Page last updated: 2024-08-23

levocabastine and sr 142948

levocabastine has been researched along with sr 142948 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gendron, L; Giddings, AM; Gilmour, BP; Longpre, JM; Olepu, S; Runyon, SP; Sarret, P; Thomas, JB; Warner, KR; Wiethe, RW; Zhang, Y1
Boigegrain, R; Durant, F; Gully, D; Labeeuw, B; Longfils, G; Quéré, L1
Greengard, P; Higashi, H; Maeda, H; Matsuyama, S; Nishi, A1
Fukui, R; Higashi, H; Matsuyama, S; Nishi, A1

Other Studies

4 other study(ies) available for levocabastine and sr 142948

ArticleYear
Identification of 1-({[1-(4-fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane carboxylic acid as a selective nonpeptide neurotensin receptor type 2 compound.
    Journal of medicinal chemistry, 2014, Jun-26, Volume: 57, Issue:12

    Topics: Analgesics; Animals; Calcium; CHO Cells; Cricetulus; Cyclohexanecarboxylic Acids; Drug Partial Agonism; Pyrazoles; Radioligand Assay; Rats; Receptors, Neurotensin; Structure-Activity Relationship

2014
X-ray structural characterization of SR 142948, a novel potent synthetic neurotensin receptor antagonist.
    Bioorganic & medicinal chemistry letters, 1998, Mar-17, Volume: 8, Issue:6

    Topics: Animals; Crystallography, X-Ray; Mice; Models, Molecular; Piperidines; Protein Conformation; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin

1998
Neurotensin regulates DARPP-32 thr34 phosphorylation in neostriatal neurons by activation of dopamine D1-type receptors.
    Journal of neurochemistry, 2002, Volume: 81, Issue:2

    Topics: Animals; Cobalt; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Glutamine; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Phosphorylation; Piperidines; Pyrazoles; Quinolines; Receptors, Dopamine D1; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin

2002
Regulation of DARPP-32 Thr75 phosphorylation by neurotensin in neostriatal neurons: involvement of glutamate signalling.
    The European journal of neuroscience, 2003, Volume: 18, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Anesthetics, Local; Animals; Benzazepines; Dizocilpine Maleate; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Glutamic Acid; Histamine H1 Antagonists; Immunoblotting; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Piperidines; Pyrazoles; Quinolines; Raclopride; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin; Threonine; Time Factors

2003