabgi, P; Labbé-Jullié, C; Martinez, J; Richard, F1
Gendron, L; Giddings, AM; Gilmour, BP; Longpre, JM; Olepu, S; Runyon, SP; Sarret, P; Thomas, JB; Warner, KR; Wiethe, RW; Zhang, Y1
Alonso, R; Beaudet, A; Faure, MP; Nouel, D; Quirion, R; St Pierre, JA1
Botto, JM; Guillemare, E; Mazella, J; Vincent, JP1
Forgez, P; Lombet, A; Rostène, W; Yamada, M1
Laissue, JA; Reubi, JC; Schaer, JC; Waser, B1
Greengard, P; Higashi, H; Maeda, H; Matsuyama, S; Nishi, A1
Garcia-Marin, L; Jensen, RT; Leyton, J; Moody, TW1
Beaudet, A; Gallo-Payet, N; Gendron, L; Kilian, P; Nguyen, HM; Payet, MD; Sarret, P1
Fukui, R; Higashi, H; Matsuyama, S; Nishi, A1
Bredeloux, P; Costentin, J; Dubuc, I1
Abderrahmani, A; Béraud-Dufour, S; Brau, F; Coppola, T; Mazella, J; Noel, J; Waeber, G1
Arnaiz, GR; Ordieres, MG; Rosin, C1
Hugel, S; Kadiri, N; Rodeau, JL; Schlichter, R1
Bogdański, P; Krauss, H; Maćkowiak, P; Nowak, D; Piątek, J1

Other Studies

16 other study(ies) available for levocabastine and sr 48692

ArticleYear
Stable expression of the mouse levocabastine-sensitive neurotensin receptor in HEK 293 cell line: binding properties, photoaffinity labeling, and internalization mechanism.
    Biochemical and biophysical research communications, 1998, Feb-13, Volume: 243, Issue:2

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Cell Line; Endocytosis; Gene Expression Regulation; Humans; Iodine Radioisotopes; Kinetics; Mice; Molecular Sequence Data; Neurotensin; Peptides; Photoaffinity Labels; Piperidines; Protein Binding; Receptors, Neurotensin; Signal Transduction; Transfection

1998
Agonism, inverse agonism, and neutral antagonism at the constitutively active human neurotensin receptor 2.
    Molecular pharmacology, 2001, Volume: 60, Issue:6

    Topics: Amino Acid Sequence; Animals; COS Cells; Histamine H1 Antagonists; Humans; Molecular Sequence Data; Neurotensin; Piperidines; Pyrazoles; Quinolines; Receptors, Neurotensin; Sequence Homology, Amino Acid; Transfection

2001
Identification of 1-({[1-(4-fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane carboxylic acid as a selective nonpeptide neurotensin receptor type 2 compound.
    Journal of medicinal chemistry, 2014, Jun-26, Volume: 57, Issue:12

    Topics: Analgesics; Animals; Calcium; CHO Cells; Cricetulus; Cyclohexanecarboxylic Acids; Drug Partial Agonism; Pyrazoles; Radioligand Assay; Rats; Receptors, Neurotensin; Structure-Activity Relationship

2014
Differential binding profile and internalization process of neurotensin via neuronal and glial receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Mar-01, Volume: 17, Issue:5

    Topics: Animals; Animals, Newborn; Binding Sites; Cells, Cultured; Cerebral Cortex; Coculture Techniques; Endocytosis; GTP-Binding Proteins; Mesencephalon; Nerve Tissue Proteins; Neuroglia; Neurons; Neurotensin; Piperidines; Protein Binding; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Signal Transduction; Tegmentum Mesencephali; Tyrosine 3-Monooxygenase

1997
Effects of SR 48692 on neurotensin-induced calcium-activated chloride currents in the Xenopus oocyte expression system: agonist-like activity on the levocabastine-sensitive neurotensin receptor and absence of antagonist effect on the levocabastine insensi
    Neuroscience letters, 1997, Feb-28, Volume: 223, Issue:3

    Topics: Animals; Calcium; Chlorides; Electric Conductivity; Female; Mice; Neurotensin; Oocytes; Piperidines; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin

1997
Distinct functional characteristics of levocabastine sensitive rat neurotensin NT2 receptor expressed in Chinese hamster ovary cells.
    Life sciences, 1998, Volume: 62, Issue:23

    Topics: Animals; Calcium; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Neurotensin; Oligopeptides; Piperidines; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin; Signal Transduction; Transfection

1998
Neurotensin receptors in human neoplasms: high incidence in Ewing's sarcomas.
    International journal of cancer, 1999, Jul-19, Volume: 82, Issue:2

    Topics: Animals; Bone Neoplasms; Humans; Neoplasm Proteins; Neoplasms; Neurotensin; Organ Specificity; Peptide Fragments; Piperidines; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin; RNA, Messenger; RNA, Neoplasm; Sarcoma, Ewing

1999
Neurotensin regulates DARPP-32 thr34 phosphorylation in neostriatal neurons by activation of dopamine D1-type receptors.
    Journal of neurochemistry, 2002, Volume: 81, Issue:2

    Topics: Animals; Cobalt; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Glutamine; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Phosphorylation; Piperidines; Pyrazoles; Quinolines; Receptors, Dopamine D1; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin

2002
Neurotensin causes tyrosine phosphorylation of focal adhesion kinase in lung cancer cells.
    European journal of pharmacology, 2002, May-10, Volume: 442, Issue:3

    Topics: Binding, Competitive; Cell Division; Cytochalasin D; Dose-Response Relationship, Drug; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Humans; Lung Neoplasms; Neurotensin; Nucleic Acid Synthesis Inhibitors; Peptide Fragments; Phosphorylation; Piperidines; Protein-Tyrosine Kinases; Pyrazoles; Quinolines; Receptors, Neurotensin; Tumor Cells, Cultured; Tyrosine

2002
Pharmacology and functional properties of NTS2 neurotensin receptors in cerebellar granule cells.
    The Journal of biological chemistry, 2002, Sep-27, Volume: 277, Issue:39

    Topics: Aniline Compounds; Animals; Binding Sites; Binding, Competitive; Calcium; Cerebellum; Clathrin; Cytosol; Dose-Response Relationship, Drug; Fluorescent Dyes; Histamine H1 Antagonists; Inhibitory Concentration 50; Male; Microscopy, Confocal; Piperidines; Polymerase Chain Reaction; Protein Binding; Pyrazoles; Quinolines; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Receptors, Neurotensin; Receptors, Presynaptic; Reverse Transcriptase Polymerase Chain Reaction; RNA; Time Factors; Xanthenes

2002
Regulation of DARPP-32 Thr75 phosphorylation by neurotensin in neostriatal neurons: involvement of glutamate signalling.
    The European journal of neuroscience, 2003, Volume: 18, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Anesthetics, Local; Animals; Benzazepines; Dizocilpine Maleate; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Glutamic Acid; Histamine H1 Antagonists; Immunoblotting; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Piperidines; Pyrazoles; Quinolines; Raclopride; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin; Threonine; Time Factors

2003
Interactions between NTS2 neurotensin and opioid receptors on two nociceptive responses assessed on the hot plate test in mice.
    Behavioural brain research, 2006, Dec-15, Volume: 175, Issue:2

    Topics: Analgesia; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Histamine H1 Antagonists, Non-Sedating; Injections, Intraventricular; Ligands; Male; Mice; Morphine; Neurotensin; Pain Threshold; Piperidines; Pyrazoles; Quinolines; Reaction Time; Receptors, Neurotensin; Receptors, Opioid

2006
Neurotensin is a regulator of insulin secretion in pancreatic beta-cells.
    The international journal of biochemistry & cell biology, 2010, Volume: 42, Issue:10

    Topics: Animals; Calcium Signaling; Cell Line; Cyclic AMP-Dependent Protein Kinases; Cytoprotection; Enzyme Activation; Insulin; Insulin Secretion; Insulin-Secreting Cells; Neurotensin; Piperidines; Protein Kinase C-alpha; Protein Kinase C-epsilon; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin

2010
Neurotensin decreases high affinity [3H]-ouabain binding to cerebral cortex membranes.
    Regulatory peptides, 2011, Dec-10, Volume: 172, Issue:1-3

    Topics: Animals; Cerebral Cortex; Male; Neurotensin; Ouabain; Piperidines; Protein Binding; Pyrazoles; Quinolines; Rats; Rats, Wistar; Receptors, Neurotensin

2011
Neurotensin inhibits background K+ channels and facilitates glutamatergic transmission in rat spinal cord dorsal horn.
    The European journal of neuroscience, 2011, Volume: 34, Issue:8

    Topics: Animals; Benzophenanthridines; Excitatory Postsynaptic Potentials; Glutamic Acid; Neurotensin; Oligopeptides; Patch-Clamp Techniques; Pertussis Toxin; Piperidines; Posterior Horn Cells; Potassium Channels; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Signal Transduction; Synapses; Synaptic Transmission

2011
In vivo investigations of neurotensin receptors in adipocytes, hepatocytes and enterocytes of rat.
    Annals of agricultural and environmental medicine : AAEM, 2011, Volume: 18, Issue:2

    Topics: Adipocytes; Adipose Tissue; Animals; Antigen-Antibody Reactions; Cell Membrane; Enterocytes; Hepatocytes; Histamine H1 Antagonists, Non-Sedating; Intestine, Small; Iodine Radioisotopes; Isotope Labeling; Liver; Male; Neurotensin; Piperidines; Pyrazoles; Quinolines; Rats; Rats, Wistar; Receptors, Neurotensin

2011